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2279

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866 (38.0%)
Target
1100 (48.3%)
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Halaman 35 / 46
Prochlorperazine Approved DB00433
small molecule | CAS: 58-38-8

Prochlorperazine, also known as compazine, is a piperazine phenothiazine and first-generation antipsychotic drug that is used for the treatment of severe nausea and vomiting, as well as short-term management of psychotic disorders such as generalized non-psyc…

Kategori:
AntiemeticsAntipsychotic AgentsAntipsychotic Agents (First Generation [Typical]) +28
Target Protein:
D(2) dopamine receptorHistamine H1 receptorAlpha-1 adrenergic receptors +1
Waktu ParuhFollowing intraveno…
Vol. DistribusiIn a preliminary ph…
KlirensThe mean plasma cle…
Genetik -
Progesterone Approved DB00396
small molecule | CAS: 57-83-0

Progesterone is a hormone that occurs naturally in females, and is essential for endometrial receptivity, embryo implantation, and the successful establishment of pregnancy. A low progesterone concentration or an insufficient response to progesterone can caus…

Kategori:
Adrenal Cortex HormonesBCRP/ABCG2 InducersBCRP/ABCG2 Inhibitors +47
Target Protein:
Progesterone receptorMineralocorticoid receptorEstrogen receptor +7
Waktu ParuhAbsorption half-lif…
Vol. DistribusiWhen administered v…
Klirens**Apparent clearanc…
Genetik -
biotech | CAS: 67422-14-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBlood Glucose Lowering AgentsHormones +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prolease-r-hFSH DB05826
biotech

Prolease-r-hFSH is a recombinant human follicle stimulating hormone (r-hFSH) with Alkermes' ProLease injectable sustained release drug delivery technology. It provides patients with long term therapeutic benefit from a single administration rather than multip…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prolectin-M DB16521
small molecule

Prolectin-M is a (1-6)-alpha-D-mannopyranose[L31338] and acts as an antagonist of galectin.[L31343] It is being investigated in the clinical trial NCT04512027 (Prolectin-M in COVID-19 Patients Having Mild to Moderate Symptoms Not Requiring Oxygen Support. (Pr…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propagermanium DB17608
small molecule | CAS: 12758-40-6

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAntineoplastic AgentsElements +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propiomazine Approved DB00777
small molecule | CAS: 362-29-8

Propiomazine, an atypical antipsychotic agent, is used to treat both negative and positive symptoms of schizophrenia, acute mania with bipolar disorder, agitation, and psychotic symptoms in dementia. Future uses may include the treatment of obsessive-compulsi…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +20
Target Protein:
Histamine H1 receptorMuscarinic acetylcholine receptorAlpha-1A adrenergic receptor +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propofol Approved DB00818
small molecule | CAS: 2078-54-8

Propofol is an intravenous anaesthetic agent used for induction and maintenance of general anaesthesia. IV administration of propfol is used to induce unconsciousness after which anaesthesia may be maintained using a combination of medications. Recovery from …

Kategori:
Agents Causing Muscle ToxicityAgents that produce hypertensionAgents that reduce seizure threshold +32
Target Protein:
Gamma-aminobutyric acid receptor subunit beta-2Gamma-aminobutyric acid receptor subunit beta-3GABA(A) Receptor +2
Waktu ParuhInitial distributio…
Vol. Distribusi* 60 L/kg [healthy …
Klirens* 23 - 50 mL/kg/min…
Genetik -
small molecule | CAS: 41598-07-6

The principal cyclooxygenase metabolite of arachidonic acid. It is released upon activation of mast cells and is also synthesized by alveolar macrophages. Among its many biological actions, the most important are its bronchoconstrictor, platelet-activating-fa…

Kategori:
AutacoidsBiological FactorsEicosanoids +7
Target Protein:
Prostaglandin D2 receptorProstaglandin F2-alpha receptorProstaglandin E2 receptor EP1 subtype +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protamine sulfate Approved DB09141
biotech | CAS: 9009-65-8

Since it's earliest discovery in salmon rine sperm heads in the late 1800's to its formal introduction via US FDA approval in 1939, protamine sulfate has occupied an important therapeutic niche as perhaps the only viable option for reversing the anticoagulant…

Kategori:
Amino Acids, Peptides, and ProteinsAntiheparin AgentsHematologic Agents +5
Waktu ParuhThe half-life of pr…
Vol. DistribusiIn a study group of…
KlirensIn a study group of…
Genetik -
Protein C Approved DB11312
biotech

Protein C is an endogenously occurring plasma protein that plays a key role within the coagulation cascade. Protein C is a zymogen, or enzyme precursor, of a vitamin K-dependent anticoagulant glycoprotein (serine protease) that is synthesized in the liver. It…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsBiological Factors +15
Target Protein:
Coagulation factor VCoagulation factor VIII
Waktu ParuhInitial half life =…
Vol. DistribusiVolume of distribut…
KlirensCL = 0.0533 dL/kg/h
Genetik -
Protein S human Approved DB13149
biotech

Protein S human is a vitamin K-dependent plasma glycoprotein which has antcoagulant properties [A19561]. It serves as a negative feedback mechanism in the coagulation cascade.

