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1977

Total database: 17430
Struktur (SMILES)
1074 (54.3%)
Target
1046 (52.9%)
Genomik
39 (2.0%)
Referensi
1977 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (1977)

Halaman 39 / 40
Velpatasvir Approved DB11613
small molecule | CAS: 1377049-84-7

Velpatasvir is a Direct-Acting Antiviral (DAA) medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized in…

Kategori:
Acids, AcyclicAnti-Infective AgentsAntiinfectives for Systemic Use +22
Target Protein:
Nonstructural protein 5A
Waktu Paruh15h [FDA Label].
Vol. Distribusi1.4-1.6 L/kg [A191…
KlirensEstimated 0.12 L/h/…
Genetik -
Venanprubart DB18891
biotech | CAS: 2635407-50-8

Venanprubart is under investigation in clinical trial NCT05781451 (Anti-btla Agonist Therapy in Subjects With Primary Sjogren's Syndrome).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Venlafaxine Approved DB00285
small molecule | CAS: 93413-69-5

Venlafaxine is an antidepressant and a serotonin and norepinephrine reuptake inhibitor (SNRI). Its active metabolite, [desvenlafaxine], works by blocking the reuptake of serotonin and norepinephrine, which are key neurotransmitters in mood regulation. Venlafa…

Kategori:
Agents producing tachycardiaAgents that reduce seizure thresholdAmines +39
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporterSodium-dependent dopamine transporter
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +2
Waktu ParuhThe apparent elimin…
Vol. DistribusiThe apparent volume…
KlirensMean ± SD plasma ap…
Genetik 5 Varian
Vercirnon DB15250
small molecule | CAS: 698394-73-9

Vercirnon is a novel, orally active anti-inflammatory agent that targets a chemokine receptor protein implicated in both Crohn's disease and ulcerative colitis, the two principal forms of IBD. It is under investigation in clinical trial NCT01611805 (Japanese …

Kategori:
AmidesSulfonesSulfur Compounds
Target Protein:
C-C chemokine receptor type 9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vericiguat Approved DB15456
small molecule | CAS: 1350653-20-1

Vericiguat is a direct stimulator of soluble guanylate cyclase (sGC) used in the management of systolic heart failure to reduce mortality and hospitalizations.[L31153] A key component of the NO-sGC-cGMP signaling pathway that helps to regulate the cardiovascu…

Kategori:
BCRP/ABCG2 SubstratesCardiac TherapyGuanylate Cyclase Stimulators +8
Target Protein:
Retinal guanylyl cyclase 1Guanylate cyclase soluble subunit beta-1
Waktu ParuhIn patients with he…
Vol. DistribusiIn healthy subjects…
KlirensVericiguat is a low…
Genetik -
Verubecestat DB12285
small molecule | CAS: 1286770-55-5

Verubecestat is under investigation for the treatment of Alzheimer's Disease, Prodromal Alzheimer's disease, and Amnestic Mild Cognitive Impairment. Verubecestat is Merck’s investigational oral ?-site amyloid precursor protein cleaving enzyme (BACE1 or ? …

Kategori:
Sulfur CompoundsThiazines
Target Protein:
Beta-secretase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Vespula pensylvanica venom protein is an extract of Vespula pensylvanica venom. Vespula pensylvanica venom protein is used in allergenic testing.

Kategori:
Bee and Wasp VenomCell-mediated ImmunityIncreased Histamine Release +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Vespula vulgaris venom protein is an extract of Vespula vulgaris venom. Vespula vulgaris venom protein is used in allergenic testing.

