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6694

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4518 (67.5%)
Target
3751 (56.0%)
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81 (1.2%)
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6694 (100.0%)

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Halaman 42 / 134
Crotalus atrox antivenin Approved DB13892
biotech

Each year it is estimated there are 45,000 snakebites in the US and 300,000 to 400,000 bites worldwide. About 8000 of these snakebites involve venomous snake species. The majority of people bitten are males and about 50% occur in the age group of 18 to 28 [F1…

Kategori:
AntiveninsPassively Acquired ImmunityVenom Neutralization
Waktu Paruh12-23 hours [F113]
Vol. Distribusi-
Klirens-
Genetik -
biotech

Crotalus scutulatus antivenin is derived and purified immunoglobulin fragments obtained from other domestic animals such as sheep previously immunized with Crotalus scutulatus (also known as the _Mojave rattlesnake_ [L2856]). The final purified antivenin …

Kategori:
AntiveninsPassively Acquired ImmunityVenom Neutralization
Waktu ParuhApproximately 15 ho…
Vol. Distribusi0.3 L/kg [FDA label]
Klirens32 mL/min (approxim…
Genetik -
Crotamiton Approved DB00265
small molecule | CAS: 483-63-6

Crotamiton is a scabicidal and antipruritic agent available as a cream or lotion for topical use only. It is a colorless to slightly yellowish oil, having a faint amine-like odor. It is miscible with alcohol and with methanol.

Kategori:
AgrochemicalsAminesAniline Compounds +6
Target Protein:
Transient receptor potential cation channel subfamily V member 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Crovalimab Approved DB16128
biotech | CAS: 1917321-26-6

Crovalimab is a humanized monoclonal antibody and complement C5 inhibitor.[L50908] It consists of two heavy chains (451 amino acid residues each) and two light chains (217 amino acid residues each).[L50908] First developed by Chugai Pharmaceutical, in collabo…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntineoplastic and Immunomodulating Agents +7
Target Protein:
Complement C5
Waktu ParuhThe mean estimated …
Vol. DistribusiThe mean central an…
KlirensIn PNH treatment-na…
Genetik -
Crozbaciclib DB18081
small molecule | CAS: 2099128-41-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CRS-3123 DB12262
small molecule | CAS: 1013915-71-3

CRS3123 has been used in trials studying the treatment of Clostridial Infection and Clostridium Difficile Colitis.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CRx-139 DB05744
small molecule

CRx-139 is an oral synergistic combination drug candidates with novel mechanisms of action targeting multiple biological pathways simultaneously. It is a dissociated steroid designed to enhance the immuno-modulatory activity of a low-dose glucocorticoid stero…

Target Protein:
Tumor necrosis factorInterleukin-6C-reactive protein +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cry5B DB17783
biotech

Cry5B is a pore-forming crystal protein produced by and derived from the soil bacterium _Bacillus thuringiensis_. With demonstrated anthelmintic properties, it has been investigated in the treatment of parasitic intestinal infections.[A259372, A259377]

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Cryptenamine Approved DB00785
small molecule | CAS: 1356-18-9

Cryptenamine is a mixture of closely related hypotensive alkaloids from Veratrum album (Liliaceae). It has been used in the treatment of hypertension but has largely been replaced by drugs with fewer adverse effects. Cryptenamine has a marked and re-producibl…

Kategori:
AlkaloidsAntihypertensive AgentsCardiovascular Agents +3
Target Protein:
Muscarinic acetylcholine receptor M2Beta adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CT-011 DB05916
biotech

CT-011 is a humanized monoclonal antibody directed against a B7 family-associated protein, in patients with advanced haematological malignancies. It is directed against human PD-1 (programmed cell death 1; PDCD1), with immunomodulating and antitumor activitie…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntineoplastic Agents +7
Target Protein:
Programmed cell death protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CTA018 DB05024
small molecule

CTA018 is a member of a new class of vitamin D analogues with a dual mechanism of action, called Vitamin D Signal Amplifiers. This proprietary new drug is both a potent inhibitor of CYP24 (the enzyme responsible for the breakdown of vitamin D) and a potent ac…

Target Protein:
1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrialVitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CTS-1027 DB08490
small molecule | CAS: 193022-04-7

CTS-1027 has been used in trials studying the treatment of Hepatitis C and Chronic Hepatitis C Virus Infection.

