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2279

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Halaman 43 / 46
biotech | CAS: 1808916-28-0

Tralesinidase alfa is a chimeric fusion protein comprised of recombinant human NAGLU and a modified human insulin-like growth factor 2. It is being investigated for the treatment of mucopolysaccharidosis type IIIB (MPS IIIB), also known as Sanfilippo syndrome…

Kategori:
Amino Acids, Peptides, and Proteinsbeta-N-AcetylhexosaminidasesBiological Factors +12
Waktu Paruh-
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Tralokinumab Approved DB12169
biotech | CAS: 1044515-88-9

Atopic dermatitis (AD) is an inflammatory skin disorder that causes skin inflammation, skin barrier dysfunction, and chronic pruritus.[A242432] It is estimated to affect up to 20% of adults and children worldwide, and is frequently associated with other atopi…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAmino Acids, Peptides, and ProteinsAntibodies +9
Target Protein:
Interleukin-13
Waktu ParuhThe half-life of tr…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of tr…
Genetik -
Tranilast DB07615
small molecule | CAS: 53902-12-8

Tranilast is an antiallergic drug developed by Kissei Pharmaceuticals. In 1982, it was approved in Japan and South Korea for the management of bronchial asthma. Indications for keloid and hypertrophic scar were added in 1993. It has been used for the treatmen…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAminobenzoates +23
Target Protein:
Steryl-sulfataseHistamine H1 receptorHematopoietic prostaglandin D synthase
Waktu Paruh-
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biotech | CAS: 721946-42-5

Deskripsi belum tersedia.

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Trastuzumab Approved DB00072
biotech | CAS: 180288-69-1

Produced in CHO cell cultures, trastuzumab is a recombinant IgG1 kappa, humanized monoclonal antibody [A40276] that selectively binds with high affinity in a cell-based assay (Kd = 5 nM) to the extracellular domain of the human epidermal growth factor recepto…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +21
Target Protein:
Receptor tyrosine-protein kinase erbB-2
Gen Terkait:
ERBB2
Waktu ParuhThe terminal half-l…
Vol. Distribusi-
KlirensThe predicted stead…
Genetik 1 Varian
biotech | CAS: 1642152-40-6

Trastuzumab duocarmazine is under investigation in clinical trial NCT03262935 (SYD985 vs. Physician's Choice in Participants With Her2-positive Locally Advanced or Metastatic Breast Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Waktu Paruh-
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TRC093 DB06356
biotech

TRC093 is a recombinant humanized IgG1k monoclonal antibody.

Target Protein:
Collagen alpha-4(IV) chain
Waktu Paruh-
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Tremelimumab Approved DB11771
biotech | CAS: 745013-59-6

Tremelimumab, formerly known as ticilimumab, is a fully human IgG2 monoclonal antibody directed against cytotoxic T-lymphocyte-associated antigen 4 (CTLA-4). CTLA-4 is a cell surface receptor expressed on activated T cells to act as a negative regulator for T…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Cytotoxic T-lymphocyte protein 4
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Trenonacog alfa DB13201
biotech | CAS: 1232401-60-3

Human coagulation factor IX (EC 3.4.21.22, Christmas factor, plasma thromboplastin component), produced in CHO cells.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +5
Waktu Paruh-
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Tretinoin Approved DB00755
small molecule | CAS: 302-79-4

Tretinoin, also known as all-trans-retinoic acid (ATRA), is a naturally occurring derivative of [vitamin A] (retinol).[A257474] It is an oxidation product in the physiological pathway of vitamin A metabolism.[A257689] In human circulation, tretinoin is normal…

Kategori:
Agents that produce hypertensionAlkenesAnti-Acne Preparations +37
Target Protein:
Retinoic acid receptor alphaRetinoic acid receptor betaRetinoic acid receptor gamma +13
Waktu ParuhThe terminal elimin…
Vol. DistribusiTretinoin is rapidl…
KlirensNo information is a…
Genetik -
Triamterene Approved DB00384
small molecule | CAS: 396-01-0