Kategori:
Allergenic ExtractsBee and Wasp VenomCell-mediated Immunity +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vestronidase alfa Approved DB12366
biotech | CAS: 1638194-78-1

Vestronidase alfa, or vestronidase alfa-vjbk, is a recombinant human lysosomal beta glucuronidase that is a purified enzyme produced by recombinant DNA technology in a Chinese hamster ovary cell line. The enzyme is a homotetramer consisted of 4 monomers with …

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes +3
Waktu ParuhAfter repeated dosi…
Vol. DistribusiAfter repeated dosi…
KlirensAfter repeated dosi…
Genetik -
VG161 DB18469
biotech

VG161 is an oncolytic virus therapy under investigation for the treatment of cholangiocarcinoma.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vibegron Approved DB14895
small molecule | CAS: 1190389-15-1

Vibegron is a potent, selective beta-3 adrenergic receptor (?3) agonist that relaxes the detrusor smooth muscle of the bladder, thereby increasing bladder capacity.[L28305] Vibegron was first approved in Japan in September 2018 for the treatment of overactive…

Kategori:
Adrenergic AgonistsAdrenergic beta-3 Receptor AgonistsAdrenergic beta-Agonists +10
Target Protein:
Beta-3 adrenergic receptor
Waktu ParuhThe terminal plasma…
Vol. DistribusiThe mean apparent v…
KlirensThere is limited in…
Genetik -
Vibostolimab DB16420
biotech | CAS: 2231305-30-7

Vibostolimab is under investigation in clinical trial NCT04303169 (Substudy 02C: Safety and Efficacy of Pembrolizumab in Combination With Investigational Agents or Pembrolizumab Alone in Participants With Stage III Melanoma Who Are Candidates for Neoadjuvant …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1704499-30-8

_Vibrio cholerae_ CVD 103-HgR strain live antigen is a component of Vaxchora, an oral vaccine for immunization against _Vibrio cholerae_ serogroup O1.[L12801] Cholera is an acute bacterial disease of the small intestine caused by _Vibrio cholerae_, which is g…

Kategori:
Bacterial VaccinesBiological ProductsComplex Mixtures +3
Waktu ParuhPharmacokinetic inf…
Vol. DistribusiPharmacokinetic inf…
KlirensPharmacokinetic inf…
Genetik -
VidPrevtyn Beta Approved DB16427
biotech

VidPrevtyn Beta is an adjuvanted, recombinant COVID-19 vaccine developed collaboratively by GlaxoSmithKline (GSK) and Sanofi Pasteur.[L49691] It comprises a recombinant SARS-CoV-2 spike protein (B.1.351 strain) - produced by recombinant DNA technology using a…

Kategori:
Biological ProductsComplex MixturesCOVID-19 Vaccines +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vilastobart DB19327
biotech | CAS: 2760549-50-4

Vilastobart is under investigation in clinical trial NCT04896697 (Vilastobart (XTX101) Monotherapy and Vilastobart and Atezolizumab Combination Therapy in Advanced Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vilazodone Approved DB06684
small molecule | CAS: 163521-12-8

Vilazodone is a novel compound with combined high affinity and selectivity for the 5-hydroxytryptamine (5-HT) transporter and 5-HT(1A) receptors[Label,A177622]. Vilazodone may also be associated with less sexual dysfunction and weight gain[A6947]. Vilazodone …

Kategori:
Agents that produce hypertensionAntidepressive AgentsAntidepressive Agents Indicated for Depression +26
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 1A
Waktu Paruh25 hours[Label,A384…
Vol. DistribusiVilazodone's volume…
KlirensClearance of vilazo…
Genetik -
Vincristine Approved DB00541
small molecule | CAS: 57-22-7

Vincristine is an antitumor vinca alkaloid isolated from Vinca Rosea. It is marketed under several brand names, many of which have different formulations such as Marqibo (liposomal injection) and Vincasar. Vincristine is indicated for the treatment of acute l…

Kategori:
Agents Causing Muscle ToxicityAlkaloidsAntimitotic Agents +33
Target Protein:
Tubulin beta chainTubulin alpha-4A chain
Waktu ParuhWhen intravenously …
Vol. DistribusiWithin 15 to 30 min…
Klirens-
Genetik -
Vindesine Approved DB00309
small molecule | CAS: 53643-48-4

Vinblastine derivative with antineoplastic activity against cancer. Major side effects are myelosuppression and neurotoxicity. Vindesine is used extensively in chemotherapy protocols (antineoplastic combined chemotherapy protocols).

