Hasil Filter

11793

Total database: 17430
Struktur (SMILES)
8607 (73.0%)
Target
6418 (54.4%)
Genomik
102 (0.9%)
Referensi
11793 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (11793)

Halaman 44 / 236
Ardeparin Approved DB00407
small molecule | CAS: 9005-49-6

Ardeparin, marketed under the US trade name Normiflo, is a low molecular weight heparin (LMWH) anticoagulant used for the prevention of postoperative venous thrombosis. Ardeparin is derived via peroxide degradation of heparin extracted from porcine intestinal…

Kategori:
Agents causing hyperkalemiaAnticoagulantsCarbohydrates +7
Target Protein:
Antithrombin-IIIHeparin cofactor 2
Waktu ParuhElimination half-li…
Vol. Distribusi-
Klirens-
Genetik -
Arecoline DB04365
small molecule | CAS: 63-75-2

An alkaloid obtained from the betel nut (Areca catechu), fruit of a palm tree. It is an agonist at both muscarinic and nicotinic acetylcholine receptors. It is used in the form of various salts as a ganglionic stimulant, a parasympathomimetic, and a vermifuge…

Kategori:
AlkaloidsCholinergic AgentsCholinergic Agonists +3
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arformoterol Approved DB01274
small molecule | CAS: 67346-49-0

Arformoterol is a bronchodilator. It works by relaxing muscles in the airways to improve breathing. Arformoterol inhalation is used to prevent bronchoconstriction in people with chronic obstructive pulmonary disease, including chronic bronchitis and emphysema…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +21
Target Protein:
Beta-2 adrenergic receptor
Waktu ParuhIn COPD patients gi…
Vol. Distribusi-
KlirensIn healthy male sub…
Genetik -
ARG098 DB06338
biotech

ARG098 (anti-Fas IgM monoclonal antibody) was studied in a Phase I clinical trial in 2007 involving patients with rheumatoid arthritis.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ARG201 DB06621
biotech

ARG201, a bovine-derived Type I collagen, aims to induce immune tolerance in patients with Diffuse Systemic Scleroderma (dcSSc). This drug was investigated in the completed clinical trial NCT0000567 (Multicenter Phase II Trial of Oral Type I Bovine Collagen i…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Argadin DB04350
small molecule | CAS: 289665-92-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Chitotriosidase-1Endochitinase B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Argatroban Approved DB00278
small molecule | CAS: 74863-84-6

Argatroban is a direct, selective thrombin inhibitor. The American College of Cardiologists (ACC) recommend using bivalirudin or argatroban in patients who have had, or at risk for, heparin induced thrombocytopenia (HIT) and are undergoing percutaneous corona…

Kategori:
AmidesAmino AcidsAmino Acids, Basic +22
Target Protein:
Prothrombin
Waktu Paruh39 and 51 minutes
Vol. Distribusi* 174 mL/kg * 12.1…
Klirens* 5.1 L/kg/hr [infu…
Genetik -
Argifin DB03632
small molecule | CAS: 243975-37-3

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsChitinases, antagonists & inhibitorsPeptides
Target Protein:
Chitotriosidase-1Endochitinase B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 7675-83-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Basic +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arginine PCA DB16025
small molecule | CAS: 56265-06-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Argininosuccinate lyaseArgininosuccinate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arhalofenate DB11811
small molecule | CAS: 24136-23-0

Arhalofenate has been investigated for the treatment of Gout and Hyperuricemia.

Kategori:
AcetatesAcids, AcyclicAcids, Carbocyclic +1
Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arimoclomol Approved DB05025
small molecule | CAS: 289893-25-0

Arimoclomol is a hydroxylamine derivative [A264414] and a heat-shock protein-70 (HSP70) co-inducer.[L51384] Arimoclomol was approved by the FDA on September 20, 2024, making it the first treatment for Niemann-Pick disease, type C (NPC).[L51389] It is also bei…

Kategori:
AminesMATE 1 SubstratesMATE 2 Substrates +3
Waktu ParuhThe elimination hal…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent c…
Genetik -
Aripiprazole Approved DB01238
small molecule | CAS: 129722-12-9

Aripiprazole is an atypical antipsychotic orally indicated for the treatment of schizophrenia, bipolar I, major depressive disorder, irritability associated with autism, and Tourette's.[L45859] It is also indicated as an injection for agitation associated wit…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +48
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 1A +35
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe steady-state vo…
KlirensThe clearance of ar…
Genetik -
Aripiprazole lauroxil Approved DB14185
small molecule | CAS: 1259305-29-7

Aripiprazole lauroxil is a long-acting injectable atypical antipsychotic drug used in the treatment of schizophrenia in adult patients. It is a prodrug of [aripiprazole], which acts as a partial agonist at the D2 and 5-HT1A receptors, and as an antagonist at …

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +29
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 1A5-hydroxytryptamine receptor 2A +22
Waktu ParuhThe mean aripiprazo…
Vol. DistribusiBased on population…
KlirensIn rats, the cleara…
Genetik -
Arketamine DB19150
small molecule | CAS: 33643-49-1