Triamterene (2,4,7-triamino-6-phenylpteridine) is a potassium-sparing diuretic that is used in the management of hypertension. It works by promoting the excretion of sodium ions and water while decreasing the potassium excretion in the distal part of the neph…

Kategori:
Agents causing hyperkalemiaCardiovascular AgentsCytochrome P-450 CYP1A2 Substrates +15
Target Protein:
Amiloride-sensitive sodium channel subunit gammaAmiloride-sensitive sodium channel subunit alphaAmiloride-sensitive sodium channel subunit beta +1
Waktu ParuhThe half-life of th…
Vol. DistribusiIn a pharmacolineti…
KlirensThe total plasma cl…
Genetik -
Tricaine DB11552
small molecule | CAS: 582-33-2

Tricaine (as tricaine methanesulfonate) is white powder used for anesthesia, sedation, or euthanasia of fish. It is also the only anesthetic licensed in the United States for use in fin fish that are intended for human consumption.

Kategori:
Acids, CarbocyclicAnestheticsBenzene Derivatives +3
Waktu Paruh-
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Trichloroethylene Approved DB13323
small molecule | CAS: 79-01-6

Trichloroethylene is a halocarbon commonly used as an industrial solvent, not to be confused with the similar 1,1,1-trichloroethane, also known as chlorothene. It has been sold under a variety of trade names including Trimar and Trilene and used as a volatile…

Kategori:
Agents that produce hypertensionAnestheticsAnesthetics, General +8
Waktu Paruh-
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Triclabendazole Approved DB12245
small molecule | CAS: 68786-66-3

Triclabendazole, manufactured by Novartis pharmaceuticals, is an antihelminthic drug that was approved by the FDA in February 2019 for the treatment of fascioliasis in humans.[FDA label, L5452] Fascioliasis is a parasitic infection often caused by the helmi…

Kategori:
AnthelminticsAnti-Infective AgentsAntihelminthic +34
Target Protein:
CruzipainExcretory Secretory (ES) proteins
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe apparent volume…
Klirens-
Genetik -
Tridecactide DB15687
small molecule | CAS: 22006-64-0

Tridecactide, also known as alpha-corticotropin 1-13, is a deacetylated and deaminated alpha-melanocyte stimulating hormone, which may have antipyretic, anti-inflammatory, and antimicrobial effects.[A203210] Tridecactide, along with [metenkefalin], are under …

Kategori:
Experimental Unapproved Treatments for COVID-19Melanocyte-Stimulating Hormones
Waktu Paruh-
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Tridolgosir DB02034
small molecule | CAS: 72741-87-8

An indolizidine alkaloid from the plant Swainsona canescens that is a potent alpha-mannosidase inhibitor. Swainsonine also exhibits antimetastatic, antiproliferative, and immunomodulatory activity.

Target Protein:
Alpha-mannosidase 2
Waktu Paruh-
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Triethylenetetramine Approved DB06824
small molecule | CAS: 112-24-3

Triethylenetatramine (TETA), also known as trientine, is a potent and selective copper (II)-selective chelator. It is a structural analog of linear polyamine compounds, [spermidine] and [spermine]. TETA was first developed in Germany in 1861 and its chelating…

Kategori:
Alimentary Tract and MetabolismAminesChelating Agents +11
Target Protein:
Carbonic anhydrase 14
Waktu ParuhThe mean terminal h…
Vol. DistribusiTETA is widely dist…
KlirensIn healthy adult vo…
Genetik -
Trimethobenzamide Approved DB00662
small molecule | CAS: 138-56-7

Trimethobenzamide is a novel antiemetic which prevents nausea and vomiting in humans. Its actions are unclear but most likely involves the chemoreceptor trigger zone (CTZ). In dogs pretreated with trimethobenzamide HCl, the emetic response to apomorphine is i…

Kategori:
Acids, CarbocyclicAmidesAminoalkyl Ethers +10
Target Protein:
D(2) dopamine receptor
Waktu ParuhThe mean eliminatio…
Vol. Distribusi-
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TRK-250 DB18500
biotech

TRK-250 is a small interfering RNA agent that targets human transforming growth factor-beta 1 (TGF-?1) messenger RNA.

