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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 44 / 272
?A?–Gas6 DB17069
biotech

?A?–Gas6 is a chimeric fusion protein being investigated in preclinical studies as an immunotherapeutic agent for Alzheimer's disease (AD). It is made of a single chain variable fragment (scFv) of an Amyloid ? (A?)-targeting monoclonal antibody fused with a t…

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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Stromelysin-1
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A-16L DB18270
biotech | CAS: 410527-75-2

Deskripsi belum tersedia.

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A-620223 DB07330
small molecule | CAS: 272769-49-0

Deskripsi belum tersedia.

Target Protein:
Poly [ADP-ribose] polymerase 1
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A-674563 DB08568
small molecule | CAS: 552325-73-2

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingPyrazoles
Target Protein:
RAC-alpha serine/threonine-protein kinasecAMP-dependent protein kinase catalytic subunit alphacAMP-dependent protein kinase inhibitor alpha
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biotech | CAS: 1470038-56-2

A-dmDT390-bisFv(UCHT1) is under investigation in clinical trial NCT02943642 (Safety and Effectiveness of A-dmdt390-bisfv(ucht1) Fusion Protein in Subjects With Mycosis Fungoides).

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A166 DB17413
biotech

A166 is an antibody-drug conjugate composed of a novel cytotoxic drug (Duo-5, anti-microtubule agent) site-specifically conjugated to an anti-HER2 antibody (trastuzumab) via a stable protease-cleavable valine citrulline linker.

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AAG-1 DB17199
small molecule | CAS: 1204408-18-3

Deskripsi belum tersedia.

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AAV-CNGB3 DB18344
biotech

AAV-CNGB3 is an adenovirus associated viral vector serotype 8 containing the human CNGB3 gene.

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AAV-RPE65 DB18343
biotech

AAV-RPE65 is an adenovirus associated viral vector serotype 5 containing the human RPE65 gene

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AAV1-FS344 DB17855
biotech

AAV1-FS344 is an investigational gene therapy developed by Milo Biotechnology to deliver follistatin, a potent myostatin inhibitor. It is being investigated for the treatment of Duchenne Muscular Dystrophy, Becker Muscular Dystrophy, and inclusion body myosit…

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biotech

Deskripsi belum tersedia.

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AB-001 DB18009
small molecule | CAS: 2663700-89-6

Deskripsi belum tersedia.

Kategori:
Bridged-Ring CompoundsCycloparaffinsHeterocyclic Compounds, Fused-Ring
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AB-201 DB18629
biotech

AB-201 is a CAR-NK cell therapy targeted against HER2.[L48340] It is under investigation for the treatment of HER2-positive cancers, including breast and gastric carcinomas.

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AB-22 DB18296
small molecule | CAS: 1463913-43-0

Deskripsi belum tersedia.

Target Protein:
Sphingosine 1-phosphate receptor 2
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AB-8939 DB17115
small molecule | CAS: 1974336-09-8

Deskripsi belum tersedia.

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AB-G023 DB18576
biotech

AB-G023 is a solution stable glucagon analog

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Abacavir Approved DB01048
small molecule | CAS: 136470-78-5

Abacavir (ABC) is a powerful nucleoside analog reverse transcriptase inhibitor (NRTI) used to treat HIV and AIDS. Chemically, it is a synthetic carbocyclic nucleoside and is the enantiomer with 1S, 4R absolute configuration on the cyclopentene ring. In vivo, …

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +22
Target Protein:
Reverse transcriptase/RNaseHGag-Pol polyprotein
Gen Terkait:
HCP5
Waktu Paruh1.54 ± 0.63 hours
Vol. Distribusi* 0.86 ± 0.15 L/kg …
Klirens* 0.80 ± 0.24 L/hr/…
Genetik 1 Varian
Abafungin DB06395
small molecule | CAS: 129639-79-8

Deskripsi belum tersedia.

Kategori:
Antifungal AgentsAzole AntifungalsSulfur Compounds
Target Protein:
Lanosterol 14-alpha demethylase
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Abaloparatide Approved DB05084
biotech | CAS: 247062-33-5

Abaloparatide is an N-terminal analog of parathyroid hormone-related protein (PTHrP) [A256778] and an agonist at the parathyroid hormone type 1 (PTH1) receptor.[L740] It is a synthetic 34 amino acid peptide with 41% homology to human parathyroid hormone 1-34 …

Kategori:
Amino Acids, Peptides, and ProteinsAnalogs/DerivativesBiological Factors +13
Target Protein:
Parathyroid hormone/parathyroid hormone-related peptide receptor
Waktu ParuhThe mean half-life …
Vol. DistribusiThe volume of distr…
KlirensThe mean apparent t…
Genetik -
Abametapir Approved DB11932
small molecule | CAS: 1762-34-1

Abametapir is a novel pediculicidal metalloproteinase inhibitor used to treat infestations of head lice.[L15153] The life cycle of head lice (_Pediculus capitis_) is approximately 30 days, seven to twelve of which are spent as eggs laid on hair shafts near th…

