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11793

Total database: 17430
Struktur (SMILES)
8607 (73.0%)
Target
6418 (54.4%)
Genomik
102 (0.9%)
Referensi
11793 (100.0%)

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Hasil Pencarian (11793)

Halaman 41 / 236
Amylopectin DB14927
small molecule | CAS: 9037-22-3

Amylopectin is under investigation in clinical trial NCT01708694 (Role of Slowly Digesible Starch on Diabetes Risk Factors).

Kategori:
CarbohydratesDietary CarbohydratesGlucans +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Amylose DB15216
small molecule | CAS: 9005-82-7

Amylose is under investigation in clinical trial NCT01027325 (Resistant Starch Insulin Sensitivity Trial).

Kategori:
CarbohydratesDietary CarbohydratesGlucans +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AN-2718 DB12810
small molecule | CAS: 174672-06-1

An2718 has been used in trials studying Tinea Pedis.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AN-9 DB05103
small molecule | CAS: 122110-53-6

Pivaloyloxymethyl butyrate (AN-9), an acyloxyalkyl ester prodrug of butyric acid (BA), exhibited low toxicity and significant anticancer activity in vitro and in vivo. It shows greater potency than BA at inducing malignant cell differentiation and tumor growt…

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Target Protein:
Histone deacetylase 1Apoptosis regulator Bcl-2Caspase-8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AN2898 DB16039
small molecule | CAS: 906673-33-4

AN2898 is under investigation in clinical trial NCT01301508 (Efficacy and Safety of AN2898 and AN2728 Topical Ointments to Treat Mild-to-moderate Atopic Dermatitis).

Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4D3',5'-cyclic-AMP phosphodiesterase 4B3',5'-cyclic-AMP phosphodiesterase 4A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ANA975 DB06490
small molecule | CAS: 847453-47-8

ANA975 is a toll-like receptor 7 agonist that is developed for the treatment of hepatitis C.

Target Protein:
Toll-like receptor 7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anacaulase Approved DB17449
biotech

Anacaulase (anacaulase-bcdb) is a mixture of proteolytic enzymes extracted from the stems of pineapple plants (_Ananas comosus_ [L.] Merr.). It is mostly composed (80-95% w/w) of proteins such as stem bromelain, ananain, jacalin-like lectin, bromelain inhibit…

Kategori:
Administration, TopicalCysteine EndopeptidasesCytochrome P-450 CYP2C8 Inhibitors +9
Target Protein:
Alpha-1-antichymotrypsinAlpha-2-macroglobulin
Waktu ParuhThe mean eliminatio…
Vol. Distribusi-
Klirens-
Genetik -
Anacetrapib DB06630
small molecule | CAS: 875446-37-0

Deskripsi belum tersedia.

Kategori:
Anticholesteremic AgentsCholesterol Ester Transfer Proteins, antagonists & inhibitorsHypolipidemic Agents +2
Target Protein:
Cholesteryl ester transfer protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anagliptin DB12417
small molecule | CAS: 739366-20-2

Anagliptin is under investigation for the treatment of LDL Cholesterol, Coronary Disease, Diabetes Mellitus, Glycosylated Hemoglobin, and Dipeptidyl-Peptidase 4 Inhibitors.

Kategori:
Agents causing angioedemaBlood Glucose Lowering AgentsDPP-IV Inhibitors +2
Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anagrelide Approved DB00261
small molecule | CAS: 68475-42-3

Anagrelide is a platelet-reducing agent used to lower dangerously elevated platelet levels (i.e. to treat thrombocythemia) in patients with myeloproliferative neoplasms.[L14153] It is an oral imidazoquinazoline that was first approved for use in the US in 199…

Kategori:
Agents producing tachycardiaAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +18
Target Protein:
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A
Waktu ParuhThe t<sub>1/2</sub>…
Vol. Distribusi-
Klirens-
Genetik -
Anakinra Approved DB00026
biotech | CAS: 143090-92-0

