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12560

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9109 (72.5%)
Target
6912 (55.0%)
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109 (0.9%)
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12560 (100.0%)

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Halaman 42 / 252
Alflorex Approved DB18507
biotech

Alflorex is a probiotic with 35624 cultures, part of the Bifidobacterium longum.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alflutinib DB16087
small molecule | CAS: 1869057-83-9

Alflutinib is under investigation in clinical trial NCT03452592 (Efficacy and Safety of Alflutinib in Locally Advanced or Metastatic Non-small Cell Lung Cancer Patients With T790M).

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alfuzosin Approved DB00346
small molecule | CAS: 81403-80-7

Benign prostatic hyperplasia (BPH) refers to a benign growth or hyperplasia of the prostate and leads to lower urinary tract symptoms in men, such as urgency, frequency and changes to urine flow. The prevalence of BPH is as high as 50%-60% for males in their …

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +17
Target Protein:
Alpha-1 adrenergic receptorsAlpha-1A adrenergic receptorAlpha-1B adrenergic receptor +1
Waktu ParuhThe apparent elimin…
Vol. DistribusiThe volume of distr…
KlirensExercise caution if…
Genetik -
Algestone DB18000
small molecule | CAS: 595-77-7

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesContraceptive Agents, FemaleContraceptive Agents, Hormonal +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 24356-94-3

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesAlgestoneAnti-Inflammatory Agents +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alginic acid Approved DB13518
small molecule | CAS: 9005-32-7

Alginic acid, also referred to as algin or alginate, is a hydrophilic or anionic polysaccharide isolated from certain brown seaweed (_Phacophycae_) via alkaline extraction. It is present in cell walls of brown algae where it forms a viscous gel when binding w…

Kategori:
Acids, AcyclicAcids, AldehydicAlginates +11
Waktu ParuhThis pharmacokineti…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Alglucerase Approved DB00088
biotech | CAS: 143003-46-7

Human Beta-glucocerebrosidase or Beta-D-glucosyl-N-acylsphingosine glucohydrolase E.C. 3.2.1.45. 497 residue protein with N-linked carbohydrates, MW=59.3 kD. Alglucerase is prepared by modification of the oligosaccharide chains of human Beta-glucocerebrosidas…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +6
Target Protein:
Glucocerebroside
Waktu Paruh3.6-10.4 min
Vol. Distribusi* 49.4 to 282.1 mL/…
Klirens-
Genetik -
Alglucosidase alfa Approved DB01272
biotech | CAS: 420784-05-0

Aglucosidase alfa consists of the human enzyme acid alpha-glucosidase (GAA) which is essential for the degradation of glygogen to glucose in lysosomes. It is encoded by the most predominant of nine observed haplotypes of this gene. Aglucosidase alfa is produc…

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes +5
Target Protein:
Cation-dependent mannose-6-phosphate receptorGlycogen
Waktu Paruh2.3 ± 0.4 ho…
Vol. Distribusi* 96 ± 16 mL/kg [20…
Klirens* 25+/- 4 mL/hr/kg …
Genetik -
Alicaforsen DB06224
small molecule | CAS: 185229-68-9

Deskripsi belum tersedia.

Kategori:
Gastrointestinal AgentsImmunologic FactorsNucleic Acids, Nucleotides, and Nucleosides +3
Target Protein:
Intercellular adhesion molecule 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alintegimod DB18879
small molecule | CAS: 1378535-08-0

Alintegimod is under investigation in clinical trial NCT06362369 (A Study of Oral 7HP349 (Alintegimod) in Combination With Ipilimumab Followed by Nivolumab Monotherapy).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alipogene tiparvovec Approved DB13521
biotech | CAS: 929881-05-0

Alipogene tiparvovec is an adeno-associated viral vector of serotype 1-based gene therapy that delivers the Ser(447)X variant of the human lipoprotein lipase (LPL) gene. It is being investigated for the treatment of lipoprotein lipase (LPL) deficiency.[A25979…

