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2279

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Halaman 38 / 46
SAR422459 DB17908
biotech

SAR422459 is a Lentiviral Vector Containing The Human Abca4 Gene that is currently being investigated to treat Stargardt disease.

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small molecule | CAS: 110880-55-2

Sar9, Met (O2)11-Substance P is a neurokinin-1 receptor agonist. It is an analog of the naturally occurring human neuropeptide Substance P, which can be found throughout the body, including in the airways of humans and many other species.

Kategori:
Amino Acids, Peptides, and ProteinsAutacoidsBiological Factors +11
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Sarafloxacin DB11491
small molecule | CAS: 98105-99-8

Sarafloxacin is a quinolone antibiotic drug, which was discontinued by its manufacturer, Abbott Laboratories, before receiving approval for use in the US or Canada.

Kategori:
4-QuinolonesAnti-Bacterial AgentsCytochrome P-450 CYP1A2 Inhibitors +8
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Sarecycline Approved DB12035
small molecule | CAS: 1035654-66-0

Sarecycline is a semi-synthetic derivative of tetracycline that was initially discovered by Paratek Pharmaceuticals from Boston, MA but then licensed to Warner Chilcott of Rockaway, NJ in July of 2007 [A40005]. After completing various phase-II and phase-III …

Kategori:
Anti-Acne PreparationsAnti-Acne Preparations for Systemic UseAnti-Bacterial Agents +7
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent o…
Genetik -
Sargramostim Approved DB00020
biotech | CAS: 123774-72-1

Sargramostim is a human recombinant granulocyte macrophage colony-stimulating factor (GM-CSF) expressed in yeast. It is a glycoprotein that is 127 residues. Substitution of Leu23 leads to a difference from native protein.

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +14
Target Protein:
Granulocyte-macrophage colony-stimulating factor receptor subunit alphaInterleukin-3 receptor subunit alphaCytokine receptor common subunit beta +2
Waktu Paruh-
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Klirens* 420 mL/min/m2 [No…
Genetik -
Sarilumab Approved DB11767
biotech | CAS: 1189541-98-7

Sarilumab is a fully human anti-interleukin 6 (IL-6) receptor monoclonal IgG1 antibody that binds to both membrane-bound and soluble IL-6 receptor forms, thus blocking the cis- and trans-inflammatory signalling cascades of IL-6.[A27262] Sarilumab was develope…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +22
Target Protein:
Interleukin-6 receptor subunit alphaHigh affinity immunoglobulin gamma Fc receptor ILow affinity immunoglobulin gamma Fc region receptor II-a +3
Waktu ParuhThe half-life will …
Vol. DistribusiIn patients with rh…
KlirensSarilumab is not el…
Genetik -
Sarracenia Purpurea Approved DB13965
biotech

_Sarracenia purpurea_, commonly known as the purple pitcher plant, northern pitcher plant, turtle socks, or side-saddle flower, is a perennial carnivorous plant in the family _Sarraceniaceae_. _Sarracenia purpurea_ attract and trap insects within their pitche…

Kategori:
Miscellaneous Analgesics and Antipyretics
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
biotech

SARS-CoV-2 mRNA vaccine (ARCoV) is a novel mRNA coronavirus vaccine that consists of a lipid nanoparticle-encapsulated mRNA encoding the receptor binding domain of SARS-CoV-2[A220048]. It is the first COVID-19 mRNA vaccine to be approved for clinical trials …

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biotech

Bimervax is an adjuvanted non-mRNA COVID-19 vaccine utilizing a SARS-CoV-2 recombinant spike (S) protein receptor binding domain (RBD) fusion heterodimer.[L48902] It is intended to elicit protection against Omicron XBB.1.5, one of the dominant circulating SAR…

Kategori:
COVID-19 VaccinesVaccinesViral Vaccines
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Saruplase DB13646
biotech | CAS: 99149-95-8

Deskripsi belum tersedia.

Kategori:
Agents causing angioedemaAmino Acids, Peptides, and ProteinsAnticoagulants +16
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Satralizumab Approved DB15762
biotech | CAS: 1535963-91-7

Satralizumab is a recombinant humanized monoclonal antibody targeted against human interleukin-6 (IL-6) receptors, similar to [tocilizumab], which is produced in Chinese hamster ovary cells and based on an IgG2 framework.[L15536] Satralizumab is used in the t…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Interleukin-6 receptor subunit alpha
Waktu ParuhThe terminal half-l…
Vol. DistribusiSatralizumab is sub…
KlirensThe total clearance…
Genetik -
SB 224289 DB17052
small molecule | CAS: 180083-23-2

