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11793

Total database: 17430
Struktur (SMILES)
8607 (73.0%)
Target
6418 (54.4%)
Genomik
102 (0.9%)
Referensi
11793 (100.0%)

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Hasil Pencarian (11793)

Halaman 36 / 236
Alendronic acid Approved DB00630
small molecule | CAS: 66376-36-1

Alendronic acid is a second generation bisphosphonate that is used for the treatment of some forms of osteoperosis and Paget's disease[FDA Label][A959,A203111]. It functions by preventing resorption of bone[FDA Label][A959].

Kategori:
Agents Causing Muscle ToxicityBisphosphonatesBone Density Conservation Agents +5
Target Protein:
Farnesyl pyrophosphate synthaseHydroxylapatiteTyrosine-protein phosphatase non-receptor type 4 +3
Waktu ParuhDue to alendronic a…
Vol. Distribusi28L[FDA Label].
Klirens71mL/min[FDA Label].
Genetik -
Aleplasinin DB12635
small molecule | CAS: 481629-87-2

Aleplasinin has been investigated in Alzheimer Disease.

Target Protein:
Plasminogen activator inhibitor 1Plasminogen activator inhibitor 2Plasma serine protease inhibitor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Alethine DB05800
small molecule | CAS: 646-08-2

Alethine is studied in the treatment of cancer. It belongs to a family of chemicals called disulfides. It is a low molecular weight disulfide that has been shown to exhibit in vivo antitumor activity in murine myeloma and melanoma models.

Kategori:
AminesEthylaminesMercaptoethylamines +2
Waktu Paruh-
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Alexitol sodium DB15908
small molecule | CAS: 66813-51-2

Deskripsi belum tersedia.

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Alfacalcidol Approved DB01436
small molecule | CAS: 41294-56-8

Alfacalcidol, or 1-alpha-hydroxycholecalciferol or 1-alpha-hydroxyvitamin D3, is a non-endogenous analogue of [vitamin D].[A234044] It plays an essential function in calcium homeostasis and bone metabolism. Alfacaldisol is activated by the enzyme 25-hydroxyla…

Kategori:
Alimentary Tract and MetabolismBone Density Conservation AgentsCholestanes +13
Target Protein:
Vitamin D3 receptor25-hydroxyvitamin D-1 alpha hydroxylase, mitochondrialRetinoic acid receptor RXR-alpha
Waktu ParuhThe half-life of al…
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 473553-86-5

Alferminogene tadenovec, Cardium’s lead product candidate, is being developed for the potential treatment of myocardial ischemia that gives rise to angina symptoms associated with coronary heart disease. Alferminogene tadenovec represents a new therapeutic cl…

Kategori:
Antianginal AgentsVasodilating Agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alfimeprase DB04919
biotech | CAS: 259074-76-5

Alfimeprase is a recombinant analog of fibrolase. Fibrolase is a zinc-containing metalloproteinase isolated from the venom of the southern copperhead snake (<i>Agkistrodon contortrix contortrix</i>). It is a small protein that contains 203 residues (Randolph …

Kategori:
EndopeptidasesEnzymesEnzymes and Coenzymes +3
Target Protein:
Fibrinogen alpha chainFibrinogen beta chain
Waktu Paruh-
Vol. Distribusi-
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Alflorex Approved DB18507
biotech

Alflorex is a probiotic with 35624 cultures, part of the Bifidobacterium longum.

Waktu Paruh-
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Alflutinib DB16087
small molecule | CAS: 1869057-83-9

Alflutinib is under investigation in clinical trial NCT03452592 (Efficacy and Safety of Alflutinib in Locally Advanced or Metastatic Non-small Cell Lung Cancer Patients With T790M).

