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3253

Total database: 17430
Struktur (SMILES)
2451 (75.3%)
Target
1833 (56.3%)
Genomik
35 (1.1%)
Referensi
3253 (100.0%)

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Hasil Pencarian (3253)

Halaman 44 / 66
OMS-824 DB17874
small molecule | CAS: 1207549-69-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Onalespib DB06306
small molecule | CAS: 912999-49-6

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +3
Target Protein:
Heat shock protein HSP 90-alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Onapristone DB12637
small molecule | CAS: 96346-61-1

Onapristone has been used in trials studying the treatment of Prostate Cancer, Recurrent Prostate Cancer, Metastatic Prostate Cancer, Androgen-independent Prostate Cancer, and Progesterone Receptor Positive Tumor: Max 1 Line of Prior Chemotherapy, no Prior Ho…

Kategori:
Antineoplastic AgentsFertility AgentsFertility Agents, Female +5
Target Protein:
Progesterone receptorGlucocorticoid receptorAdhesion G-protein coupled receptor D1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Onatasertib DB12570
small molecule | CAS: 1228013-30-6

Onatasertib (CC-223) has been used in trials studying the treatment and basic science of Multiple Myeloma, Glioblastoma Multiforme, HepatoCellular Carcinoma, Non-small Cell Lung Cancer, and Diffuse Large B-Cell Lymphoma, among others.

Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ondelopran DB12585
small molecule | CAS: 676501-25-0

Ondelopran has been used in trials studying the treatment of Alcohol Dependence.

Kategori:
AminesBenzene DerivativesBenzyl Compounds +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ONL-1204 DB18239
biotech | CAS: 2040964-58-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ONO-7579 DB17236
small molecule | CAS: 1622212-25-2

Deskripsi belum tersedia.

Kategori:
Enzyme InhibitorsProtein Kinase Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Opaganib DB12764
small molecule | CAS: 915385-81-8

Opaganib, also known as ABC294640, is a selective [sphingosine kinase-2 (SK2)](https://go.drugbank.com/polypeptides/Q9NRA0) inhibitor that is orally administered.[L27436] This drug has potential anticancer, anti-inflammatory, and antiviral activities, with po…

Kategori:
Bridged-Ring CompoundsCycloparaffins
Target Protein:
Sphingosine kinase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Opevesostat DB18818
small molecule | CAS: 2231294-96-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Opipramol DB12930
small molecule | CAS: 315-72-0

Opipramol has been used in trials studying the treatment of Dementia, Depression, Schizophrenia, Anxiety Disorders, and Psychosomatic Disorders.

Kategori:
Adrenergic AgentsAgents that produce hypertensionAgents that reduce seizure threshold +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orantinib DB12072
small molecule | CAS: 252916-29-3

Orantinib has been used in trials studying the treatment of Lung Cancer, Breast Cancer, Kidney Cancer, Gastric Cancer, and Prostate Cancer, among others.

Kategori:
Acids, AcyclicAlkaloidsEnzyme Inhibitors +9
Target Protein:
Vascular endothelial growth factor receptor 2Aurora kinase AFibroblast growth factor receptor 1 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ORE-1001 DB12271
small molecule | CAS: 305335-31-3

ORE1001 has been used in trials studying the treatment of Mild to Moderate Ulcerative Colitis. It is an ACE2 inhibitor.

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Peptides, and Proteins
Target Protein:
Angiotensin-converting enzyme 2Carboxypeptidase N catalytic chainCarboxypeptidase N subunit 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oregovomab DB04964
biotech | CAS: 213327-37-8

Oregovomab is a murine monoclonal antibody that attaches to the tumor-associated antigen CA125.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Target Protein:
Mucin-16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orforglipron DB18964
small molecule | CAS: 2212020-52-3

Orforglipron is under investigation in clinical trial NCT06010004 (A Long-term Safety Study of Orforglipron (LY3502970) in Participants With Type 2 Diabetes).

Kategori:
Oxazoles
Target Protein:
Glucagon-like peptide 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ORG-25435 DB12312
small molecule | CAS: 256456-73-2

Org 25435 has been used in trials studying the treatment of Anaesthesia.