SB-224289 is a small molecule with a high affinity for human 5-HT1B receptors.[A253122]

Kategori:
Piperidines
Target Protein:
5-hydroxytryptamine receptor 1B
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SB-559448 DB05930
small molecule

SB-559448 is a small-molecule drug that mimics the activity of thrombopoietin (TPO), a protein factor that promotes growth and production of blood platelets. This drug is developed by GlaxoSmithKline and used to treat Thrombocytopenia.Thrombocytopenia (decrea…

Target Protein:
Thrombopoietin receptor
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SBT101 DB18139
biotech

SBT101 is a non-replicating recombinant adeno-associated virus serotype 9 (AAV9) gene therapy vector containing the human adenosine triphosphate (ATP)-binding cassette (ABC) sub-family D member 1 (ABCD1) gene.

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scAAV9.U7.ACCA DB18582
biotech

scAAV9.U7.ACCA is a non-replicating recombinant adeno-associated virus vector containing 4 antisense sequences designed to target exon 2 in the human DMD gene under the control of U7 small nuclear non-coding RNA. Developed by Nationwide Children’s Hospital, i…

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SCH-58500 DB17416
biotech

SCH-58500 is a recombinant replication-deficient adenovirus vector carrying the human p53 gene.

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SCIB1 DB18439
biotech

SCIB1 is an investigational cancer vaccine being developed by Scancell Ltd. It is being investigated for the treatment of melanoma. It consists of plasmid DNA molecules that express a modified antibody in human cells, working to stimulate the patient's T cell…

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biotech

Centruroides (scorpion) Immune F(ab')2 (equine) is a purified preparation of immune globulin F(ab’)2 fragments that are derived from plasma of the horses immunized with venom of *C. noxius*, *C. l. limpidus*, *C. l. tecomanus*, and *C. s. suffusus*. It is int…

Kategori:
AntiveninsPassively Acquired ImmunityVenom Neutralization
Waktu Paruh159 ± 57 h [FDA lab…
Vol. DistribusiSteady state: 13.6 …
Klirens83.5 ± 38.4 ml/Hr […
Genetik -
scyllo-inositol DB03106
small molecule | CAS: 488-59-5

An isomer of glucose that has traditionally been considered to be a B vitamin although it has an uncertain status as a vitamin and a deficiency syndrome has not been identified in man. (From Martindale, The Extra Pharmacopoeia, 30th ed, p1379) Inositol phosph…

Kategori:
AlcoholsCarbohydratesStereoisomerism +1
Target Protein:
Lysosomal acid glucosylceramidase1-phosphatidylinositol phosphodiesteraseCDP-diacylglycerol--inositol 3-phosphatidyltransferase +1
Waktu Paruh-
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SEA-BCMA DB18309
biotech | CAS: 2115084-53-0

Deskripsi belum tersedia.

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SEA-CD70 DB17555
biotech

SEA-CD70 is an investigational humanized, non-fucosylated monoclonal antibody targeting CD70. SEA-CD70 is under investigation in clinical trial NCT04227847 (A Safety Study of SEA-CD70 in Patients With Myeloid Malignancies).

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Secnidazole Approved DB12834
small molecule | CAS: 3366-95-8

Secnidazole is a second-generation 5-nitroimidazole antimicrobial agent. It is structurally related to other 5-nitroimidazoles, including [DB00916] and [DB00911], but displays improved oral absorption and a longer terminal elimination half-life than other dru…

Kategori:
Anti-Infective AgentsAntibacterials for Systemic UseAntiinfectives for Systemic Use +18
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe apparent volume…
KlirensThe total body clea…
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Secretin human Approved DB09532
biotech | CAS: 108153-74-8

Human secretin is a gastrointestinal peptide hormone that regulates secretions in the stomach, pancreas, and liver. The hormone is produced from the enterochromaffin cells in the duodenum in response to the duodenal content with the pH less than 4.5 [L1875]. …

Kategori:
Amino Acids, Peptides, and ProteinsDiagnostic AgentsGastrointestinal Agents +11
Target Protein:
Secretin receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of sy…
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Secukinumab Approved DB09029
biotech | CAS: 1229022-83-6

Secukinumab is a fully human monoclonal IgG1/? antibody against interleukin-17A (IL-17A), a proinflammatory cytokine implicated in various chronic immune-mediated inflammatory disorders, such as plaque psoriasis.[L39600] By blocking the actions of IL-17A, sec…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntibodies +14
Target Protein:
Interleukin-17A
Waktu ParuhThe half-life range…
Vol. DistribusiThe mean volume of …
KlirensThe mean systemic c…
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Segesterone acetate Approved DB14583
small molecule | CAS: 7759-35-5