Kategori:
Adeno-associated Viral Vector TherapiesLipid Modifying AgentsLipid Modifying Agents, Plain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alirinetide DB17007
biotech | CAS: 725715-18-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alirocumab Approved DB09302
biotech | CAS: 1245916-14-6

Alirocumab is a biopharmaceutical that obtained FDA approval in July 2015 as a second line treatment for high cholesterol in adults whose LDL-cholesterol (LDL-C) is not controlled by the combination of diet and statin treatment. It is a human monoclonal antib…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +20
Target Protein:
Proprotein convertase subtilisin/kexin type 9
Waktu ParuhIn monotherapy, the…
Vol. DistribusiAlirocumab is mainl…
Klirens-
Genetik -
Alisertib DB05220
small molecule | CAS: 1028486-01-2

Alisertib is a novel aurora A kinase inhibitor under investigation for the treatment of various forms of cancer.

Kategori:
Protein Kinase Inhibitors
Target Protein:
Aurora kinase A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aliskiren Approved DB09026
small molecule | CAS: 173334-57-1

Aliskiren is the first drug in the renin inhibitor drug class and is used for the treatment of hypertension.[A203624] It was developed by Speedel and Novartis and initially approved by the FDA in early 2007.[L14018] Aliskiren has been proven to efficacious in…

Kategori:
Acids, AcyclicAgents Acting on the Renin-Angiotensin SystemAgents causing hyperkalemia +14
Target Protein:
Renin
Waktu ParuhPlasma half-life fo…
Vol. DistribusiUnchanged aliskiren…
KlirensAliskiren is partia…
Genetik -
Alisporivir DB12139
small molecule | CAS: 254435-95-5

Alisporivir has been used in trials studying the treatment of Hepatitis C and Chronic Hepatitis C.

Kategori:
Amino Acids, Peptides, and ProteinsCyclosporin DerivativesPeptides +1
Target Protein:
Guided entry of tail-anchored proteins factor CAMLG
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alitretinoin Approved DB00523
small molecule | CAS: 5300-03-8

An important regulator of gene expression during growth and development, and in neoplasms. Tretinoin, also known as retinoic acid and derived from maternal vitamin A, is essential for normal growth; and embryonic development. An excess of tretinoin can be ter…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAlkenesAntineoplastic Agents +19
Target Protein:
Retinoic acid receptor alphaRetinoic acid receptor RXR-alphaRetinoic acid receptor beta +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alizapride DB01425
small molecule | CAS: 59338-93-1

Alizapride is a dopamine antagonist that is capable of demonstrating both prokinetic and antiemetic effects. This kind of pharmacological activity makes it effective for use in the treatment of various kinds of nausea and vomiting, including that which may oc…

Kategori:
Alimentary Tract and MetabolismAntiemeticsAutonomic Agents +7
Target Protein:
D(2) dopamine receptor
Waktu Paruh3 hours
Vol. Distribusi-
Klirens-
Genetik -
ALK-4290 DB15269
small molecule | CAS: 1251528-23-0

ALK-4290 is under investigation in clinical trial NCT03558061 (Evaluate the Effects and Safety of ALK4290 in Patients With Newly Diagnosed Wet Age-Related Macular Degeneration).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Alkaline Phosphatase (AP) is an oral treatment and has a very favorable side-effect profile. AP only acts locally in the colon to reduce the continuous inflammation of the colon by endotoxin from Gram-negative bacteria and extracellular ATP in UC patients.

Kategori:
EnzymesEnzymes and CoenzymesEsterases +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ALKS 27 DB05752
small molecule

ALKS 27 is an inhaled formulation of trospium chloride for the treatment of chronic obstructive pulmonary disease (COPD). Study showed that ALKS 27 was well-tolerated over a wide dose range, with no dose-limited effects observed.

Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ALKS 29 DB05723
small molecule

ALKS 29 is a new product candidate for the treatment of alcohol dependence. It is being developed by Alkermes, Inc.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Allantoin Approved DB11100
small molecule | CAS: 97-59-6

Allantoin is a substance that is endogenous to the human body and also found as a normal component of human diets [FDA Label]. In healthy human volunteers, the mean plasma concentration of allantoin is about 2-3 mg/l. During exercise, the plasma allantoin con…

Kategori:
AmidesBasic Ointments and ProtectantsDermatologicals +5
Waktu ParuhWhen studied in cat…
Vol. Distribusi-
KlirensSome studies sugges…
Genetik -
biotech

Allenrolfea occidentalis pollen is the pollen of the Allenrolfea occidentalis plant. Allenrolfea occidentalis pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Allicin DB11780
small molecule | CAS: 539-86-6

Allicin has been used in trials studying the treatment of Follicular Lymphoma.

Kategori:
AcidsAcids, NoncarboxylicAnions +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 947331-05-7

Allisartan isoproxil is under investigation in clinical trial NCT03264352 (Intervention for High-normal Blood Pressure in Adults With Type 2 Diabetes).

Kategori:
Agents Acting on the Renin-Angiotensin SystemAngiotensin II receptor antagonistsAngiotensin II Type 1 Receptor Blockers +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ALLO-605 DB18641
biotech

ALLO-605 is an allogeneic turbo chimeric antigen receptor (Turbocar) T Cell therapy targeting B Cell maturation antigen (BCMA).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
ALLO-715 DB18640
biotech

ALLO-715 is an allogeneic chimeric antigen receptor T Cell therapy targeting B cell maturation antigen (BCMA).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Allobarbital DB13577
small molecule | CAS: 52-43-7

Deskripsi belum tersedia.

Kategori:
Barbiturates, PlainCentral Nervous System DepressantsHypnotics and Sedatives +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Cardiosphere-derived cells (CDCs) are derived from human neonatal heart tissue with a distinct antigenic profile (CD105+, CD45-, and CD90low). They exert their effects by secreting exosomes: nanometer-sized, membrane-bound vesicles used for the purpose of cel…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Stratagraft (allogeneic cultured keratinocytes and dermal fibroblasts in murine collagen-dsat) is an allogeneic cellularized scaffold product used for the treatment of adults with thermal burns containing intact dermal elements for which surgical intervention…

Kategori:
FibroblastsKeratinocytes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

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Vol. Distribusi-
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Genetik -
biotech

ORBCEL-C™ is the trade name of a product composed of highly purified stromal cells derived from the human umbilical cord. The isolated cells are expanded in culture and are able to be used allogenically -- meaning that one donor’s cells can be given to other …

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Vol. Distribusi-
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Genetik -
biotech

Umbilical-cord derived MSCs are currently being tested for numerous clinical applications due to their immunosuppressive and anti-inflammatory properties. In comparison to bone-marrow derived MSCs, these cells are more resilient, easier to extract, and genera…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Human olfactory mucosa-derived mesenchymal stem cells (OM-MSCs) reside in an accessible location of the nasal cavity and have properties of multipotency and high proliferation, which contributes to high potential for regenerative medicine. In humans, OM-MSCs …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alloin Approved DB15477
small molecule | CAS: 8015-61-0

Deskripsi belum tersedia.

Kategori:
AnthracenesAnthraquinonesBiological Products +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Allolactose DB04116
small molecule | CAS: 645-03-4

Deskripsi belum tersedia.

