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11793

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8607 (73.0%)
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6418 (54.4%)
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102 (0.9%)
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11793 (100.0%)

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Hasil Pencarian (11793)

Halaman 42 / 236
small molecule | CAS: 118-92-3

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +2
Target Protein:
L-amino-acid oxidaseD-amino-acid oxidase
Waktu Paruh-
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Genetik -
Anthrax vaccine Approved DB11003
biotech

Anthrax vaccine is a vaccine used for the pre- or post-exposure prophylaxis of disease in those at high risk of, suspected or confirmed exposure to *Bacillus anthracis*. It is subcutaneously or intramuscularly administered. It is derived from cell-free filtra…

Kategori:
Actively Acquired ImmunityAnthrax VaccinesBacterial Vaccines +6
Waktu ParuhLimited information…
Vol. DistribusiLimited information…
KlirensLimited information…
Genetik -
biotech

A macrocyclic peptide (BMS-986189) with activity in binding and functional assays comparable to a PD-L1 antibody.

Kategori:
Immune Checkpoint Inhibitors
Target Protein:
Programmed cell death 1 ligand 1
Waktu Paruh-
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Genetik -
biotech

Anti-SARS-CoV-2 equine immunoglobulin fragments, also known as INOSARS, is a polyvalent passive immunization being tested in the clinical trial NCT04514302 (Safety and Efficacy of Anti-SARS-CoV-2 Equine Antibody Fragments (INOSARS) for Hospitalized Patients W…

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Genetik -
biotech

Anti-SARS-CoV-2 IgY are chicken egg antibodies to SARS-CoV-2 which have the potential to provide temporary protection against the virus when administered as intranasal drops.[L27381] To create these antibodies, chickens are injected in the chest with the spik…

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Genetik -
biotech

Hyperimmune immunoglobulin to SARS-CoV-2 (hIVIG) is obtained from the plasma of patients who recover from COVID-19 and develop neutralizing antibodies.[L27521] Anti-coronavirus immunoglobulin is derived from [COVID-19 convalescent plasma](https://go.drugbank.…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +8
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Genetik -
biotech

Anti-SARS-COV-2 REGN-COV2 is a combination of novel antibodies designed by Regeneron for both the prevention and treatment of SARS-COV-2, the virus that causes COVID-19. This drug is a combination of the antibodies REGN10933 and REGN10987, derived from human…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +10
Target Protein:
Spike glycoprotein
Waktu Paruh-
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Genetik -
biotech | CAS: 1628187-15-4

Antihemophilic Factor (Recombinant), PEGylated, was approved by the FDA in December 2016 as the product _Adynovate_ [FDA label]. Antihemophilic Factor (Recombinant), PEGylated, is a recombinant full-length human coagulation factor VIII (2,332 amino acids w…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +14
Target Protein:
von Willebrand factor
Waktu Paruh14.69 ± 3.79h for a…
Vol. DistribusiAt steady state: 0.…
Klirens2.27 ± 0.84 for adu…
Genetik -
Antihemophilic factor human Approved DB13192
biotech

Antihemophilic factor human, also known as Coagulation Factor VIII or Anti-Hemophilic Factor (AHF), is a non-recombinant, lyophilized concentrate of coagulation factor VIII, an endogenous protein and essential component of the coagulation cascade. Antihemophi…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +11
Target Protein:
Coagulation factor IXCoagulation factor X
Waktu ParuhThe mean half-life …
Vol. DistribusiThe pharmacokinetic…
KlirensThe reported cleara…
Genetik -
biotech | CAS: 139076-62-3

Human recombinant antihemophilic factor (AHF) or Factor VIII, 2332 residues, glycosylated, produced by CHO cells

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +12
Target Protein:
Coagulation factor XCoagulation factor IXvon Willebrand factor +8
Waktu Paruh8.4-19.3 hrs
Vol. Distribusi-
Klirens* 4.1 mL/h•kg [Prev…
Genetik -
Antimony DB13110
small molecule | CAS: 7440-36-0

Antimony has been used in trials studying the treatment of Cutaneous Leishmaniasis.