Kategori:
Antiparasitic Products, Insecticides and RepellentsCytochrome P-450 CYP1A2 InhibitorsCytochrome P-450 CYP1A2 Inhibitors (strength unknown) +13
Waktu ParuhThe elimination hal…
Vol. DistribusiData regarding the …
KlirensThe clearance and e…
Genetik -
Abarelix Approved DB00106
small molecule | CAS: 183552-38-7

Synthetic decapeptide antagonist to gonadotropin releasing hormone (GnRH). It is marketed by Praecis Pharmaceuticals as Plenaxis. Praecis announced in June 2006 that it was voluntarily withdrawing the drug from the market.

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating AgentsEndocrine Therapy +4
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu Paruh13.2 ± 3.2 d…
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Abatacept Approved DB01281
biotech | CAS: 332348-12-6

Abatacept is a soluble fusion protein, which links the extracellular domain of human cytotoxic T-lymphocyte-associated antigen 4 (CTLA-4) to the modified Fc (hinge, CH2, and CH3 domains) portion of human immunoglobulin G1 (IgG1).[L20504,L42715] Structurally, …

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntibodies +18
Target Protein:
T-lymphocyte activation antigen CD80T-lymphocyte activation antigen CD86Cytotoxic T-lymphocyte protein 4
Waktu Paruh16.7 (12-23) days i…
Vol. Distribusi* 0.07 L/kg [RA Pat…
Klirens* 0.23 mL/h/kg [Hea…
Genetik -
ABBV-744 DB19199
small molecule | CAS: 2138861-99-9

Deskripsi belum tersedia.

Target Protein:
Bromodomain-containing protein 3Bromodomain-containing protein 2Bromodomain-containing protein 4
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ABBV-CLS-7262 DB18407
small molecule

Deskripsi belum tersedia.

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Abciximab Approved DB00054
biotech | CAS: 143653-53-6

Abciximab is a Fab fragment of the chimeric human-murine monoclonal antibody 7E3. Abciximab binds to the glycoprotein (GP) IIb/IIIa receptor of human platelets and inhibits platelet aggregation by preventing the binding of fibrinogen, von Willebrand factor, a…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
Integrin beta-3Integrin alpha-IIbLow affinity immunoglobulin gamma Fc region receptor II-a +2
Waktu ParuhFollowing intraveno…
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Abediterol DB12100
small molecule | CAS: 915133-65-2

Abediterol has been used in trials studying the treatment of Asthma, Chronic Obstructive Pulmonary Disease (COPD), and Chronic Obstructive Pulmonary Disease (COPD) and Asthma.

Kategori:
Adrenergic AgonistsAdrenergic beta-2 Receptor AgonistsAdrenergic beta-Agonists +4
Target Protein:
Beta-2 adrenergic receptor
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Abelacimab DB16682
biotech | CAS: 2098724-83-3

Abelacimab is under investigation in clinical trial NCT04755283 (Safety and Tolerability of Abelacimab (MAA868) vs. Rivaroxaban in Patients With Atrial Fibrillation).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Abemaciclib Approved DB12001
small molecule | CAS: 1231929-97-7

Abemaciclib is an antitumor agent and dual inhibitor of cyclin-dependent kinases 4 (CDK4) and 6 (CDK6) that are involved in the cell cycle and promotion of cancer cell growth in case of unregulated activity. On September 28, 2017, FDA granted approval of abem…

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +36
Target Protein:
Cyclin-dependent kinase 4Cyclin-dependent kinase 6
Waktu ParuhThe mean plasma eli…
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Abeprazan DB16078
small molecule | CAS: 1902954-60-2

Abeprazan is under investigation in clinical trial NCT04341454 (Study to Evaluate the Efficacy and Safety of DWP14012 in Patients With Acute or Chronic Gastritis).

Kategori:
Gastrointestinal Agents
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Abequolixron DB17146
small molecule | CAS: 610318-54-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene Derivatives
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Abequose DB02590
small molecule | CAS: 56816-60-5

Deskripsi belum tersedia.

Kategori:
CarbohydratesMonosaccharides
Target Protein:
Tail fiber protein
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Abetimus DB06662
biotech | CAS: 167362-48-3

Abetimus was developed by La Jolla Pharmaceuticals as an immunosuppressant but was never marketed in American or Europe despite application for marketing authorization in the mid-2000s.

