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3253

Total database: 17430
Struktur (SMILES)
2451 (75.3%)
Target
1833 (56.3%)
Genomik
35 (1.1%)
Referensi
3253 (100.0%)

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Halaman 37 / 66
Malacidin A DB14051
biotech

Malacidin A, along with [DB14052], is a member of a class of chemicals made by bacteria found in soil that can kill Gram-positive bacteria [A33312]. Malacidins are 10-member macrocycle lipopeptides discovered via gene sequencing and bioinformatic analysis. Wh…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +3
Target Protein:
NAM/NAG peptide subunits of peptidoglycan
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Malacidin B DB14052
small molecule

Malacidin B, along with [DB14051], is a member of a class of chemicals made by bacteria found in soil that can kill Gram-positive bacteria [A33312]. Malacidins are 10-member macrocycle lipopeptides discovered via gene sequencing and bioinformatic analysis. Wh…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +3
Target Protein:
NAM/NAG peptide subunits of peptidoglycan
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Malathion Approved DB00772
small molecule | CAS: 121-75-5

Malathion is a parasympathomimetic organophosphate compound that is used as an insecticide for the treatment of head lice. Malathion is an irreversible cholinesterase inhibitor and has low human toxicity.

Kategori:
AgrochemicalsAntiparasitic Products, Insecticides and RepellentsCholinergic Agents +19
Target Protein:
CholinesteraseAcetylcholinesterase
Waktu Paruh8-24 hours
Vol. Distribusi-
Klirens-
Genetik -
Malic acid DB12751
small molecule | CAS: 6915-15-7

Malic acid has been used in trials studying the treatment of Xerostomia, Depression, and Hypertension.

Kategori:
Acids, AcyclicDicarboxylic AcidsHydroxy Acids
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Maltodextrin DB12583
small molecule | CAS: 9050-36-6

Deskripsi belum tersedia.

Kategori:
Carbohydrates
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Maltotetraose DB02237
small molecule | CAS: 34612-38-9

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsCarbohydrates +5
Target Protein:
Glucan 1,4-alpha-maltotetraohydrolaseNeopullulanase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mangafodipir Approved DB06796
small molecule | CAS: 155319-91-8

Mangafodipir is a contrast agent used as a diagnostic tool administered intravenously to enhance contrast in magnetic resonance imaging (MRI) of the liver and pancreas. This drug is made up of paramagnetic manganese (II) ions combined with the chelating agent…

Kategori:
AcetatesAcids, AcyclicAmines +15
Waktu ParuhThe mean initial pl…
Vol. DistribusiThe volume of distr…
KlirensThe approximate tot…
Genetik -
Manganese gluconate Approved DB11141
small molecule | CAS: 6485-39-8

Manganese gluconate is a manganese salt of gluconic acid with the chemical formula C12H22MnO14 x 2H2O. It is typically obtained by reacting manganese carbonate with gluconic acid in aqueous medium and then crystallizing the product to form a slightly pink pow…

Kategori:
Acids, AcyclicCarbohydratesHydroxy Acids +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mannitol busulfan Approved DB12097
small molecule | CAS: 1187-00-4

Mm has been used in trials studying the treatment of Cocaine Dependence and Diabetes Mellitus, Type 2.

Kategori:
Agents causing hyperkalemia
Waktu Paruh-
Vol. Distribusi-
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Mannose DB12907
small molecule | CAS: 3458-28-4

Mannose is under investigation for the basic science of IUGR and Pregnancy.

Kategori:
CarbohydratesHexosesMonosaccharides
Waktu Paruh-
Vol. Distribusi-
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Mant-Adp DB03126
small molecule

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAdenine NucleotidesAminobenzoates +8
Target Protein:
Myosin-14
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Mapatumumab DB18945
biotech | CAS: 658052-09-6

Mapatumumab is under investigation in clinical trial NCT00094848 (Study of TRM-1 (TRAIL-R1 Monoclonal Antibody) in Subjects With Relapsed or Refractory Non-hodgkin's Lymphoma (NHL)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
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Maplirpacept DB18441
biotech

Maplirpacept is a recombinant fusion protein consisting of the CD47-binding domain of human signal regulatory protein alpha (SIRPa) linked to the IgG4 Fc region of human IgG.