Kategori:
AminesHydroxy AcidsHydroxylamines
Target Protein:
Stromelysin-1Interstitial collagenase72 kDa type IV collagenase +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CTT-1057 DB14965
small molecule | CAS: 1628717-55-4

CTT-1057 is under investigation in clinical trial NCT03427476 (CTT1057, a Small Molecular Inhibitor of PSMA, as a Novel Imaging Agent of Neovascularization in Renal Cell Carcinoma).

Waktu Paruh-
Vol. Distribusi-
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CTx-PDE6b DB17858
biotech

CTx-PDE6b is an adeno-associated virus (AAV) based gene therapy designed to deliver a full-length non-mutated copy of the functional human _PDE6b_ gene. Being commercialied by Coave Therapeutics, it is being investigated for the treatment of retinitis pigment…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cudetaxestat DB18203
small molecule | CAS: 1782070-21-6

Deskripsi belum tersedia.

Target Protein:
Autotaxin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Culex pipiens Approved DB14165
biotech

Culex pipiens allergenic extract is used in allergenic testing.

Kategori:
Non-Standardized Insect Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 13479-54-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, Peptides, and Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cupric oxide Approved DB11134
small molecule | CAS: 1317-38-0

Cupric oxide, or copper (II) oxide, is an inorganic compound with the chemical formula CuO. Cupric oxide is used as a precursor in many copper-containing products such as wood preservatives and ceramics. Cupric oxide may be found in over-the-counter vitamin-m…

Kategori:
Diet, Food, and NutritionElementsFood +6
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiFollowing exposure …
KlirensNo pharmacokinetic …
Genetik -
Cupric sulfate Approved DB06778
small molecule | CAS: 7758-98-7

Cupric sulfate is a salt created by treating cupric oxide with sulfuric acid. This forms as large, bright blue crystals containing five molecules of water (CuSO4?5H2O) and is also known as _blue vitriol_. The anhydrous salt is created by heating the hydrate t…

Kategori:
AntidotesAutonomic AgentsCentral Nervous System Agents +10
Waktu ParuhThe biological half…
Vol. DistribusiThe body of a 70 kg…
Klirens-
Genetik -
Curcuma aromatica root oil Approved DB11301
biotech | CAS: 94349-73-2

Curcuma aromatica root oil is obtained from the roots of *Curcuma aromatica*, or more commonly called wild tumeric, via steamed distillation. *Curcuma aromatica* belongs to the family Zingiberaceae. The wild ginger has been used as a cosmetic herbal where its…

Kategori:
Biological ProductsPlant OilsPlant Preparations
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

_Curcuma xanthorrhiza_ oil is extracted from _Curcuma xanthorrhiza_ Roxb., a member of the ginger family (_Zingiberaceae_) that is widely distributed in the region of Southeastern Asia [A33162]. _Curcuma xanthorrhiza_ is also known as Javanese Turmeric or Te…

Waktu ParuhThere are no pharma…
Vol. DistribusiThere are no pharma…
KlirensThere are no pharma…
Genetik -
Curcumin Approved DB11672
small molecule | CAS: 458-37-7

Curcumin, also known as diferuloylmethane, is an active component in the golden spice turmeric (Curcuma longa) and in [Curcuma xanthorrhiza oil]. It is a highly pleiotropic molecule that exhibits antibacterial, anti-inflammatory, hypoglycemic, antioxidant, wo…

Kategori:
AlkanesAnalgesicsAnalgesics, Non-Narcotic +29
Target Protein:
Cytochrome P450 3A4Nitric oxide synthase, inducibleCarbonic anhydrase 14 +18
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiFollowing oral admi…
KlirensNo pharmacokinetic …
Genetik -
Cusatuzumab DB15100
biotech | CAS: 1864871-20-4

CD70 is a ligand expressed on the surface of activated lymphocytes and mature dendritic cells that, in its binding to CD27 receptors, plays an important role in cell proliferation and survival. An overexpression of CD70 can result in the proliferation of mali…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Target Protein:
CD70 antigen
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CV-8102 DB19184
biotech