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsBiological Factors +8
Target Protein:
Coagulation factor VCoagulation factor XVitamin K-dependent protein C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prothrombin Approved DB11311
biotech | CAS: 9001-26-7

Prothrombin Complex Concentrate (Human), is indicated for the urgent reversal of acquired coagulation factor deficiency induced by Vitamin K antagonist (VKA, e.g., warfarin) therapy in adult patients with acute major bleeding.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +7
Target Protein:
Fibrinogen alpha chainFibrinogen beta chainCoagulation factor XIII A chain +1
Waktu ParuhApproximately 60h […
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 139-85-5

Also known as protocatechuic aldehyde, protocatechualdehyde is a naturally-occuring phenolic aldehyde that is found in barley, green cavendish bananas, grapevine leaves and root of the herb S. miltiorrhiza [A27224]. Protocatechualdehyde possesses antiprolifer…

Kategori:
AldehydesAnticoagulantsBenzene Derivatives +2
Target Protein:
Amine oxidase [flavin-containing] B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PRX-ASL DB17679
biotech

PRX-ASL is an intracellular enzyme replacement therapy designed to replace the missing or defective enzyme in patients with argininosuccinate lyase deficiency.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PTR-01 DB17900
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pucotenlimab Approved DB17552
biotech | CAS: 2403647-03-8

Pucotenlimab is a recombinant humanized anti-PD-1 monoclonal antibody. It received its first global approval in China in July 2022 for the treatment of solid tumours.[A257296] It is being investigated in other cancers.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pulocimab DB18938
biotech | CAS: 2428381-49-9

Pulocimab is under investigation in clinical trial NCT06341335 (A Study of Ak104/placebo Plus Ak109/placebo and Paclitaxel in Gastric or Gastroesophageal Junction Adenocarcinoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pyrantel Approved DB11156
small molecule | CAS: 15686-83-6

Pyrantel is a pyrimidine-derivative anthelmintic agent for the oral treatment of various parasitic worm infections including ascariasis, hookworm infections, enterobiasis (pinworm infection), trichostrongyliasis, and trichinellosis [L1904]. Pyrantel was in…

Kategori:
AnthelminticsAnti-Infective AgentsAntinematodal Agents +12
Target Protein:
G-protein coupled receptor 35Muscarinic acetylcholine receptor M1
Waktu ParuhIn pigs, following …
Vol. Distribusi-
Klirens-
Genetik -
Pyrethrum extract Approved DB11087
biotech | CAS: 8003-34-7

Pyrethrum is the crude extract form obtained from flowers of the plant Chrysanthemum cinerariifolium. Pyrethrin refers to a more refined extract of pyrethrum. While pyrethrum extract is composed of 6 esters, both organic compounds mediate insecticidal activit…

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingCyclopentane Monoterpenes +6
Target Protein:
Nuclear receptor subfamily 1 group I member 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pyridoxine Approved DB00165
small molecule | CAS: 65-23-6

Pyridoxine is the 4-methanol form of vitamin B6, an important water-soluble vitamin that is naturally present in many foods. As its classification as a vitamin implies, Vitamin B6 (and pyridoxine) are essential nutrients required for normal functioning of man…

Kategori:
Alimentary Tract and MetabolismAnalogs/DerivativesAntiinfectives for Systemic Use +10
Target Protein:
Aromatic-L-amino-acid decarboxylasePyridoxal kinase
Waktu ParuhThe total adult bod…
Vol. DistribusiPyridoxine main act…
Klirens-
Genetik -
Pyruvic acid Approved DB00119
small molecule | CAS: 127-17-3

An intermediate compound in the metabolism of carbohydrates, proteins, and fats. In thiamine deficiency, its oxidation is retarded and it accumulates in the tissues, especially in nervous structures. (From Stedman, 26th ed)

Kategori:
Dietary SupplementsKeto AcidsPyruvates +1
Target Protein:
Carbonic anhydrase 44-aminobutyrate aminotransferase, mitochondrialMonocarboxylate transporter 4 +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
QR-334 DB05473
small molecule

