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14494

Total database: 17430
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14494 (100.0%)

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Halaman 40 / 290
Afimetoran DB16580
small molecule | CAS: 2171019-55-7

Afimetoran is an immunomodulator and an antagonist of toll-like receptors 7 and 8.[L32018, L32023] It is also is under investigation in clinical trial NCT04269356 (Study to Assess the Way the Body Absorbs, Distributes, Breaks Down and Eliminates Radioactive B…

Target Protein:
Toll-like receptor 7Toll-like receptor 8
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Afimoxifene DB04468
small molecule | CAS: 68392-35-8

Afimoxifene (4-Hydroxytamoxifen, trade name TamoGel) is a new estrogen inhibitor under investigation for a variety of estrogen-dependent conditions, including cyclic breast pain and gynecomastia. TamoGel is formulated using Enhanced Hydroalcoholic Gel (EHG) T…

Kategori:
AndrostanesAndrostenesAndrostenols +12
Target Protein:
Estrogen receptorTrefoil factor 1Steroid hormone receptor ERR1 +4
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Aflibercept Approved DB08885
biotech | CAS: 862111-32-8

Aflibercept is a recombinant protein composed of the binding domains of two human vascular endothelial growth factor (VEGF) receptors, VEGFR1 and VEGFR2, fused with the Fc region of human immunoglobulin gamma 1 (IgG1).[A261130] Structurally, Aflibercept is a …

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +16
Target Protein:
Vascular endothelial growth factor A, long formPlacenta growth factorVascular endothelial growth factor B
Waktu ParuhFor the intravitrea…
Vol. DistribusiThe volume of distr…
KlirensFollowing an hour o…
Genetik -
AFM-13 DB17404
biotech

Deskripsi belum tersedia.

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AFN-1252 DB12658
small molecule | CAS: 620175-39-5

AFN-1252 has been used in trials studying the treatment of Cellulitis, Burn Infection, Wound Infection, Cutaneous Abscess, and Skin and Subcutaneous Tissue Bacterial Infections.

Kategori:
Heterocyclic Compounds, Fused-RingPyrans
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Afuresertib DB11648
small molecule | CAS: 1047644-62-1

Afuresertib has been used in trials studying the treatment of Cancer and Neoplasms, Haematologic.

Kategori:
AminesPolyaminesSulfur Compounds
Target Protein:
RAC-alpha serine/threonine-protein kinase
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AG-702 DB05836
biotech

AG-702 is a recombinant human heat shock protein also known as stress protein. It is also known as HSPs, which are a group of proteins that are induced when a cell undergoes various types of environmental stresses like heat, cold and oxygen deprivation. HSPs …

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AG-858 DB05502
biotech

AG-858 (autologous heat-shock protein 70 peptide vaccine) is a recombinant cancer vaccine made with tumor-derived heat shock protein 70 (HSP70) peptide complexes. HSP70 associates with antigenic peptides, transporting them into antigen presenting cells (APC)…

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AG0301-COVID19 DB15856
biotech

AG0301-COVID19 is a vaccine candidate developed by AnGes Inc. and Osaka University. The candidate is a plasmid DNA vaccine developed using an intradermal gene transfer method targeting the SARS-CoV-2 spike protein. The gene transfer method increases the effic…

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AG0302-COVID19 DB16435
biotech

Sponsored by Anges, Inc. in Japan, the AG0302-COVID19 is a DNA-based vaccine that recently completed Phase I/II trials (NCT04527081)[A226813, L30548].

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AGA2115 DB17840
biotech

AGA2115 is a humanized bispecific antibody neutralizing both sclerostin and Dickkopf-1. Developed by Angitia Biopharmaceuticals, AGA2115 is being investigated for the treatment of osteogenesis imperfect.[L46646]

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Agalsidase alfa Approved DB15874
biotech

Agalsidase alfa is a recombinant human ?-galactosidase A similar to [agalsidase beta]. While patients generally do not experience a clinically significant difference in outcomes between the two drugs, some patients may experience greater benefit with agalsida…

Kategori:
Alimentary Tract and Metabolismalpha-Galactosidase, antagonists & inhibitorsAmino Acids, Peptides, and Proteins +9
Target Protein:
Globotriaosylceramide
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance for d…
Genetik -
Agalsidase beta Approved DB00103
biotech

Agalsidase beta is a recombinant human ?-galactosidase A similar to [agalsidase alfa]. While patients generally do not experience a clinically significant difference in outcomes between the two drugs, some patients may experience greater benefit with agalsida…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsEnzymes +7
Target Protein:
Globotriaosylceramide
Waktu Paruhagalsidase beta has…
Vol. DistribusiA 1 mg/kg dose of a…
KlirensA 1 mg/kg dose of a…
Genetik -
small molecule | CAS: 910562-20-8

Aganepag isopropyl is under investigation in clinical trial NCT01110499 (Safety and Efficacy of AGN-210961 Ophthalmic Solution Compared With Bimatoprost Ophthalmic Solution in Patients With Glaucoma or Ocular Hypertension).

