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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 37 / 236
biotech | CAS: 1621271-62-2

Aglatimagene besadenovec is under investigation in clinical trial NCT00638612 (AdV-tk Therapy With Surgery and Chemoradiation for Pancreas Cancer (PaTK01)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Agmatine DB08838
small molecule | CAS: 306-60-5

Agmantine is a natural metabolite of the amino acid arginine. It is formed when arginine is decarboxylated by the enzyme arginine decarboxylase and is found naturally in ragweed pollen, ergot fungi, octopus muscle, herring sperm, sponges, and the mammalian br…

Kategori:
Agents causing hyperkalemiaAmidinesAntiarrhythmic agents +12
Target Protein:
Alpha-2C adrenergic receptorNischarinAcetylcholine receptor subunit alpha +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AGN-201904 DB13135
small molecule | CAS: 651729-53-2

Agn 201904 has been used in trials studying the prevention of Peptic Ulcer.

Kategori:
2-PyridinylmethylsulfinylbenzimidazolesBenzimidazolesHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Agomelatine Approved DB06594
small molecule | CAS: 138112-76-2

Agomelatine is structurally closely related to melatonin. Agomelatine is a potent agonist at melatonin receptors and an antagonist at serotonin-2C (5-HT2C) receptors, tested in an animal model of depression. Agomelatine was developed in Europe by Servier Labo…

Kategori:
AcetatesAcids, AcyclicAmides +15
Target Protein:
5-hydroxytryptamine receptor 2CMelatonin receptor type 1AMelatonin receptor type 1B
Waktu Paruh<2 hours
Vol. Distribusi-
Klirens-
Genetik -
Agrostis gigantea top Approved DB14757
biotech

Agrostis gigantea top is the flowering part of the Agrostis gigantea plant. Agrostis gigantea top is mainly used in allergenic testing.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AGS-004 DB05742
small molecule

AGS-004 is a personalized RNA-loaded dendritic cellbased immunotherapy that is designed to stimulate the patient’s immune system to target and destroy the patient’s own unique viral burden. Non-personalized HIV immunotherapies are unable to raise cytotoxic T…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AGS-005 DB05741
small molecule

AGS-005 is a personalized dendritic cell-based immunotherapy, with optimized immune response characteristics, that is designed to stimulate the patient's immune system to target and destroy the patient's cancer cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AGS-16C3F DB17551
biotech

AGS 16C3F is an intravenously administered, anti-ectonucleotide pyrophosphatase/phosphodiesterase 3 (ENPP3) antibody-drug conjugate. AGS-16C3F is under investigation in clinical trial NCT02639182 (A Study of AGS-16C3F vs. Axitinib in Metastatic Renal Cell Car…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AGS-499 DB18058
small molecule | CAS: 1092372-02-5

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesTelomerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AGT-182 DB17630
biotech

AGT-182 is an investigational enzyme replacement therapy engineered by the fusion of the iduronate-2-sulfatase (IDS) enzyme and a human insulin receptor monoclonal antibody.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AGT-184 DB17691
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AGTC-401 DB18432
biotech

AGTC-401 is a recombinant adeno-associated virus vector expressing the cyclic nucleotide gated channel beta subunit (rAAV-CNGB3).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2417550-70-8

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AIC100 DB17350
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 3031-94-5

5-Aminoimidazole-4-carboxamide ribonucleotide (AICAR) is an intermediate in the generation of inosine monophosphate and analog of adenosine monophosphate (AMP) that is capable of stimulating AMP-dependent protein kinase (AMPK) activity. AICAR has been used cl…

Kategori:
Blood Glucose Lowering AgentsImidazolesNucleic Acids, Nucleotides, and Nucleosides +1
Target Protein:
Bifunctional purine biosynthesis protein ATIC
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AIM-102 DB16176
small molecule | CAS: 551936-17-5

AIM-102 is under investigation in clinical trial NCT01501942 (Efficacy, Safety, Tolerability, Pharmacodynamics and Pharmacokinetics of Oral Administration of AIM-102 in Patients With Mild to Moderate Allergic Asthma).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
AIT-034 DB06106
small molecule | CAS: 138117-48-3

AIT-034 is a distinct chemical analog of hypoxanthine and pyrollidone that has been demonstrated in animal studies to enhance memory and to reverse memory deficits in severely impaired animals that do not respond to Neotrofin. AIT-034 does not induce the prod…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ajmaline Approved DB01426
small molecule | CAS: 4360-12-7

An alkaloid found in the root of Rauwolfia serpentina, among other plant sources. It is a class Ia antiarrhythmic agent that apparently acts by changing the shape and threshold of cardiac action potentials. Ajmaline produces potent sodium channel blocking eff…

Kategori:
Ajmaline and derivativesAlkaloidsAntiarrhythmic agents +16
Target Protein:
Sodium channel protein type 5 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ajoene DB17735
small molecule | CAS: 92285-01-3

Deskripsi belum tersedia.

