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3253

Total database: 17430
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2451 (75.3%)
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1833 (56.3%)
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35 (1.1%)
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3253 (100.0%)

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Halaman 42 / 66
Nemolizumab Approved DB15252
biotech | CAS: 1476039-58-3

Nemolizumab is a humanized monoclonal modified immunoglobulin 2 (IgG2) antibody directed against interleukin-31 receptor alpha (IL-31RA),[L51159] which is an endogenous cytokine implicated in the pathophysiology of various skin inflammatory disorders.[A264254…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAmino Acids, Peptides, and ProteinsAntibodies +10
Target Protein:
Interleukin-31 receptor subunit alpha
Waktu ParuhThe estimated termi…
Vol. DistribusiThe estimated volum…
KlirensThe estimated syste…
Genetik -
biotech | CAS: 2315268-27-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NEO-212 DB17100
small molecule | CAS: 1361198-79-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Neosaxitoxin DB12989
small molecule | CAS: 64296-20-4

Neosaxitoxin is under investigation in clinical trial NCT01786655 (Safety Study of Long-Acting Local Anesthetic).

Kategori:
AgrochemicalsBacterial ToxinsBiological Factors +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nepadutant DB12538
small molecule | CAS: 183747-35-5

Nepadutant has been used in trials studying the treatment of Colic, Infantile Colic, and Infantile Functional Gastrointestinal Disorders.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Asthmatic AgentsAutonomic Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nepicastat DB12979
small molecule | CAS: 173997-05-2

Nepicastat has been investigated for the treatment of Cocaine Dependence and Posttraumatic Stress Disorder.

Kategori:
Dopamine beta-Hydroxylase, antagonists & inhibitorsSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nerinetide DB12595
biotech | CAS: 500992-11-0

Na 1 is under investigation in clinical trial NCT00728182 (Evaluating Neuroprotection in Aneurysm Coiling Therapy).

Kategori:
Amino Acids, Peptides, and ProteinsNeuroprotective Agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nerispirdine DB12714
small molecule | CAS: 119229-65-1

Nerispirdine has been used in trials studying the treatment of Neuritis, Optic Nerve, and Multiple Sclerosis.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Voltage-gated inwardly rectifying potassium channel KCNH2Sodium channel protein type 11 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nerofe DB14786
small molecule | CAS: 1311294-45-7

Nerofe is under investigation in clinical trial NCT03059615 (A Phase 2a, Open-Label, Two Stage Study of Nerofe or Nerofe With Doxorubicin in Subjects With AML or MDS).

Kategori:
Amino Acids, Peptides, and Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 9061-61-4

Nerve Growth Factor has been used in trials studying the prevention and treatment of Mental Handicap, Alzheimer's Disease, Traumatic Brain Injury, Cerebral Palsy Children, and Delayed Speech Development, among others.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nesiritide Approved DB04899
biotech | CAS: 124584-08-3

Nesiritide is a medication used to treat acutely decompensated congestive heart failure with dyspnea at rest or with minimal exertion (such as talk, eating or bathing). Nesiritide is a 32 amino acid recombinant human B-type natriuretic peptide.

Kategori:
Amino Acids, Peptides, and ProteinsCardiac TherapyCardiovascular Agents +11
Target Protein:
Atrial natriuretic peptide receptor 1Atrial natriuretic peptide receptor 2Atrial natriuretic peptide receptor 3
Waktu ParuhApproximately 18 mi…
Vol. Distribusi* 0.19 L/kg
Klirens* 9.2 mL/min/k [pat…
Genetik -
Nesvacumab DB15330
biotech | CAS: 1296818-77-3

Nesvacumab is under investigation in clinical trial NCT01997164 (Study of Intravitreal (IVT) REGN910-3 and IVT REGN910 in Patients With Either Neovascular (Wet) Age Related Macular Degeneration (AMD) or Diabetic Macular Edema (DME)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Netarsudil Approved DB13931
small molecule | CAS: 1254032-66-0

A Rho kinase inhibitor with norepinephrine transport inhibitory activity that reduces production of aqueous As of December 18, 2017 the FDA approved Aerie Pharmaceutical's Rhopressa (netarsudil ophthalmic solution) 0.02% for the indication of reducing elev…

Kategori:
Acids, CarbocyclicAlanineAmino Acids +8
Target Protein:
Rho-associated protein kinase 1Rho-associated protein kinase 2Sodium-dependent noradrenaline transporter
Waktu ParuhThe half-life of ne…
Vol. DistribusiAs netarsudil and i…
KlirensThe clearance of ne…
Genetik -
Netazepide DB12355
small molecule | CAS: 155488-25-8

Netazepide has been used in trials studying the prevention and treatment of Dyspepsia, Hypergastrinaemia, Barrett's Esophagus, ECL-cell Hyperplasia, and Rebound Hyperacidity, among others.

