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11778

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8554 (72.6%)
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6383 (54.2%)
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96 (0.8%)
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11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 41 / 236
biotech | CAS: 2416824-55-8

Alunacedase alfa is a recombinant and soluble glycosylated form of human ACE2. This recombinant version of the enzyme has antihypertensive and potential antineoplastic activities.

Kategori:
Amino Acids, Peptides, and ProteinsCarboxypeptidasesEnzymes +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alvelestat DB11863
small molecule | CAS: 848141-11-7

Alvelestat has been investigated for the basic science of Chronic Obstructive Pulmonary Disease.

Kategori:
Leukocyte Elastase, antagonists & inhibitorsPyridinesSulfur Compounds
Target Protein:
Neutrophil elastase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alvespimycin DB12442
small molecule | CAS: 467214-20-6

Alvespimycin is a derivative of geldanamycin and heat shock protein (HSP) 90 inhibitor. It has been used in trials studying the treatment of solid tumor in various cancer as an antitumor agent. In comparison to the first HSP90 inhibitor tanespimycin, it exhib…

Kategori:
AmidesHSP90 Heat-Shock ProteinsLactams +1
Target Protein:
Heat shock protein HSP 90-alpha
Waktu ParuhThe half-life acros…
Vol. DistribusiAt the maximum tole…
KlirensThe mean clearance …
Genetik -
Alvimopan Approved DB06274
small molecule | CAS: 156053-89-3

Alvimopan is a peripherally acting ? opioid antagonist. It is used to avoid postoperative ileus following small or large bowel resection and accelerates the gastrointestinal recovery period.

Kategori:
Alimentary Tract and MetabolismDrugs for ConstipationGastrointestinal Agents +3
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor
Waktu Paruh10 to 17 hours (gut…
Vol. Distribusi* 30±10 L
Klirens* 402 ± 89 mL/min
Genetik -
biotech | CAS: 137487-62-8

Alvircept Sudotox has been used in trials studying the treatment of HIV Infections.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ALX-009 DB17916
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AM336 DB06563
biotech | CAS: 247207-64-3

Leconotide (development codes CNSB004 and AM336) is an omega-conotoxin peptide known for its analgesic properties, which work by blocking neuronal voltage-sensitive calcium channels. It was investigated as a potential treatment for various pain conditions.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAntiarrhythmic agents +17
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amantadine Approved DB00915
small molecule | CAS: 768-94-5

An antiviral that is used in the prophylactic or symptomatic treatment of influenza A. It is also used as an antiparkinsonian agent, to treat extrapyramidal reactions, and for postherpetic neuralgia. The mechanisms of its effects in movement disorders are not…

Kategori:
Adamantane DerivativesAdamantanesAnalgesics +25
Target Protein:
Matrix protein 2Glutamate receptor ionotropic, NMDA 3AD(2) dopamine receptor +3
Waktu ParuhMean half-lives ran…
Vol. Distribusi* 3 to 8 L/kg [heal…
Klirens* 0.2 - 0.3 L/hr/kg…
Genetik -
biotech

Amaranthus tuberculatus pollen allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ambazone DB13697
small molecule | CAS: 539-21-9

Deskripsi belum tersedia.

Kategori:
AmidinesAnti-Infective Agents, LocalGuanidines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ambenonium Approved DB01122
small molecule | CAS: 7648-98-8

Ambenonium is a cholinesterase inhibitor. It is used in the management of myasthenia gravis.

Kategori:
AminesAutonomic AgentsBenzylammonium Compounds +9
Target Protein:
Acetylcholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ambrisentan Approved DB06403
small molecule | CAS: 177036-94-1

Ambrisentan is an orally active selective type A endothelin receptor antagonist indicated for the treatment of pulmonary arterial hypertension. It is approved in Europe, Canada and the United States for use as a single agent to improve exercise ability and de…

Kategori:
Acids, CarbocyclicAntihypertensive AgentsAntihypertensives for Pulmonary Arterial Hypertension +15
Target Protein:
Endothelin-1 receptorEndothelin receptor type B
Waktu ParuhAmbrisentan has a t…
Vol. DistribusiAmbrisentan has a l…
KlirensThe mean oral clear…
Genetik -
Ambrosia ambrosioides pollen Approved DB10947
biotech

Ambrosia ambrosioides pollen is the pollen of the Ambrosia ambrosioides plant. Ambrosia ambrosioides pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Pollen Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Ambrosia confertiflora pollen is the pollen of the Ambrosia confertiflora plant. Ambrosia confertiflora pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ambrosia deltoidea pollen Approved DB10765
biotech

Ambrosia deltoidea pollen is the pollen of the Ambrosia deltoidea plant. Ambrosia deltoidea pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Pollen Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ambrosia dumosa pollen Approved DB10871
biotech

Ambrosia dumosa pollen is the pollen of the Ambrosia dumosa plant. Ambrosia dumosa pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Pollen Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ambrosia psilostachya pollen Approved DB10387
biotech

Ambrosia psilostachya pollen is the pollen of the Ambrosia psilostachya plant. Ambrosia psilostachya pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Pollen Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ambroxol Approved DB06742
small molecule | CAS: 18683-91-5

Ambroxol is a secretolytic agent used in the treatment of respiratory diseases associated with viscid or excessive mucus. It is the active ingredient of Mucosolvan, Lasolvan or Mucoangin. The substance is a mucoactive drug with several properties including se…

Kategori:
Adrenergics for Systemic UseAminesAnesthetics +13
Waktu Paruh7-12 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 96989-76-3

Deskripsi belum tersedia.

