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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
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11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 44 / 236
small molecule | CAS: 1224-78-8

Deskripsi belum tersedia.

Kategori:
AlkenesBiological FactorsCarotenoids +9
Waktu Paruh-
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Genetik -
Anifrolumab Approved DB11976
biotech | CAS: 1326232-46-5

Anifrolumab, or MEDI-546, is a type 1 interferon receptor (IFNAR) inhibiting IgG1? monoclonal antibody indicated in the treatment of adults with moderate to severe systemic lupus erythematosus.[A237074,L34929] The standard therapy for systemic lupus erythemat…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Interferon alpha/beta receptor 1
Waktu ParuhThe serum eliminati…
Vol. DistribusiBased on population…
KlirensFollowing the admin…
Genetik -
Aniline DB06728
small molecule | CAS: 62-53-3

Aniline, phenylamine or aminobenzene is an organic compound with the formula C6H5NH2. Consisting of an amine attached to a benzene ring, aniline is the prototypical aromatic amine. Being a precursor to many industrial chemicals, its main use is in the manufac…

Kategori:
AminesCarcinogensCytochrome P-450 CYP2E1 Substrates +3
Target Protein:
Kallikrein-1Albumin
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

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Aniracetam DB04599
small molecule | CAS: 72432-10-1

Compound with anti-depressive properties used as a mental performance enhancer.

Kategori:
Antidepressive AgentsCentral Nervous System AgentsCentral Nervous System Depressants +6
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2AGlutamate receptor 2 +1
Waktu Paruh1-2.5 hours
Vol. Distribusi-
Klirens-
Genetik -
Anise oil DB15776
biotech | CAS: 8007-70-3

Deskripsi belum tersedia.

Kategori:
AngiospermsApiaceaeBiological Products +10
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Anisindione Approved DB01125
small molecule | CAS: 117-37-3

Anisindione is a synthetic anticoagulant and an indanedione derivative. Its anticoagulant action is mediated through the inhibition of the vitamin K-mediated gamma-carboxylation of precursor proteins that are critical in forming the formation of active procoa…

Kategori:
IndansIndenes
Target Protein:
Vitamin K-dependent gamma-carboxylaseProthrombin
Waktu ParuhNot Known
Vol. Distribusi-
Klirens-
Genetik -
Anisodamine DB11785
small molecule | CAS: 55869-99-3

Anisodamine has been investigated for the treatment of Intestinal Diseases.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic Antagonists +29
Target Protein:
Beta-1 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anisomycin DB07374
small molecule | CAS: 22862-76-6

Anisomycin (sometimes known as flagecidin), is an antibiotic retrieved from the bacteria _Streptomyces griseolus_. This drug acts to inhibit bacterial protein and DNA synthesis.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntiparasitic Agents +5
Target Protein:
Ribosomal protein uL16-likeLarge ribosomal subunit protein uL13Large ribosomal subunit protein uL14 +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anisotropine methylbromide Approved DB00517
small molecule | CAS: 80-50-2

Anisotropine methylbromide is a quaternary ammonium compound. Its use as treatment adjunct in peptic ulcer has been replaced by the use of more effective agents. Depending on the dose, anisotropine methylbromide may reduce the motility and secretory activity …

Kategori:
Agents producing tachycardiaAlkaloidsAnticholinergic Agents +5
Target Protein:
Muscarinic acetylcholine receptor M5Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2 +1
Waktu ParuhNot Known
Vol. Distribusi-
Klirens-
Genetik -
Anistreplase Approved DB00029
biotech | CAS: 81669-57-0

Human tissue plasminogen activator, purified, glycosylated, 527 residues purified from CHO cells. Eminase is a lyophilized (freeze-dried) formulation of anistreplase, the p-anisoyl derivative of the primary Lys-plasminogen-streptokinase activator complex (a c…

Kategori:
Agents causing angioedemaAmino Acids, Peptides, and ProteinsAnticoagulants +15
Target Protein:
PlasminogenFibrinogen alpha chainPlasminogen activator inhibitor 1
Waktu Paruh-
Vol. Distribusi-
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Anivamersen DB16089
biotech | CAS: 959716-29-1

Anivamersen is under investigation in clinical trial NCT01848106 (A Study to Determine the Efficacy and Safety of REG1 Compared to Bivalirudin in Patients Undergoing PCI).