Kategori:
AmidesBenzazepinesBenzene Derivatives +2
Target Protein:
Gastrin/cholecystokinin type B receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Netivudine DB12606
small molecule | CAS: 84558-93-0

Netivudine has been used in trials studying the treatment of Chickenpox and HIV Infections.

Kategori:
Anti-Infective AgentsAntiviral AgentsArabinonucleosides +4
Target Protein:
DNA polymerase catalytic subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nevirapine Approved DB00238
small molecule | CAS: 129618-40-2

A potent, non-nucleoside reverse transcriptase inhibitor (NNRTI) used in combination with nucleoside analogues for treatment of Human Immunodeficiency Virus Type 1 (HIV-1) infection and AIDS. Structurally, nevirapine belongs to the dipyridodiazepinone chemica…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +39
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Waktu Paruh45 hours
Vol. Distribusi* 1.21 ± 0.09 L/kg …
Klirens-
Genetik -
Nialamide Approved DB04820
small molecule | CAS: 51-12-7

Withdrawn from the Canadian, US, and UK markets in 1963 due to interactions with food products containing tyrosine.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +11
Target Protein:
Amine oxidase [flavin-containing] BAmine oxidase [flavin-containing] ACatechol O-methyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nicoboxil Approved DB12911
small molecule | CAS: 13912-80-6

Nicoboxil has been investigated for the treatment of Acute Low Back Pain, where it is typically considered an effective and safe therapeutic option. Nevertheless, it is predominantly found paired with nonivamide as a combination topical analgesic product wher…

Kategori:
Drugs that are Mainly Renally ExcretedPyridines
Waktu ParuhThe half-life of es…
Vol. DistribusiDespite the fact th…
KlirensThe elimination of …
Genetik -
Nicotine Approved DB00184
small molecule | CAS: 54-11-5

Nicotine is highly toxic alkaloid. It is the prototypical agonist at nicotinic cholinergic receptors where it dramatically stimulates neurons and ultimately blocks synaptic transmission. Nicotine is also important medically because of its presence in tobacco …

Kategori:
Agents producing tachycardiaAlkaloidsAutonomic Agents +40
Target Protein:
Neuronal acetylcholine receptor subunit alpha-4Neuronal acetylcholine receptor subunit alpha-7Neuronal acetylcholine receptor subunit beta-2 +10
Waktu ParuhCotinine has a half…
Vol. Distribusi* 2 to 3 L/kg
Klirens* 1.2 L/min [health…
Genetik -
Nikkomycin Z DB12939
small molecule | CAS: 59456-70-1

Nikkomycin Z has been used in trials studying the treatment and basic science of Coccidioidomycosis.

Kategori:
Anti-Infective AgentsAntifungal AgentsCarbohydrates +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nilutamide Approved DB00665
small molecule | CAS: 63612-50-0

Nilutamide is an antineoplastic hormonal agent primarily used in the treatment of prostate cancer. Nilutamide is a pure, nonsteroidal anti-androgen with affinity for androgen receptors (but not for progestogen, estrogen, or glucocorticoid receptors). Conseque…

Kategori:
Androgen Receptor AntagonistsAndrogen Receptor InhibitorsAntiandrogens +18
Target Protein:
Androgen receptor
Waktu Paruh38.0-59.1 hours
Vol. Distribusi-
Klirens-
Genetik -
Nilvadipine Approved DB06712
small molecule | CAS: 75530-68-6

Nilvadipine is a calcium channel blocker (CCB) for the treatment of hypertension.

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntihypertensive Agents +27
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent calcium channel subunit alpha-2/delta-1Voltage-dependent L-type calcium channel subunit beta-2 +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nimesulide Approved DB04743
small molecule | CAS: 51803-78-2

Nimesulide is a relatively COX-2 selective, non-steroidal anti-inflammatory drug (NSAID) with analgesic and antipyretic properties. Its approved indications are the treatment of acute pain, the symptomatic treatment of osteoarthritis and primary dysmenorrhoea…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +25
Target Protein:
Prostaglandin G/H synthase 2Tumor necrosis factor ligand superfamily member 10Lactotransferrin +1
Waktu Paruh1.8–4.7 hours
Vol. Distribusi-
Klirens-
Genetik -
Nimorazole DB12172
small molecule | CAS: 6506-37-2

Nimorazole has been used in trials studying the treatment of Hypoxia, Radiotherapy, Hypoxic Modification, Gene Profile, Gene Signature, and Head and Neck Squamous Cell Carcinoma, among others.