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Aganirsen DB15369
biotech | CAS: 1146887-67-3

Aganirsen is under investigation in clinical trial NCT02947867 (Trial of Aganirsen in iCRVO Patients at Risk of Developing NVG).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
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Agatolimod DB15018
biotech | CAS: 207623-20-9

Agatolimod is under investigation in clinical trial NCT00471471 (Vaccine Therapy in Treating Patients With Recurrent Stage III or Stage IV Melanoma That Cannot Be Removed by Surgery).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
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Agave sisalana fiber Approved DB10712
biotech

Agave sisalana fiber is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Agerafenib DB15068
small molecule | CAS: 1188910-76-0

Agerafenib is under investigation in clinical trial NCT03052569 (Expanded Access to RXDX-105 for Cancers With RET Alterations).

Kategori:
AmidesBenzene DerivativesEnzyme Inhibitors +3
Target Protein:
Proto-oncogene tyrosine-protein kinase receptor RetSerine/threonine-protein kinase B-raf
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AGF-94 DB18023
small molecule | CAS: 136784-51-5

Deskripsi belum tersedia.

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AGG-523 DB15460
small molecule | CAS: 920289-29-8

AGG-523 is under investigation in clinical trial NCT00380900 (Study Evaluating the Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of Multiple Ascending Doses in Healthy subjects and in subjects with osteoarthritis).

Target Protein:
A disintegrin and metalloproteinase with thrombospondin motifs 5
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AGI-1096 DB05840
small molecule

AGI-1096 is a novel oral antioxidant and selective anti-inflammatory agent that is being developed to address the accelerated inflammation of grafted blood vessels, known as transplant arteritis, common in chronic organ transplant rejection.

Kategori:
Acids, AcyclicBenzene DerivativesFatty Acids +2
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AGI-134 DB19005
small molecule | CAS: 1821461-84-0

AGI-134 is under investigation in clinical trial NCT03593226 (Study to Evaluate Safety & Tolerability of AGI-134 in Solid Tumour).

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AGIL-FA DB16973
biotech

Deskripsi belum tersedia.

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biotech

Agkistrodon piscivorus antivenin is derived and purified immunoglobulin fragments obtained from other domestic animals such as sheep previously immunized with Agkistrodon piscivorus (_Cottonmouth_ or _Water Moccasin snake_). The final purified antivenin produ…

Kategori:
AntiveninsPassively Acquired ImmunityVenom Neutralization
Target Protein:
Group 10 secretory phospholipase A2
Waktu Paruh12 to 23 hours [FDA…
Vol. Distribusi-
KlirensSystemic clearance …
Genetik -
biotech | CAS: 1621271-62-2

Aglatimagene besadenovec is under investigation in clinical trial NCT00638612 (AdV-tk Therapy With Surgery and Chemoradiation for Pancreas Cancer (PaTK01)).

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Agmatine DB08838
small molecule | CAS: 306-60-5

Agmantine is a natural metabolite of the amino acid arginine. It is formed when arginine is decarboxylated by the enzyme arginine decarboxylase and is found naturally in ragweed pollen, ergot fungi, octopus muscle, herring sperm, sponges, and the mammalian br…

Kategori:
Agents causing hyperkalemiaAmidinesAntiarrhythmic agents +12
Target Protein:
Alpha-2C adrenergic receptorNischarinAcetylcholine receptor subunit alpha +4
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AGN-201904 DB13135
small molecule | CAS: 651729-53-2

Agn 201904 has been used in trials studying the prevention of Peptic Ulcer.

Kategori:
2-PyridinylmethylsulfinylbenzimidazolesBenzimidazolesHeterocyclic Compounds, Fused-Ring +3
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Agomelatine Approved DB06594
small molecule | CAS: 138112-76-2

Agomelatine is structurally closely related to melatonin. Agomelatine is a potent agonist at melatonin receptors and an antagonist at serotonin-2C (5-HT2C) receptors, tested in an animal model of depression. Agomelatine was developed in Europe by Servier Labo…

Kategori:
AcetatesAcids, AcyclicAmides +15
Target Protein:
5-hydroxytryptamine receptor 2CMelatonin receptor type 1AMelatonin receptor type 1B
Waktu Paruh<2 hours
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AGRO100 DB04998
biotech | CAS: 301636-59-9

AGRO100 is an oligonucleotide that functions as an aptamer and binds to nucleolin, a protein found intranuclear in all cells, but uniquely expressed on the surface of tumor cells. Such binding leads to internalization of the complex, and a strong anti-prolife…

Kategori:
Aptamers, NucleotideNucleic Acids, Nucleotides, and NucleosidesNucleotides +2
Target Protein:
NF-kappa-B essential modulator
Waktu Paruh-
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Agrostis gigantea pollen Approved DB10403
biotech

Agrostis gigantea pollen is the pollen of the Agrostis gigantea plant. Agrostis gigantea pollen is mainly used in allergenic testing.