Kategori:
AlkaloidsAntimitotic AgentsAntineoplastic Agents +19
Target Protein:
Tubulin beta-1 chain
Waktu Paruh24 hours.
Vol. Distribusi-
Klirens-
Genetik -
Vinflunine Approved DB11641
small molecule | CAS: 162652-95-1

Vinflunine is a third-generation member of the vinca alkaloid family with anti-tumour actions. It was first described in 1998 at the Pierre Fabre research center in France. Like other vinca agents, vinflunine is an anti-mitotic agent that induces a cell cycle…

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +14
Target Protein:
Tubulin beta chain
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe terminal volume…
KlirensThe total blood cle…
Genetik -
Vintafolide DB05168
small molecule | CAS: 742092-03-1

Vintafolide is a folate-targeted chemotherapeutic conjugate (folate vitamin + vinca alkaloid) in clinical stage development as a treatment for folate-receptor positive cancers.

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +9
Target Protein:
Folate receptor alphaFolate receptor betaFolate receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Viralym-C DB17975
biotech

Viralym-C is an investigational T-cell immunotherapy developed by ViraCyte. It consists of Human Leukocyte Antigen (HLA)-matched cytomegalovirus (CMV)-specific T lymphocytes. It was granted FDA orphan designation in January 2017 and investigated for the treat…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vismodegib Approved DB08828
small molecule | CAS: 879085-55-9

Vismodegib is an orally active small molecule that inhibits the hedgehog signaling pathway by binding to and inhibiting the transmembrane protein smoothened homologue (SMO).[A258613,A258618,L45803] It was discovered by high-throughput screening of a library o…

Kategori:
AmidesAminesAniline Compounds +18
Target Protein:
Protein smoothened
Waktu ParuhThe half-life of vi…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Visugromab DB18894
biotech | CAS: 2556646-63-8

Visugromab is under investigation in clinical trial NCT06059547 (Neoadjuvant Immunotherapy in Combination With the Anti-gdf-15 Antibody Visugromab (CTL-002) for Treatment of Muscle Invasive Bladder Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vitespen DB06400
biotech | CAS: 492448-75-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiological ProductsComplex Mixtures +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VLTS-589 DB05430
small molecule

VLTS-589 consists of plasmid encoding the angiomatrix protein Del-1 in conjunction with poloxamer 188 for the treatment of peripheral vascular disease.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VLTS-934 DB05597
small molecule

VLTS-934 was developed by Valentis inc. for the treatment of Peripheral Arterial Disease (PAD). It was under investigation in clinical trial NCT00113009 (Trial of VLTS-934 in Subjects With Intermittent Claudication Secondary to Peripheral Arterial Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2490556-51-7

Vobramitamab duocarmazine is under investigation in clinical trial NCT05551117 (A Study of Vobramitamab Duocarmazine in Participants With Metastatic Castration Resistant Prostate Cancer and Other Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Voclosporin Approved DB11693
small molecule | CAS: 515814-01-4

Lupus nephritis (LN) is a type of glomerulonephritis occurring in patients with systemic lupus erythematosus (SLE). LN is a significant cause of renal failure, morbidity, and death in patients with SLE. Within 10 years of being diagnosed with SLE, 5-20% of …

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating AgentsCalcineurin Inhibitor Immunosuppressant +16
Target Protein:
Guided entry of tail-anchored proteins factor CAMLGProtein phosphatase 3 catalytic subunit alphaCalcineurin subunit B type 1 +1
Waktu ParuhThe average termina…
Vol. DistribusiThe apparent volume…
KlirensThe mean apparent s…
Genetik -
Volagidemab DB16421
biotech | CAS: 1233956-13-2

Volagidemab is under investigation in clinical trial NCT03117998 (Multiple Dose Study to Evaluate the Efficacy, Safety and Pharmacodynamics of REMD-477 in Subjects With Type 1 Diabetes Mellitus).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Volanesorsen Approved DB15067
biotech | CAS: 915430-78-3

