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3253

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2451 (75.3%)
Target
1833 (56.3%)
Genomik
35 (1.1%)
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3253 (100.0%)

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Halaman 35 / 66
Levobunolol Approved DB01210
small molecule | CAS: 47141-42-4

A nonselective beta-adrenoceptor antagonist used in the treatment of glaucoma.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +22
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptor
Waktu Paruh20 hours
Vol. Distribusi-
Klirens-
Genetik -
Levobupivacaine Approved DB01002
small molecule | CAS: 27262-47-1

Levobupivacaine is an amino-amide local anaesthetic drug belonging to the family of n-alkylsubstituted pipecoloxylidide. It is the S-enantiomer of bupivacaine. Levobupivacaine hydrochloride is commonly marketed by AstraZeneca under the trade name Chirocaine.…

Kategori:
AmidesAminesAnesthetics +15
Target Protein:
Sodium channel protein type 10 subunit alpha
Waktu Paruh3.3 hours
Vol. Distribusi66.91 ±18.23 L [aft…
Klirens39.06 ±13.29 L/h [a…
Genetik -
Levodopa Approved DB01235
small molecule | CAS: 59-92-7

Levodopa is a prodrug of dopamine that is administered to patients with Parkinson's due to its ability to cross the blood-brain barrier[Label]. Levodopa can be metabolised to dopamine on either side of the blood-brain barrier and so it is generally administer…

Kategori:
AminesAmino AcidsAmino Acids, Aromatic +21
Target Protein:
D(1A) dopamine receptorD(1B) dopamine receptorD(2) dopamine receptor +2
Waktu Paruh2.3 hours for orall…
Vol. Distribusi168L for orally inh…
KlirensIntravenously admin…
Genetik -
small molecule | CAS: 99291-25-5

Levodropropizine is under investigation in clinical trial NCT01573663 (A Drug-Drug Interaction Study of Ambroxol and Levodropropizine).

Kategori:
AlcoholsAntitussive AgentsCentral Nervous System Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levofloxacin Approved DB01137
small molecule | CAS: 100986-85-4

Levofloxacin is a fluoroquinolone antibiotic and the optical S-(-) isomer of racemic [ofloxacin].[A190663] It reportedly carries 8 to 128-fold more activity against both gram-negative and gram-positive bacteria compared to R-(+)-ofloxacin[A190663] and remains…

Kategori:
4-QuinolonesAlimentary Tract and MetabolismAnti-Bacterial Agents +35
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +1
Waktu ParuhThe average termina…
Vol. DistribusiLevofloxacin is wid…
KlirensThe average apparen…
Genetik -
Levoglucose DB12970
small molecule | CAS: 921-60-8

Levoglucose has been used in trials studying the diagnostic of Bowel Cleansing Prior to Colonoscopy.

Kategori:
CarbohydratesCompounds used in a research, industrial, or household settingDiet, Food, and Nutrition +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levoketoconazole Approved DB05667
small molecule | CAS: 142128-57-2

Cushing's syndrome (CS) is underpinned by chronic hypercortisolism leading to multisystem morbidity, including effects on the cardiovascular and endocrine systems, metabolic syndrome with accompanying changes in body composition, neuropsychiatric effects, cha…

Kategori:
Adrenal Cortex HormonesAntiadrenal PreparationsAnticorticosteroids +32
Target Protein:
Steroid 17-alpha-hydroxylase/17,20 lyaseCytochrome P450 11B1, mitochondrialCytochrome P450 11B2, mitochondrial +2
Waktu ParuhLevoketoconazole ha…
Vol. DistribusiLevoketoconazole ha…
Klirens-
Genetik -
Levomefolic acid Approved DB11256
small molecule | CAS: 31690-09-2

Levomefolic acid (INN) is the metabolite of folic acid (Vitamin B9) and it is a predominant active form of folate found in foods and in the blood circulation, accounting for 98% of folates in human plasma [A19276]. It is transported across the membranes inclu…

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +10
Waktu ParuhThe mean eliminatio…
Vol. DistribusiCirculates in its f…
Klirens-
Genetik -
Levomenol Approved DB13153
small molecule | CAS: 23089-26-1

