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6694

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4518 (67.5%)
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3751 (56.0%)
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81 (1.2%)
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6694 (100.0%)

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Halaman 36 / 134
Ceftobiprole medocaril Approved DB14733
small molecule | CAS: 376653-43-9

Ceftobiprole medocaril is a prodrug of [ceftobiprole], a fifth-generation semisynthetic cephalosporin antibacterial. Ceftobiprole is a broad-spectrum agent with demonstrated activity against both Gram-positive and Gram-negative bacteria, including antibiotic-…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +11
Target Protein:
MecAPenicillin-binding protein 2BPenicillin-binding protein 2X
Waktu ParuhThe half-life of ac…
Vol. DistribusiThe steady-state vo…
KlirensThe mean clearance …
Genetik -
Ceftolozane Approved DB09050
small molecule | CAS: 689293-68-3

Ceftolozane is a semi-synthetic broad-spectrum fifth generation cephalosporin.[L6685] It was approved by the FDA in 2014 for use in combination with [Tazobactam] for the treatment of serious infections, such as intra-abdominal infections and complicated urina…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +8
Target Protein:
Penicillin-binding protein 1BCell division proteinPenicillin-binding protein 1C +2
Waktu Paruh2.77 hours on day 1…
Vol. Distribusi13.5 L.[L41618] Tis…
KlirensThe renal clearance…
Genetik -
Ceftriaxone Approved DB01212
small molecule | CAS: 73384-59-5

Ceftriaxone is a broad-spectrum third-generation cephalosporin antibiotic.[A215582] It has a very long half-life compared to other cephalosporins and is high penetrable into the meninges[A215582], eyes[A215647], and inner ear[A215627]. Ceftriaxone has broader…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +15
Target Protein:
Penicillin-binding protein 2BSolute carrier family 22 member 11Solute carrier family 22 member 6 +2
Waktu ParuhThe elimination hal…
Vol. DistribusiThe apparent volume…
KlirensThe plasma clearanc…
Genetik -
Cefuroxime Approved DB01112
small molecule | CAS: 55268-75-2

Broad-spectrum cephalosporin antibiotic resistant to beta-lactamase. It has been proposed for infections with gram-negative and gram-positive organisms, gonorrhea, and haemophilus.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +12
Target Protein:
Penicillin-binding protein 1A
Waktu ParuhApproximately 80 mi…
Vol. Distribusi-
Klirens-
Genetik -
Celastrol DB18736
small molecule | CAS: 34157-83-0

Celastrol is a pentacyclic triterpenoid isolated from the root extracts of _Tripterygium wilfordii_.[L50567]

Kategori:
TerpenesTripterygiumTriterpenes
Target Protein:
Interleukin-1 betaTumor necrosis factor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Celecoxib Approved DB00482
small molecule | CAS: 169590-42-5

Celecoxib, a selective cyclooxygenase-2 (COX-2) inhibitor, is a nonsteroidal anti-inflammatory drug (NSAID) which is known for its decreased risk of causing gastrointestinal bleeding compared to other NSAIDS.[A181544] It is used to manage symptoms of various …

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +41
Target Protein:
Prostaglandin G/H synthase 2Signal transducer and activator of transcription 3Sialidase-1 +4
Gen Terkait:
CYP2C9
Waktu ParuhThe effective half-…
Vol. DistribusiThe apparent volume…
KlirensApparent clearance …
Genetik 1 Varian
Celiprolol Approved DB04846
small molecule | CAS: 56980-93-9

Celiprolol is indicated for the management of mild to moderate hypertension and effort-induced angina pectoris. It is simultaneously a selective ?1 receptor antagonist, a ?2 receptor partial agonist and a weak ?2 receptor antagonist. In 2010 a clinical trial …

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic Antagonists +30
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorBeta-3 adrenergic receptor +3
Waktu Paruh5 hours
Vol. DistribusiThe distribution vo…
KlirensCleared by both ren…
Genetik -
Celtis occidentalis pollen Approved DB10472
biotech

