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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 39 / 252
small molecule

Deskripsi belum tersedia.

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Genetik -
small molecule | CAS: 58-64-0

Deskripsi belum tersedia.

Kategori:
Adenine NucleotidesHeterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
P2Y purinoceptor 6Transient receptor potential cation channel subfamily M member 4P2Y purinoceptor 12
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Adenosine phosphate Approved DB00131
small molecule | CAS: 61-19-8

Adenosine phosphate, or adenylic acid, is an adenine nucleotide containing one phosphate group esterified to the sugar moiety in the 2'-, 3'-, or 5'-position. Adenosine phosphate was withdrawn by the FDA since it was considered neither safe nor ef…

Kategori:
Adenine NucleotidesDietary SupplementsHeterocyclic Compounds, Fused-Ring +6
Target Protein:
5'-AMP-activated protein kinaseAdenosine kinase5'-AMP-activated protein kinase subunit beta-1 +11
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small molecule

Deskripsi belum tersedia.

Target Protein:
Eosinophil cationic proteinRibonuclease pancreaticNon-secretory ribonuclease
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small molecule

Deskripsi belum tersedia.

Target Protein:
Nuclease P1
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small molecule

Deskripsi belum tersedia.

Kategori:
Vanadates
Target Protein:
Bifunctional 3'-phosphoadenosine 5'-phosphosulfate synthase 1
Waktu Paruh-
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small molecule

Deskripsi belum tersedia.

Target Protein:
Adenosine 5'-monophosphoramidase HINT1
Waktu Paruh-
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small molecule

Serves as the glycosyl donor for formation of bacterial glycogen, amylose in green algae, and amylopectin in higher plants. [PubChem]

Target Protein:
ADP-L-glycero-D-manno-heptose-6-epimerase
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small molecule

Deskripsi belum tersedia.

Target Protein:
Diadenosine hexaphosphate hydrolase
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small molecule

Deskripsi belum tersedia.

Target Protein:
Acetyl-coenzyme A synthetase
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small molecule

Deskripsi belum tersedia.

Target Protein:
Adenylate cyclase
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small molecule

Deskripsi belum tersedia.

Target Protein:
Folylpolyglutamate synthase
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small molecule

Deskripsi belum tersedia.

Target Protein:
Insulin receptorFolylpolyglutamate synthaseChemotaxis protein CheA +11
Waktu Paruh-
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small molecule

Deskripsi belum tersedia.

Target Protein:
NAD-dependent protein deacylase sirtuin-5, mitochondrialp-hydroxybenzoate hydroxylaseADP-ribose pyrophosphatase +8
Waktu Paruh-
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biotech

Deskripsi belum tersedia.

Kategori:
Actively Acquired ImmunityAdenovirus VaccinesLive Human Adenovirus Type 7 Vaccine +3
Waktu Paruh-
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Adenovirus/PNP DB17175
biotech

Deskripsi belum tersedia.

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small molecule

Deskripsi belum tersedia.

Target Protein:
Ribonuclease pancreatic
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small molecule | CAS: 1985-21-3

Deskripsi belum tersedia.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Target Protein:
Diphtheria toxin
Waktu Paruh-
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ADH-1 DB05485
biotech

Adherex's biotechnology compound, ADH-1, targets N-cadherin, a protein present on certain tumor cells and established tumor blood vessels. ADH-1 is currently in clinical development in a combination program with a range of chemotherapeutic agents to investiga…

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ADH-503 DB17133
small molecule | CAS: 2055362-74-6

Deskripsi belum tersedia.