Waktu Paruh-
Vol. Distribusi-
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Mapracorat DB12041
small molecule | CAS: 887375-26-0

Mapracorat has been investigated for the treatment of Eczema and Atopic Dermatitis.

Kategori:
AlcoholsFatty AlcoholsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Glucocorticoid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2760218-55-9

Maridebart Cafraglutide is under investigation in clinical trial NCT05669599 (Dose-ranging Study to Evaluate the Efficacy, Safety, and Tolerability of AMG 133 in Adult Subjects With Overweight or Obesity, With or Without Type 2 Diabetes Mellitus).

Waktu Paruh-
Vol. Distribusi-
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Martinostat DB14979
small molecule | CAS: 1629052-58-9

Martinostat is under investigation in clinical trial NCT03721211 (Imaging With [11C]Martinostat in Breast Cancer).

Kategori:
AminesBridged-Ring CompoundsCarbon Radioisotopes +3
Target Protein:
Histone deacetylase 7Histone deacetylase 9Histone deacetylase 8 +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Masilukast DB16227
small molecule | CAS: 136564-68-6

Masilukast is under investigation in clinical trial NCT01740986 (Safety and Efficacy of SA09012 in Asthma).

Target Protein:
Cysteinyl leukotriene receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Matairesinol DB04200
small molecule | CAS: 580-72-3

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesBenzyl CompoundsPlants
Target Protein:
Dehydrogenase/reductase SDR family member 4-like 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mavatrep DB12875
small molecule | CAS: 956274-94-5

Mavatrep has been used in trials studying the treatment of Osteoarthritis, Knee.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Transient receptor potential cation channel subfamily V member 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mavelertinib DB16228
small molecule | CAS: 1776112-90-3

Mavelertinib is under investigation in clinical trial NCT02349633 (Study for Patients With NSCLC EGFR Mutations (Del 19 or L858R +/- T790M)).

Waktu Paruh-
Vol. Distribusi-
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Mavoglurant DB13004
small molecule | CAS: 543906-09-8

Mavoglurant has been used in trials studying the treatment of Patient Diagnosed With OCD and and Resistant to SSRI Treatment (Failed SSRI Over 12 Weeks at Appropriate Doses).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Metabotropic glutamate receptor 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mavrilimumab DB12534
biotech | CAS: 1085337-57-0

Mavrilimumab has been investigated for the treatment of Rheumatoid Arthritis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MAX-40279 DB15191
small molecule | CAS: 2070931-57-4

MAX-40279 is under investigation in clinical trial NCT03412292 (MAX-40279 in Subjects With Acute Myelogenous Leukemia (AML)).

Waktu Paruh-
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Mazorelvimab DB17767
biotech | CAS: 2419087-89-9

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
biotech

MB-102 are autologous T cells genetically modified to express CD123-specific, hinge-optimized CD28-costimulatory chimeric receptor and a truncated human epidermal growth factor receptor.

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MBP-091 DB17741
biotech

MBP-091 is a monoclonal antibody being investigated for the treatment of Marburg virus disease (MVD) caused by infection with Marburg virus (MARV).[L46212]

Waktu Paruh-
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MBT-0312 DB05880
small molecule

MediGene's newly acquired drug candidates MBT-0312 aim at a novel method of cancer therapy by "starving out" tumors.

Waktu Paruh-
Vol. Distribusi-
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MBX-2982 DB12345
small molecule | CAS: 1037792-44-1

MBX-2982 has been used in trials studying the treatment of Diabetes.

Kategori:
Sulfur Compounds
Target Protein:
Glucose-dependent insulinotropic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mebeverine Approved DB12554
small molecule | CAS: 3625-06-7

Mebeverine has been investigated for the treatment of Irritable Bowel Syndrome and Post-cholecystectomy Gastrointestinal Spasms.