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Waktu Paruh-
Vol. Distribusi-
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Alfuzosin Approved DB00346
small molecule | CAS: 81403-80-7

Benign prostatic hyperplasia (BPH) refers to a benign growth or hyperplasia of the prostate and leads to lower urinary tract symptoms in men, such as urgency, frequency and changes to urine flow. The prevalence of BPH is as high as 50%-60% for males in their …

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +17
Target Protein:
Alpha-1 adrenergic receptorsAlpha-1A adrenergic receptorAlpha-1B adrenergic receptor +1
Waktu ParuhThe apparent elimin…
Vol. DistribusiThe volume of distr…
KlirensExercise caution if…
Genetik -
Algestone DB18000
small molecule | CAS: 595-77-7

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesContraceptive Agents, FemaleContraceptive Agents, Hormonal +14
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 24356-94-3

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesAlgestoneAnti-Inflammatory Agents +13
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Alginic acid Approved DB13518
small molecule | CAS: 9005-32-7

Alginic acid, also referred to as algin or alginate, is a hydrophilic or anionic polysaccharide isolated from certain brown seaweed (_Phacophycae_) via alkaline extraction. It is present in cell walls of brown algae where it forms a viscous gel when binding w…

Kategori:
Acids, AcyclicAcids, AldehydicAlginates +11
Waktu ParuhThis pharmacokineti…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Alglucerase Approved DB00088
biotech | CAS: 143003-46-7

Human Beta-glucocerebrosidase or Beta-D-glucosyl-N-acylsphingosine glucohydrolase E.C. 3.2.1.45. 497 residue protein with N-linked carbohydrates, MW=59.3 kD. Alglucerase is prepared by modification of the oligosaccharide chains of human Beta-glucocerebrosidas…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +6
Target Protein:
Glucocerebroside
Waktu Paruh3.6-10.4 min
Vol. Distribusi* 49.4 to 282.1 mL/…
Klirens-
Genetik -
Alglucosidase alfa Approved DB01272
biotech | CAS: 420784-05-0

Aglucosidase alfa consists of the human enzyme acid alpha-glucosidase (GAA) which is essential for the degradation of glygogen to glucose in lysosomes. It is encoded by the most predominant of nine observed haplotypes of this gene. Aglucosidase alfa is produc…

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes +5
Target Protein:
Cation-dependent mannose-6-phosphate receptorGlycogen
Waktu Paruh2.3 &plusmn; 0.4 ho…
Vol. Distribusi* 96 ± 16 mL/kg [20…
Klirens* 25+/- 4 mL/hr/kg …
Genetik -
ALGRX 1207 DB06482
small molecule

ALGRX 1207 is a topical local anesthetic that acts by binding to the fast sodium channel. ALGRX 1207 entered clinical trials for cutaneous neuropathic pain, such as chemotherapy-induced neuropathy, in 2006. It was being developed by Anesiva, but trials have h…

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Alicaforsen DB06224
small molecule | CAS: 185229-68-9

Deskripsi belum tersedia.

Kategori:
Gastrointestinal AgentsImmunologic FactorsNucleic Acids, Nucleotides, and Nucleosides +3
Target Protein:
Intercellular adhesion molecule 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alidornase alfa DB18144
biotech | CAS: 1788036-49-6

Deskripsi belum tersedia.

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Alimemazine Approved DB01246
small molecule | CAS: 84-96-8

A phenothiazine derivative that is used as an antipruritic.

Kategori:
Antihistamines for Systemic UseAntipruriticsAntipsychotic Agents +13
Target Protein:
Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
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Alintegimod DB18879
small molecule | CAS: 1378535-08-0

Alintegimod is under investigation in clinical trial NCT06362369 (A Study of Oral 7HP349 (Alintegimod) in Combination With Ipilimumab Followed by Nivolumab Monotherapy).

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Alipogene tiparvovec Approved DB13521
biotech | CAS: 929881-05-0

Alipogene tiparvovec is an adeno-associated viral vector of serotype 1-based gene therapy that delivers the Ser(447)X variant of the human lipoprotein lipase (LPL) gene. It is being investigated for the treatment of lipoprotein lipase (LPL) deficiency.[A25979…

Kategori:
Adeno-associated Viral Vector TherapiesLipid Modifying AgentsLipid Modifying Agents, Plain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alirinetide DB17007
biotech | CAS: 725715-18-4

Deskripsi belum tersedia.