Kategori:
Antineoplastic and Immunomodulating AgentsImmunologic FactorsImmunosuppressive Agents +4
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Abexinostat DB12565
small molecule | CAS: 783355-60-2

Abexinostat has been used in trials studying the treatment of Sarcoma, Lymphoma, Leukemia, Lymphocytic, and Hodgkin Disease, among others. It is a novel, broad-spectrum hydroxamic acid-based inhibitor of histone deacetylase (HDAC) with potential antineoplasti…

Kategori:
AminesAntineoplastic AgentsEnzyme Inhibitors +6
Target Protein:
Histone deacetylase 1Histone deacetylase
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ABG-023 DB18829
biotech

ABG-023 is a glucagon analog which is soluble and solution-stable.[L50778]

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ABH001 DB16177
small molecule | CAS: 502-97-6

ABH001 is under investigation in clinical trial NCT01749306 (A Study of the Efficacy and Safety of ABH001 in the Treatment of Patients With Epidermolysis Bullosa Who Have Wounds That Are Not Healing).

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Abicipar Pegol DB12258
biotech | CAS: 1327278-94-3

Abicipar Pegol has been used in trials studying the treatment of Macular Edema and Macular Degeneration.

Kategori:
Amino Acids, Peptides, and ProteinsAntineovascularisation AgentsOcular Vascular Disorder Agents +5
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Abiprubart DB19333
biotech | CAS: 2765071-95-0

Abiprubart is being evaluated for its efficacy and safety in participants with Sjögren's Disease in clinical trial NCT06531395

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Abiraterone Approved DB05812
small molecule | CAS: 154229-19-3

Abiraterone is a potent, irreversible, and selective inhibitor of 17 ?hydroxylase/C17,20-lyase (CYP17), an enzyme expressed in testicular, adrenal, and prostatic tumour tissues, to regulate androgen biosynthesis.[A3811, A260880, L40968] Abiraterone was first …

Kategori:
AndrostanesAndrostenesAntineoplastic Agents +32
Target Protein:
Steroid 17-alpha-hydroxylase/17,20 lyase
Waktu ParuhIn patients with mC…
Vol. DistribusiThe mean (± SD) app…
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Abituzumab DB12775
biotech | CAS: 1105038-73-0

Abituzumab has been used in trials studying the treatment of Prostate Cancer Metastatic.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Abivertinib DB15327
small molecule | CAS: 1557267-42-1

Abivertinib is a tyrosine kinase inhibitor targeted against mutant forms of both human epidermal growth factor receptor (EGFR) and Bruton's tyrosine kinase (BTK).[L17383] It has been investigated for use in the treatment of non-small cell lung cancer (NSCLC) …

Kategori:
Acids, AcyclicAcrylatesAmides +4
Target Protein:
Epidermal growth factor receptorTyrosine-protein kinase BTK
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ABO-201 DB17951
biotech

Deskripsi belum tersedia.

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ABP-700 DB15411
small molecule | CAS: 1446482-29-6

ABP-700 is under investigation in clinical trial NCT02800590 (Study to Investigate the Safety and Efficacy of 3 Dosing Regimens of ABP-700 for Procedural Sedation in Adult Participants Undergoing Colonoscopy).

Kategori:
GABA AgentsGABA AgonistsGABA-A Receptor Agonists +1
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Abrilumab DB15076
biotech | CAS: 1342290-43-0

Abrilumab is under investigation in clinical trial NCT01290042 (Study to Evaluate Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of AMG 181.).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Abrocitinib Approved DB14973
small molecule | CAS: 1622902-68-4

Abrocitinib is an oral small-molecule inhibitor of Janus kinase 1 (JAK1). Janus kinases are intracellular enzymes involved in transduction pathways that regulate hematopoiesis and immune cell function.[L39774] The Janus kinase (JAK)–signal transducer and acti…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAmidesCytochrome P-450 CYP2B6 Substrates +17
Target Protein:
Tyrosine-protein kinase JAK1Tyrosine-protein kinase JAK2Tyrosine-protein kinase JAK3 +1
Waktu ParuhThe mean eliminatio…
Vol. DistribusiAfter intravenous a…
KlirensThere is no informa…
Genetik -
Abscisic Acid DB16829
small molecule | CAS: 21293-29-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAlkenesCarotenoids +11
Waktu Paruh-
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ABSK-012 DB18035
small molecule | CAS: 2271209-99-3

Deskripsi belum tersedia.

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ABSK-091 DB18442
small molecule | CAS: 1035270-39-3

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesAntineoplastic Agents +2
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ABT-072 DB15156
small molecule | CAS: 1132936-00-5

ABT-072 is under investigation in clinical trial NCT00890318 (A Study in Healthy Adult Subjects to Evaluate the Safety, Tolerability, and Pharmacokinetic Profiles of Multiple Doses of ABT-072 Used to Treat Hepatitis C).

Kategori:
AmidesPyrimidinesPyrimidinones +2
Target Protein:
Genome polyprotein
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ABT-341 DB08044
small molecule | CAS: 913623-69-5

ABT-341 is a potent and selective DPP-4 inhibitor with a structure very similar to sitagliptin (in 2D; the 3D structure is significantly different). [A39406]

Kategori:
Benzene DerivativesEnzyme InhibitorsProtease Inhibitors
Target Protein:
Dipeptidyl peptidase 4
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