Kategori:
Agents Causing Muscle ToxicityAgents producing tachycardiaAlimentary Tract and Metabolism +10
Target Protein:
Muscarinic acetylcholine receptor M5
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Mecasermin Approved DB01277
biotech | CAS: 68562-41-4

Mecasermin contains recombinant-DNA-engineered human insulin-like growth factor-1 (rhIGF-1)[FDA Label]. IGF-1 consists of 70 amino acids in a single chain with three intramolecular disulfide bridges and a molecular weight of 7649 daltons. The amino acid seque…

Kategori:
Amino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and AnaloguesBiological Factors +15
Target Protein:
Insulin-like growth factor 1 receptorInsulin-like growth factor-binding protein 3Insulin receptor +1
Waktu ParuhMean half life of 5…
Vol. Distribusi* 0.257 ± 0.073 L/k…
KlirensClearance of Mecase…
Genetik -
Mecasermin rinfabate Approved DB14751
biotech | CAS: 478166-15-3

Mecasermin rinfabate is approved for severe primary insulin-like growth factor (IGF) deficiency or in patients with GH gene deletion who have developed antibodies to growth hormone (GH)[A176020]. Mecasermin rinfabate is similar to [DB01277] in that both drugs…

Kategori:
Anterior Pituitary Lobe Hormones and AnaloguesPituitary and Hypothalamic Hormones and AnaloguesSomatropin and Somatropin Agonists +1
Target Protein:
Insulin-like growth factor 1 receptorInsulin receptorCation-independent mannose-6-phosphate receptor
Waktu ParuhHalf life ranges fr…
Vol. DistribusiApproximately 1000m…
KlirensClearance ranges fr…
Genetik -
biotech | CAS: 2460400-64-8

Mecbotamab vedotin is an anti-Axl humanized monoclonal antibody conjugated to monomethyl auristatin E using a cleavable linker (CAB-Axl-ADC).[A255212]

Waktu Paruh-
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Meclocycline DB13092
small molecule | CAS: 2013-58-3

Meclocycline is under investigation in clinical trial NCT00385515 (Efficacy of SNX-1012 in the Treatment of Oral Mucositis) [L797].

Kategori:
Anti-Acne PreparationsAnti-Acne Preparations for Topical UseAnti-Bacterial Agents +5
Target Protein:
30S ribosomal protein S7
Waktu ParuhHalf life estimated…
Vol. DistribusiEstimated Vd of 121…
Klirens-
Genetik -
Mecobalamin Approved DB03614
small molecule | CAS: 13422-55-4

Deskripsi belum tersedia.

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansCorrinoids +4
Target Protein:
Methionine synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Medazepam DB13437
small molecule | CAS: 2898-12-6

Deskripsi belum tersedia.

Kategori:
Anti-Anxiety AgentsAnticonvulsantsBenzazepines +17
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MEDI3506 DB16473
biotech | CAS: 2376858-66-9

Tozorakimab (MEDI3506), developed by AstraZeneca, was investigated in multiple clinical trials to evaluate its safety, tolerability, efficacy, and pharmacokinetics across various conditions. These trials include NCT03096795 (completed; healthy participants, C…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
Interleukin-33
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MEDI6012 DB14833
biotech

Recombinant human lecithin:cholesterol acyltransferase is under investigation in clinical trial NCT03578809 (A Study to Evaluate the Safety and Efficacy of MEDI6012 in Acute ST Elevation Myocardial Infarction).

Waktu Paruh-
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Medium-chain triglycerides Approved DB13959
small molecule | CAS: 438544-49-1

Medium-chain triglycerides (MCTs) are triglycerides made up of a glycerol backbone and three fatty acids with an aliphatic tail of six to 12 carbon atoms. MCTs are found in natural foods, such as coconut oil, palm kernel oil, and raw coconut meat. In the body…

Kategori:
LipidsOilsParenteral Nutrition Solutions +1
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe apparent volume…
KlirensThe clearance of me…
Genetik -
Medrogestone Approved DB09124
small molecule | CAS: 977-79-7

Medrogestone (INN), also known as 6,17?-dimethyl-6-dehydroprogesterone, is a progestational agent derived from 17-methylprogesterone. It was conceived as an alternative for an orally effective contraceptive option.[A31526] It was developed by Ayerst, approved…

Kategori:
Adrenal Cortex HormonesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +10
Target Protein:
Progesterone receptor
Waktu ParuhThe half-life of me…
Vol. Distribusi-
Klirens-
Genetik -
Melarsomine DB11528
small molecule | CAS: 128470-15-5

Melarsomine is a trypanocidal agent marketed by Merial under the trade name Immiticide. It is the only FDA-approved treatment for adult heartworm infection in dogs, however, is is not approved for use in dogs with late-stage infection.