Bisabolol, or more formally ?-(?)-bisabolol or also known as levomenol, (-)-alpha-Bisabolol is found in fats and oils. (-)-alpha-Bisabolol is isolated from essential oil of Matricaria chamomilla (German chamomile) (-)-alpha-Bisabolol belongs to the family of …

Kategori:
Biological ProductsComplex MixturesLipids +7
Waktu Paruh-
Vol. DistribusiTo demonstrate the …
Klirens-
Genetik -
Levomenthol Approved DB00825
small molecule | CAS: 2216-51-5

Menthol is a covalent organic compound made synthetically or obtained from peppermint or other mint oils. Forming clear or white waxy, crystalline substance, menthol is typically solid at room temperature. (-)-Menthol is the naturally-occurring and main form …

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntipruritics +16
Target Protein:
Transient receptor potential cation channel subfamily M member 8Transient receptor potential cation channel subfamily A member 1Transient receptor potential cation channel subfamily V member 3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levomethadone DB13515
small molecule | CAS: 125-58-6

Deskripsi belum tersedia.

Kategori:
Drugs Used in Addictive DisordersDrugs Used in Opioid DependenceNervous System
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levonorgestrel Approved DB00367
small molecule | CAS: 797-63-7

Levonorgestrel (LNG) is a synthetic progestogen similar to [Progesterone] used in contraception and hormone therapy.[A181988,T659] Also known as Plan B, it is used as a single agent in emergency contraception, and as a hormonal contraceptive released from an …

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +23
Target Protein:
Progesterone receptor3-oxo-5-alpha-steroid 4-dehydrogenase 1Estrogen receptor +3
Waktu ParuhThe elimination hal…
Vol. DistribusiOne pharmacokinetic…
KlirensClearance was found…
Genetik -
small molecule | CAS: 1390631-57-8

Lexaptepid pegol has been used in trials studying the treatment of Anemia, Inflammation, Chronic Diseases, End Stage Renal Disease, and Anemia of Chronic Disease.

Kategori:
Anti-Inflammatory AgentsNucleic Acids, Nucleotides, and NucleosidesNucleotides +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LGD-6972 DB14779
small molecule | CAS: 1207989-09-0

LGD-6972 is under investigation in clinical trial NCT01919684 (Study to Evaluate Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of LGD-6972 in Healthy Subjects and Subjects With Type 2 Diabetes Mellitus).

Kategori:
Acids, CarbocyclicAlkanesAlkanesulfonic Acids +7
Target Protein:
Glucagon receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LGH-447 DB14943
small molecule | CAS: 1210608-43-7

LGH-447 is under investigation in clinical trial NCT02160951 (Dose Escalation Study of LGH447 in Japanese Patients With Relapsed and/or Refractory Hematologic Malignancies).

Target Protein:
Serine/threonine-protein kinase pim-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Licogliflozin DB15048
small molecule | CAS: 1291094-73-9

Licogliflozin is under investigation in clinical trial NCT03320941 (A Dose-finding Study to Evaluate the Change in Weight After Treatment With LIK066 in Japanese Patients With Obesity).

Kategori:
AlcoholsBlood Glucose Lowering AgentsCarbohydrates +2
Target Protein:
Sodium/glucose cotransporter 1Sodium/glucose cotransporter 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1401812-88-1

Lifastuzumab vedotin is under investigation in clinical trial NCT01363947 (Safety and Pharmacokinetics of Escalating Doses of DNIB0600A in Participants With Non-Small Cell Lung Cancer (NSCLC) and Platinum Resistant Ovarian Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lifibrol DB12448
small molecule | CAS: 96609-16-4

Lifibrol has been used in trials studying the basic science of Hyperlipoproteinemia and Hypercholesterolemia.

Kategori:
Acids, CarbocyclicAlcoholsBenzene Derivatives +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ligustrazine DB19074
small molecule | CAS: 1124-11-4

Ligustrazine is under investigation in clinical trial NCT05942352 (Clinical Study of Ligustrazine in Treating Alcohol Addiction).