CV-8102 is under investigation in clinical trial NCT03203005 (IMA970A Plus CV8102 in Very Early, Early and Intermediate Stage Hepatocellular Carcinoma Patients).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CVac Approved DB17351
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
CVnCoV DB15844
biotech

The CVnCov Vaccine (or CV07050101) is in development by CureVac AG. The vaccine uses mRNA technology to create a protein associated with SARS-CoV2, and upon administration and replication, to initiate subsequent immune responses in the body. As of June 2020, …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CVnCoV Vaccine DB15843
biotech

The CVnCov Vaccine (or CV07050101) is in development by CureVac AG. The vaccine uses mRNA technology to create a protein associated with SARS-CoV2, and upon administration and replication, to initiate subsequent immune responses in the body. As of June 2020, …

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CX-046684 Approved DB19414
biotech

CX-046684 is a COVID-19 mRNA vaccine encoding the pre-fusion stabilized Spike glycoprotein (S) of the SARS-CoV-2 Omicron variant lineage KP.2. It is the active ingredient of the 2024-2025 formulation of Moderna's Spikevax vaccine.[L40074]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CX-717 DB05047
small molecule | CAS: 867276-98-0

CX-717 is an ampakine compound previously investigated for the treatment of Attention-Deficit/Hyperactivity Disorder (ADHD) and Alzheimer's disease.

Target Protein:
Neurotrophic factor BDNF precursor formGlutamate receptor 1Glutamate receptor 2 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CXA-10 DB15026
small molecule | CAS: 875685-46-4

CXA-10 is under investigation in clinical trial NCT03422510 (FIRSTx - A Study of Oral CXA-10 in Primary Focal Segmental Glomerulosclerosis (FSGS)).

Kategori:
Anti-Inflammatory AgentsFatty AcidsFatty Acids, Monounsaturated +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CY 1899 DB17797
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CY301 DB06382
biotech

CY301 (Simplivir) is an investigational gene silencing compound developed by CytoGenix for the treatment of HSV.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cyamemazine DB09000
small molecule | CAS: 3546-03-0

Cyamemazine (Tercian), also known as cyamepromazine, is a typical antipsychotic drug of the phenothiazine class used primarily in the treatment of schizophrenia and psychosis-associated anxiety. Cyamemazine actually behaves like an atypical antipsychotic, due…

Kategori:
Anti-Anxiety AgentsAntidepressive AgentsAntipsychotic Agents +16
Target Protein:
5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 1A5-hydroxytryptamine receptor 7 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cyanamide DB02679
small molecule | CAS: 420-04-2

A cyanide compound which has been used as a fertilizer, defoliant and in many manufacturing processes. It often occurs as the calcium salt, sometimes also referred to as cyanamide. The citrated calcium salt is used in the treatment of alcoholism. [PubChem]

Kategori:
CarbodiimidesCyanidesImines +1
Target Protein:
Cathepsin KCarbonic anhydrase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cyanocinnoline DB02882
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cyanocobalamin Approved DB00115
small molecule | CAS: 68-19-9

Cyanocobalamin (commonly known as Vitamin B12) is a highly complex, essential vitamin, owing its name to the fact that it contains the mineral, cobalt. This vitamin is produced naturally by bacteria [A175276], and is necessary for DNA synthesis and cellular e…

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansCorrinoids +10
Target Protein:
Methionine synthaseMethylmalonyl-CoA mutase, mitochondrialMethionine synthase reductase +3
Waktu ParuhApproximately 6 day…
Vol. DistribusiCobalamin is distri…
KlirensDuring vitamin load…
Genetik -
Cyanocobalamin Co-57 Approved DB09385
small molecule | CAS: 13115-03-2

Deskripsi belum tersedia.