Celtis occidentalis pollen is the pollen of the Celtis occidentalis plant. Celtis occidentalis pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cemiplimab Approved DB14707
biotech | CAS: 1801342-60-8

Cemiplimab is a fully human monoclonal antibody that works against programmed death receptor-1 (PD-1), which is a negative regulator of T cell function. By blocking PD-1, cemiplimab works to enhance T cell-mediated antitumour responses.[L39804] Cemiplimab …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
Programmed cell death protein 1
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensCemiplimab clearanc…
Genetik -
Cenegermin Approved DB13926
biotech | CAS: 1772578-74-1

Cenegermin is a human beta-nerve growth factor (beta-ngf)-(1-118)- peptide (non-covalent dimer) produced in escherichia coli. It received European Union Approval in July 2017 for the treatment of moderate to severe neurotrophic keratitis. Cenegermin received …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +7
Target Protein:
High affinity nerve growth factor receptorTumor necrosis factor receptor superfamily member 16
Waktu ParuhHalf-life data spec…
Vol. DistribusiAfter eye drop admi…
KlirensAlthough the system…
Genetik -
Cenersen DB15455
biotech | CAS: 415168-49-9

Cenersen is under investigation in clinical trial NCT02243124 (A Study of Aezea® (Cenersen) in Transfusion Dependent Anemia Associated With Myelodysplastic Syndrome (MDS)).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cenicriviroc DB11758
small molecule | CAS: 497223-25-3

Cenicriviroc has been used in trials studying the treatment of HIV-infection/AIDS, AIDS Dementia Complex, Nonalcoholic Steatohepatitis, Human Immunodeficiency Virus, and HIV-1-Associated Cognitive Motor Complex.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +4
Target Protein:
C-C chemokine receptor type 5C-C chemokine receptor type 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Centhaquine DB16122
small molecule | CAS: 57961-90-7

Centhaquine is under investigation in clinical trial NCT04045327 (Efficacy of PMZ-2010 (Centhaquine) a Resuscitative Agent for Hypovolemic Shock).

Kategori:
Adrenergic and Dopaminergic AgentsCardiac Stimulants Excl. Cardiac GlycosidesCardiac Therapy
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CEP-9722 DB14882
small molecule | CAS: 916574-83-9

CEP-9722 is under investigation in clinical trial NCT01345357 (Study of CEP-9722 in Combination With Gemcitabine and Cisplatin in Patients With Advanced Solid Tumors or Mantle Cell Lymphoma).

Kategori:
Acids, CarbocyclicHeterocyclic Compounds, Fused-RingImides +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cephalexin Approved DB00567
small molecule | CAS: 15686-71-2

Cephalexin is the first of the first generation cephalosporins.[A179071,A179074] This antibiotic contains a beta lactam and a dihydrothiazide.[A179071] Cephalexin is used to treat a number of susceptible bacterial infections through inhibition of cell wall s…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +23
Target Protein:
Penicillin-binding protein 3Penicillin-binding protein 2aPenicillin-binding protein 1b +2
Waktu ParuhThe half life of ce…
Vol. Distribusi5.2-5.8L.[A179068]
KlirensClearance from one …
Genetik -
Cephaloglycin Approved DB00689
small molecule | CAS: 3577-01-3

A cephalorsporin antibiotic that is no longer commonly used.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +7
Target Protein:
Penicillin-binding protein 1B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cephalosporin C DB03313
small molecule | CAS: 61-24-5

Deskripsi belum tersedia.