Anakinra is a recombinant human interleukin-1 (IL-1) receptor antagonist (IL-1Ra) composed of 153 amino acid residues. Unlike native human IL-1Ra, anakinra has an additional methionine residue at the amino terminus. This drug binds to the IL-1 receptor, compe…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +12
Target Protein:
Interleukin-1 receptor type 1
Waktu ParuhIn patients with rh…
Vol. DistribusiIn adult subjects w…
KlirensIn patients with rh…
Genetik -
Anamorelin DB06645
small molecule | CAS: 249921-19-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +2
Target Protein:
Growth hormone secretagogue receptor type 1Lysosomal alpha-glucosidaseNeutral alpha-glucosidase AB +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anaritide DB17613
biotech | CAS: 95896-08-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsDiureticsHormones +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anastrozole Approved DB01217
small molecule | CAS: 120511-73-1

Anastrozole is a non-steroidal aromatase inhibitor (AI), similar to [letrozole], used to decrease circulating estrogen levels in the treatment of postmenopausal women with estrogen-responsive breast cancer.[L8863] Anastrozole is also related to [exemestane], …

Kategori:
Antineoplastic AgentsAntineoplastic Agents, HormonalAntineoplastic and Immunomodulating Agents +30
Target Protein:
Aromatase
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensAnastrozole's clear…
Genetik -
Anbenitamab DB18411
biotech | CAS: 2367012-88-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ANC-501 DB18907
small molecule | CAS: 1370444-22-6

ANC-501 is under investigation in clinical trial NCT05439603 (ANC-501 in the Treatment of Adults With Major Depressive Disorder).

Kategori:
AcetatesAcids, AcyclicAmides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ancestim Approved DB09103
biotech | CAS: 163545-26-4

Ancestim is a non-glycosylated recombinant methionyl human stem cell factor. It is a 166 amino acid protein produced by E. coli with an amino acid sequence that is identical to the natural sequence predicted from human DNA sequence analysis, except for the ad…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +8
Target Protein:
Mast/stem cell growth factor receptor Kit
Waktu ParuhIn clinical trials,…
Vol. DistribusiPreclinical reports…
KlirensThe apparent cleara…
Genetik -
Ancrod Approved DB05099
biotech | CAS: 9046-56-4

Ancrod, marketed as Viprinex, is a defibrinogenating agent derived from Malayan pit viper venom. The defribrinogenation of blood results in an anticoagulant effect. Currently, Viprinex®/ancrod is not approved or marketed in any country, but is being investiga…

Kategori:
AnticoagulantsBiological FactorsBlood and Blood Forming Organs +18
Target Protein:
Fibrinogen alpha chain
Waktu Paruh3 to 5 hours
Vol. Distribusi-
Klirens-
Genetik -
Andecaliximab DB17564
biotech | CAS: 1518996-49-0

Andecaliximab is a monoclonal antibody directed against matrix metallopeptidase 9 (MMP9). Andecaliximab is under investigation in clinical trial NCT03631836 (Phase I Study of Monoclonal Antibondy (GS) 5745, an Matix Metalloproteinase 9 (MMP9) Mab Inhibitor, i…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Andexanet alfa Approved DB14562
biotech | CAS: 1262449-58-0

Andexanet alfa is a recombinant human coagulation Factor Xa that promotes blood coagulation. It was developed by Portola Pharmaceuticals and was approved in in May 2018. It is marketed as Andexxa for intravenous injection or infusion and is indicated for the …

Kategori:
Amino Acids, Peptides, and ProteinsAntidotesBiological Factors +12
Target Protein:
Tissue factor pathway inhibitor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensClearance for andex…
Genetik -
Andrographolide DB05767
small molecule | CAS: 5508-58-7

Andrographolide (HMPL-004) is a botanical product extracted from a herb that occurs naturally in China. The herb has an extensive history of use in TCM for the treatment of upper respiratory tract infections and other inflammatory and infectious diseases.

Kategori:
AcanthaceaeAnalgesicsAnalgesics, Non-Narcotic +25
Target Protein:
Tumor necrosis factorInterleukin-1 betaInterleukin-6 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Androstanedione DB01561
small molecule | CAS: 846-46-8

Deskripsi belum tersedia.

Target Protein:
17-beta-hydroxysteroid dehydrogenase type 1Steroid Delta-isomerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Androstenedione DB01536
small molecule | CAS: 63-05-8

A delta-4 C19 steroid that is produced not only in the testis, but also in the ovary and the adrenal cortex. Depending on the tissue type, androstenedione can serve as a precursor to testosterone as well as estrone and estradiol.

