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2279

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Halaman 40 / 46
biotech

Mesenchymal stem cells (MSCs) exert their therapeutic effects through multiple modalities, including paracrine factors such as exosomes. Exosomes are nanometer-sized, membrane-bound vesicles secreted for the purpose of cell-cell communication. Once secreted i…

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Streptomycin Approved DB01082
small molecule | CAS: 57-92-1

Streptomycin, an antibiotic derived from _Streptomyces griseus_, was the first aminoglycoside to be discovered and used in practice in the 1940s.[A233325,A233390] Selman Waksman and eventually Albert Schatz were recognized with the Nobel Prize in Medicine for…

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAminoglycoside Antibacterials +16
Target Protein:
16S ribosomal RNA23S ribosomal RNA30S ribosomal protein S12 +3
Waktu ParuhStreptomycins serum…
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Strimvelis DB17594
biotech

Deskripsi belum tersedia.

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STRO-001 DB17224
biotech

Deskripsi belum tersedia.

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STX-100 DB16334
biotech | CAS: 1439902-67-6

STX-100 is under investigation in clinical trial NCT01371305 (STX-100 in Patients With Idiopathic Pulmonary Fibrosis (IPF)).

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Succinic acid Approved DB00139
small molecule | CAS: 110-15-6

A water-soluble, colorless crystal with an acid taste that is used as a chemical intermediate, in medicine, the manufacture of lacquers, and to make perfume esters. It is also used in foods as a sequestrant, buffer, and a neutralizing agent. (Hawley's Condens…

Kategori:
Acids, AcyclicDicarboxylic AcidsDietary Supplements +3
Target Protein:
Succinate-semialdehyde dehydrogenase, mitochondrialSuccinate receptor 1
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Sucralfate Approved DB00364
small molecule | CAS: 54182-58-0

Sucralfate is a medication that is widely used to prevent and treat a number of diseases in the gastrointestinal tract such as duodenal ulcers [FDA label], gastro-esophageal reflux disease (GERD), gastritis, peptic ulcer disease, stress ulcer, in addition to …

Kategori:
Alimentary Tract and MetabolismAluminium CompoundsAluminum Complex +14
Target Protein:
Pepsin A-5Fibroblast growth factor 2Pro-epidermal growth factor +1
Waktu ParuhThe half-life is no…
Vol. DistribusiThis drug is absorb…
KlirensSucralfate contains…
Genetik -
Sufentanil Approved DB00708
small molecule | CAS: 56030-54-7

Sufentanil is an opioid analgesic that is used as an adjunct in anesthesia, in balanced anesthesia, and as a primary anesthetic agent. It is administered by the intravenous, epidural and sublingual routes. Also known as _Dsuvia_, the sublingual form is u…

Kategori:
Adjuvants, AnesthesiaAgents that produce hypertensionAnalgesics +25
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiSufentanil has a di…
KlirensThe total plasma cl…
Genetik -
Sugemalimab DB16641
biotech | CAS: 2256084-03-2

Sugemalimab is a fully human, full-length IgG4 monoclonal anti-PD-L1 antibody discovered by CStone Pharmaceuticals and being investigated against relapsed or refractory extranodal natural killer (NK)/T-cell lymphoma (R/R ENKTL) in adult patients and T-cell ly…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
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Sulesomab Approved DB13976
biotech | CAS: 167747-19-5

Market product is Tc99m-labeled murine antibody fragment for nuclear imaging of activated granulocytes.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
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Sulfacytine Approved DB01298
small molecule | CAS: 17784-12-2

Sulfacytine is a short-acting sulfonamide. The sulfonamides are synthetic bacteriostatic antibiotics with a wide spectrum against most gram-positive and many gram-negative organisms. However, many strains of an individual species may be resistant. Sulfonamide…

Kategori:
AmidesAminesAniline Compounds +5
Target Protein:
Dihydropteroate synthase
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Sulfadimethoxine Approved DB06150
small molecule | CAS: 122-11-2

Sulfadimethoxine is a sulfonamide antibiotic. Sulfadimethoxine is used to treat many infections, including treatment of respiratory, urinary tract, enteric, and soft tissue infections. It is most frequently used in veterinary medicine, although it is approved…

Kategori:
AmidesAminesAniline Compounds +16
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Sulfasalazine Approved DB00795
small molecule | CAS: 599-79-1

Sulfasalazine is an anti-inflammatory drug structurally related to salicylates and other non-steroidal anti-inflammatory drugs. It is indicated for managing inflammatory diseases such as ulcerative colitis and rheumatoid arthritis (RA).[L39065, A255582] Metab…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAlimentary Tract and Metabolism +23
Target Protein:
Broad substrate specificity ATP-binding cassette transporter ABCG2Transcription factor RelBTranscription factor p65 +12
Waktu ParuhThe observed plasma…
Vol. DistribusiFollowing intraveno…
KlirensThe calculated clea…
Genetik -
small molecule | CAS: 297-83-6

Sulfobromophthalein or otherwise called bromsulphthalein is used as a test of liver function in humans [A174970].