Kategori:
CarbohydratesDisaccharidesOligosaccharides +1
Target Protein:
Beta-galactosidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Allopurinol Approved DB00437
small molecule | CAS: 315-30-0

Gout is a disease that occurs by the deposition of monosodium urate crystals (MSU) in body tissues, especially around joints [A175942]. This disease has been well-documented in historical medical records and appears in the biographies of several prominent, h…

Kategori:
Antigout PreparationsAntimetabolitesAntioxidants +12
Target Protein:
Xanthine dehydrogenase/oxidase
Gen Terkait:
HCP5
Waktu ParuhThe plasma half-lif…
Vol. DistribusiAllopurinol and oxy…
KlirensSince allopurinol a…
Genetik 1 Varian
small molecule | CAS: 16220-07-8

Allopurinol riboside is a nucleoside analogue of [allopurinol] with a beta-D-ribofuranosyl moiety at the 1-position.

Kategori:
Anti-Infective AgentsAntiparasitic AgentsAntiprotozoals +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Allovectin-7 DB17439
biotech | CAS: 190857-15-9

Allovectin-7 or allovectin-7(r) is a lipid complex that contains the DNA sequences encoding HLA-B7 and beta-2 microglobulin. It was discontinued after it failed to improve the objective response rate or overall survival versus first-line chemotherapy in malig…

Kategori:
LiposomesNucleic AcidsNucleic Acids, Nucleotides, and Nucleosides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Allylprodine DB01542
small molecule | CAS: 25384-17-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Allysine DB02571
small molecule | CAS: 6665-12-9

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAdipatesAmino Acids +3
Target Protein:
Glutaminase-asparaginase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ALM201 DB17206
biotech

ALM201 is an anti-angiogenic synthetic peptide identified from the endogenous human protein, FKBPL. It is being investigated in the treatment of various cancers.[A254556]

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Almasilate Approved DB13595
small molecule | CAS: 71205-22-6

Almasilate is a buffering antacid that has been used in peptic ulcers and dyspepsia. It is a crystalline polyhydrate of aluminium/magnesium silicate and mediates its buffering activity by binding hydrogen ions within the polymer. However its therapeutic effic…

Kategori:
Alimentary Tract and MetabolismAluminum and magnesium containing antacidsAntacids +6
Waktu ParuhReadily accessible …
Vol. DistribusiThe distribution of…
KlirensReadily accessible …
Genetik -
Almitrine Approved DB01430
small molecule | CAS: 27469-53-0

Almitrine is a respiratory stimulant that enhances respiration by acting as an agonist of peripheral chemoreceptors located on the carotid bodies. It is used in the treatment of chronic obstructive pulmonary disease. It is also reported to have a potentially …

Kategori:
AlkaloidsCentral Nervous System AgentsCompounds used in a research, industrial, or household setting +12
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Almond Approved DB10500
biotech

Almond allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Almonertinib DB16640
small molecule | CAS: 1899921-05-1

Almonertinib is a third-generation EGFR tyrosine kinase inhibitor targeting EGFR-sensitizing and T790M resistance mutations.[A231859, A231864, A231869] It is being investigated against advanced or metastatic EGFR-mutated non-small cell lung cancer (NSCLC).[A2…

Kategori:
Acids, AcyclicAcrylatesAmides +1
Target Protein:
Epidermal growth factor receptorReceptor protein-tyrosine kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Almorexant DB06673
small molecule | CAS: 871224-64-5

Deskripsi belum tersedia.

Kategori:
AcetatesAcids, AcyclicAmides +1
Target Protein:
Orexin/Hypocretin receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Almotriptan Approved DB00918
small molecule | CAS: 154323-57-6

Almotriptan is a triptan drug for the treatment of migraine headaches. Almotriptan is in a class of medications called selective serotonin receptor agonists. It works by narrowing blood vessels in the brain, stopping pain signals from being sent to the brain,…

Kategori:
Agents that produce hypertensionAminesAnalgesics +30
Target Protein:
5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 1B
Gen Terkait:
GNB3
Waktu Paruh3-4 hours
Vol. Distribusi* 180 to 200 L
Klirens* 57 L/h [healthy] …
Genetik 1 Varian
Menampilkan 2051–2100 dari 12560
Sebelumnya Halaman 42 / 252 Berikutnya