QR-334 is under investigation for the treatment of sialorrhea. Sialorrhea is an excess secretion of saliva produced by the salivary glands, resulting in drooling. No pharmaceutical interventions currently exist to treat sialorrhea. The symptom is associated w…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quaternium-15 Approved DB14198
small molecule | CAS: 4080-31-3

Quaternium-15 is a quaternary ammonium salt used as a surfactant and preservative in many products including cosmetics. It is an anti-microbial agent by virtue of being a formaldehyde releaser, however this can also cause contact dermatitis, a symptom of an a…

Kategori:
AminesBridged-Ring CompoundsCell-mediated Immunity +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quercetin DB04216
small molecule | CAS: 117-39-5

Quercetin is a flavonol widely distributed in plants. It is an antioxidant, like many other phenolic heterocyclic compounds. Glycosylated forms include RUTIN and quercetrin.

Kategori:
AntioxidantsBCRP/ABCG2 InhibitorsBenzopyrans +26
Target Protein:
Signal transducer and activator of transcription 3Lysophosphatidylcholine acyltransferase 2Lysophosphatidylcholine acyltransferase 1 +29
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Queuine DB14732
small molecule | CAS: 72496-59-4

Queuine is a derivative of [7-Deazaguanine]. Bacteria possess the exclusive ability to synthesize queuine, which is then salvaged and passed on to plants and animals. Quantities of queuine have been found in tomatoes, wheat, coconut water, and milk from human…

Kategori:
Heterocyclic Compounds, Fused-RingPurinesPurinones
Waktu ParuhData regarding the …
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Quisovalimab DB16482
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-30490 DB09179
small molecule | CAS: 60618-49-7

R-30490 is an opioid related to carfentanil used as an animal tranquilizer. It was first synthesized by Janssen Pharmaceutica as part of a structure-activity relationship study of fentanly and its derivatives. R-30490 was found to be the most selective agonis…

Kategori:
Piperidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-851 DB05747
small molecule

R-851 is part of the family of immune response modifier (IRM) and it acts in a novel way to stimulate the human body's immnune system to attack virus-infected cells and tumor cells. It is expected to be topical treatment for cervical displasia and cervical hi…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
rAAV9-hNAGLU DB18415
biotech

rAAV9-hNAGLU consists of a recombinant AAV9 expressing human alpha-N-acetylglucosaminidase.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

IMOGAM Rabies Pasteurized is indicated for post-exposure prophylaxis in persons suspected of exposure to rabies, who have not previously received a complete immunization regimen with a cell culture produced rabies vaccine. Persons previously vaccinated wit…

Kategori:
Human Rabies Immune GlobulinsSerumVaccines
Target Protein:
Rabies Virus Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Inactivated rabies virus antigen B is a component of rabies vaccines used for pre- and post-exposure prophylaxis against rabies.[L12795]

Kategori:
Actively Acquired ImmunityAntiinfectives for Systemic UseImmune Sera +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RAD 502 DB17328
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Radotermin DB19127
biotech | CAS: 575458-75-2

Radotermin is under investigation in clinical trial NCT01182337 (A Clinical Trial to Evaluate the Safety, Tolerability and Preliminary Effectiveness of Single Administration Intradiscal Rhgdf-5 for the Treatment of Early Stage Lumbar Disc Degeneration).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ragifilimab DB18853
biotech | CAS: 2207590-51-8

Ragifilimab is under investigation in clinical trial NCT04225039 (Anti-gitr/anti-pd1/stereotactic Radiosurgery, in Recurrent Glioblastoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Raloxifene Approved DB00481
small molecule | CAS: 84449-90-1

Raloxifene is a second generation selective estrogen receptor modulator (SERM) that mediates anti-estrogenic effects on breast and uterine tissues, and estrogenic effects on bone, lipid metabolism, and blood coagulation.[A4979,T28] Exhibiting tissue-specific …

Kategori:
BCRP/ABCG2 SubstratesBenzene DerivativesBenzylidene Compounds +23
Target Protein:
Estrogen receptorEstrogen receptor betaSerpin B9 +1
Waktu ParuhThe average plasma …
Vol. DistribusiFollowing oral admi…
KlirensFollowing intraveno…
Genetik -
Raltitrexed Approved DB00293
small molecule | CAS: 112887-68-0

Raltitrexed (brand name Tomudex®) is a chemotherapy drug manufactured AstraZeneca Company, is an antimetabolite used in chemotherapy. It is an inhibitor of thymidylate synthase.