Kategori:
Allergenic ExtractsCell-mediated ImmunityGrass Pollen Allergen Extracts +4
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Agrostis gigantea top Approved DB14757
biotech

Agrostis gigantea top is the flowering part of the Agrostis gigantea plant. Agrostis gigantea top is mainly used in allergenic testing.

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Agrostis stolonifera pollen Approved DB10962
biotech

Agrostis stolonifera pollen is the pollen of the Agrostis stolonifera plant. Agrostis stolonifera pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityGrass Pollen Allergen ExtractsIncreased Histamine Release +2
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AGS-004 DB05742
small molecule

AGS-004 is a personalized RNA-loaded dendritic cellbased immunotherapy that is designed to stimulate the patient’s immune system to target and destroy the patient’s own unique viral burden. Non-personalized HIV immunotherapies are unable to raise cytotoxic T…

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AGS-005 DB05741
small molecule

AGS-005 is a personalized dendritic cell-based immunotherapy, with optimized immune response characteristics, that is designed to stimulate the patient's immune system to target and destroy the patient's cancer cells.

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AGS-16C3F DB17551
biotech

AGS 16C3F is an intravenously administered, anti-ectonucleotide pyrophosphatase/phosphodiesterase 3 (ENPP3) antibody-drug conjugate. AGS-16C3F is under investigation in clinical trial NCT02639182 (A Study of AGS-16C3F vs. Axitinib in Metastatic Renal Cell Car…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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AGT-182 DB17630
biotech

AGT-182 is an investigational enzyme replacement therapy engineered by the fusion of the iduronate-2-sulfatase (IDS) enzyme and a human insulin receptor monoclonal antibody.

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AGTC-401 DB18432
biotech

AGTC-401 is a recombinant adeno-associated virus vector expressing the cyclic nucleotide gated channel beta subunit (rAAV-CNGB3).

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AGTC-402 DB18433
biotech

AGTC-402 is a recombinant adeno-associated virus vector expressing the cyclic nucleotide gated channel alpha subunit (CNGA3).

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AGuIX DB18189
biotech

AGuIX is an investigational brand product consisting of a polysiloxane matrix and gadolinium chelates. It is under development as a radiosensitizer to be used during radiation treatment of malignant glioma.

Kategori:
ElementsLanthanoid Series ElementsMetals +2
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biotech | CAS: 2417550-70-8

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
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AI-128 DB05841
small molecule

AI-128 is the first human demonstration of sustained release drug administration in the lung. AI-128 consists of slowly dissolving microspheres designed to control where drug particles go in the lung and how quickly they release their drug.

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AI-850 DB05842
small molecule

AI-850 is a Cremophor(R)-free formulation of paclitaxel, the active ingredient in Taxol(R), a product used to treat a variety of solid tumors.

Kategori:
CyclodecanesCycloparaffinsDiterpenes +2
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AIC100 DB17350
biotech

Deskripsi belum tersedia.

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small molecule | CAS: 3031-94-5

5-Aminoimidazole-4-carboxamide ribonucleotide (AICAR) is an intermediate in the generation of inosine monophosphate and analog of adenosine monophosphate (AMP) that is capable of stimulating AMP-dependent protein kinase (AMPK) activity. AICAR has been used cl…

Kategori:
Blood Glucose Lowering AgentsImidazolesNucleic Acids, Nucleotides, and Nucleosides +1
Target Protein:
Bifunctional purine biosynthesis protein ATIC
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Ailanthus altissima pollen Approved DB10452
biotech

Ailanthus altissima pollen is the pollen of the Ailanthus altissima plant. Ailanthus altissima pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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AIM-102 DB16176
small molecule | CAS: 551936-17-5

AIM-102 is under investigation in clinical trial NCT01501942 (Efficacy, Safety, Tolerability, Pharmacodynamics and Pharmacokinetics of Oral Administration of AIM-102 in Patients With Mild to Moderate Allergic Asthma).

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AIT-034 DB06106
small molecule | CAS: 138117-48-3

AIT-034 is a distinct chemical analog of hypoxanthine and pyrollidone that has been demonstrated in animal studies to enhance memory and to reverse memory deficits in severely impaired animals that do not respond to Neotrofin. AIT-034 does not induce the prod…

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Ajmaline Approved DB01426
small molecule | CAS: 4360-12-7

An alkaloid found in the root of Rauwolfia serpentina, among other plant sources. It is a class Ia antiarrhythmic agent that apparently acts by changing the shape and threshold of cardiac action potentials. Ajmaline produces potent sodium channel blocking eff…

Kategori:
Ajmaline and derivativesAlkaloidsAntiarrhythmic agents +16
Target Protein:
Sodium channel protein type 5 subunit alpha
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Ajoene DB17735
small molecule | CAS: 92285-01-3

Deskripsi belum tersedia.

Kategori:
AnionsAnti-Infective AgentsAntifungal Agents +9
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AK106-001616 DB16058
small molecule | CAS: 590416-75-4

AK106-001616 is under investigation in clinical trial NCT01285752 (A Study of AK106-001616 in Patients With Rheumatoid Arthritis (RA)).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +3
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