Kategori:
Agents that reduce seizure thresholdAmidesbeta-Lactams +4
Target Protein:
Penicillin-binding protein 1bPeptidoglycan synthase FtsIPenicillin-binding protein 1A +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CER-001 DB18538
biotech

CER-001 is a negatively charged lipoprotein particle comprising human recombinant apolipoprotein A-I and two phospholipids: sphingomyelin and dipalmitoylphosphatidylglycerol.[L48290] It is under investigation for the treatment of lecithin-cholesterol acyltran…

Kategori:
Amino Acids, Peptides, and ProteinsApolipoproteinsApolipoproteins A +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceramide NP DB14111
small molecule | CAS: 100403-19-8

Ceramide NP is a lipid molecule included in a group of lipid molecules called ceramides. Ceramides are major lipid components in the stratum corneum of the human skin. Ceramide 3 consists of a phytosphingosine backbone N-acylated with a saturated fatty acid (…

Kategori:
AntigensAntigens, NeoplasmBiological Factors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CERE-110 DB05898
biotech

CERE-110 is a gene-therapy product that involves in vivo delivery of nerve growth factor (NGF) genes through an adeno-associated viral vector (AAV) delivery system. This drug is developed by Ceregene and currently under phase I of clinical trial.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CERE-120 DB05637
biotech | CAS: 1148126-35-5

CERE-120 is an investigational drug consisting of an adeno-associated virus (AAV) that was engineered to carry the human gene for neurturin, a neurotrophic (growth) factor. It was under investigation in clinical trials for the treatment of Parkinson's Disease.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1509916-03-3

Cergutuzumab amunaleukin is under investigation in clinical trial NCT02004106 (A Study to Evaluate Safety, Pharmacokinetics, and Efficacy of RO6895882 in Participants With Advanced and/or Metastatic Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceritinib Approved DB09063
small molecule | CAS: 1032900-25-6

Ceritinib is used for the treatment of adults with anaplastic lymphoma kinase (ALK)-positive metastatic non-small cell lung cancer (NSCLC) following failure (secondary to resistance or intolerance) of prior crizotinib therapy. About 4% of patients with NSCLC …

Kategori:
Anaplastic lymphoma kinase (ALK) inhibitorsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +25
Target Protein:
ALK tyrosine kinase receptor
Waktu ParuhThe terminal half l…
Vol. DistribusiThe apparent volume…
KlirensThe geometric mean …
Genetik -
Cerliponase alfa Approved DB13173
biotech | CAS: 151662-36-1

Cerliponase alfa is a hydrolytic lysosomal N-terminal tripeptidyl peptidase-1 (TPP1).[L51319] On April 27, 2017, cerliponase alfa was first approved by the FDA as the first treatment for neuronal ceroid lipofuscinosis type 2 (CLN2), also known as TPP1 deficie…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsEnzymes +6
Target Protein:
Cation-independent mannose-6-phosphate receptor
Waktu ParuhFollowing intravent…
Vol. DistribusiFollowing intravent…
KlirensFollowing intravent…
Genetik -
Certolizumab pegol Approved DB08904
biotech | CAS: 428863-50-7

Certolizumab pegol is a pegylated monoclonal antibody against the tumor necrosis factor-alpha (TNF-alpha).[A176585] It is formed with a humanized Fab fragment of 50 kDa, from an IgG 1 isotype, fused to a 40 kDa polyethylene glycol moiety replacing the Fc anti…

Kategori:
Agents reducing cytokine levelsAlcoholsAmino Acids, Peptides, and Proteins +31
Target Protein:
Tumor necrosis factor
Waktu ParuhThe circulatory hal…
Vol. DistribusiCertolizumab pegol …
KlirensThe clearance rate …
Genetik -
Cerulenin DB01034
small molecule | CAS: 17397-89-6

Cerulenin is an antifungal agent whose activity interferes with or otherwise acts to prevent the formation of fatty acids and sterols. In fatty acid synthesis, reported to bind in equimolar ratio to b-keto-acyl-ACP synthase. In sterol synthesis, inhibits HMG-…

Kategori:
AmidesAnti-Infective AgentsAntifungal Agents +3
Target Protein:
3-oxoacyl-[acyl-carrier-protein] synthase 13-oxoacyl-[acyl-carrier-protein] synthase 23-oxoacyl-[acyl-carrier-protein] synthase 3 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceruletide Approved DB00403
small molecule | CAS: 17650-98-5

Caerulein is a specific decapeptide similar in action and composition to the natural gastrointestinal peptide hormone cholecystokinin. It exerts stimulatory effects on the gastric, biliary, and pancreatic secretion, as well as on certain smooth muscles.