Kategori:
Benzene Derivatives
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ORG-25935 DB12220
small molecule | CAS: 1147011-84-4

Org 25935 has been used in trials studying the treatment of Alcoholism, Schizophrenia, and Panic Disorder.

Kategori:
Naphthalenes
Target Protein:
Sodium- and chloride-dependent glycine transporter 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orilanolimab DB15312
biotech | CAS: 2066544-85-0

Orilanolimab is under investigation in clinical trial NCT03075878 (A Safety Study of SYNT001 in Subjects With Chronic, Stable Warm Autoimmune Hemolytic Anemia (WAIHA)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oritavancin Approved DB04911
small molecule | CAS: 171099-57-3

Oritavancin is a glycopeptide antibiotic used for the treatment of skin infections. It was developed by The Medicines Company (acquired by Novartis).[L12858] Oritavancin was initially approved by the FDA in 2014 and formulated to combat susceptible gram-posit…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +24
Target Protein:
Dihydropteroate synthasePeptidoglycan precursorsBacterial cell wall peptide bridging segments +1
Waktu ParuhThe average termina…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of or…
Genetik -
ORM-12741 DB12057
small molecule | CAS: 610782-82-6

ORM-12741 has been used in trials studying the basic science and treatment of Alzheimer's Disease.

Kategori:
Adrenergic alpha-2 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +2
Target Protein:
Alpha-2C adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ORM-13070 C-11 DB15324
small molecule | CAS: 1227170-74-2

ORM-13070 C-11 is under investigation in clinical trial NCT00735774 (Suitability of 11C-ORM-13070 as a PET Tracer).

Kategori:
Carbon Radioisotopes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ornithine Approved DB00129
small molecule | CAS: 70-26-8

Produced during the urea cycle, ornithine is an amino acid produced from the splitting off of urea from arginine. L-Ornithine allows for the disposal of excess nitrogen and acts as a precursor of citrulline and arginine.

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids, Basic +9
Target Protein:
Ornithine aminotransferase, mitochondrialOrnithine transcarbamylase, mitochondrialArginase-1 +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ORP-101 DB16072
small molecule | CAS: 1820753-68-1

ORP-101 is under investigation in clinical trial NCT04129619 (A Comparison of the Effects of ORP-101 Versus Placebo in Adult Patients With Irritable Bowel Syndrome With Diarrhea (IBS-D)).

Target Protein:
Mu-type opioid receptorKappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orteronel DB12066
small molecule | CAS: 566939-85-3

Orteronel has been investigated for the treatment of Prostate Cancer.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Orvepitant DB12427
small molecule | CAS: 579475-18-6

Orvepitant has been used in trials studying the treatment of Depressive Disorder, Depressive Disorder, Major, Post-Traumatic Stress Disorder, and Posttraumatic Stress Disorder (PTSD).

Kategori:
Antidepressive AgentsCentral Nervous System Depressants
Target Protein:
Substance-P receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OSE-2101 DB17122
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oseltamivir Approved DB00198
small molecule | CAS: 196618-13-0

Oseltamivir (marketed as the product Tamiflu?), is an antiviral neuraminidase inhibitor used for the treatment and prophylaxis of infection with influenza viruses A (including pandemic H1N1) and B. Oseltamivir exerts its antiviral activity by inhibiting the a…

Kategori:
AcetamidesAcetatesAmides +8
Target Protein:
NeuraminidaseSialidase-1Sialidase-2
Waktu ParuhPlasma concentratio…
Vol. DistribusiThe mean volume of …
KlirensRenal clearance (18…
Genetik -
OSI-027 DB12387
small molecule | CAS: 936890-98-1

OSI-027 has been used in trials studying the treatment of Any Solid Tumor or Lymphoma.

Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Osilodrostat Approved DB11837
small molecule | CAS: 928134-65-0

Osilodrostat is an inhibitor of 11?-hydroxylase (also referred to as CYP11B1), the enzyme that catalyzes the final step in the biosynthesis of endogenous cortisol.[L12123] It is used to lower circulating cortisol levels in the treatment of Cushing's disease, …

Kategori:
Antiadrenal PreparationsAnticorticosteroidsCortisol Synthesis Inhibitors +32
Target Protein:
Cytochrome P450 11B1, mitochondrialCytochrome P450 11B2, mitochondrial
Waktu ParuhThe elimination hal…
Vol. DistribusiThe median apparent…
KlirensData regarding the …
Genetik -
Osoresnontrine DB16274
small molecule | CAS: 1189767-28-9

Osoresnontrine is under investigation in clinical trial NCT02281773 (A Study to Investigate the Efficacy, Safety and Tolerability of Four Different Doses of BI 409306 Compared to Placebo Given for 12 Weeks in Patients With Schizophrenia on Stable Antipsychoti…

Kategori:
Enzyme InhibitorsPhosphodiesterase Inhibitors
Target Protein:
High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ospemifene Approved DB04938
small molecule | CAS: 128607-22-7

Ospemifene is a new selective non-hormonal estrogen receptor modulator (SERM) that is used for the treatment of moderate to severe dyspareunia, a symptom of vulvar and vaginal atrophy, due to menopause. FDA approved on February 26, 2013.

Kategori:
Benzene DerivativesBenzylidene CompoundsCytochrome P-450 CYP2B6 Substrates +14
Target Protein:
Estrogen receptor
Waktu ParuhTerminal half-life …
Vol. Distribusi448 L
KlirensTotal body clearanc…
Genetik -
Osugacestat DB12006
small molecule | CAS: 1401066-79-2

Osugacestat (BMS-906024) has been used in trials studying the treatment of Cancer, Lymphoblastic Leukemia, Acute T-cell, and Precursor T-Cell Lymphoblastic Lymphoma.

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OT-730 DB16112
small molecule | CAS: 870809-51-1

OT-730 is under investigation in clinical trial NCT00753168 (Phase 1-2 Evaluation of OT-730 Eye Drops in Reducing the Intraocular Pressure in Patients With Ocular Hypertension or Open-angle Glaucoma).

Target Protein:
Beta-3 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OTOF-GT DB18129
biotech

OTOF-GT is a dual vector AAV gene therapy being investigated for the restoration of hearing loss associated with otoferlin deficiency.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OTX-008 DB13123
small molecule | CAS: 286936-40-1

OTX008 has been used in trials studying the treatment of Solid Tumors.

Target Protein:
Galectin-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ovatodiolide DB19264
small molecule | CAS: 3484-37-5

Ovatodiolide is under investigation in clinical trial NCT04220411 (A Study for AR100DP1 in Mild to Moderate Atopic Dermatitis (AD)).

Kategori:
Terpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1254-35-9

Oxabolone cipionate is the C17? cypionate ester and a prodrug of [DB01500]. A synthetic anabolic-androgenic (AAS) steroid, it is a derivative of 19-nortestosterone (nandrolone). It is considered as a performance enhancing drug thus is prohibited from use in s…

Kategori:
Alimentary Tract and MetabolismAnabolic Agents for Systemic UseAnabolic Steroids +11
Waktu Paruh-
Vol. Distribusi-
KlirensThe elimination on …
Genetik -
Oxamniquine Approved DB01096
small molecule | CAS: 21738-42-1

An anthelmintic with schistosomicidal activity against Schistosoma mansoni, but not against other Schistosoma spp. Oxamniquine causes worms to shift from the mesenteric veins to the liver where the male worms are retained; the female worms return to the mesen…

Kategori:
AnthelminticsAnti-Infective AgentsAntihelminthic +15
Target Protein:
DNA
Waktu Paruh1-2.5 hours
Vol. Distribusi-
Klirens-
Genetik -
Oxaprotiline DB09307
small molecule | CAS: 56433-44-4

Oxaprotiline is a norepinephrine reuptake inhibitor of the tetracyclic antidepressant family that is related to maprotiline. This drug was never marketed. Oxaprotiline is a racemic mixture of the isomers levoprotiline and dextroprotiline. Levoprotiline is the…

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAnthracenes +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxaprozin Approved DB00991
small molecule | CAS: 21256-18-8

Oxaprozin is a non-narcotic, non-steroidal anti-inflammatory drug (NSAID), used to relieve the inflammation, swelling, stiffness, and joint pain associated with osteoarthritis and rheumatoid arthritis.