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Trolamine salicylate Approved DB11079
small molecule | CAS: 2174-16-5

Trolamine salicylate is an organic compound or a salt formed between triethanolamine and salicylic acid. Triethanolamine neutralizes the acidity of the salicylic acid. It is a topical analgesic used for temporary relief of minor pain associated with arthritis…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAnti-Inflammatory Agents +11
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. DistribusiTopical administrat…
Klirens-
Genetik -
Tromantadine Approved DB13288
small molecule | CAS: 53783-83-8

Tromantadine is marketed as Viru-Merz in the Czech Republic [L5740]. It is an antiviral used in the treatment of herpes zoster and simplex.

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +5
Waktu Paruh-
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Trospium Approved DB00209
small molecule | CAS: 47608-32-2

Trospium is an antispasmodic agent used to treat the symptoms of overactive bladder, a condition that causes the bladder muscles to contract uncontrollably.[L6208] An overactive bladder leads to an increased urge to urinate, frequent urination, and sometimes,…

Kategori:
Acids, CarbocyclicAgents producing tachycardiaAlimentary Tract and Metabolism +22
Target Protein:
Muscarinic acetylcholine receptor M5Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M1
Waktu ParuhThe half-life of tr…
Vol. DistribusiThe volume of distr…
KlirensThe total apparent …
Genetik -
TRX1 DB05863
biotech

TRX1 is a humanized antibody that binds to the CD4 receptor found on a subset of T cells. TRX1 is being developed for the potential treatment of autoimmune diseases in collaboration with Genentech, Inc. TolerRx is currently conducting a Phase I clinical study…

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TSHA-102 DB18599
biotech

TSHA-102 is a recombinant serotype 9 adeno-associated virus encoding a codon-optimized human MECP2 gene.

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TSHA-105 DB18328
biotech

TSHA-105 is an adeno-associated virus serotype 9 (AAV9) vector with an engineered transgene encoding the human SLC13A5 protein.

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TSHA-118 DB16996
biotech

TSHA-118 is a self-complementary AAV9 gene replacement therapy designed to express a human codon-optimized CLN1 transgene for the treatment of CLN1 disease.

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TT 173 DB17717
biotech

TT 173 is a Modified Human Tissue Factor currently being investigated to treat bleeding disorders such as hemophilia and von Willebrand disease, as well as bleeding episodes in cutaneous injuries or dental procedures.

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TTAX01 DB17928
biotech

TTAX01 is a cryopreserved human umbilical cord product being developed by TissueTech.[L47246]

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TTP889 DB05131
small molecule

TTP889, an orally bioavailable selective inhibitor of the intrinsic coagulation pathway, is being developed as an anticoagulant for the treatment of thromboembolic disorders. TTP889 is the only known selective small molecule inhibitor of Factor IX, a key enzy…

Target Protein:
Coagulation factor IX
Waktu Paruh20 hours
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 92129-86-7

Tuberculin Purified Protein Derivative (PPD) is a sterile aqueous solution of a purified protein fraction for intradermal administration as an aid in the diagnosis of tuberculosis. The diagnostic test is commonly referred to as the Mantoux test which serves t…

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Bacterial +12
Target Protein:
Toll-like receptor 2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Tulisokibart DB18719
biotech | CAS: 2648504-55-4

PRA023 is a humanized monoclonal antibody directed to vascular endothelial growth inhibitor, also known as tumour necrosis factor (TNF)-like ligand 1A (TL1A) and TNF superfamily member 15. It is being investigated for ulcerative colitis.