Kategori:
Benzene DerivativesColoring AgentsCompounds used in a research, industrial, or household setting +7
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Sulisobenzone DB11185
small molecule | CAS: 4065-45-6

Sulisobenzone is approved by the FDA in concentrations of up to 10% and in Canada, is approved by Health Canada at the same concentrations [F38]. It works to filter out both UVA and UVB rays, protecting the skin from sun UV damage [L2153]. The UV-filter s…

Kategori:
Benzene DerivativesDrugs that are Mainly Renally ExcretedKetones +1
Target Protein:
Skin epithelial cells
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Sumanirole DB06477
small molecule | CAS: 179386-43-7

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
D(2) dopamine receptorD(3) dopamine receptorD(4) dopamine receptor
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Suramin DB04786
small molecule | CAS: 145-63-1

A polyanionic compound with an unknown mechanism of action. It is used parenterally in the treatment of African trypanosomiasis and it has been used clinically with diethylcarbamazine to kill the adult Onchocerca. (From AMA Drug Evaluations Annual, 1992, p164…

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAnti-Infective AgentsAntinematodal Agents +12
Target Protein:
HeparanaseP2Y purinoceptor 2NAD-dependent protein deacylase sirtuin-5, mitochondrial +5
Waktu ParuhApproximately 36 to…
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Suratadenoturev DB18672
biotech | CAS: 1268642-13-2

Suratadenoturev is a gene-modified oncolytic adenovirus expressing the telomerase reverse transcriptase gene.

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Susoctocog alfa Approved DB11606
biotech | CAS: 1339940-90-7

Intravenous susoctocog alfa is a recombinant, B-domain deleted, porcine sequence antihaemophilic factor VIII (FVIII) product that has recently been approved for the treatment of bleeding episodes in adults with acquired haemophilia A (AHA). AHA is a rare blee…

Kategori:
Blood and Blood Forming OrgansBlood Coagulation FactorsHemostatics
Target Protein:
von Willebrand factor
Waktu ParuhThe terminal half-l…
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
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Sutimlimab Approved DB14996
biotech | CAS: 2049079-64-1

Cold agglutinin disease (CAD) is a type of autoimmune hemolytic anemia (AIHA) in which autoantibodies directed against red blood cell surface antigens cause hemolysis at low (3-4°C) temperatures.[A245154,L40114] This cold subtype accounts for approximately 15…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Complement C1s subcomponent
Waktu ParuhAt the approved rec…
Vol. DistribusiAt steady-state, th…
KlirensAt the approved rec…
Genetik -
SVV-001 DB06129
biotech

SVV-001 is investigated for use/treatment in cancer/tumors and lung cancer. SVV-001 is a solid. SVV-001 (Seneca Valley Virus) is a novel native picornavirus being developed as a systemically deliverable oncolytic virus for treatment of human cancers with neur…

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Syagrus romanzoffiana pollen Approved DB10482
biotech

Syagrus romanzoffiana pollen is the pollen of the Syagrus romanzoffiana plant. Syagrus romanzoffiana pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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SYNB1020 DB17667
biotech

SYNB1020 is an engineered strain of _Escherichia coli_ Nissle 1917 developed by Synlogic Inc. It was initially designed to convert ammonia to L-arginine [A258838] and granted orphan designation by the FDA for the treatment of urea cycle disorders in August 20…

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SynOV1.1 DB17539
biotech

SynOV1.1 is an investigational cancer immunotherapy developed by SyngenTech. It is a recombinant oncolytic adenovirus, controlled by synthetic gene circuit, encoding the human immunostimulating factor cytokine granulocyte-macrophage colony-stimulating factor …

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small molecule

Synthetic conjugated estrogens A are composed of a blend of the following nine synthetic estrogenic substances: estrone sulfate, sodium equilin sulfate, sodium 17?-dihydroequilin sulfate, sodium 17?-estradiol sulfate, sodium 17?­ dihydroequilin sulfate, sodiu…

Kategori:
Cytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 SubstratesCytochrome P-450 Substrates +7
Target Protein:
Estrogen receptor
Waktu ParuhThe half life of ba…
Vol. DistribusiThe distribution of…
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small molecule | CAS: 746658-13-9

Synthetic conjugated estrogens, B tablets contain a blend of ten synthetic estrogenic substances. The estrogenic substances are: sodium estrone sulfate, sodium equilin sulfate, sodium 17?-dihydroequilin sulfate, sodium 17?-estradiol sulfate, sodium 17?­ dihyd…

Kategori:
Cytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 SubstratesCytochrome P-450 Substrates +7
Target Protein:
Estrogen receptor
Waktu ParuhThe half life of ba…
Vol. DistribusiThe distribution of…
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TA-CIN DB05809
biotech

TA-CIN is a subunit vaccine comprising L2/E6/E7 proteins from Human Papillomavirus (HPV16), designed to generate a strong cellular immune response against HPV-infected cells.