Kategori:
AlkaloidsAminesAniline Compounds +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amcasertib DB14866
small molecule | CAS: 1129403-56-0

Amcasertib is under investigation in clinical trial NCT02483247 (A Study of BBI503 in Combination With Selected Anti-Cancer Therapeutics in Adult Patients With Advanced Cancer).

Target Protein:
Platelet-derived growth factor receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amcipatricin DB12333
small molecule | CAS: 143483-67-4

Amcipatricin has been used in trials studying the treatment of Cryptococcosis or Aspergillosis Infections. Amcipatricin (as amcipatricin diascorbate; SPK-843) is a water-soluble partricin derivative patented by SPA Societa Prodotti Antibiotici S.p.A. and deve…

Kategori:
AlkenesHydrocarbons, Acyclic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amdinocillin DB01163
small molecule | CAS: 32887-01-7

Amidinopenicillanic acid derivative with broad spectrum antibacterial action. It is poorly absorbed if given orally and is used in urinary infections and typhus. Amdinocillin is not available in the United States.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 2aPenicillin-binding protein 2Penicillin-binding protein 3 +3
Waktu ParuhApproximately 1 hou…
Vol. Distribusi-
Klirens-
Genetik -
AME-527 DB05879
biotech

AME-527 is a humanized monoclonal antibody that recognizes human TNF-alpha (hTNF-alpha) with high affinity and specificity. AME-527 was generated by protein engineering and identified from a library of antibody variants based on its improved binding propertie…

Target Protein:
Tumor necrosis factor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amedalin DB09188
small molecule | CAS: 22136-26-1

Amedalin is a selective norepinephrine reuptake inhibitor developed in the 1970s. It has no significant effect on reuptake of serotonin and dopamine and no antihistamine or anticholinergic properties. This drug was never marketed.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amediplase DB06679
biotech | CAS: 151912-11-7

Amediplase is a recombinant chimeric plasminogen activator, consisting of the kringle 2 domain from the A-chain of tissue plasminogen activator (t-PA) and the carboxy terminal region of pro-urokinase. [MeSH]

Kategori:
Agents causing angioedemaAmino Acids, Peptides, and ProteinsAnticoagulants +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amelubant DB06248
small molecule | CAS: 346735-24-8

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicReceptors, Leukotriene B4, antagonists & inhibitors
Target Protein:
Leukotriene B4 receptor 1Leukotriene B4 receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amenamevir DB11701
small molecule | CAS: 841301-32-4

Amenamevir has been used in trials studying the treatment of Herpes Zoster, Herpes Simplex, Herpes Genitalis, and Safety of Amenamevir.

Kategori:
Antiinfectives for Systemic UseAntiviral AgentsAntivirals for Systemic Use +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 30578-37-1

Deskripsi belum tersedia.

Kategori:
Adrenergic and Dopaminergic AgentsCardiac Stimulants Excl. Cardiac GlycosidesCardiac Therapy
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amfenac DB15911
small molecule | CAS: 51579-82-9

Deskripsi belum tersedia.

Kategori:
Acids, Carbocyclic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AMG 108 DB05545
biotech | CAS: 877879-38-4

AMG 108 was investigated for use as an antirheumatic agent.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AMG 424 DB17357
biotech

AMG 424 is a novel, humanized, anti-CD3/CD38 bispecific monoclonal antibody being investigated for multiple myeloma.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AMG-119 DB17363
biotech

AMG-119 are CAR-T cells targeting delta-like ligand 3 (DLL3).[A254811]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AMG-208 DB08079
small molecule | CAS: 1002304-34-8

AMG-208 has been used in trials studying the treatment of Cancer, Tumors, Oncology, Prostate Cancer, and Oncology Patients, among others.

Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AMG-222 DB06011
small molecule | CAS: 913978-37-7

Deskripsi belum tersedia.

Kategori:
Agents causing angioedemaBenzocycloheptenesBlood Glucose Lowering Agents +1
Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AMG-319 DB16879
small molecule | CAS: 1608125-21-8

Deskripsi belum tersedia.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AMG-337 DB15639
small molecule | CAS: 1173699-31-4

AMG-337 is under investigation in clinical trial NCT03147976 (QUILT-3.036: AMG 337 in Subjects With Advanced or Metastatic Solid Tumors).

Kategori:
Antineoplastic AgentsPyridines
Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AMG-900 DB17197
small molecule | CAS: 945595-80-2

Deskripsi belum tersedia.