Target Protein:
Tumor necrosis factor ligand superfamily member 15
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Tunicamycin DB13172
small molecule | CAS: 11089-65-9

Tunicamycin is a mixture of homologous nucleoside antibiotics that inhibits the UDP-HexNAc: polyprenol-P HexNAc-1-P family of enzymes. One member of this family is the enzyme GlcNAc phosphotransferase (GPT), which catalyzes the transfer of N-acetylglucosamine…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsNucleic Acids, Nucleotides, and Nucleosides +3
Waktu Paruh-
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Tuparstobart DB19118
biotech | CAS: 2649466-03-3

Tuparstobart is under investigation in clinical trial NCT05287113 (Study of Retinfanlimab in Combination With INCAGN02385 and INCAGN02390 as First-line Treatment in Participants With Pd-l1-positive (CPS ? 1) Recurrent/metastatic Squamous Cell Carcinoma of the…

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Turoctocog alfa Approved DB09109
biotech | CAS: 1192451-26-5

Turoctocog alfa is a recombinant factor VIII (rFVIII) with a truncated B-domain made from the sequence coding for 10 amino acids from the N-terminus and 11 amino acids from the C-terminus of the naturally occurring B-domain. Turoctocog alfa is produced in Chi…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +5
Target Protein:
Coagulation factor IXCoagulation factor XProthrombin
Waktu ParuhIn pre-clinical stu…
Vol. DistribusiIn pre-clinical stu…
KlirensIn pre-clinical stu…
Genetik -
Turoctocog alfa pegol Approved DB14738
biotech | CAS: 1309086-46-1

Turoctocog alfa pegol is a pegylated version of [turoctocog alfa]. Novo Nordisk's brand name Esperoct (turoctocog alfa pegol, N8-GP) was approved by the US FDA on February 19, 2019. Fundamentally, the N8-GP moiety is identical to [turoctocog alfa], a recom…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +5
Target Protein:
Coagulation factor IXCoagulation factor XProthrombin +1
Waktu ParuhThe mean plasma hal…
Vol. DistribusiThe mean volume of …
KlirensThe mean clearance …
Genetik -
Tuvirumab DB17752
biotech | CAS: 138660-97-6

Deskripsi belum tersedia.

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TVN-102 DB16990
biotech

Deskripsi belum tersedia.

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Tyrothricin Approved DB13503
small molecule | CAS: 1404-88-2

Tyrothricin is an antibiotic peptide complex produced and extracted from the aerobic Gram-positive bacillus Brevibacillus parabrevis [L4019, L4021, A32851] which was previously categorized as Bacillus brevis and Bacillus aneurinolyticus [A36353]. This complex…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +9
Target Protein:
Phospholipid membraneAcetylcholinesteraseBeta-galactosidase
Waktu Paruh-
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UB-612 DB16444
biotech

The UB-612 COVID-19 vaccine was developed by United Biomedical Inc Asia in Taipei as the first COVID-19 “multi-tope” protein-peptide vaccine made up of eight rationally designed components[L30653]. The vaccine incorporates a strong S1-RBD component linked to …

Kategori:
Biological ProductsComplex MixturesVaccines +1
Waktu Paruh-
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Ubidecarenone Approved DB09270
small molecule | CAS: 303-98-0

Ubidecarenone, also called coenzyme Q10, is a 1,4-benzoquinone. From its name (Q10), the Q refers to the constitutive quinone group, and 10 is related to the number of isoprenyl subunits in its tail.[A7874] It is a powerful antioxidant, a lipid-soluble and es…

Kategori:
Agents Causing Muscle ToxicityBenzoquinonesCardiac Therapy +13
Target Protein:
NADH dehydrogenase [ubiquinone] flavoprotein 3, mitochondrialSuccinate dehydrogenase [ubiquinone] flavoprotein subunit, mitochondrial
Waktu ParuhThe pharmacokinetic…
Vol. DistribusiUbidecarenone is di…
KlirensIn preclinical stud…
Genetik -
Ubiquinol Approved DB11340
small molecule | CAS: 992-78-9