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Tabelecleucel Approved DB17072
biotech

Tabelecleucel is an innovative therapy that uses Epstein-Barr virus (EBV)-specific allogeneic cytotoxic T cells (CTLs). It is produced by mixing T-cells with B-cells that have been infected with the Epstein-Barr virus (EBV). Both T-cells and B-cells are obtai…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsAntineoplastic cell and gene therapy
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Tafasitamab Approved DB15044
biotech | CAS: 1422527-84-1

Tafasitamab is a humanized, CD19-directed cytolytic monoclonal antibody intended for the treatment of B-cell malignancies.[L15302] It is produced using recombinant DNA technology in Chinese hamster ovary cells, and contains an IgG1/2 hybrid Fc-domain which ha…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +13
Target Protein:
B-lymphocyte antigen CD19
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe total volume of…
KlirensThe clearance of ta…
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Tafluprost Approved DB08819
small molecule | CAS: 209860-87-7

A prostaglandin analogue ester prodrug used topically (as eye drops) to control the progression of glaucoma and in the management of ocular hypertension. Chemically, tafluprost is a fluorinated analog of prostaglandin F2-alpha. Tafluprost was approved for use…

Kategori:
Antiglaucoma Preparations and MioticsAutacoidsBiological Factors +13
Target Protein:
Prostaglandin F2-alpha receptor
Waktu Paruh-
Vol. DistribusiThe highest concent…
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Tafolecimab DB16336
biotech | CAS: 2225109-03-3

Tafolecimab is under investigation in clinical trial NCT04031742 (A Study to Evaluate Safety and Efficacy of IBI306, a PCSK9 Monoclonal Antibody in Chinese Subjects With Homozygous Familial Hypercholesterolemia).

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Tagitanlimab DB18221
biotech | CAS: 2417649-97-7

Deskripsi belum tersedia.

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Tagraxofusp Approved DB14731
biotech | CAS: 2055491-00-2

Tagraxofusp is a CD123-directed cytotoxin. It is a fusion protein composed of a human interleukin-3 (IL-3) that is genetically fused to the catalytic and translocation domains of truncated diphtheria toxin (DT) produced in _Escherichia coli_.[A253762, A253887…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +7
Target Protein:
Interleukin-3 receptor subunit alpha
Waktu ParuhThe mean (SD) termi…
Vol. DistribusiFollowing administr…
KlirensMean clearance (SD)…
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TAK-611 DB17644
biotech

TAK-611, formerly known as SHP611, is a recombinant human arylsulfatase A. First developed by Takeda, it is being investigated for the treatment of metachromatic leukodystrophy.

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biotech | CAS: 1580555-26-5

Talditercept alfa is under investigation in clinical trial NCT03039686 (Clinical Trial to Evaluate the Efficacy, Safety, and Tolerability of RO7239361 in Ambulatory Boys With Duchenne Muscular Dystrophy).

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Taliglucerase alfa Approved DB08876
biotech | CAS: 37228-64-1

Taliglucerase alfa is the recombinant active form of the human lysosomal enzyme, ?-glucocerebrosidase. It was approved in 2012 and is marketed under the name Elelyso for use in patients with type 1 Gaucher's disease.

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +7
Target Protein:
Glucocerebroside
Waktu ParuhThe half life is be…
Vol. DistribusiThe steady state vo…
KlirensThe systemic cleara…
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Talimogene laherparepvec Approved DB13896
biotech | CAS: 1187560-31-1

Talimogene laherparepvec is an oncolytic treatment used in local treatment of unresectable cutaneous, subcutaneous, and nodal lesions in patients with recurrent melanoma. It is a genetically administered herpes simplex virus 1 (HSV-1) that expresses human cyt…

Kategori:
AlphaherpesvirinaeAntineoplastic AgentsAntineoplastic Agents, Immunological +9
Target Protein:
Granulocyte-macrophage colony-stimulating factor
Waktu ParuhReadily accessible …
Vol. DistribusiTalimogene laherpar…
KlirensAlthough readily ac…
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TALL-104 DB17360
biotech

Deskripsi belum tersedia.