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AdimrSC-2f DB16436
biotech

The AdimrSC-2f (SARS-CoV-2) vaccine is developed through Adimmune Corporation, the only influenza vaccine manufacturer with both EU GMP and US FDA certification in Asia[L30553]. A phase I study (NCT04522089) will investigate the safety and immunogenicity of t…

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Adinazolam DB00546
small molecule | CAS: 37115-32-5

Adinazolam (Deracyn®) is a benzodiazepine derivative with anxiolytic, anticonvulsant, sedative, and antidepressant properties. Adinazolam was first developed to enhance the antidepressant effects of [alprazolam]. It has never been approved by the FDA for clin…

Kategori:
Anti-Anxiety AgentsAntidepressive AgentsBenzazepines +12
Target Protein:
Translocator proteinGABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu ParuhLess than 3 hours.
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Adiphenine Approved DB15795
small molecule | CAS: 64-95-9

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAnticholinergic AgentsPhenylacetates
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Adipiplon DB06579
small molecule | CAS: 840486-93-3

Adipiplon is an nonbenzodiazepine anxiolytic developed by Neurogen Corporation. It is known by the standardized identifier NG2-73.

Kategori:
Anti-Anxiety AgentsCentral Nervous System AgentsCentral Nervous System Depressants +5
Target Protein:
GABA(A) Receptor Benzodiazepine Binding SiteGamma-aminobutyric acid receptor subunit alpha-3
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biotech

Adipose mesenchymal stem cells (AMSCs) are MSCs derived from adipose tissue, which is more accessible and less painful than stem cells extracted from most other sources. Autologous stem cells are those derived from a patient’s own cells while allogeneic stem …

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ADL 10-0101 DB05443
small molecule

ADL 10-0101 is a peripheral kappa opioid agonist analgesic product candidate. Preclinical trials of ADL 10-0101 have suggested that the compound may be effective for the treatment of inflammatory pain, itch and visceral pain. Because ADL 10-0101 does not cros…

Target Protein:
Kappa-type opioid receptor
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ADL-5859 DB18910
small molecule | CAS: 850305-06-5

ADL-5859 is under investigation in clinical trial NCT00626275 (Study Evaluating the Analgesic Efficacy and Safety of ADL5859 in Participants With Rheumatoid Arthritis).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +4
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ADL5859 DB05050
small molecule

ADL5859 is a novel, oral compound that targets the Delta opioid receptor. Delta receptor agonists are thought to offer benefits over other approaches to the management of pain.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +4
Target Protein:
Delta-type opioid receptor
Waktu Paruh-
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biotech | CAS: 2143579-02-4

Adlinacogene civaparvovec is an investigational _in vivo_ genome editing therapeutic product. It uses proprietary zinc finger nuclease (ZFN) genome editing to insert into the DNA of liver cells a copy of the F9 gene, which controls the production of Factor IX…

Kategori:
Adeno-associated Viral Vector Therapies
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Adomeglivant DB11704
small molecule | CAS: 1488363-78-5

Adomeglivant has been investigated for the basic science of Type 2 Diabetes.

Kategori:
Benzene Derivatives
Target Protein:
Glucagon receptor
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Adomiparin DB06005
small molecule | CAS: 9005-49-6

Deskripsi belum tersedia.

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ADP-597 DB12084
small molecule | CAS: 897732-93-3

JNJ-38431055 has been used in trials studying the treatment of Diabetes Mellitus, Type 2.

Target Protein:
Glucose-dependent insulinotropic receptor
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AdPEDF DB05138
biotech

AdPEDF is under development for the treatment of wet age-related macular degeneration (AMD). It has been shown to rapidly elevate the intraocular AdPEDF protein levels in the eye, inhibit abnormal blood vessel growth, and cause abnormal blood vessels to regre…

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Adrabetadex DB15146
small molecule | CAS: 128446-35-5

Adrabetadex is under investigation in clinical trial NCT03887533 (Combined Intrathecal and Intravenous VTS-270 Therapy for Liver and Neurological Disease Associated With Niemann-Pick Disease, Type C1).

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Adrafinil DB08925
small molecule | CAS: 63547-13-7

Adrafinil is a mild central nervous system stimulating drug typically employed to relieve excessive sleepiness and inattention in geriatric patients. It is also been used off-label to prevent fatigue or falling asleep for extended periods of time. Adrafinil d…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-Agonists +10
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Adrenalone DB13394
small molecule | CAS: 99-45-6

Deskripsi belum tersedia.