Kategori:
ElementsMetalloidsMetals +1
Waktu Paruh-
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small molecule | CAS: 91531-30-5

Antineoplaston A10 has been used in trials studying the treatment of Sarcoma, Lymphoma, Lung Cancer, Liver Cancer, and Kidney Cancer, among others.

Kategori:
AcetamidesAmidesBenzene Derivatives +1
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Antipain DB15251
small molecule | CAS: 37691-11-5

Antipain is a serine/cysteine protease inhibitor originally isolated from various strains of actinomycetes.[A214481] Early studies investigated the potential for antipain to alter DNA damage and chromosomal aberrations in irradiated cells or those treated wit…

Kategori:
Amino Acids, Peptides, and ProteinsEnzyme InhibitorsOligopeptides +2
Waktu Paruh-
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Antipyrine Approved DB01435
small molecule | CAS: 60-80-0

An analgesic and antipyretic that has been given by mouth and as ear drops. Antipyrine is often used in testing the effects of other drugs or diseases on drug-metabolizing enzymes in the liver. (From Martindale, The Extra Pharmacopoeia, 30th ed, p29)

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +30
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh-
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Antithrombin Alfa Approved DB11166
biotech | CAS: 84720-88-7

Antithrombin Alfa is a recombinant antithrombin , an anticoagulant, that is used for the prevention of thromboembolic events in patients that have hereditary deficiency of antithrombin in high risk situations.

Kategori:
AnticoagulantsDecreased Coagulation Factor ActivityFactor Xa Inhibitors +2
Target Protein:
ProthrombinCoagulation factor X
Waktu ParuhDose of: 50IU/kg: …
Vol. DistribusiDose of: 50IU/kg: …
KlirensDose of: 50IU/kg: …
Genetik -
biotech | CAS: 1311281-25-0

Antithrombin gamma is under investigation in clinical trial NCT04182373 (KW-3357 Study in Patients With Early Onset Severe Preeclampsia).

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Antithrombin III human Approved DB11598
biotech | CAS: 9000-94-6

A plasma alpha 2 glycoprotein that accounts for the major antithrombin activity of normal plasma and also inhibits several other enzymes. It is a member of the serpin superfamily.

Kategori:
Alpha-GlobulinsAmino Acids, Peptides, and ProteinsAnticoagulants +18
Target Protein:
Antithrombin-III
Waktu Paruh2.5 - 3.8 hs
Vol. DistribusiDistributed into pl…
Klirens-
Genetik -
biotech | CAS: 308067-60-9

Rabbit anti-thymocyte globulin. Thymoglobulin is a polyclonal antibody that suppresses certain types of immune cells responsible for acute organ rejection in transplant patients. Thymoglobulin is a mixture of antibodies intended to bind to various cell surfac…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibody-Surface Protein Interactions +22
Target Protein:
Major histocompatibility complex class I-related gene proteinIntegrin alpha-LT-lymphocyte activation antigen CD86 +6
Waktu Paruh2-3 days, may incre…
Vol. Distribusi-
Klirens-
Genetik -
Antroquinonol DB12326
small molecule | CAS: 1010081-09-0

Antroquinonol has been used in trials studying the treatment of Hyperlipidemias, Non-small Cell Lung Cancer, and Non-small Cell Lung Cancer Stage IV.

Kategori:
BenzoquinonesCoenzymesEnzymes and Coenzymes +1
Target Protein:
DNA (cytosine-5)-methyltransferase 1
Waktu Paruh-
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Genetik -
biotech | CAS: 2636710-07-9

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ANX-005 DB16977
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
ANZ-100 DB05967
small molecule

Deskripsi belum tersedia.

Target Protein:
KiSS-1 receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Anzurstobart DB17547
biotech | CAS: 2543693-10-1

Anzurstobart is a monoclonal antibody directed against signal-regulatory protein alpha (SIRP?) on monocytes and macrophages to potently block the CD47-SIRP? interaction. It is being investigated for cancers.