Kategori:
Protein Kinase InhibitorsPyridazines
Target Protein:
Aurora kinase CAurora kinase BAurora kinase A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AMGN-0007 DB06511
biotech

Recombinant osteoprotegerin (AMGN-0007) is a recombinant OPG construct developed as a potential therapeutic agent in the treatment of bone disease.

Kategori:
Amino Acids, Peptides, and ProteinsMembrane ProteinsProteins +1
Target Protein:
Tumor necrosis factor ligand superfamily member 11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amidephrine DB16623
small molecule | CAS: 37571-84-9

Deskripsi belum tersedia.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-Agonists +4
Target Protein:
Alpha-2C adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amifampridine Approved DB11640
small molecule | CAS: 54-96-6

Amifampridine, or 3,4-diaminopyridine (3,4-DAP), is a quaternary ammonium compound that blocks presynaptic potassium channels, and subsequently prolongs the action potential and increases presynaptic calcium concentrations [A33863]. It was first discovered in…

Kategori:
AminesAminopyridinesMembrane Transport Modulators +7
Target Protein:
Potassium voltage-gated channel subfamily A member 1
Waktu ParuhThe average elimina…
Vol. DistribusiIn healthy voluntee…
KlirensOverall clearance o…
Genetik -
Amifostine Approved DB01143
small molecule | CAS: 20537-88-6

A phosphorothioate proposed as a radiation-protective agent. It causes splenic vasodilation and may block autonomic ganglia.

Kategori:
Compounds used in a research, industrial, or household settingCytoprotective AgentDetoxifying Agents for Antineoplastic Treatment +9
Target Protein:
Alkaline phosphatase, germ cell type
Waktu Paruh8 minutes
Vol. Distribusi-
Klirens-
Genetik -
Amikacin Approved DB00479
small molecule | CAS: 37517-28-5

Amikacin is a semi-synthetic aminoglycoside antibiotic that is derived from kanamycin A.[FDA label] Amikacin is synthesized by acylation with the l-(-)-?-amino-?-hydroxybutyryl side chain at the C-1 amino group of the deoxystreptamine moiety of kanamycin A.[A…

Kategori:
Aminoglycoside AntibacterialsAnti-Bacterial AgentsAnti-Infective Agents +7
Target Protein:
30S ribosomal protein S12
Waktu ParuhThe plasma eliminat…
Vol. Distribusi* 24 L (28% of body…
KlirensThe mean serum clea…
Genetik -
Amiloride Approved DB00594
small molecule | CAS: 2609-46-3

A pyrazine compound inhibiting sodium reabsorption through sodium channels in renal epithelial cells. This inhibition creates a negative potential in the luminal membranes of principal cells, located in the distal convoluted tubule and collecting duct. Negati…

Kategori:
Acid Sensing Ion Channel BlockersAgents causing hyperkalemiaCardiovascular Agents +11
Target Protein:
Amiloride-sensitive sodium channel subunit alphaAmiloride-sensitive sodium channel subunit betaAmiloride-sensitive sodium channel subunit gamma +6
Waktu ParuhPlasma half-life va…
Vol. Distribusi-
Klirens-
Genetik -
Amiloxate Approved DB11207
small molecule | CAS: 71617-10-2

Amiloxate is an EMA-approved chemical UV-filter found in over-the-counter sunscreen products at concentrations up to 10%m [F35]. It is often referred to as isoamyl 4-methoxycinnamate or isoamyl p-methoxycinnamate. Amiloxate is a cinnamic acid derivative with …

Kategori:
Acids, CarbocyclicSunscreen Agents
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Aminaphthone DB13039
small molecule | CAS: 14748-94-8

Aminaftone has been investigated for the treatment of Cockett Syndrome, May-Thurner Syndrome, and Iliac Vein Obstruction.

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amineptine DB04836
small molecule | CAS: 57574-09-1

The Food and Drug Administration suspended the marketing authorisation for Survector in 1999 and France withdrew it from the market, however several developing countries continued to produce it up until 2005.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +11
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporterSodium-dependent serotonin transporter
Waktu Paruh48 minutes for the …
Vol. Distribusi-
Klirens-
Genetik -
Amino acids DB09393
small molecule | CAS: 65072-01-7

Mixture of amino acids ; used for parenteral nutrition in infants.

Kategori:
Amino Acid Hypertonic SolutionAmino AcidsAmino Acids, Peptides, and Proteins +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aminoanthracene DB01976
small molecule | CAS: 62813-37-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aminocandin DB05128
small molecule | CAS: 227472-48-2

Aminocandin is a new representative of the echinocandins that could potentially affect the cellular morphology and metabolic status of Candida albicans cells within biofilms.

Kategori:
Amino Acids, Peptides, and ProteinsEchinocandin AntifungalLipids +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aminoflavone DB19077
small molecule | CAS: 165179-35-1

Aminoflavone is under investigation in clinical trial NCT01015521 (Efficacy Study of Aminoflavone Prodrug to Treat Breast Cancer).

Kategori:
BenzopyransChromonesHeterocyclic Compounds, Fused-Ring +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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