Kategori:
CoagulantsNucleic Acids, Nucleotides, and NucleosidesNucleotides +1
Waktu Paruh-
Vol. Distribusi-
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Anlotinib DB11885
small molecule | CAS: 1058156-90-3

Anlotinib has been investigated for the treatment of Non-small Cell Lung Cancer and Metastatic Colorectal Cancer.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Proto-oncogene tyrosine-protein kinase Src
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anpocogin DB06552
biotech

Recombinant nematode anticoagulant protein c2 (rNAPc2) is a specific inhibitor of tissue factor (TF)/factor VIIa complex with novel antithrombotic activity. [A175642]

Target Protein:
Coagulation factor VIITissue factorCoagulation factor X
Waktu ParuhOver 50 hours
Vol. Distribusi-
Klirens-
Genetik -
Anselamimab DB17492
biotech | CAS: 2414866-63-8

Deskripsi belum tersedia.

Waktu Paruh-
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Ansofaxine DB15052
small molecule | CAS: 916918-80-4

Ansofaxine is under investigation in clinical trial NCT02271412 (Multiple Ascending Dose Study in Healthy Subjects to Evaluate the Safety, Tolerability, and Pharmacokinetics of LY03005).

Waktu Paruh-
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Genetik -
Ansuvimab Approved DB16385
biotech | CAS: 2375952-29-5

Infection with pathogenic filoviruses, such as _Zaire ebolavirus_ (Ebola virus, EBOV), can cause severe hemorrhagic fever in humans, resulting in frequent outbreaks with case fatality rates as high as 90%.[A225933, A225938] Virtually all steps of the EBOV lif…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +13
Target Protein:
Envelope glycoprotein
Waktu ParuhThe half-life of an…
Vol. DistribusiThe steady-state vo…
KlirensThe clearance of an…
Genetik -
Antazoline Approved DB08799
small molecule | CAS: 91-75-8

Antazoline is a 1st generation antihistamine with anticholinergic activity. It is used to relieve nasal congestion. It is also formulated as eye drops with naphazoline to relieve allergic conjunctivitis.

Kategori:
Anti-Allergic AgentsAntiallergic Agents, Excl. CorticosteroidsAntihistamines for Systemic Use +8
Target Protein:
Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anthralin Approved DB11157
small molecule | CAS: 1143-38-0

Anthralin (1,8?dihydroxy?9anthrone, dithranol) is an older anti-psoriatic agent that was first synthesized as a derivative of chrysarobin, obtained from the araroba tree in Brazil over 100 years ago. Adverse effects of anthralin include irritation and discolo…

Kategori:
AnthracenesAntipsoriaticsAntipsoriatics for Topical Use +2
Target Protein:
Keratin, type II cytoskeletal 2 epidermalKeratin, type I cytoskeletal 12C-Jun-amino-terminal kinase-interacting protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Anthrax immune globulin is a human antibody given with antibiotics for the treatment of anthrax. It is derived from the plasma of humans immunized with BioThrax (adsorbed anthrax vaccine), which is then further purified. Available as the product Anthrasil (FD…

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsHuman Immunoglobulin +5
Target Protein:
Protective antigen
Waktu Paruh24.3 days
Vol. Distribusi5714.8 mL
Klirens174.2 mL/day
Genetik -
Anthrax vaccine Approved DB11003
biotech