Volanesorsen is an antisense oligonucleotide that binds to apoC-III mRNA to prevent its translation.[L16621] It is indicated to treat familial chylomicronemia, a genetic condition that prevents breakdown of triglycerides and chylomicrons.[L16621] This drug is…

Kategori:
CarbohydratesGlycosidesLipid Modifying Agents +4
Target Protein:
Apolipoprotein C-III
Waktu ParuhVolanesorsen has a …
Vol. DistribusiThe volume of distr…
KlirensThe exact rate of c…
Genetik -
biotech | CAS: 2092457-20-8

Volrubigene ralaparvovec is under investigation in clinical trial NCT03223194 (Gene Transfer Clinical Study in Crigler-najjar Syndrome).

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Von Willebrand factor human Approved DB13133
biotech | CAS: 109319-16-6

The human von Willebrand factor (vWF) is a human plasma-derived vWF, an endogenous large multimeric plasma glycoprotein involved in hemostasis. It serves a dual role in hemostasis by mediating platelet adhesion and aggregation at the site of blood vessel inju…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +8
Target Protein:
Coagulation factor VIIICollagen alpha-1(I) chainAsialoglycoprotein receptor 1 +1
Waktu ParuhIn patients with Ty…
Vol. DistribusiThe volume of distr…
KlirensIn patients with Ty…
Genetik -
Vonoprazan Approved DB11739
small molecule | CAS: 881681-00-1

Vonoprazan is a potassium-competitive acid blocker (PCAB) that inhibits H<sup>+</sup>, K<sup>+</sup>-ATPase-mediated gastric acid secretion. PCABs represent an alternative to proton-pump inhibitors for the treatment of acid-related disorders. Unlike proton-pu…

Kategori:
Alimentary Tract and MetabolismAmidesCytochrome P-450 CYP2B6 Substrates +17
Target Protein:
Hydrogen potassium ATPase
Waktu ParuhVonoprazan has an e…
Vol. DistribusiVonoprazan has an a…
KlirensVonoprazan has an a…
Genetik -
Vopratelimab DB15378
biotech | CAS: 2039148-04-2

Vopratelimab is under investigation in clinical trial NCT02904226 (JTX-2011 Alone and in Combination With Anti-PD-1 or Anti-CTLA-4 in Subjects With Advanced and/or Refractory Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Voretigene neparvovec Approved DB13932
biotech | CAS: 1646819-03-5

Voretigene Neparvovec-rzyl (VN-rzyl) is an adeno-associated virus vector-based gene therapy.[L1094] An adeno-associated virus is a small virus that infects humans and other primates. It is not pathogenic and it causes a very mild immune response. This type of…

Kategori:
Adeno-associated Viral Vector TherapiesOphthalmologicalsSensory Organs
Target Protein:
Retinoid isomerohydrolase
Waktu ParuhBased on the pharma…
Vol. DistribusiVN-rzyl was shown t…
KlirensAccording to the ki…
Genetik -
Vorolanib DB15247
small molecule | CAS: 1013920-15-4

Vorolanib is under investigation in clinical trial NCT03904719 (CM082 and JS001 in Patients With Advanced Small-cell Lung Cancer (SCLC)).

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vortioxetine Approved DB09068
small molecule | CAS: 508233-74-7

Vortioxetine is an antidepressant medication indicated for the treatment of major depressive disorder (MDD). It is classified as a serotonin modulator and stimulator (SMS) as it has a multimodal mechanism of action towards the serotonin neurotransmitter syste…

Kategori:
Agents that produce hypertensionAnti-Anxiety AgentsAntidepressive Agents +30
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 3A5-hydroxytryptamine receptor 7 +4
Waktu ParuhMean terminal half­…
Vol. DistribusiThe apparent volume…
Klirens-
Genetik -
Voruciclib DB15157
small molecule | CAS: 1000023-04-0

Voruciclib is under investigation in clinical trial NCT03547115 (A Phase 1 Study of Voruciclib in Subjects With B-Cell Malignancies or AML).