Segesterone acetate is a steroidal progestin or synthetic progesterone and a 19-norprogesterone derivative with no CH3 group radical in position 6 [A37048]. In animal studies, segesterone acetate was shown to be one of the most potent progestins [A37090]. It …

Kategori:
Adrenal Cortex HormonesContraceptive Agents, FemaleContraceptive Agents, Hormonal +24
Target Protein:
Progesterone receptorAndrogen receptorGlucocorticoid receptor
Waktu ParuhThe mean (SD) half …
Vol. DistribusiThe volume of distr…
KlirensNo pharmacokinetic …
Genetik -
Selamectin DB11459
small molecule | CAS: 220119-17-5

Selamectin is a topical parasiticide and antihelminthic used on dogs and cats to treat and prevent infections of heartworms, fleas, ear mites, sarcoptic mange, and certain types of ticks in dogs as well as prevent heartworms, fleas, ear mites, hookworms, and …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntiparasitic Agents +7
Waktu Paruh-
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Selenic acid Approved DB11068
small molecule | CAS: 7783-08-6

Selenic acid is an organic compound with the chemical formula H2SeO4. It may be found in over-the-counter daily dietary supplements as a source of [DB11135], an essential trace mineral for human health.

Kategori:
Alimentary Tract and MetabolismAntioxidantsBiological Factors +10
Waktu ParuhFollowing single or…
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
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Selenious acid Approved DB11127
small molecule | CAS: 7783-00-8

Selenious acid is the acid form of sodium selenite, a form of selenium [L1910]. Selenium is an essential trace element and antioxidant. It is a cofactor metabolic enzyme regulation. It also plays an important role in maintaining the general health of tissu…

Kategori:
Alimentary Tract and MetabolismBlood and Blood Forming OrgansBlood Substitutes and Perfusion Solutions +14
Waktu Paruh30 days in beagle d…
Vol. DistribusiFollowing oral inta…
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Selenium Approved DB11135
small molecule | CAS: 7782-49-2

Selenium is a trace metal in the human body particularly important as a component of glutathione peroxidase, an important enzyme in the prevention of cellular damage by free radicals and reactive oxygen species [FDA Label]

Kategori:
Alimentary Tract and MetabolismAntioxidantsBiological Factors +14
Waktu ParuhHalf life was obser…
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Selenomethionine Approved DB11142
small molecule | CAS: 3211-76-5

Selenomethionine is a naturally occuring amino acid in some plant materials such as cereal grains, soybeans and enriched yeast but it cannot be synthesized from animals or humans. It can be produced from post-structural modifications. *In vivo*, selenomethion…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsOrganoselenium Compounds +1
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Seletracetam DB05885
small molecule | CAS: 357336-74-4

Seletracetam is a pyrrolidone derivative and with a structural similarity to newer generation antiepileptic drug levetiracetam. It binds to the same target as levetiracetam but with higher affinity and has shown potent seizure suppression in models of acquire…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +6
Target Protein:
Synaptic vesicle glycoprotein 2AVoltage-dependent N-type calcium channel subunit alpha-1BGlycine receptor (alpha-1/beta)
Waktu ParuhApproximately 8 hou…
Vol. DistribusiThe volume of distr…
KlirensThe total apparent …
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Selpercatinib Approved DB15685
small molecule | CAS: 2152628-33-4

Selpercatinib is a kinase inhibitor with enhanced specificity for RET tyrosine kinase receptors (RTKs) over other RTK classes.[A202055, A202052, L13604] Enhanced RET (Rearranged during transfection) oncogene expression is a hallmark of many cancers. Although …

Kategori:
Agents that produce hypertensionAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +19
Target Protein:
Proto-oncogene tyrosine-protein kinase receptor RetVascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 3 +3
Waktu ParuhSelpercatinib has a…
Vol. DistribusiSelpercatinib has a…
KlirensSelpercatinib has a…
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Semaglutide Approved DB13928
small molecule | CAS: 910463-68-2

Semaglutide is a glucagon-like peptide 1 (GLP-1) analog used to manage type 2 diabetes along with lifestyle changes, such as dietary restrictions and increased physical activity.[A31421,L8681] Other members of this drug class include [Exenatide] and [Liraglut…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +11
Target Protein:
Glucagon-like peptide 1 receptor
Waktu ParuhOne of the major pr…
Vol. DistribusiThe volume of distr…
KlirensThe clearance rate …
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Sennosides DB11365
small molecule | CAS: 517-43-1

Sennosides (also known as senna glycoside or senna) is a medication used to treat constipation[FDA Label][L771] and empty the large intestine before surgery. The medication is taken by mouth or via the rectum[FDA Label]. It typically begins working in minutes…

Kategori:
Alimentary Tract and MetabolismAnthracenesAnthraquinones +13
Target Protein:
Aquaporin-3Reverse transcriptase/RNaseH
Waktu ParuhThe half life of ra…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ra…
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Sepantronium DB17062
small molecule | CAS: 753440-91-4

Sepantronium is a compound that suppresses survivin expression in a dose and time-dependent manner, and causes broad-range apoptosis.[A253167]

Kategori:
NaphthalenesQuinones
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Seractide acetate Approved DB09334
biotech | CAS: 39295-97-1

Seractide acetate is the acetate salt of full length human corticotropin.