Kategori:
Radioactive Diagnostic AgentRadiopharmaceutical Activity
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cyanocobalamin Co-60 Approved DB09387
small molecule | CAS: 13422-53-2

Cyanocobalamin Co-60 is an analog of Vitamin B12 labeled with Co60. Cyanocobalamin Co-60 was used for the diagnosis of pernicious anemia, but now it is withdrawn from the market in the US for unknown reasons.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cyclacillin Approved DB01000
small molecule | CAS: 3485-14-1

A cyclohexylamido analog of penicillanic acid.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +8
Target Protein:
Penicillin-binding protein 1APenicillin-binding protein 3Penicillin binding protein 2a +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cyclandelate Approved DB04838
small molecule | CAS: 456-59-7

A direct-acting smooth muscle relaxant used to dilate blood vessels. It may cause gastrointestinal distress and tachycardia. Cyclandelate is not approved for use in the U.S. or Canada, but is approved in various European countries.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAntiarrhythmic agents +10
Target Protein:
Voltage-dependent calcium channel subunit alpha-2/delta-1Liver carboxylesterase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 60-92-4

Cyclic adenosine monophosphate (cAMP, cyclic AMP or 3'-5'-cyclic adenosine monophosphate) is a molecule that is important in many biological processes; it is derived from adenosine triphosphate (ATP).

Kategori:
Adenine NucleotidesCyclic AMPHeterocyclic Compounds, Fused-Ring +8
Target Protein:
Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 2cAMP-dependent protein kinase type I-alpha regulatory subunitcAMP-dependent protein kinase type II-beta regulatory subunit +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cyclic GMP DB02315
small molecule | CAS: 7665-99-8

Cyclic guanosine monophosphate (Cyclic GMP) is a guanine nucleotide containing one phosphate group which is esterified to the sugar moiety in both the 3'- and 5'-positions. It is a cellular regulatory agent and has been described as a second messenger…

Kategori:
Guanine NucleotidesHeterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and Nucleosides +5
Target Protein:
cGMP-dependent 3',5'-cyclic phosphodiesterasePotassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 2cAMP-dependent protein kinase type I-alpha regulatory subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cyclizine Approved DB01176
small molecule | CAS: 82-92-8

A histamine H1 antagonist given by mouth or parenterally for the control of postoperative and drug-induced vomiting and in motion sickness. (From Martindale, The Extra Pharmacopoeia, 30th ed, p935)

Kategori:
AntiemeticsAntihistamines for Systemic UseAutonomic Agents +15
Target Protein:
Histamine H1 receptorSulfotransferase 1E1
Waktu Paruh20 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 97011-16-0

NA-831 (Traneurocin), is under investigation in two clinical trials: NCT03538522 (completed, for mild cognitive impairment and Alzheimer’s disease) and NCT04452565 (unknown status, combination therapy with Atazanavir and Dexamethasone for COVID-19).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Chitinase B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cyclobenzaprine Approved DB00924
small molecule | CAS: 303-53-7

Cyclobenzaprine, a centrally-acting muscle relaxant, was first synthesized in 1961[A185039] and has been available for human use since 1977.[A184982] It was initially studied for use as antidepressant given its structural similarity to tricyclic antidepressan…

Kategori:
Agents that reduce seizure thresholdAntidepressive AgentsBenzocycloheptenes +23
Target Protein:
Alpha-2C adrenergic receptor5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2B +7
Waktu ParuhThe effective half-…
Vol. DistribusiThe volume of distr…
KlirensThe approximate pla…
Genetik -
Cyclobutyrol DB13493
small molecule | CAS: 512-16-3

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAlimentary Tract and MetabolismBile and Liver Therapy +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cyclocreatine DB17624
small molecule | CAS: 35404-50-3

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntineoplastic Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 701-97-3

Deskripsi belum tersedia.

Target Protein:
Aromatic-amino-acid aminotransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cyclohexanol DB03703
small molecule | CAS: 108-93-0

Monohydroxy derivatives of cyclohexanes that contain the general formula R-C6H11O. They have a camphorlike odor and are used in making soaps, insecticides, germicides, dry cleaning, and plasticizers. [PubChem]

Kategori:
AlcoholsCyclohexanesCycloparaffins +3
Target Protein:
Beta-lactamaseAll-trans-retinol dehydrogenase [NAD(+)] ADH1B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cycloleucine DB04620
small molecule | CAS: 52-52-8

Cycloleucine is non-metabolisable amino acid formed by cyclization of leucine. It is also a specific and reversible inhibitor of nucleic acid methylation and widely used in biochemical experiments.

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +2
Target Protein:
Glutamate receptor ionotropic, NMDA 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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