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Genetik -
AO-176 DB18287
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
AOC 1001 DB18620
biotech | CAS: 2653183-66-3

Delpacibart (AOC 1001) is being investigated in a global study for the treatment of Myotonic Dystrophy type 1 (DM1) in clinical trial NCT06411288

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AOC-1020 DB18621
biotech

AOC-1020 is an antibody oligonucleotide conjugate, comprised of a human transferrin receptor 1 targeting, effector function null, humanized IgG1 antibody, a MCC maleimide linker, and a double-stranded siRNA oligonucleotide targeting DUX4.

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AOD9604 DB06388
small molecule | CAS: 221231-10-3

AOD9604 is a synthetic analogue of the lipolytic domain of human growth hormone, being investigated for the treatment of obesity.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +8
Waktu Paruh-
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Genetik -
AP-001 DB18511
small molecule | CAS: 660430-03-5

Deskripsi belum tersedia.

Kategori:
Dietary FatsDietary Fats, UnsaturatedFats +6
Waktu Paruh-
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Genetik -
AP-102 DB18206
small molecule | CAS: 846569-60-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AP-22408 DB01830
small molecule | CAS: 268741-43-1

Deskripsi belum tersedia.

Target Protein:
Proto-oncogene tyrosine-protein kinase SrcTyrosine-protein kinase Lck
Waktu Paruh-
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Genetik -
AP5346 DB04992
small molecule

AP5346 is designed to target a diaminocyclohexane platinum (Pt) moiety to tumors through pH-sensitive linkage to a 25 kDa hydroxypropylmethacrylamide polymer. It is being pursued by Access Pharmaceuticals, Inc.

Kategori:
Organometallic Compounds
Target Protein:
DNA
Waktu Paruh-
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Genetik -
Apadamtase alfa Approved DB15164
biotech | CAS: 2086325-24-6

Thrombotic thrombocytopenic purpura (TTP) is a rare blood clotting disorder characterized by thrombocytopenia, microangiopathic hemolytic anemia, and various degrees of organ damage.[A262076] It may be inherited (congenital TTP; cTTP) or acquired due to autoa…

Kategori:
ADAM ProteinsADAMTS ProteinsAmino Acids, Peptides, and Proteins +12
Target Protein:
von Willebrand factor
Waktu ParuhFollowing the intra…
Vol. Distribusi-
Klirens-
Genetik -
Apadenoson DB05009
small molecule | CAS: 250386-15-3

Apadenoson is a selective A2a adenosine receptor agonist designed for use as a pharmacologic stress agent in cardiac perfusion imaging studies. It is developed by Bristol-Myers Squibb and is in phase II of clinical trials.

Kategori:
Acids, CarbocyclicAdenosine A receptor agonistsAdenosine A2 Receptor Agonists +7
Target Protein:
Adenosine receptor A2a
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apalutamide Approved DB11901
small molecule | CAS: 956104-40-8

Apalutamide is a potent androgen receptor (AR) antagonist that selectively binds to the ligand-binding domain of AR and blocks AR nuclear translocation or binding to androgen response elements [A31846]. It has been used in trials studying the treatment of Pro…

Kategori:
Androgen Receptor InhibitorsAntiandrogensAntineoplastic Agents +28
Target Protein:
Androgen receptorGABA(A) Receptor
Waktu ParuhThe mean effective …
Vol. DistribusiThe mean apparent v…
KlirensThe CL/F of apaluta…
Genetik -
biotech | CAS: 2097132-02-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Apararenone DB15024
small molecule | CAS: 945966-46-1

Apararenone is under investigation in clinical trial NCT02531568 (Drug Interaction Study of Warfarin and MT-3995).

Kategori:
AmidesSulfonesSulfur Compounds
Waktu Paruh-
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Genetik -
Apatorsen DB06094
biotech | CAS: 1002331-21-6

Apatorsen is a second generation antisense drug which in preclinical experiments, inhibits production of Heat Shock Protein 27 (Hsp27) a cell survival protein found at elevated levels in many human cancers including prostate, lung, breast, ovarian, bladder, r…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
Heat shock protein beta-1
Waktu Paruh-
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Genetik -
Apaziquone DB12593
small molecule | CAS: 114560-48-4

Apaziquone has been investigated for the treatment of Bladder Cancer and Bladder Neoplasms.