Arketamine is under investigation in clinical trial NCT05414422 (A Randomized, Placebo-controlled, Double-blind Study to Assess Safety and Efficacy of PCN-101 in TRD).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ARM-210 DB16944
small molecule | CAS: 1467605-57-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Armodafinil Approved DB06413
small molecule | CAS: 112111-43-0

Armodafinil is the enantiopure of the wakefulness-promoting agent modafinil (Provigil), and is indicated to improve wakefulness in adult patients with excessive sleepiness associated with obstructive sleep apnea (OSA), narcolepsy, or shift work disorder (SWD)…

Kategori:
Benzene DerivativesBenzhydryl CompoundsCentral Nervous System Agents +21
Target Protein:
Alpha-1D adrenergic receptorSodium-dependent dopamine transporter
Waktu ParuhTerminal half-life …
Vol. DistribusiApparent volume of …
KlirensThe oral clearance …
Genetik -
Arnica montana DB14297
biotech | CAS: 8057-65-6

Arnica montana is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsAsteraceaeBiological Products +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ARO-ANG3 DB17626
biotech

ARO-ANG3 is a subcutaneously administered RNA interference (RNAi)-based investigational medicine targeting angiopoietin-like protein 3 (ANGPTL3). It was granted an orphan drug designation for the treatment of homozygous familial hypercholesterolemia (HoFH).[L…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ARO-APOC3 DB17625
biotech

ARO-APOC3 is an investigational RNAi therapeutic targeting apolipoprotein C-III (APOC3). It received an Orphan Drug designation by the FDA for the treatment of familial chylomicronemia syndrome.[L45864]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arotinoid acid DB02877
small molecule | CAS: 71441-28-6

Arotinoid acid is a retinoic acid analog which acts as a selective RAR agonist.

Kategori:
Acids, CarbocyclicAlkenesBenzene Derivatives +9
Target Protein:
Retinoic acid receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arotinolol DB09204
small molecule | CAS: 68377-92-4

Arotinolol is an alpha- and beta-receptor blocker developed in Japan. It is a thiopropanolamine with a tertiary butyl moiety. It has been studied for its potential to be an antihypertensive therapy.[T87] Artinolol is being developed by Sumitomo Pharmaceutical…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +11
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorAlpha-1 adrenergic receptors
Waktu ParuhThe reported half-l…
Vol. DistribusiThe stereospecifici…
Klirens-
Genetik -
ARQ 171 DB06034
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ARRY-502 DB16053
small molecule | CAS: 1202891-16-4

ARRY-502 is under investigation in clinical trial NCT01561690 (A Study of ARRY-502 in Patients With Persistent Asthma).

Target Protein:
Prostaglandin D2 receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arsanilic acid DB03006
small molecule | CAS: 98-50-0

An arsenical which has been used as a feed additive for enteric conditions in pigs and poultry. It causes blindness and is ototoxic and nephrotoxic in animals. [PubChem]

Kategori:
Adjuvants, ImmunologicAlkenesAnti-Infective Agents +10
Target Protein:
Lysozyme C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arsenic trioxide Approved DB01169
small molecule | CAS: 1327-53-3

Arsenic trioxide is a chemotherapeutic agent of idiopathic function used to treat leukemia that is unresponsive to first line agents. It is suspected that arsenic trisulfide induces cancer cells to undergo apoptosis. In general, arsenic is known to be a natur…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsArsenicals +16
Target Protein:
Inhibitor of nuclear factor kappa-B kinase subunit betaThioredoxin reductase 1, cytoplasmicTranscription factor Jun +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arsenite ion DB18509
small molecule | CAS: 15502-74-6

Deskripsi belum tersedia.

Kategori:
AnionsArsenicalsElectrolytes +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arsenous acid DB04456
small molecule | CAS: 13464-58-9

Deskripsi belum tersedia.

Kategori:
AnionsArsenicalsElectrolytes +1
Target Protein:
Arsenate reductaseArsenical pump-driving ATPase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arsthinol DB08928
small molecule | CAS: 119-96-0

Arsthinol (INN) is an antiprotozoal agent that was first synthesized by Ernst A.H. Friedheim in 1949 via the complexing of acetarsol with 2,3-dimercaptopropanol. It has since been demonstrated that the agent possesses activity against amoebas and yaws. Consid…

Kategori:
Antiparasitic Products, Insecticides and RepellentsAntiprotozoalsArsenicals
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artefenomel DB11809
small molecule | CAS: 1029939-86-3

Artefenomel has been investigated for the treatment of Malaria.