Kategori:
Anti-Infective AgentsAntiparasitic AgentsAntiparasitic Products, Insecticides and Repellents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Niraparib Approved DB11793
small molecule | CAS: 1038915-60-4

Niraparib is an orally active poly (ADP-ribose) polymerase (PARP) inhibitor. By blocking the enzymes responsible for DNA repair, niraparib induces cytotoxicity in cancer cells.[L43277] Niraparib is selective towards PARP-1 and PARP-2.[A253248] First approved …

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +20
Target Protein:
Poly [ADP-ribose] polymerase 1Poly [ADP-ribose] polymerase 2
Waktu ParuhFollowing multiple …
Vol. DistribusiThe average (±SD) a…
KlirensIn a population pha…
Genetik -
Nirogacestat Approved DB12005
small molecule | CAS: 1290543-63-3

Nirogacestat is a small-molecule gamma-secretase inhibitor that was investigated as a potential treatment for desmoid tumors. Desmoid tumors are typically characterized by aberrant activation in Notch signaling.[A262556] Interaction between the notch receptor…

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Peptides, and Proteins +20
Target Protein:
Gamma-secretase subunit APH-1BNicastrinPresenilin-1 +3
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe apparent volume…
KlirensThe apparent system…
Genetik -
Nirsevimab Approved DB16258
biotech | CAS: 1989556-22-0

Nirsevimab (MEDI8897) is a recombinant human immunoglobulin G1 kappa (IgG1?) monoclonal antibody used to prevent respiratory syncytial virus (RSV) lower respiratory tract disease in neonates and infants.[L44146] It binds to the prefusion conformation of the R…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Fusion glycoprotein F0Fusion glycoprotein F0Fusion glycoprotein F0
Waktu ParuhThe terminal half-l…
Vol. DistribusiFor an infant weigh…
KlirensFor an infant weigh…
Genetik -
Nisin Z DB19122
biotech | CAS: 137061-46-2

Nisin Z is under investigation in clinical trial NCT06097468 (Nisin in Oral Cavity Squamous Cell Carcinoma (OCSCC)).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nitrite Approved DB12529
small molecule | CAS: 14797-65-0

Nitrite is under investigation for the treatment of Heart Failure.

Kategori:
AnionsElectrolytesIons +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nitroaspirin DB12445
small molecule | CAS: 175033-36-0

Nitroaspirin has been investigated for the treatment of Intermittent Claudication.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +19
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nitrous acid Approved DB09112
small molecule | CAS: 7782-77-6

Nitrous acid (as sodium nitrite) is used as part of an intravenous mixture with sodium thiosulfate to treat cyanide poisoning. It is on the World Health Organization's List of Essential Medicines, a list of the most important medications needed in a basic hea…

Kategori:
AcidsAcids, NoncarboxylicAnions +16
Target Protein:
Hemoglobin subunit alphaHemoglobin subunit betaMyoglobin
Waktu ParuhHalf life of 0.4-0.…
Vol. Distribusi-
Klirens-
Genetik -
Nivocasan DB12720
small molecule | CAS: 908253-63-4

Nivocasan has been used in trials studying the treatment of HCV Infection and Nonalcoholic Steatohepatitis.

Target Protein:
Caspase-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nivolumab Approved DB09035
biotech | CAS: 946414-94-4

Nivolumab is a fully human IgG4 antibody targeting the immune checkpoint programmed death receptor-1 (PD-1).[L12129] This antibody was produced entirely in mice and grafted onto human kappa and IgG4 Fc region with the mutation _S228P_ for additional stability…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntibodies +20
Target Protein:
Programmed cell death protein 1Programmed cell death 1 ligand 1
Waktu ParuhThe serum half life…
Vol. DistribusiThe volume of distr…
KlirensThe estimated clear…
Genetik -
NKTT-120 DB17730
biotech

NKTT-120 is a recombinant humanized IgG1k monoclonal antibody to human invariant T cell receptor (iTCR).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NM-3 DB12818
small molecule | CAS: 181427-78-1

NM-3 has been used in trials studying the treatment of Neoplasms.

Target Protein:
Vascular endothelial growth factor A, long formVascular endothelial growth factor BVascular endothelial growth factor C +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nolasiban DB16259
small molecule | CAS: 1477482-19-1

Nolasiban is under investigation in clinical trial NCT03081208 (Phase 3 Placebo Controlled Study of Nolasiban to Improve Pregnancy Rates in Women Undergoing IVF/ICSI).