Kategori:
Antiplatelet agentsCardiovascular AgentsVasodilating Agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Limaprost DB09211
small molecule | CAS: 74397-12-9

Limaprost (as Limaprost alfadex; CAS number 88852-12-4) is an oral prostaglandin E1 analog. Prostaglandins act on a variety of cells such as vascular smooth muscle cells causing constriction or dilation, on platelets causing aggregation or disaggregation and …

Kategori:
AnticoagulantsAutacoidsBiological Factors +11
Target Protein:
Prostaglandin E2 receptor EP2 subtypeProstaglandin E2 receptor EP1 subtypeProstaglandin E2 receptor EP3 subtype +1
Waktu ParuhThe mean half life …
Vol. Distribusi-
KlirensMean total clearanc…
Genetik -
Linaclotide Approved DB08890
small molecule | CAS: 851199-59-2

Linaclotide is a synthetic 14-amino acid cyclic peptide [A260271] and first-in-class guanylate cyclase-C (G-CC) agonist.[A260271, L47211] Linaclotide is structurally related to human guanylin and uroguanylin, paracrine peptide hormones that are endogenous act…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsDrugs for Constipation +7
Target Protein:
Guanylyl cyclase C
Waktu ParuhThere is no availab…
Vol. DistribusiGiven that linaclot…
KlirensNo information is a…
Genetik -
Linagliptin Approved DB08882
small molecule | CAS: 668270-12-0

Linagliptin is a DPP-4 inhibitor developed by Boehringer Ingelheim for the treatment of type II diabetes [L9557]. Linagliptin differs from other DPP-4 inhibitors in that it has a non-linear pharmacokinetic profile, is not primarily eliminated by the renal sys…

Kategori:
Agents causing angioedemaAlimentary Tract and MetabolismBlood Glucose Lowering Agents +24
Target Protein:
Dipeptidyl peptidase 4
Waktu ParuhThe terminal half l…
Vol. DistribusiA single intravenou…
KlirensTotal clearance of …
Genetik -
Linezolid Approved DB00601
small molecule | CAS: 165800-03-3

Linezolid is a synthetic antibiotic which is used for the treatment of infections caused by aerobic Gram-positive bacteria. Its effects are bacteriostatic against both enterococci and staphylococci and bactericidal against most isolates of streptococci.[L3296…

Kategori:
AcetamidesAcetatesAcids, Acyclic +22
Target Protein:
23S ribosomal RNA
Waktu ParuhThe elimination hal…
Vol. DistribusiAt steady-state, th…
KlirensTotal clearance of …
Genetik -
Linoleic acid Approved DB14104
small molecule | CAS: 60-33-3

Deskripsi belum tersedia.

Kategori:
Fatty AcidsFatty Acids, EssentialFatty Acids, Omega-6 +3
Target Protein:
Fatty acid-binding protein, adipocyte
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 20196-64-9

Liothyronine I-131 has been used in trials studying the treatment of Tricuspid Atresia and Heart Defects, Congenital.

Kategori:
Thyroxine-binding globulin substrates
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lipoic acid Approved DB00166
small molecule | CAS: 1200-22-2

A vitamin-like antioxidant.

Kategori:
Alimentary Tract and MetabolismAntioxidantsBiological Factors +15
Target Protein:
Lipoyl amidotransferase LIPT1, mitochondrialSodium-dependent multivitamin transporterLipoyl synthase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lipotecan DB17385
small molecule | CAS: 1432468-79-5

Deskripsi belum tersedia.

Kategori:
Alkaloids
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 8046-19-3

Deskripsi belum tersedia.

Kategori:
Biological ProductsComplex MixturesPharmaceutical Preparations +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lisavanbulin DB15224
small molecule | CAS: 1263384-43-5

Lisavanbulin is under investigation in clinical trial NCT02895360 (Phase 1/2a Study of BAL101553 as 48-hour Infusions in Patients With Advanced Solid Tumors or Recurrent Glioblastoma).