Kategori:
Acids, AcyclicAgents causing hyperkalemiaAgents that produce hypertension +22
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh54.9 hours
Vol. Distribusi* 11 to 17 L/70 kg
Klirens-
Genetik -
Oxatomide Approved DB12877
small molecule | CAS: 60607-34-3

Oxatomide has been used in trials studying the treatment of Muscular Dystrophy, Duchenne.

Kategori:
Anti-Allergic AgentsAnti-Asthmatic AgentsAntihistamines for Systemic Use +8
Target Protein:
Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxetacaine Approved DB12532
small molecule | CAS: 126-27-2

Oxetacaine, also called oxethazaince, is a potent surface analgesic with the molecular formula N, N-bis-(N-methyl-N-phenyl-t-butyl-acetamide)-beta-hydroxyethylamine that conserves its unionized form at low pH levels. Its actions have shown to relieve dysphagi…

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAnestheticsAnesthetics, Local +5
Target Protein:
Gastrin
Waktu ParuhOxetacaine presents…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Oxitropium DB12086
small molecule | CAS: 99571-64-9

Oxitropium has been investigated for the treatment of Pulmonary Disease, Chronic Obstructive.

Kategori:
Agents producing tachycardiaAlkaloidsAnticholinergic Agents +9
Target Protein:
Muscarinic acetylcholine receptor M5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 19771-63-2

Procysteine has been used in trials studying the treatment of HIV Infections.

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Cyclic +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxycodone Approved DB00497
small molecule | CAS: 76-42-6

Oxycodone is a semisynthetic opioid analgesic derived from thebaine in Germany in 1917.[A178696] It is currently indicated as an immediate release product for moderate to severe pain and as an extended release product for chronic moderate to severe pain requi…

Kategori:
AlkaloidsAnalgesicsCentral Nervous System Agents +21
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor
Waktu ParuhThe apparent elimin…
Vol. Distribusi2.6L/kg.[Label]
KlirensTotal plasma cleara…
Genetik -
Oxymetholone Approved DB06412
small molecule | CAS: 434-07-1

Oxymetholone is a synthetic anabolic steroid marketed under the brand name Anapolon by Hoffmann La Roche Limitedand used in the treatment of osteoporosis, anaemia, and as an agent to stimulate muscle growth in malnourished or underdeveloped patients. Anabolic…

Kategori:
Alimentary Tract and MetabolismAnabolic AgentsAnabolic Agents for Systemic Use +20
Target Protein:
Androgen receptorNatriuretic peptides B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxyphenbutazone Approved DB03585
small molecule | CAS: 129-20-4

Oxyphenbutazone was withdrawn from the Canadian market in March 1985 due to concerns regarding bone marrow suppression.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +20
Target Protein:
AlbuminGroup IIE secretory phospholipase A2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxyphencyclimine Approved DB00383
small molecule | CAS: 125-53-1

Oxyphencyclimine is an anticholinergic drug (trade name Daricon) used in treating peptic ulcers.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnticholinergic Agents +3
Target Protein:
Muscarinic acetylcholine receptor M5Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxyphenisatin DB04823
small molecule | CAS: 125-13-3

A laxative that undergoes enterohepatic circulation. It may cause jaundice.

Kategori:
Alimentary Tract and MetabolismContact LaxativesDrugs for Constipation +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ozagrel DB12017
small molecule | CAS: 82571-53-7

Ozagrel has been used in trials studying the treatment of Dry Eye Syndromes.

Kategori:
Acids, AcyclicAcrylatesCardiovascular Agents +6
Target Protein:
Mitogen-activated protein kinase 14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 2151–2200 dari 3253
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