Target Protein:
Adrenocorticotropic hormone receptor
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Serelaxin DB05794
biotech | CAS: 99489-94-8

Recombinant human relaxin is a hormone produced during pregnancy that facilitates the birth process by causing a softening and lengthening of the cervix and the pubic symphysis (the place where the pubic bones come together).It is a heterodimer protein secret…

Kategori:
Cardiac TherapyVasodilators Used in Cardiac Diseases
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Sermorelin Approved DB00010
biotech | CAS: 86168-78-7

Sermorelin acetate is the acetate salt of an amidated synthetic 29-amino acid peptide (GRF 1-29 NH 2 ) that corresponds to the amino-terminal segment of the naturally occurring human growth hormone-releasing hormone (GHRH or GRF) consisting of 44 amino acid r…

Kategori:
Amino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and AnaloguesDiagnostic Agents +13
Target Protein:
Growth hormone-releasing hormone receptor
Waktu Paruh11-12 min
Vol. Distribusi-
Klirens-
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Serplulimab DB17451
biotech | CAS: 2231029-82-4

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsMonoclonal antibodies and antibody drug conjugates +1
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Seviprotimut-L DB16328
biotech

Seviprotimut-L is under investigation in clinical trial NCT01546571 (Study of a Melanoma Vaccine in Stage Iib, Iic, and III Melanoma Patients).

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Sevirumab DB17771
biotech | CAS: 138660-96-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
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SGN-B6A DB18377
biotech | CAS: 2764774-91-4

Sigvotatug vedotin (SGN-B6A) is a humanized immunoglobulin G1 anti-integrin beta-6 monoclonal antibody conjugated to monomethyl auristatin E.

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Siagoside DB12351
small molecule | CAS: 100345-64-0

Siagoside (Sygen, AGF 2) has been investigated for the treatment of Parkinson Disease. It is a naturally occurring substance in the nerve cell’s membrane that is thought to play a role in cell growth, development, and repair. Siagoside completed phase 2 trial…

Kategori:
Acidic GlycosphingolipidsCarbohydratesGangliosides +7
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Sibeprenlimab DB18919
biotech | CAS: 2382896-07-1

Sibeprenlimab is under investigation in clinical trial NCT05248659 (Phase 2/3 Open-label Trial of Sibeprenlimab in the Treatment of Immunoglobulin a Nephropathy).

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Sibrotuzumab DB06474
biotech

Sibrotuzumab is a humanized monoclonal antibody directed against fibroblast activation protein (FAP). It is used to treat cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Prolyl endopeptidase FAP
Waktu Paruh-
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Sifalimumab DB12773
biotech | CAS: 1006877-41-3

Sifalimumab is a fully human monoclonal antibody targeting interferon-alpha. The levels of interferon-alpha are elevated in many patients with active systemic lupus erythematosus (SLE, or lupus) and other autoimmune disorders, and may be associated with disea…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Interferon alpha-2
Waktu Paruh-
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SIG-001 DB17826
biotech

SIG-001 is a cultured human retinal pigment epithelial cell line (ARPE-19) genetically modified with a non-viral vector to express B domain deleted human factor VIII protein, encapsulated within two-layer modified alginate spheres.

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SIG-007 DB17710
biotech

SIG-007 is a gene therapy that consists of cells that are genetically modified with a non-viral vector to express human alpha-galactosidase A. Developed by Sigilon Therapeutics, t is being investigated for the treatment of Fabry Disease.[L46153]

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SIG-205 DB18548
biotech

SIG-205 is a Cultured human retinal pigment epithelial cells (ARPE-19) genetically modified with a non-viral vector to express human native alpha-L-iduronidase enzyme (hIDUA), encapsulated within two-layer modified alginate spheres

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SIG-207 DB18547
biotech

SIG-207 is a Cultured human retinal pigment epithelial cells (ARPE-19) genetically modified with a non-viral vector to express Human alpha-galactosidase A (alpha-Gal A), encapsulated within two-layer modified alginate spheres

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