Kategori:
AminesHydroxylamines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nolatrexed DB12912
small molecule | CAS: 147149-76-6

Nolatrexed is under investigation in clinical trial NCT00012324 (Nolatrexed Dihydrochloride Compared With Doxorubicin in Treating Patients With Recurrent or Unresectable Liver Cancer).

Kategori:
AntimetabolitesAntineoplastic AgentsEnzyme Inhibitors +5
Target Protein:
Thymidylate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nomacopan DB14991
biotech | CAS: 875125-19-2

Nomacopan is under investigation in clinical trial NCT03427060 (Coversin in PNH in Patients With Resistance to Eculizumab Due to Complement C5 Polymorphisms).

Kategori:
Recombinant Protein Inhibitor of Complement Factor 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nona-arginine DB12648
small molecule | CAS: 143413-47-2

Nona-arginine is under investigation in clinical trial NCT00264706 (PolyArginine Treated vEiN grafTs (PATENT)).

Kategori:
Amino Acids, Peptides, and ProteinsFurin, antagonists & inhibitorsPeptides
Target Protein:
Nitric oxide synthase, inducible
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nonacog beta pegol Approved DB13933
biotech | CAS: 1175512-71-6

Nonacog beta pegol is a recombinant coagulation factor IX derivative. It is produced without animal-derived materials and with an attached 40kDa polyethylene glycol (PEG) molecule for peptide activation by a site-directed glycoPEGylation. Once activated, the …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +10
Target Protein:
Coagulation factor VIICoagulation factor VIIICoagulation factor X
Waktu ParuhThe mean half-life …
Vol. DistribusiThe volume of distr…
KlirensMean clearance in c…
Genetik -
Nonoxynol-9 Approved DB06804
small molecule | CAS: 26027-38-3

Nonoxynol-9 (N-9) is a typical surfactant used as a vaginal spermicide. Spermicides are locally acting non-hormonal contraceptives. When present in the vagina during intercourse, they immobilize/inactivate/damage and/or kill sperms without eliciting systemic …

Kategori:
Adrenal Cortex HormonesAlcoholsAntispermatogenic Agents +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NOP-1A DB15208
small molecule | CAS: 1283095-70-4

NOP-1A is under investigation in clinical trial NCT01198197 (PET Brain and Whole Body Distribution Studies for Nociceptin/Orphanin FQ Peptide (NOP) Receptor Using [11C]NOP-1A).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Norepinephrine Approved DB00368
small molecule | CAS: 51-41-2

Precursor of epinephrine that is secreted by the adrenal medulla and is a widespread central and autonomic neurotransmitter. Norepinephrine is the principal transmitter of most postganglionic sympathetic fibers and of the diffuse projection system in the brai…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +34
Target Protein:
Alpha-1A adrenergic receptorAlpha-1B adrenergic receptorAlpha-1D adrenergic receptor +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Norethandrolone DB12787
small molecule | CAS: 52-78-8

Norethandrolone is under investigation in clinical trial NCT00700544 (Treatment Outcome in Elderly Patients).

Kategori:
Alimentary Tract and MetabolismAnabolic AgentsAnabolic Agents for Systemic Use +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 156126-12-4

Deskripsi belum tersedia.

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Noscapine Approved DB06174
small molecule | CAS: 128-62-1

Deskripsi belum tersedia.

Kategori:
AlkaloidsAntitussive AgentsCentral Nervous System Agents +12
Target Protein:
Sigma non-opioid intracellular receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NP-50301 DB05662
small molecule

NP-50301 is an ophthalmic therapeutic eye drop treating post-menopausal Dry Eye Syndrome (DES). It is being developed by Nascent Pharmaceuticals. It is estimated that about 30% of postmenopausal women suffer symptoms of DES, which accounts for over 12 million…

Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NP2 DB06308
small molecule

NP2 is a replication defective HSV-1 based gene transfer vector engineered to express human preproenkephalin. It was under investigation in clinical trial NCT01291901 (NP2 Enkephalin For Treatment of Intractable Cancer Pain).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NS-398 DB14060
small molecule | CAS: 123653-11-2

NS-398 is a COX-2 inhibitor. It was developed as part of the mechanistic study of the cyclooxygenases.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +14
Target Protein:
Prostaglandin G/H synthase 2Cyclooxygenase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NSI-189 DB16230
small molecule | CAS: 1270138-40-3

NSI-189 is under investigation in clinical trial NCT02695472 (Study of NSI-189 for Major Depressive Disorder).

Kategori:
AminesPyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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