Waktu Paruh-
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Melarsoprol DB12864
small molecule | CAS: 494-79-1

Melarsoprol is under investigation in clinical trial NCT00330148 (Randomized Clinical Trial of Three Drug Combinations for Late-Stage Gambiense Human African Trypanosomiasis).

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAnti-Infective AgentsAntiparasitic Agents +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meloxicam Approved DB00814
small molecule | CAS: 71125-38-7

Meloxicam is a nonsteroidal anti-inflammatory drug (NSAID) used to relieve various types of pain, including pain caused by musculoskeletal conditions, osteoarthritis, and rheumatoid arthritis.[A190189] With a longer half-life than most other NSAIDS, it is a f…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +28
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhThe half-life of me…
Vol. DistribusiThe volume of distr…
KlirensAfter an oral dose,…
Genetik -
Melphalan flufenamide Approved DB16627
small molecule | CAS: 380449-51-4

Melphalan flufenamide, also known as melflufen or J1, is a prodrug of [melphalan].[A230123,L32173] Melphalan flufenamide is more readily uptaken by cells than melphalan, and is cleaved to the active metabolite by aminopeptidases.[A230123] _In vitro_ models sh…

Kategori:
Alkylating ActivityAlkylating DrugsAmino Acids +12
Target Protein:
DNA
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean volume of …
KlirensThe mean clearance …
Genetik -
Menaquinone 7 DB13075
small molecule | CAS: 2124-57-4

Menaquinone 7 is under investigation in clinical trial NCT00402974 (The Effect of Vitamin K Supplementation on Osteocalcin Carboxylation in Healthy Children).

Kategori:
CoagulantsDiterpenesHematologic Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menatetrenone DB12148
small molecule | CAS: 863-61-6

Menatetrenone has been used in trials studying the treatment of Diabetes, Osteoporosis, Prediabetic State, and Hepatocellular Carcinoma.

Kategori:
CoagulantsDiterpenesDrugs Affecting Bone Structure and Mineralization +12
Target Protein:
Cruzipain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menotropins Approved DB00032
biotech | CAS: 9002-68-0

Menotropins contains follicle stimulating hormone (FSH) and luteinizing hormone (LH) purified from the urine of postmenopausal women. It is used as a fertility medication that is injected either subcutaneously or intramuscularly. It is composed of LH with 2 …

Kategori:
Amino Acids, Peptides, and ProteinsBiological ProductsComplex Mixtures +14
Target Protein:
Follicle-stimulating hormone receptorLutropin-choriogonadotropic hormone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menthol Approved DB14123
small molecule | CAS: 1490-04-6

Deskripsi belum tersedia.

Kategori:
AlcoholsAntipruriticsCyclohexane Monoterpenes +9
Target Protein:
Transient receptor potential cation channel subfamily M member 8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menthyl salicylate Approved DB11201
small molecule | CAS: 89-46-3

Menthyl salicylate is an ester of menthol and salicylic acid [L2808]. This product is used to treat minor aches and pains of the muscles/joints (e.g., arthritis, backache, sprains) [L2810].

Kategori:
Anti-Inflammatory AgentsAnti-Inflammatory Agents, Non-Steroidal
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mepartricin DB13633
small molecule | CAS: 11121-32-7

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAlkenesAnti-Bacterial Agents +19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mephentermine Approved DB01365
small molecule | CAS: 100-92-5

A sympathomimetic agent with mainly indirect effects on adrenergic receptors. It is used to maintain blood pressure in hypotensive states, for example, following spinal anesthesia. Although the central stimulant effects of mephentermine are much less than tho…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +17
Target Protein:
Alpha adrenergic receptorD(2) dopamine receptorBeta adrenergic receptor
Waktu Paruh17 to 18 hours.
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 1801–1850 dari 3253
Sebelumnya Halaman 37 / 66 Berikutnya