Kategori:
17-KetosteroidsAdrenal Cortex HormonesAndrostanes +12
Target Protein:
Aromatase17-beta-hydroxysteroid dehydrogenase type 13 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 1 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anecortave DB12081
small molecule | CAS: 10184-70-0

Anecortave is under investigation in clinical trial NCT00691717 (Anecortave Acetate Safety in Patients With Open-Angle Glaucoma or Ocular Hypertension).

Kategori:
11-Hydroxycorticosteroids17-HydroxycorticosteroidsAdrenal Cortex Hormones +17
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 7753-60-8

Anecortave acetate (Retaane) is an analog of cortisol acetate; among the modifications to the steroid are the removal of the 11ß hydroxyl OH group and an addition of a 21-acetate group. As a result of these modifications, anecortave acetate lacks the typical …

Kategori:
11-Hydroxycorticosteroids17-HydroxycorticosteroidsAngiogenesis Inhibitors +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anethole Approved DB15916
small molecule | CAS: 4180-23-8

Deskripsi belum tersedia.

Kategori:
AlkenesAllyl CompoundsBenzene Derivatives +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anethole trithione Approved DB13853
small molecule | CAS: 532-11-6

Anethole trithione (ATT) appears to have a broad range of unique functions, from increasing salivary secretion to help treat xerostomia [A27165, A32618, A32620, A32621], to demonstrating an ability to inhibit carcinogenesis by increasing the activity of elect…

Kategori:
Alimentary Tract and MetabolismAnisolesBenzene Derivatives +10
Target Protein:
Protein-glutamine gamma-glutamyltransferase 2
Waktu ParuhDespite the medicat…
Vol. DistribusiDespite the medicat…
KlirensDespite the medicat…
Genetik -
biotech | CAS: 1375258-01-7

Anetumab ravtansine is under investigation in clinical trial NCT03455556 (Anetumab Ravtansine and Atezolizumab in Treating Participants With Advanced Non-small Cell Lung Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibody-drug Conjugates +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anfibatide DB15094
biotech | CAS: 1622134-89-7

Anfibatide is under investigation in clinical trial NCT01585259 (Anfibatide Phase Ib-IIa Clinical Trial).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsComplex Mixtures +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ANG1005 DB18167
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsCyclodecanesCycloparaffins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Angelica sinensis root is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngelicaAngiospermsApiaceae +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 53-73-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAngiotensinsAutacoids +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 38390-45-3

Anhydrovinblastine has been used in trials studying the treatment of Unspecified Adult Solid Tumor, Protocol Specific.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anidulafungin Approved DB00362
biotech | CAS: 166663-25-8

Anidulafungin or Eraxis is an anti-fungal drug manufactured by Pfizer that gained approval by the Food and Drug Administration (FDA) in February 21, 2006; it was previously known as LY303366. There is preliminary evidence that it has a similar safety profile …

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntifungal Agents +6
Target Protein:
1,3-beta-glucan synthase component FKS11,3-beta-glucan synthase component GSC2
Waktu Paruh40-50 hours
Vol. Distribusi* 30 to 50 L
Klirens* 1 L/h
Genetik -
Anifrolumab Approved DB11976
biotech | CAS: 1326232-46-5

Anifrolumab, or MEDI-546, is a type 1 interferon receptor (IFNAR) inhibiting IgG1? monoclonal antibody indicated in the treatment of adults with moderate to severe systemic lupus erythematosus.[A237074,L34929] The standard therapy for systemic lupus erythemat…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Interferon alpha/beta receptor 1
Waktu ParuhThe serum eliminati…
Vol. DistribusiBased on population…
KlirensFollowing the admin…
Genetik -
Aniline DB06728
small molecule | CAS: 62-53-3

Aniline, phenylamine or aminobenzene is an organic compound with the formula C6H5NH2. Consisting of an amine attached to a benzene ring, aniline is the prototypical aromatic amine. Being a precursor to many industrial chemicals, its main use is in the manufac…

Kategori:
AminesCarcinogensCytochrome P-450 CYP2E1 Substrates +3
Target Protein:
Kallikrein-1Albumin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anise oil DB15776
biotech | CAS: 8007-70-3

Deskripsi belum tersedia.