Anthrax vaccine is a vaccine used for the pre- or post-exposure prophylaxis of disease in those at high risk of, suspected or confirmed exposure to *Bacillus anthracis*. It is subcutaneously or intramuscularly administered. It is derived from cell-free filtra…

Kategori:
Actively Acquired ImmunityAnthrax VaccinesBacterial Vaccines +6
Waktu ParuhLimited information…
Vol. DistribusiLimited information…
KlirensLimited information…
Genetik -
biotech

Integrins are important adhesion molecules that regulate tumor and endothelial cell survival, proliferation and migration. The integrin alpha5beta1 has been shown to play a critical role during angiogenesis. anti-alpha5beta1 integrin antibody inhibits angioge…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Deskripsi belum tersedia.

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Genetik -
biotech

Deskripsi belum tersedia.

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Genetik -
biotech

Deskripsi belum tersedia.

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biotech

A macrocyclic peptide (BMS-986189) with activity in binding and functional assays comparable to a PD-L1 antibody.

Kategori:
Immune Checkpoint Inhibitors
Target Protein:
Programmed cell death 1 ligand 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Anti-SARS-CoV-2 equine immunoglobulin fragments, also known as INOSARS, is a polyvalent passive immunization being tested in the clinical trial NCT04514302 (Safety and Efficacy of Anti-SARS-CoV-2 Equine Antibody Fragments (INOSARS) for Hospitalized Patients W…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Anti-SARS-CoV-2 IgY are chicken egg antibodies to SARS-CoV-2 which have the potential to provide temporary protection against the virus when administered as intranasal drops.[L27381] To create these antibodies, chickens are injected in the chest with the spik…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Hyperimmune immunoglobulin to SARS-CoV-2 (hIVIG) is obtained from the plasma of patients who recover from COVID-19 and develop neutralizing antibodies.[L27521] Anti-coronavirus immunoglobulin is derived from [COVID-19 convalescent plasma](https://go.drugbank.…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Anti-SARS-COV-2 REGN-COV2 is a combination of novel antibodies designed by Regeneron for both the prevention and treatment of SARS-COV-2, the virus that causes COVID-19. This drug is a combination of the antibodies REGN10933 and REGN10987, derived from human…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +10
Target Protein:
Spike glycoprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1628187-15-4

Antihemophilic Factor (Recombinant), PEGylated, was approved by the FDA in December 2016 as the product _Adynovate_ [FDA label]. Antihemophilic Factor (Recombinant), PEGylated, is a recombinant full-length human coagulation factor VIII (2,332 amino acids w…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +14
Target Protein:
von Willebrand factor
Waktu Paruh14.69 ± 3.79h for a…
Vol. DistribusiAt steady state: 0.…
Klirens2.27 ± 0.84 for adu…
Genetik -
Antihemophilic factor human Approved DB13192
biotech

Antihemophilic factor human, also known as Coagulation Factor VIII or Anti-Hemophilic Factor (AHF), is a non-recombinant, lyophilized concentrate of coagulation factor VIII, an endogenous protein and essential component of the coagulation cascade. Antihemophi…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +11
Target Protein:
Coagulation factor IXCoagulation factor X
Waktu ParuhThe mean half-life …
Vol. DistribusiThe pharmacokinetic…
KlirensThe reported cleara…
Genetik -
biotech | CAS: 139076-62-3

Human recombinant antihemophilic factor (AHF) or Factor VIII, 2332 residues, glycosylated, produced by CHO cells

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +12
Target Protein:
Coagulation factor XCoagulation factor IXvon Willebrand factor +8
Waktu Paruh8.4-19.3 hrs
Vol. Distribusi-
Klirens* 4.1 mL/h•kg [Prev…
Genetik -
Antimony DB13110
small molecule | CAS: 7440-36-0

Antimony has been used in trials studying the treatment of Cutaneous Leishmaniasis.

Kategori:
ElementsMetalloidsMetals +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 1315-04-4

Deskripsi belum tersedia.