Kategori:
AnionsAnti-Infective AgentsAntifungal Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AK106-001616 DB16058
small molecule | CAS: 590416-75-4

AK106-001616 is under investigation in clinical trial NCT01285752 (A Study of AK106-001616 in Patients With Rheumatoid Arthritis (RA)).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AK119 DB16423
biotech

AK119 is a humanized anti-CD73 monoclonal antibody being investigated in the clinical trial NCT04516564 (A Study of AK119 (Anti-CD73 Antibody), a Treatment for COVID-19, in Healthy Subjects).[L28315]

Waktu Paruh-
Vol. Distribusi-
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AKI-001 DB07266
small molecule | CAS: 925218-37-7

AKI-001 is an aurora kinase inhibitor.

Kategori:
Heterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Target Protein:
Aurora kinase A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aklavine DB19070
small molecule | CAS: 66676-88-8

Aklavine is under investigation in clinical trial NCT03026842 (Decitabine Versus Conventional Chemotherapy for Maintenance Therapy of Acute Myeloid Leukemia With T(8;21)).

Kategori:
Adjuvants, ImmunologicAminoglycoside AntibacterialsAnthracyclines +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AKN-028 DB12746
small molecule | CAS: 1175017-90-9

AKN-028 has been used in trials studying the treatment of Acute Myeloid Leukemia.

Target Protein:
Receptor-type tyrosine-protein kinase FLT3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AKV-9 DB18061
small molecule | CAS: 1307262-15-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AL-01211 DB17654
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
AL-034 DB17471
small molecule

AL-034 (TQ-A3334) is an oral toll-like receptor 7 agonist developed for the treatment of chronic hepatitis B (CHB) viral infection.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AL-4623 DB03877
small molecule | CAS: 138890-59-2

Deskripsi belum tersedia.

Target Protein:
Carbonic anhydrase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AL5927 DB03526
small molecule

Deskripsi belum tersedia.

Target Protein:
Carbonic anhydrase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AL6528 DB04371
small molecule

Deskripsi belum tersedia.

Target Protein:
Carbonic anhydrase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AL7089A DB02220
small molecule | CAS: 220402-83-5

Deskripsi belum tersedia.

Target Protein:
Carbonic anhydrase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AL7099A DB03221
small molecule

Deskripsi belum tersedia.

Target Protein:
Carbonic anhydrase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AL7182 DB02602
small molecule

Deskripsi belum tersedia.

Target Protein:
Carbonic anhydrase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Ala-geninthiocin is a novel thiopeptide antibacterial compound derived from marine _Streptomyces_ species.[A192840] It has exhibited potent _in vitro_ activity against gram-positive bacteria including _Staphylococcus aureus_, _Bacillus subtilis_, _Mycobacteri…

Kategori:
Anti-Bacterial Agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alagebrium DB12497
small molecule | CAS: 393121-34-1

Alagebrium has been investigated for the treatment and prevention of Aging, Heart Failure, Physical Activity, Diabetic Nephropathy, and Cardiovascular Disease, among others.

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alanine DB00160
small molecule | CAS: 56-41-7

Alanine is a non-essential amino acid that occurs in high levels in its free state in plasma. It is produced from pyruvate by transamination. It is involved in sugar and acid metabolism, increases immunity, and provides energy for muscle tissue, brain, and th…

Kategori:
AlanineAmino AcidsAmino Acids, Peptides, and Proteins +3
Target Protein:
4-aminobutyrate aminotransferase, mitochondrialAlanine--glyoxylate aminotransferaseAlanine aminotransferase 1 +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 39537-23-0

Alanyl Glutamine is under investigation in clinical trial NCT00338221 (Clinical Trial of Alanyl-Glutamine or Glycine in Children With Persistent Diarrhea or Malnutrition).