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Talquetamab Approved DB16678
biotech | CAS: 2226212-40-2

Talquetamab is a IgG4-PAA bispecific G protein-coupled receptor class C group 5 member D (GPRC5D)-directed CD3 T-cell engager. It consists of two arms - anti-GPRC5D and anti-CD3 arms - linked by two interchain disulfide bonds, each arm comprising a heavy and …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntineoplastic Agents +7
Target Protein:
T-cell surface glycoprotein CD3G-protein coupled receptor family C group 5 member D
Waktu ParuhThe mean (CV%) term…
Vol. DistribusiThe geometric mean …
KlirensTalquetamab clearan…
Genetik -
Tanespimycin DB05134
small molecule | CAS: 75747-14-7

Tanespimycin, manufactured by Conforma Therapeutics is under development as a small molecule inhibitor of heat shock protein 90 (HSP90). It is developed for the treatment of several types of cancer, solid tumors or chronic myelogenous leukemia.

Kategori:
AmidesHSP90 Heat-Shock Proteins, antagonists & inhibitorsLactams +2
Target Protein:
Heat shock protein HSP 90-alphaHeat shock protein HSP 90-beta
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Tanfanercept DB19142
biotech | CAS: 2119738-70-2

Tanfanercept is under investigation in clinical trial NCT06400589 (A Study to Evaluate the Efficacy and Safety of Tanfanercept (HL036) in Dry Eye Disease).

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Tangerine peel DB14316
biotech

Tangerine peel is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Biological ProductsComplex MixturesPharmaceutical Preparations +2
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Taniraleucel DB18311
biotech

Deskripsi belum tersedia.

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Tapentadol Approved DB06204
small molecule | CAS: 175591-23-8

Tapentadol is a centrally-acting synthetic analgesic with a dual mechanism of action. It is a mu-opioid receptor agonist that also inhibits norepinephrine reuptake.[A260721, A36596] Tapentadol was first approved by the FDA on November 20, 2008. The extende…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAnalgesics +25
Target Protein:
Mu-type opioid receptorSodium-dependent noradrenaline transporterKappa-type opioid receptor +2
Waktu ParuhThe terminal half-l…
Vol. DistribusiTapentadol is widel…
KlirensThe total clearance…
Genetik -
biotech | CAS: 2411896-53-0

Tarcocimab tedromer is under investigation in clinical trial NCT06270836 (A Study to Evaluate the Efficacy and Safety of Tarcocimab Tedromer Compared With Sham Treatment in Participants With Moderately Severe to Severe Non-proliferative Diabetic Retinopathy (…

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Tarenflurbil DB05289
small molecule | CAS: 51543-40-9

Tarenflurbil is an investigational drug that was studied in patients with mild Alzheimer's disease. It is a selective amyloid lowering agent (SALA) that reduces levels of the toxic peptide amyloid beta 42 (A?42) in cultured human cells and in animal models. A…

Kategori:
Acids, AcyclicAnalgesicsAnalgesics, Non-Narcotic +11
Target Protein:
Gamma-secretase subunit APH-1BNicastrinGamma-secretase subunit APH-1A +4
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TAS-106 DB06656
small molecule | CAS: 180300-43-0

TAS-106 is a new nucleoside antimetabolite. TAS-106 has demonstrated strong antitumor activity without serious toxicity in nude rat models bearing human tumours [A31693].

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosidesPyrimidine Nucleosides +2
Target Protein:
DNA-directed RNA polymerase subunit betaDNA-directed RNA polymerase subunit beta'
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Tasquinimod DB05861
small molecule | CAS: 254964-60-8

The quinoline-3-carboxamide anti-angiogenic agent, tasquinimod, enhances the anti-prostate cancer efficacy of androgen ablation and taxotere without effecting serum PSA directly in human xenografts

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
Target Protein:
Protein S100-A9
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Taurine Approved DB01956
small molecule | CAS: 107-35-7

Taurine, whose chemical name is 2-aminoethanesulfonic acid, is one of the most abundant amino acids in several organs. It plays important role in essential biological processes.[A31396] This conditional amino acid can be either be manufactured by the body or …

Kategori:
AlkanesAlkanesulfonic AcidsAmino Acids +5
Target Protein:
Glutamate receptor ionotropic, NMDA 2BGlycine receptor subunit betaGlycine receptor subunit alpha-2 +6
Waktu ParuhOral administration…
Vol. DistribusiThe distribution of…
KlirensThe clearance rate …
Genetik -
Tauroursodeoxycholic acid Approved DB08834
small molecule | CAS: 14605-22-2

Tauroursodeoxycholic acid, also known as ursodoxicoltaurine, is a highly hydrophilic tertiary bile acid [A249070] that is produced in humans at a low concentration.[A249070] It is a taurine conjugate of [ursodeoxycholic acid] [A249065] with comparable therape…

Kategori:
Alimentary Tract and MetabolismBile acids and derivativesBile Acids and Salts +10
Target Protein:
Integrin alpha-5
Waktu Paruh-
Vol. DistribusiThere is evidence t…
Klirens-
Genetik -
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