Kategori:
Air PollutantsAnionsCough and Cold Preparations +9
Waktu Paruh-
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small molecule | CAS: 28300-74-5

Antimony potassium tartrate is a schistosomicide possibly useful against other parasites. It has irritant emetic properties and may cause lethal cardiac toxicity among other adverse effects.

Kategori:
AnthelminticsAnti-Infective AgentsAntiparasitic Agents +2
Waktu Paruh-
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Genetik -
small molecule | CAS: 91531-30-5

Antineoplaston A10 has been used in trials studying the treatment of Sarcoma, Lymphoma, Lung Cancer, Liver Cancer, and Kidney Cancer, among others.

Kategori:
AcetamidesAmidesBenzene Derivatives +1
Waktu Paruh-
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Genetik -
Antipain DB15251
small molecule | CAS: 37691-11-5

Antipain is a serine/cysteine protease inhibitor originally isolated from various strains of actinomycetes.[A214481] Early studies investigated the potential for antipain to alter DNA damage and chromosomal aberrations in irradiated cells or those treated wit…

Kategori:
Amino Acids, Peptides, and ProteinsEnzyme InhibitorsOligopeptides +2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Antithrombin Alfa Approved DB11166
biotech | CAS: 84720-88-7

Antithrombin Alfa is a recombinant antithrombin , an anticoagulant, that is used for the prevention of thromboembolic events in patients that have hereditary deficiency of antithrombin in high risk situations.

Kategori:
AnticoagulantsDecreased Coagulation Factor ActivityFactor Xa Inhibitors +2
Target Protein:
ProthrombinCoagulation factor X
Waktu ParuhDose of: 50IU/kg: …
Vol. DistribusiDose of: 50IU/kg: …
KlirensDose of: 50IU/kg: …
Genetik -
biotech | CAS: 1311281-25-0

Antithrombin gamma is under investigation in clinical trial NCT04182373 (KW-3357 Study in Patients With Early Onset Severe Preeclampsia).

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biotech | CAS: 308067-60-9

Rabbit anti-thymocyte globulin. Thymoglobulin is a polyclonal antibody that suppresses certain types of immune cells responsible for acute organ rejection in transplant patients. Thymoglobulin is a mixture of antibodies intended to bind to various cell surfac…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibody-Surface Protein Interactions +22
Target Protein:
Major histocompatibility complex class I-related gene proteinIntegrin alpha-LT-lymphocyte activation antigen CD86 +6
Waktu Paruh2-3 days, may incre…
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2636710-07-9

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
Waktu Paruh-
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Klirens-
Genetik -
ANX-005 DB16977
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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ANZ-100 DB05967
small molecule

Deskripsi belum tersedia.

Target Protein:
KiSS-1 receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Anzurstobart DB17547
biotech | CAS: 2543693-10-1

Anzurstobart is a monoclonal antibody directed against signal-regulatory protein alpha (SIRP?) on monocytes and macrophages to potently block the CD47-SIRP? interaction. It is being investigated for cancers.

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AO-176 DB18287
biotech

Deskripsi belum tersedia.

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AOC 1001 DB18620
biotech | CAS: 2653183-66-3

Delpacibart (AOC 1001) is being investigated in a global study for the treatment of Myotonic Dystrophy type 1 (DM1) in clinical trial NCT06411288

Waktu Paruh-
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AOD9604 DB06388
small molecule | CAS: 221231-10-3

AOD9604 is a synthetic analogue of the lipolytic domain of human growth hormone, being investigated for the treatment of obesity.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +8
Waktu Paruh-
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AP-001 DB18511
small molecule | CAS: 660430-03-5

Deskripsi belum tersedia.

Kategori:
Dietary FatsDietary Fats, UnsaturatedFats +6
Waktu Paruh-
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Genetik -
AP-101 DB17947
biotech

AP-101 is a recombinant human antibody directed against human misfolded superoxide dismutase 1.

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