Kategori:
Amino Acids, Peptides, and ProteinsDiagnostic AgentsOligopeptides +2
Target Protein:
Cholecystokinin receptor type AGastrin/cholecystokinin type B receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cethromycin DB06419
small molecule | CAS: 205110-48-1

Cethromycin is a 3-keto (ketolide) derivative of erythromycin A with an 11,12-carbamate group and an O-6-linked aromatic ring system.[A203369] Cethromycin represents a joint development effort by Abbott Laboratories, Taisho Pharmaceuticals, and Advanced Life …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsCytochrome P-450 CYP3A Inhibitors +15
Target Protein:
23S ribosomal RNA
Waktu ParuhCethromycin given i…
Vol. DistribusiCethromycin given i…
KlirensCethromycin clearan…
Genetik -
Cetilistat DB06586
small molecule | CAS: 282526-98-1

Cetilistat is a novel inhibitor of pancreatic lipase being developed by Alizyme for the treatment of obesity and associated co-morbidities, including type 2 diabetes.

Kategori:
Anti-Obesity AgentsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Endothelial lipaseGastric triacylglycerol lipasePancreatic triacylglycerol lipase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetirizine Approved DB00341
small molecule | CAS: 83881-51-0

Cetirizine, also commonly known as _Zyrtec_, is an orally active second-generation histamine H1 antagonist proven effective in the treatment of various allergic symptoms, such as sneezing, coughing, nasal congestion, hives, and other symptoms [A175051], [A175…

Kategori:
Anti-Allergic AgentsAntihistamines for Systemic UseCentral Nervous System Depressants +14
Target Protein:
Histamine H1 receptor
Waktu ParuhPlasma elimination …
Vol. DistribusiApparent volume of …
KlirensApparent total body…
Genetik -
Cetrelimab DB15421
biotech | CAS: 2050478-92-5

Cetrelimab is under investigation in clinical trial NCT03547037 (A Study to Evaluate the Safety, Pharmacokinetics, Pharmacodynamics, and Immunogenicity of JNJ-63723283, an Anti-Programmed Cell Death (PD)-1 Monoclonal Antibody, as Monotherapy or in Combination…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetuximab Approved DB00002
biotech | CAS: 205923-56-4

Cetuximab is a recombinant chimeric human/mouse IgG1 monoclonal antibody that competitively binds to epidermal growth factor receptor (EGFR) and competitively inhibits the binding of epidermal growth factor (EGF).[A227973] EGFR is a member of the ErbB family …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
Epidermal growth factor receptorLow affinity immunoglobulin gamma Fc region receptor III-BComplement C1q subcomponent subunit A +5
Gen Terkait:
FCGR2A FCGR3A
Waktu ParuhAfter administratio…
Vol. DistribusiThe volume of the d…
KlirensIn patients with re…
Genetik 2 Varian
Cetyl alcohol Approved DB09494
small molecule | CAS: 36653-82-4

Cetyl alcohol, also known as 1-hexadecanol or n-hexadecyl alcohol, is a 16-C fatty alcohol with the chemical formula CH3(CH2)15OH. It can be produced from the reduction of palmitic acid. Cetyl alcohol is present in a waxy white powder or flake form at room te…

Kategori:
AlcoholsDrugs that are Mainly Renally ExcretedLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 59130-69-7

Cetyl ethylhexanoate is an ester of cetyl alcohol and 2-ethylhexanoic acid. It is present in cosmetic products as a skin conditioning agent and emollient.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetyl oleate DB19454
small molecule | CAS: 22393-86-8

Deskripsi belum tersedia.

Kategori:
Fatty AcidsLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetyl palmitate DB15782
small molecule | CAS: 540-10-3

Deskripsi belum tersedia.