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Alirocumab Approved DB09302
biotech | CAS: 1245916-14-6

Alirocumab is a biopharmaceutical that obtained FDA approval in July 2015 as a second line treatment for high cholesterol in adults whose LDL-cholesterol (LDL-C) is not controlled by the combination of diet and statin treatment. It is a human monoclonal antib…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +20
Target Protein:
Proprotein convertase subtilisin/kexin type 9
Waktu ParuhIn monotherapy, the…
Vol. DistribusiAlirocumab is mainl…
Klirens-
Genetik -
Alisertib DB05220
small molecule | CAS: 1028486-01-2

Alisertib is a novel aurora A kinase inhibitor under investigation for the treatment of various forms of cancer.

Kategori:
Protein Kinase Inhibitors
Target Protein:
Aurora kinase A
Waktu Paruh-
Vol. Distribusi-
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Aliskiren Approved DB09026
small molecule | CAS: 173334-57-1

Aliskiren is the first drug in the renin inhibitor drug class and is used for the treatment of hypertension.[A203624] It was developed by Speedel and Novartis and initially approved by the FDA in early 2007.[L14018] Aliskiren has been proven to efficacious in…

Kategori:
Acids, AcyclicAgents Acting on the Renin-Angiotensin SystemAgents causing hyperkalemia +14
Target Protein:
Renin
Waktu ParuhPlasma half-life fo…
Vol. DistribusiUnchanged aliskiren…
KlirensAliskiren is partia…
Genetik -
Alitretinoin Approved DB00523
small molecule | CAS: 5300-03-8

An important regulator of gene expression during growth and development, and in neoplasms. Tretinoin, also known as retinoic acid and derived from maternal vitamin A, is essential for normal growth; and embryonic development. An excess of tretinoin can be ter…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAlkenesAntineoplastic Agents +19
Target Protein:
Retinoic acid receptor alphaRetinoic acid receptor RXR-alphaRetinoic acid receptor beta +6
Waktu Paruh-
Vol. Distribusi-
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Genetik -
ALK-4290 DB15269
small molecule | CAS: 1251528-23-0

ALK-4290 is under investigation in clinical trial NCT03558061 (Evaluate the Effects and Safety of ALK4290 in Patients With Newly Diagnosed Wet Age-Related Macular Degeneration).

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small molecule

Alkaline Phosphatase (AP) is an oral treatment and has a very favorable side-effect profile. AP only acts locally in the colon to reduce the continuous inflammation of the colon by endotoxin from Gram-negative bacteria and extracellular ATP in UC patients.

Kategori:
EnzymesEnzymes and CoenzymesEsterases +2
Waktu Paruh-
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Allantoin Approved DB11100
small molecule | CAS: 97-59-6

Allantoin is a substance that is endogenous to the human body and also found as a normal component of human diets [FDA Label]. In healthy human volunteers, the mean plasma concentration of allantoin is about 2-3 mg/l. During exercise, the plasma allantoin con…

Kategori:
AmidesBasic Ointments and ProtectantsDermatologicals +5
Waktu ParuhWhen studied in cat…
Vol. Distribusi-
KlirensSome studies sugges…
Genetik -
biotech

Beef liver allergenic extract is used in allergenic testing.

Kategori:
Non-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Allicin DB11780
small molecule | CAS: 539-86-6

Allicin has been used in trials studying the treatment of Follicular Lymphoma.

Kategori:
AcidsAcids, NoncarboxylicAnions +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 947331-05-7

Allisartan isoproxil is under investigation in clinical trial NCT03264352 (Intervention for High-normal Blood Pressure in Adults With Type 2 Diabetes).

Kategori:
Agents Acting on the Renin-Angiotensin SystemAngiotensin II receptor antagonistsAngiotensin II Type 1 Receptor Blockers +3
Waktu Paruh-
Vol. Distribusi-
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Allitinib DB18840
small molecule | CAS: 897383-62-9

Allitinib is under investigation in clinical trial NCT04671303 (To Evaluate the Efficacy and Safety of Anlotinib Combined With Allitinib in Lung Cancer).