Kategori:
AnionsAnti-Infective AgentsAntimalarials +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artemether Approved DB06697
small molecule | CAS: 71963-77-4

Artemether is an antimalarial agent used to treat acute uncomplicated malaria. It is administered in combination with lumefantrine for improved efficacy. This combination therapy exerts its effects against the erythrocytic stages of <i>Plasmodium spp.</i> and…

Kategori:
Anti-Infective AgentsAntimalarialsAntiparasitic Agents +25
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1
Waktu ParuhArtemether, 1.6 +/-…
Vol. Distribusi-
Klirens-
Genetik -
Artemin DB15438
biotech | CAS: 309758-71-2

Artemin is under investigation in clinical trial NCT01842126 (Phase 1 Subcutaneous Single and Multiple Ascending Dose Study of BG00010 (Neublastin)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artemisia absinthium pollen Approved DB10768
biotech

Artemisia absinthium pollen is the pollen of the Artemisia absinthium plant. Artemisia absinthium pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Pollen Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artemisia douglasiana pollen Approved DB10761
biotech

Artemisia douglasiana pollen is the pollen of the Artemisia douglasiana plant. Artemisia douglasiana pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artemisia ludoviciana pollen Approved DB10762
biotech

Artemisia ludoviciana pollen is the pollen of the Artemisia ludoviciana plant. Artemisia ludoviciana pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Pollen Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artemisinin DB13132
small molecule | CAS: 63968-64-9

Artemisinin has been used in trials studying the treatment of Schizophrenia, Malaria, Falciparum, and Plasmodium Falciparum.

Kategori:
Anti-Infective AgentsAntimalarialsAntiparasitic Products, Insecticides and Repellents +13
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artemisone DB16097
small molecule | CAS: 255730-18-8

Artemisone is under investigation in clinical trial NCT00936767 (Artemisone for the Treatment of Uncomplicated Falciparum Malaria in Western Cambodia).

Kategori:
Free RadicalsPeroxidesReactive Oxygen Species +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artemotil Approved DB13851
small molecule | CAS: 75887-54-6

Artemotil, also known as ?-arteether, is a semi-synthetic derivative of artemisinin and a fast acting blood schizonticide specifically indicated for the treatment of chloroquine-resistant _Plasmodium falciparum_ malaria and cerebral malaria cases.

Kategori:
AmebicidesAnti-Infective AgentsAntimalarials +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artenimol Approved DB11638
small molecule | CAS: 71939-50-9

Artenimol is an artemisinin derivative and antimalarial agent used in the treatment of uncomplicated *Plasmodium falciparum* infections [FDA Label]. It was first authorized for market by the European Medicines Agency in October 2011 in combination with [DB139…

Kategori:
Anti-Infective AgentsAntimalarialsAntiparasitic Agents +16
Target Protein:
Actin, cytoplasmic 2Alpha-aminoadipic semialdehyde dehydrogenaseAnnexin A2 +188
Waktu ParuhArtenimol was repor…
Vol. DistribusiArtenimol was obser…
KlirensArtenimol was obser…
Genetik -
Arterolane DB19027
small molecule | CAS: 664338-39-0

Arterolane is under investigation in clinical trial NCT03452475 (Comparison of Arterolane-piperaquine Versus Arterolane-piperaquine+mefloquine Versus Artemether-lumefantrine in Kenyan Children).

Kategori:
AnionsAntimalarialsAntiparasitic Products, Insecticides and Repellents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artesunate Approved DB09274
small molecule | CAS: 88495-63-0

Artesunate is indicated for the initial treatment of severe malaria.[L14099] The World Health Organization recommends artesunate as first line treatment for severe malaria.[L890] Artesunate was developed out of a need for a more hydrophilic derivative of [art…

Kategori:
Acids, AcyclicAnionsAnthelmintics +28
Target Protein:
Malaria protein EXP-1
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ar…
Genetik -
Articaine Approved DB09009
small molecule | CAS: 23964-58-1

Articaine is a dental local anesthetic. Articaine is widely used around the world and is the most popular local anesthetic in many European countries.

Kategori:
AmidesAnestheticsAnesthetics, Local +11
Target Protein:
Voltage-gated sodium channel alpha subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Artichoke Approved DB10638
biotech

Artichoke allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arverapamil DB06669
small molecule | CAS: 123932-43-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arzoxifene Approved DB06249
small molecule | CAS: 182133-25-1

Deskripsi belum tersedia.

Kategori:
Sulfur Compounds
Target Protein:
Estrogen receptorEstrogen receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ASC-618 DB18423
biotech

ASC-618 is a recombinant adeno-associated virus serotype 8 (rAAV2/8) vector expressing bioengineered B domain deleted liver-codon-optimized human factor VIII.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ASC-JM-17 DB16931
small molecule | CAS: 1039760-91-2

Deskripsi belum tersedia.

Kategori:
AlkanesBenzene DerivativesCatechols +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Asciminib Approved DB12597
small molecule | CAS: 1492952-76-7

Asciminib is a tyrosine kinase inhibitor (TKI) used in the treatment of chronic-phase Philadelphia chromosome-positive chronic myeloid leukemia (Ph+ CML). More specifically, it is an inhibitor of the ABL1 kinase activity of the BCR-ABL1 fusion protein[L38995]…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBcr-Abl Tyrosine Kinase Inhibitors +26
Target Protein:
Tyrosine-protein kinase ABL1
Waktu ParuhThe terminal elimin…
Vol. DistribusiAt steady-state, th…
KlirensThe total apparent …
Genetik -
Menampilkan 2151–2200 dari 11793
Sebelumnya Halaman 44 / 236 Berikutnya