Kategori:
Antineoplastic AgentsAzirinesHeterocyclic Compounds, Fused-Ring +2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
APD-209 DB18759
small molecule | CAS: 1261156-82-4

Deskripsi belum tersedia.

Target Protein:
Beta-2 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
APD668 DB05166
small molecule

APD668 is a novel, highly potent and orally active glucose-dependent insulinotropic receptor (GDIR) agonist intended to more efficiently stimulate insulin release by beta cells in response to elevated blood glucose levels, and to also avoid hypoglycemia.

Target Protein:
Glucose-dependent insulinotropic receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
APG-1387 DB16095
small molecule | CAS: 1570231-89-8

APG-1387 is under investigation in clinical trial NCT04568265 (A Clinical Study of APG-1387 in Combination With Entecavir in Patients With Chronic Hepatitis B).

Kategori:
AmidesSulfonesSulfur Compounds
Target Protein:
E3 ubiquitin-protein ligase XIAPBaculoviral IAP repeat-containing protein 2Baculoviral IAP repeat-containing protein 3 +3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
APG-157 DB18683
small molecule

APG-157 consists of zinflavonoids being investigated for the treatment of cancers.

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Genetik -
Aphidicolin DB17742
small molecule | CAS: 38966-21-1

Aphidicolin is an antimitotic and antiviral metabolite of the mould _Cephalosporium aphidicola_. It inhibits DNA polymerase alpha and blocks DNA replication.[A259157, A259162]

Kategori:
Anti-Infective AgentsAntiviral AgentsDiterpenes +2
Target Protein:
DNA polymerase catalytic subunit
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Apigenin DB07352
small molecule | CAS: 520-36-5

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavones +3
Target Protein:
Casein kinase II subunit alphaAldo-keto reductase family 1 member B1Cytochrome P450 1B1 +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apilimod DB05611
small molecule | CAS: 541550-19-0

Deskripsi belum tersedia.

Kategori:
HydrazinesOxazines
Target Protein:
1-phosphatidylinositol 3-phosphate 5-kinaseInterleukin-12 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Apinocaltamide DB16241
small molecule | CAS: 1838651-58-3

Apinocaltamide is under investigation in clinical trial NCT03239691 (A Study to Evaluate the Effect of ACT-709478 in Photosensitive Epilepsy Patients).

Kategori:
AcetatesAcids, AcyclicAmides +5
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Apitegromab DB16096
biotech | CAS: 2278276-46-1

Apitegromab is under investigation in clinical trial NCT03921528 (An Active Treatment Study of SRK-015 in Patients With Type 2 or Type 3 Spinal Muscular Atrophy).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Apixaban Approved DB06605
small molecule | CAS: 503612-47-3

Apixaban is an oral, direct, and highly selective factor Xa (FXa) inhibitor of both free and bound FXa, as well as prothrombinase, independent of antithrombin III for the prevention and treatment of thromboembolic diseases[Label,A6897]. It is marketed under t…

Kategori:
AnticoagulantsAntithrombinsBCRP/ABCG2 Substrates +17
Target Protein:
Coagulation factor X
Waktu Paruh12.7±8.55h[Label,A1…
Vol. DistribusiApproximately 21L[L…
Klirens3.3L/h[Label] thoug…
Genetik -
APL-502 DB17473
biotech | CAS: 2303884-58-2

APL 502 is a humanised immunoglobulin G1 (IgG1) monoclonal antibody targeting the programmed cell death-1 ligand-1 (PD-L1).

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APL-9 DB16460
small molecule

APL-9 is an investigational drug intended to centrally control the complement cascade at C3, potentially treating various diseases caused by excessive or uncontrolled complement activation. It shares the same mechanism of action as Apellis’ lead compound, peg…

Kategori:
Experimental Unapproved Treatments for COVID-19
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