Kategori:
AngiospermsApiaceaeBiological Products +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anisodamine DB11785
small molecule | CAS: 55869-99-3

Anisodamine has been investigated for the treatment of Intestinal Diseases.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic Antagonists +29
Target Protein:
Beta-1 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anisomycin DB07374
small molecule | CAS: 22862-76-6

Anisomycin (sometimes known as flagecidin), is an antibiotic retrieved from the bacteria _Streptomyces griseolus_. This drug acts to inhibit bacterial protein and DNA synthesis.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntiparasitic Agents +5
Target Protein:
Ribosomal protein uL16-likeLarge ribosomal subunit protein uL13Large ribosomal subunit protein uL14 +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anistreplase Approved DB00029
biotech | CAS: 81669-57-0

Human tissue plasminogen activator, purified, glycosylated, 527 residues purified from CHO cells. Eminase is a lyophilized (freeze-dried) formulation of anistreplase, the p-anisoyl derivative of the primary Lys-plasminogen-streptokinase activator complex (a c…

Kategori:
Agents causing angioedemaAmino Acids, Peptides, and ProteinsAnticoagulants +15
Target Protein:
PlasminogenFibrinogen alpha chainPlasminogen activator inhibitor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anivamersen DB16089
biotech | CAS: 959716-29-1

Anivamersen is under investigation in clinical trial NCT01848106 (A Study to Determine the Efficacy and Safety of REG1 Compared to Bivalirudin in Patients Undergoing PCI).

Kategori:
CoagulantsNucleic Acids, Nucleotides, and NucleosidesNucleotides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anlotinib DB11885
small molecule | CAS: 1058156-90-3

Anlotinib has been investigated for the treatment of Non-small Cell Lung Cancer and Metastatic Colorectal Cancer.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Proto-oncogene tyrosine-protein kinase Src
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Annamycin DB06420
small molecule | CAS: 92689-49-1

Deskripsi belum tersedia.

Kategori:
AnthracyclinesAntibiotics, AntineoplasticAntineoplastic Agents +4
Target Protein:
DNA topoisomerase 2-alphaDNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anpocogin DB06552
biotech

Recombinant nematode anticoagulant protein c2 (rNAPc2) is a specific inhibitor of tissue factor (TF)/factor VIIa complex with novel antithrombotic activity. [A175642]

Target Protein:
Coagulation factor VIITissue factorCoagulation factor X
Waktu ParuhOver 50 hours
Vol. Distribusi-
Klirens-
Genetik -
Anrukinzumab DB12294
biotech | CAS: 910649-32-0

Anrukinzumab has been used in trials studying the diagnostic of Asthma.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anselamimab DB17492
biotech | CAS: 2414866-63-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ansofaxine DB15052
small molecule | CAS: 916918-80-4

Ansofaxine is under investigation in clinical trial NCT02271412 (Multiple Ascending Dose Study in Healthy Subjects to Evaluate the Safety, Tolerability, and Pharmacokinetics of LY03005).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ansuvimab Approved DB16385
biotech | CAS: 2375952-29-5

Infection with pathogenic filoviruses, such as _Zaire ebolavirus_ (Ebola virus, EBOV), can cause severe hemorrhagic fever in humans, resulting in frequent outbreaks with case fatality rates as high as 90%.[A225933, A225938] Virtually all steps of the EBOV lif…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +13
Target Protein:
Envelope glycoprotein
Waktu ParuhThe half-life of an…
Vol. DistribusiThe steady-state vo…
KlirensThe clearance of an…
Genetik -
Anthoxanthum odoratum Approved DB14163
biotech

Anthoxanthum odoratum allergenic extract is used in allergenic testing.

Kategori:
Allergenic ExtractsNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anthralin Approved DB11157
small molecule | CAS: 1143-38-0

Anthralin (1,8?dihydroxy?9anthrone, dithranol) is an older anti-psoriatic agent that was first synthesized as a derivative of chrysarobin, obtained from the araroba tree in Brazil over 100 years ago. Adverse effects of anthralin include irritation and discolo…

Kategori:
AnthracenesAntipsoriaticsAntipsoriatics for Topical Use +2
Target Protein:
Keratin, type II cytoskeletal 2 epidermalKeratin, type I cytoskeletal 12C-Jun-amino-terminal kinase-interacting protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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