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +11
Target Protein:
Thymidylate synthaseThymidylate synthaseFolylpolyglutamate synthase, mitochondrial
Waktu Paruh198 hours
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2610074-57-0

Raludotatug deruxtecan is under investigation in clinical trial NCT06660654 (A Study of Raludotatug Deruxtecan in Participants With Advanced/metastatic Solid Tumors (Rejoice-pantumor01)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ramucirumab Approved DB05578
biotech | CAS: 947687-13-0

Ramucirumab is a human monoclonal antibody (IgG1) against vascular endothelial growth factor receptor 2 (VEGFR2), a type II trans-membrane tyrosine kinase receptor expressed on endothelial cells. By binding to VEGFR2, ramucirumab prevents binding of its ligan…

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +20
Target Protein:
Vascular endothelial growth factor receptor 2
Waktu Paruh15 days
Vol. Distribusi5.5 L
Klirens0.014 L/hour
Genetik -
Ranibizumab Approved DB01270
biotech | CAS: 347396-82-1

Ranibizumab is a recombinant humanized IgG1 kappa isotype monoclonal antibody fragment directed against human vascular endothelial growth factor A (VEGF-A), which is a glycoprotein implicated in the pathophysiology of age-related macular degeneration.[A2301, …

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +19
Target Protein:
Vascular endothelial growth factor A, long form
Waktu ParuhThe estimated avera…
Vol. DistribusiThe apparent volume…
KlirensIn patients with re…
Genetik -
Ranolazine Approved DB00243
small molecule | CAS: 95635-55-5

Chronic angina is a common cardiovascular condition affecting millions worldwide and causes significant disability while interfering with daily activities.[A189234] Ranolazine is a well-tolerated piperazine derivative used for the management of this condition…

Kategori:
AcetamidesAntianginal AgentsBSEP/ABCB11 Substrates +26
Target Protein:
PlasminogenSodium channel proteinInward rectifier potassium channel +4
Waktu ParuhThe apparent termin…
Vol. DistribusiThe mean apparent v…
KlirensThe reported cleara…
Genetik -
Ranpirnase DB04950
biotech | CAS: 196488-72-9

Ranpirnase is a ribonuclease enzyme found in <i>Rana pipiens</i> oocytes. It is being studied in the treatment of cancer. It is manufactured by Alfacell Corporation. It is the first ribonuclease to enter cancer clinical trials.

Kategori:
Antineoplastic AgentsEgg ProteinsEnzyme Inhibitors +6
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rapacuronium Approved DB04834
small molecule | CAS: 465499-11-0

Rapacuronium was withdrawn in 2001 in many countries due to risk of fatal bronchospasm.

Kategori:
Agents producing tachycardiaAndrostanesAndrostanols +9
Target Protein:
Muscarinic acetylcholine receptor M2
Waktu Paruh141 minutes (mean)
Vol. Distribusi-
Klirens-
Genetik -
Ravulizumab Approved DB11580
biotech | CAS: 1803171-55-2

Ravulizumab is a potent and selective complement 5 (C5) inhibitor. It is a humanized monoclonal IgG2/4 kappa antibody produced in Chinese hamster ovary (CHO) cells.[L39690] Ravulizumab was engineered from [eculizumab], another complement inhibitor, to increas…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
Complement C5
Waktu ParuhThe mean (%CV) term…
Vol. DistribusiThe mean (%CV) volu…
KlirensThe mean (%CV) clea…
Genetik -
Raxibacumab Approved DB08902
biotech | CAS: 565451-13-0

Raxibacumab is a human IgG1? monoclonal antibody that binds the protective antigen (PA) component of B. anthracis toxin. Raxibacumab has a molecular weight of approximately 146 kilodaltons. Raxibacumab is produced by recombinant DNA technology in a murine cel…

Kategori:
Amino Acids, Peptides, and ProteinsAnthrax Protective Antigen-directed AntibodyAnthrax Protective Antigen-directed Antibody Interactions +12
Target Protein:
Protective antigen
Waktu ParuhMean terminal elimi…
Vol. DistribusiSteady state volume…
KlirensClearance values we…
Genetik -
RBIO-101 DB18425
biotech

RBIO-101 is a recombinant adeno-associated virus vector encoding human CYP4V2 protein.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RC118 DB18428
biotech

RC118 is an antibody-drug conjugate that consists of a recombinant humanized IgG1 anti-Claudin18.2 monoclonal antibody conjugated to MMAE.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RC88 DB18697
biotech

RC88 is an antibody-drug conjugate comprising a humanized anti-mesothelin monoclonal antibody conjugated to monomethyl auristatin E (MMAE).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Recifercept DB17899
biotech | CAS: 2226238-09-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Alpha 1-antitrypsin is a glycoprotein primarily produced by hepatocytes, and to a lesser extent, immune system cells. Recombinant alpha 1-antitrypsin (rAAT) is produced from yeast, which unlike commercially available forms of plasma-derived AAT, eliminates th…

Target Protein:
Alpha-1-antitrypsin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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