Kategori:
Antineoplastic AgentsCarbohydratesEnzyme Inhibitors +6
Target Protein:
Cyclin-dependent kinase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Voxilaprevir Approved DB12026
small molecule | CAS: 1535212-07-7

Voxilaprevir is a Direct-Acting Antiviral (DAA) medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized i…

Kategori:
Acids, AcyclicAmidesAmino Acids +36
Target Protein:
Genome polyproteinGenome polyprotein
Waktu Paruh33 hr [FDA Label]
Vol. Distribusi-
Klirens-
Genetik -
VP025 DB05133
small molecule

VP025, a novel drug formulation based on phospholipid microparticles incorporating phosphatidylglycerol, can inhibit neuroinflammation. VP025 may inhibit immune system activation and protect motoneurons from injury. It also shows the ability to reduce inflamm…

Target Protein:
Interleukin-1 beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vunakizumab DB15154
biotech | CAS: 1792181-33-9

Vunakizumab is under investigation in clinical trial NCT03463187 (Multi-Dose Study of SHR-1314 in Subjects With Moderate-to-severe Plaque Psoriasis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vutrisiran Approved DB16699
biotech | CAS: 1867157-35-4

Vutrisiran is a double-stranded small interfering ribonucleic acid (siRNA) that targets wild-type and mutant transthyretin (TTR) messenger RNA (mRNA).[L42065] This siRNA therapeutic is indicated for the treatment of neuropathies associated with hereditary tra…

Kategori:
Antisense OligonucleotidesNervous SystemNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
Transthyretin mRNA
Waktu ParuhThe median half-lif…
Vol. DistribusiBased on a populati…
KlirensThe apparent cleara…
Genetik -
VXA-CoV2-1 DB16433
biotech

VXA-CoV2-1 is a non-replicating adenoviral vector-based oral tableted vaccine candidate that expresses a SARS-CoV-2 antigen and dsRNA adjuvant[L30493]. This oral vaccine aims to induce immunogenicity through induction of potent serum neutralizing antibodies t…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Water Approved DB09145
small molecule | CAS: 7732-18-5

Water (chemical formula: H2O) is a transparent fluid which forms the world's streams, lakes, oceans and rain, and is the major constituent of the fluids of organisms. As a chemical compound, a water molecule contains one oxygen and two hydrogen atoms that are…

Kategori:
DiluentsEENT Drugs, MiscellaneousIrrigating Solutions +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
White mustard seed Approved DB15606
biotech

White mustard seed allergenic extract is used in allergenic testing.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Wormwood Approved DB14291
biotech

Wormwood is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
LipidsOils
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
WX-UK1 DB05476
small molecule | CAS: 255374-84-6

WX-UK1 is a 3-amidinophenylalanine-based non-cytotoxic small molecule that belongs to a new class of drugs. In animal models, WX-UK1 blocks tumor cell invasion, metastasis and primary tumor growth by inhibiting serine proteases and the urokinase Plasminogen A…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +1
Target Protein:
Urokinase plasminogen activator surface receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Xanthan gum Approved DB11253
small molecule | CAS: 11138-66-2

Xanthan gum is a polysaccharide gum derived from* Xanthomonas campestris* by a pure-culture fermentation process and purified by recovery with isopropyl alcohol. The major constituents include D-glucose, D-mannose, and D-glucuronic acid. Xanthan gum is a dire…

Kategori:
AntigensAntigens, BacterialBiological Factors +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
XAV-19 DB15895
biotech

XAV-19 is an intravenous antibody-based treatment targeted towards SARS-CoV-2 and other coronaviruses[L16553,L16558]. The therapy concept is based on [COVID-19 convalescent plasma]. However, rather than using human plasma, XAV-19 is a heterologous swine glyco…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
XL019 DB05243
small molecule

XL019 is a selective inhibitor of the cytoplasmic tyrosine kinase JAK2. An IND for XL019 was filed by Exelixis in May 2007.

Target Protein:
Tyrosine-protein kinase JAK2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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