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsBlood and Blood Forming Organs +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alaproclate DB13233
small molecule | CAS: 60719-82-6

Alaproclate was developed as one of the first selective serotonin reuptake inhibitor (SSRI) antidepressants by Astra AB (now AstraZeneca) in the 1970s. Development was discontinued due to concerns over hepatotoxicity observed in animal studies. Alaproclate ha…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntidepressive Agents +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alatrofloxacin Approved DB09335
small molecule | CAS: 146961-76-4

Alatrofloxacin is a fluoroquinolone antibiotic developed by Pfizer, delivered as a mesylate salt. It was withdrawn from the U.S. market in 2001.

Kategori:
4-QuinolonesAnti-Infective AgentsEnzyme Inhibitors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Albaconazole DB12073
small molecule | CAS: 187949-02-6

Albaconazole has been used in trials studying the basic science of Onychomycosis.

Kategori:
Anti-Infective AgentsAntifungal AgentsAzole Antifungals +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 54029-12-8

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAnthelminticsAnti-Infective Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Albiglutide Approved DB09043
biotech | CAS: 782500-75-8

Albiglutide is a glucagon-like peptide-1 agonist (GLP-1) biologic drug indicated in the treatment of type 2 diabetes. It is marketed under the brands Eperzan and Tanzeum by GSK (GlaxoSmithKline). It is a dipeptidyl peptidase-4-resistant glucagon-like peptide-…

Kategori:
Alimentary Tract and MetabolismBlood Glucose Lowering AgentsDrugs Used in Diabetes +10
Target Protein:
Glucagon-like peptide 1 receptor
Waktu Paruh4-7 days.
Vol. Distribusi11 L.
Klirens67 mL/h.
Genetik -
biotech | CAS: 472960-22-8

Albumin-interferon alpha (Albuferon) is a novel, long-acting form of interferon alpha. Recombinant interferon alpha is approved for the treatment of hepatitis C, hepatitis B, and a broad range of cancers. Human Genome Sciences modified interferon alpha to imp…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Albumin human Approved DB00062
biotech | CAS: 9048-46-8

Human serum albumin is the primary protein present in human blood plasma. The main function of albumin is to maintain the oncotic pressure of blood [A33706]. It binds to water, cations (such as Ca2+, Na+ and K+), fatty acids, hormones, bilirubin, thyroxine (T…

Kategori:
AlbuminsAmino Acids, Peptides, and ProteinsBlood and Blood Forming Organs +13
Target Protein:
Nitric oxide
Waktu Paruh-
Vol. DistribusiAlbumin is distribu…
Klirens-
Genetik -
biotech

I-125 iodinated albumin is a radiolabeled albumin-based diagnostic agent used in the determination of total blood and plasma volume.[L12780]

Kategori:
Radioactive Diagnostic AgentRadiopharmaceutical Activity
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Iodinated I-131 serum albumin is a radiopharmaceutical agent used for several diagnostic purposes, including the determination of body fluid volumes and the imaging of certain tissues.[L12783]

Kategori:
Radiopharmaceutical Activity
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Albusomatropin DB12950
biotech | CAS: 1613273-96-3

Albusomatropin has been used in trials studying the treatment of Growth Hormone-Deficiency and Growth Hormone Deficiency.

Kategori:
AlbuminsAmino Acids, Peptides, and ProteinsBlood Proteins +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Albuterol Approved DB01001
small molecule | CAS: 18559-94-9

Salbutamol (Albuterol [USAN]) is a short-acting, selective beta2-adrenergic receptor agonist used in the treatment of asthma and COPD. It is 29 times more selective for beta2 receptors than beta1 receptors giving it higher specificity for pulmonary beta recep…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +27
Target Protein:
Beta-2 adrenergic receptorBeta-1 adrenergic receptorBeta-3 adrenergic receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe renal clearance…
Genetik -
Albutrepenonacog alfa Approved DB13884
biotech | CAS: 1357448-54-4

Albutrepenonacog alfa (rIX-RFP) is a recombinant fusion protein that links a recombinant coagulation factor IX (rFIX) with a recombinant human albumin (rAlbumin).[A32547] It was developed by CSL Behring Canada, Inc and approved by Health Canada on April 26, 2…

Kategori:
AlbuminsAmino Acids, Peptides, and ProteinsBiological Factors +9
Target Protein:
Coagulation factor X
Waktu ParuhThe fusion of the r…
Vol. DistribusiThe reported volume…
KlirensIn clinical trials,…
Genetik -
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