Kategori:
Acids, AcyclicAcrylatesAmides +2
Target Protein:
Epidermal growth factor receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
ALLO-605 DB18641
biotech

ALLO-605 is an allogeneic turbo chimeric antigen receptor (Turbocar) T Cell therapy targeting B Cell maturation antigen (BCMA).

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ALLO-715 DB18640
biotech

ALLO-715 is an allogeneic chimeric antigen receptor T Cell therapy targeting B cell maturation antigen (BCMA).

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Allocetra DB16424
biotech

Allocetra is a novel therapy where billions of early apoptotic cells are infused into the bloodstream of a patient, using the body's own natural regulation mechanisms to rebalance an unbalanced immune system without immune system suppression. With infusion, t…

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biotech

Stratagraft (allogeneic cultured keratinocytes and dermal fibroblasts in murine collagen-dsat) is an allogeneic cellularized scaffold product used for the treatment of adults with thermal burns containing intact dermal elements for which surgical intervention…

Kategori:
FibroblastsKeratinocytes
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biotech

Deskripsi belum tersedia.

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biotech

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biotech

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biotech

Allogeneic processed thymus tissue is used for immune reconstitution in immune disorders where the patients are severely immunocompromised due to the absence of a functional thymus, such as congenital athymia. As part of the immune system, the thymus is an or…

Waktu ParuhThe pharmacokinetic…
Vol. DistribusiThe pharmacokinetic…
KlirensThe pharmacokinetic…
Genetik -
biotech

Deskripsi belum tersedia.

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biotech

ORBCEL-C™ is the trade name of a product composed of highly purified stromal cells derived from the human umbilical cord. The isolated cells are expanded in culture and are able to be used allogenically -- meaning that one donor’s cells can be given to other …

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biotech

Deskripsi belum tersedia.

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Alloin Approved DB15477
small molecule | CAS: 8015-61-0

Deskripsi belum tersedia.

Kategori:
AnthracenesAnthraquinonesBiological Products +5
Waktu Paruh-
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Allolactose DB04116
small molecule | CAS: 645-03-4

Deskripsi belum tersedia.

Kategori:
CarbohydratesDisaccharidesOligosaccharides +1
Target Protein:
Beta-galactosidase
Waktu Paruh-
Vol. Distribusi-
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Allopurinol Approved DB00437
small molecule | CAS: 315-30-0

Gout is a disease that occurs by the deposition of monosodium urate crystals (MSU) in body tissues, especially around joints [A175942]. This disease has been well-documented in historical medical records and appears in the biographies of several prominent, h…

Kategori:
Antigout PreparationsAntimetabolitesAntioxidants +12
Target Protein:
Xanthine dehydrogenase/oxidase
Gen Terkait:
HCP5
Waktu ParuhThe plasma half-lif…
Vol. DistribusiAllopurinol and oxy…
KlirensSince allopurinol a…
Genetik 1 Varian
small molecule | CAS: 16220-07-8

Allopurinol riboside is a nucleoside analogue of [allopurinol] with a beta-D-ribofuranosyl moiety at the 1-position.

Kategori:
Anti-Infective AgentsAntiparasitic AgentsAntiprotozoals +4
Waktu Paruh-
Vol. Distribusi-
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Allosamidin DB04628
small molecule | CAS: 103782-08-7

Allosamidin exhibits extremely potent inhibitory activity against chitinases from a number of sources, particularly from <i>Candida albicans</i>, and can be utilized as potent antifungal agent.

Kategori:
AgrochemicalsAmino SugarsCarbohydrates +9
Target Protein:
Chitinase BChitinase A
Waktu Paruh-
Vol. Distribusi-
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Allspice Approved DB10669
biotech

Allspice allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
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Vol. Distribusi-
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Genetik -
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