Kategori:
Fatty AcidsLipidsPalmitic Acids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 22393-83-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetylpyridinium Approved DB11073
small molecule | CAS: 7773-52-6

Cetylpyridinium is a quaternary ammonium with broad-spectrum antiseptic properties. Its salt form, cetylpyridinium chloride, is typically found as an active ingredient in mouthwashes, toothpastes, lozenges, throat sprays, breath sprays, and nasal sprays. In t…

Kategori:
Alimentary Tract and MetabolismAnti-Infective AgentsAnti-Infective Agents, Local +19
Waktu ParuhNo readily availabl…
Vol. DistribusiNo readily availabl…
KlirensNo readily availabl…
Genetik -
Cevimeline Approved DB00185
small molecule | CAS: 107233-08-9

Cevimeline is a parasympathomimetic agent that act as an agonist at the muscarinic acetylcholine receptors M1 and M3. It is indicated by the Food and Drug Administration for the treatment of dry mouth associated with Sjögren's syndrome.

Kategori:
Autonomic AgentsCholinergic AgentsCholinergic Agonists +12
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M1
Waktu Paruh5 ± 1 hours
Vol. Distribusi* 6 L/kg
Klirens-
Genetik -
Cevostamab DB18374
biotech | CAS: 2249888-53-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CG0070 DB05148
small molecule

CG0070 is investigated in clinical trials for treating bladder cancer. CG0070 is a solid. CG0070 can potentially destroy cancer cells by two different mechanisms: direct cell killing by the virus and immune-mediated cell killing stimulated by GM-CSF. CG0070, …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CG7870 DB04981
biotech

CG7870 is an oncolytic virus therapy for prostate cancer. It is a replication-selective, prostate-specific antigen-targeted oncolytic adenovirus, for the treatment of hormone-refractory, metastatic prostate cancer.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 227016-66-2

CH-1504 L-isomer is under investigation in clinical trial NCT01116141 (A Study of CH-4051 in Patients With Rheumatoid Arthritis (RA)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chenodeoxycholic acid Approved DB06777
small molecule | CAS: 474-25-9

Chenodeoxycholic acid (or Chenodiol) is an epimer of ursodeoxycholic acid (DB01586). Chenodeoxycholic acid is a bile acid naturally found in the body. It works by dissolving the cholesterol that makes gallstones and inhibiting production of cholesterol in the…

Kategori:
Alimentary Tract and MetabolismBile Acid PreparationsBile acids and derivatives +12
Target Protein:
Bile acid receptorNuclear receptor subfamily 1 group I member 2G-protein coupled bile acid receptor 1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chicory leaf DB14376
biotech

Chicory leaf is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chiglitazar DB19023
small molecule | CAS: 743438-45-1

Chiglitazar is under investigation in clinical trial NCT06125587 (Chiglitazar/metformin in Non-obese Women With PCOS).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +3
Target Protein:
Peroxisome proliferator-activated receptor gammaPeroxisome proliferator-activated receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Chikungunya virus (CHIKV) is a member of the Alphavirus genus that was first identified in Tanzania in 1952.[A262051] It is spread primarily by the bite of infected mosquitos of the _Aedes_ genus. Infection with CHIKV causes chikungunya fever, an illness char…

Kategori:
Live vaccinesVaccinesViral Vaccines
Waktu ParuhThere is limited ph…
Vol. DistribusiThere is limited ph…
KlirensThere is limited ph…
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CHIR-124 DB06852
small molecule | CAS: 405168-58-3

CHIR-124 is a potent inhibitor of Chk1 that potentiates the cytotoxicity of topoisomerase I poisons in vitro and in vivo.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Serine/threonine-protein kinase Chk1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chitin DB15142
small molecule | CAS: 1398-61-4

Shrimp shell chitin is under investigation in clinical trial NCT00863356 (Trial of a Novel Chitosan Hemostatic Sealant in the Management of Complicated Epistaxis).

Kategori:
BiopolymersCarbohydratesChitin, antagonists & inhibitors +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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