Kategori:
AlcoholsAlimentary Tract and MetabolismAmines +16
Waktu Paruh-
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Adrenomedullin DB19102
biotech | CAS: 154835-90-2

Adrenomedullin is under investigation in clinical trial NCT06072118 (Adrenomedullin for CADASIL).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Asthmatic AgentsAntihypertensive Agents +13
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Adriforant DB15027
small molecule | CAS: 943057-12-3

Adriforant is under investigation in clinical trial NCT00992342 (A Phase 1 Study To Evaluate The Safety And Tolerability Of Different Doses Of PF-03893787 In Healthy Adult Volunteers).

Target Protein:
Histamine H4 receptor
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ADU-S100 DB14722
small molecule | CAS: 1638241-89-0

ADU-S100 (MIW815) is a synthetic cyclic dinucleotide (CDN) agonist (activator) of Stimulator of Interferon Genes (STING), a receptor crucial to activate the innate (endogenous) immune system. ADU-S100 (MIW815) activates all known human and mouse STINGs, and e…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotides
Target Protein:
Stimulator of interferon genes protein
Waktu Paruh-
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Aducanumab Approved DB12274
biotech | CAS: 1384260-65-4

Aducanumab, or BIIB037, is a monoclonal IgG1 antibody that targets extracellular amyloid-? plaques in the brain; similar to [gantenerumab], [bapineuzumab] and [solanezumab].[A235668,A235730] Aducanumab is a recombinant antibody derived from patients with slow…

Kategori:
Alzheimer Disease, drug therapyAmino Acids, Peptides, and ProteinsAmyloid Beta-directed Antibodies +11
Target Protein:
Amyloid-beta precursor protein
Waktu ParuhThe terminal half l…
Vol. DistribusiThe volume of distr…
KlirensA 10 mg/kg intraven…
Genetik -
ADVM-053 DB17592
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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ADX-10061 DB05419
small molecule | CAS: 128022-68-4

ADX10061 is a potent, selective antagonist of the dopamine D1 receptor. It is developed by Addex Pharmaceuticals for the treatment of nicotine dependence.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Neuron-specific vesicular protein calcyon
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ADX10059 DB05070
small molecule

ADX10059 is a metabotropic glutamate receptor 5 (mGluR5) negative allosteric modulator (NAM). The orally available small molecule drug candidate, which is highly specific for mGluR5, was discovered at Addex in 2003. It is developed for the treatment of GERD,…

Target Protein:
Metabotropic glutamate receptor 5
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ADXS-31164 DB17325
biotech

Deskripsi belum tersedia.

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Adze-1.17-CD40L DB18528
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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AEE-788 DB12558
small molecule | CAS: 497839-62-0

AEE788 has been used in trials studying the treatment of Cancer, Glioblastoma Multiforme, and Brain and Central Nervous System Tumors.

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, Vascular Endothelial Growth Factor, antagonists & inhibitors
Target Protein:
Fibroblast growth factor receptor 2Fibroblast growth factor receptor 3
Waktu Paruh-
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AEG35156 DB06184
small molecule

A second-generation synthetic antisense oligonucleotide with potential antineoplastic activity. AEG35156 selectively blocks the cellular expression of X-linked inhibitor of apoptosis protein (XIAP), a pivotal inhibitor of apoptosis that is overexpressed in ma…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
E3 ubiquitin-protein ligase XIAP
Waktu Paruh-
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AEM-28 DB17642
biotech

AEM-28 is a 28 amino acid mimetic of apolipoprotein E being investigated for lipid disorders, such as homozygous familial hypercholesterolemia. It possesses anti-inflammatory properties.[A258764]

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AEM-28-14 DB17643
biotech

AEM-28-14 is an analog of [AEM-28], an apolipoprotein E mimetic peptide, with a 400 percent greater cholesterol-lowering efficacy and a several-fold increase in drug tolerability.[L45909] It is being investigated for lipid disorders such as homozygous familia…

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AEOL-10150 DB05874
small molecule | CAS: 286475-30-7

AEOL 10150 is developed by Aeolus as a therapeutic agents based on its proprietary small molecule catalytic antioxidants.

Kategori:
AntioxidantsBiological FactorsCoordination Complexes +3
Target Protein:
Superoxide dismutase [Cu-Zn]
Waktu Paruh-
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