Ubiquinol (CoQH2) is a reduced form of coenzyme Q10 (CoQ10) that acts as an active antioxidant that prevents the initiation and propagation of lipid peroxidation in biological membranes and human low-density lipoprotein (LDL). It plays an essential role in ma…

Kategori:
BenzoquinonesCoenzymesEnzymes and Coenzymes +1
Waktu Paruh-
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Ubrogepant Approved DB15328
small molecule | CAS: 1374248-77-7

Ubrogepant is indicated for the acute treatment of migraine headaches with or without aura in adults.[L10926] It was approved by the FDA on December 23, 2019, and is the first oral calcitonin gene-related peptide (CGRP) receptor antagonist approved for the ac…

Kategori:
AnalgesicsAntimigraine PreparationsBCRP/ABCG2 Substrates +23
Target Protein:
Calcitonin gene-related peptide type 1 receptor
Waktu ParuhUbrogepant has an e…
Vol. DistribusiThe apparent centra…
KlirensThe apparent oral c…
Genetik -
small molecule | CAS: 2616-64-0

A nucleoside diphosphate sugar which serves as a source of glucuronic acid for polysaccharide biosynthesis. It may also be epimerized to UDP iduronic acid, which donates iduronic acid to polysaccharides. In animals, UDP glucuronic acid is used for formation o…

Kategori:
CarbohydratesGlycosidesNucleic Acids, Nucleotides, and Nucleosides +8
Target Protein:
UDP-glucose 4-epimeraseGalactosylgalactosylxylosylprotein 3-beta-glucuronosyltransferase 3UDP-glucose 6-dehydrogenase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Ularitide DB05034
small molecule | CAS: 118812-69-4

Ularitide is a synthetic form of urodilatin, a naturally occurring human natriuretic peptide that is involved in regulating blood pressure and the excretion of water and sodium from the kidneys. Urodilatin is produced in the kidney and excreted into the urine…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Asthmatic AgentsAutonomic Agents +10
Target Protein:
Atrial natriuretic peptide receptor 1
Waktu Paruh-
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Genetik -
Ulenistamab DB18291
biotech | CAS: 2415259-90-2

Deskripsi belum tersedia.

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Ulviprubart DB18281
biotech | CAS: 2569434-60-0

Deskripsi belum tersedia.

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biotech

The use of umbilical cord blood (UCB) for therapies is advantageous because of its ease of access, non-invasive collection procedures, and more plasticity for multi-differentiation. UCB contains a large source of hematopoietic stem cells (HSCs) that are capab…

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Umbralisib Approved DB14989
small molecule | CAS: 1532533-67-7

Marginal zone lymphoma is a rare, slowly progressing type of non-Hodgkin lymphoma initially treated with [rituximab] (an anti-CD20 drug), either alone or in combination with chemotherapy. Unfortunately, many patients experience a relapse or develop resistance…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP1A2 Substrates +9
Target Protein:
Casein kinase I isoform epsilonPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformTyrosine-protein kinase ABL1
Waktu ParuhThe effective half-…
Vol. DistribusiThe average apparen…
KlirensThe average apparen…
Genetik -
Unasnemab DB18837
biotech | CAS: 2379805-59-9

Unasnemab is under investigation in clinical trial NCT04683848 (Study to Assess the Efficacy and Safety of MT-3921 in Subjects With Acute Traumatic Cervical Spinal Cord Injury).

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Undecylenic acid Approved DB11117
small molecule | CAS: 112-38-9

Undecylenate, or undecylenic acid, is an unsaturated fatty acid with a terminal double bond that is derived from castor oil. Undecylenic acid is also found naturally in the human sweat. It is used as a precursor in the manufacture of aromatic chemicals, polym…

Kategori:
Antifungals for Dermatological UseAntifungals for Topical UseDermatologicals +4
Target Protein:
Calpain-1 catalytic subunit
Waktu ParuhNo information rega…
Vol. DistribusiNo information rega…
KlirensNo information rega…
Genetik -
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