Kategori:
Antineoplastic AgentsAntineoplastic Agents, ImmunologicalHeterocyclic Compounds, Fused-Ring +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lisdexamfetamine Approved DB01255
small molecule | CAS: 608137-32-2

Lisdexamfetamine is a prodrug of [dextroamphetamine], a central nervous system stimulant known as d-amphetamine,[A40246] covalently attached to the naturally occurring amino acid L-lysine.[A2230] Lisdexamfetamine is the first chemically formulated prodrug sti…

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAmines +17
Target Protein:
Trace amine-associated receptor 1
Waktu ParuhPlasma concentratio…
Vol. DistribusiDextroamphetamine, …
Klirens-
Genetik -
Lisofylline DB12406
small molecule | CAS: 100324-81-0

Lisofylline has been investigated for the treatment of Type 1 Diabetes Mellitus.

Kategori:
Adjuvants, ImmunologicAnalgesicsAnalgesics, Non-Narcotic +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 29126-50-9

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicDermatologicalsDicarboxylic Acids +2
Target Protein:
Inositol monophosphatase 2Inositol monophosphatase 1Glycogen synthase kinase-3 beta +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Livmoniplimab DB18939
biotech | CAS: 2412004-88-5

Livmoniplimab is under investigation in clinical trial NCT06109272 (A Study to Assess the Dose, Adverse Events, and Change in Disease Activity of Livmoniplimab as an Intravenous (IV) Solution in Combination With Budigalimab as an IV Solution in Adult Particip…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LM-030 DB18283
small molecule | CAS: 1122484-55-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lobucavir DB12531
small molecule | CAS: 127759-89-1

Lobucavir has been used in trials studying the treatment of HIV Infections and Cytomegalovirus Infections.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +10
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lodoxamide Approved DB06794
small molecule | CAS: 53882-12-5

Lodoxamide is a mast-cell stabilizer for topical administration into the eye. Mast-cell stabilizers, first one approved being cromolyn sodium, are used in treatment of ocular hypersensitivity reactions such as vernal conjunctivitis. These conditions often req…

Kategori:
Acids, AldehydicAlcoholsAmino Acids +13
Waktu ParuhElimination half-li…
Vol. Distribusi-
Klirens-
Genetik -
Lometrexol DB12769
small molecule | CAS: 106400-81-1

Lometrexol has been used in trials studying the treatment of Lung Cancer, Drug/Agent Toxicity by Tissue/Organ, and Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
AntimetabolitesAntineoplastic AgentsCoenzymes +9
Target Protein:
Dihydrofolate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lomitapide Approved DB08827
small molecule | CAS: 182431-12-5

Lomitapide is a microsomal triglyceride transfer protein (MTP) inhibitor used in homozygous familial hypercholesterolemia (HoFH) patients. It is marketed under the name Juxtapid (R).

Kategori:
Cytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Inhibitors +17
Target Protein:
Microsomal triglyceride transfer protein large subunit
Waktu ParuhLomitapide half-lif…
Vol. DistribusiThe steady state vo…
Klirens-
Genetik -
Lomustine Approved DB01206
small molecule | CAS: 13010-47-4

An alkylating agent of value against both hematologic malignancies and solid tumors.

Kategori:
Alkylating ActivityAlkylating DrugsAmides +17
Target Protein:
DNAStathmin-4
Waktu ParuhApproximately 94 mi…
Vol. Distribusi-
Klirens-
Genetik -
Lomvastomig DB19060
biotech | CAS: 2648840-52-0

Lomvastomig is under investigation in clinical trial NCT04785820 (A Study of Lomvastomig (RO7121661) and Tobemstomig (RO7247669) Compared With Nivolumab in Participants With Advanced or Metastatic Squamous Cell Carcinoma of the Esophagus).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lonaprisan DB16221
small molecule | CAS: 211254-73-8

Lonaprisan is under investigation in clinical trial NCT00555919 (ZK 230211 in Postmenopausal Woman With Metastatic Breast Cancer).

Kategori:
EstranesFused-Ring CompoundsHydrocarbons, Fluorinated +2
Target Protein:
Progesterone receptorGlucocorticoid receptorAndrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lonoctocog alfa Approved DB13998
biotech | CAS: 1388129-63-2

Deskripsi belum tersedia.

Kategori:
Hemostatics
Target Protein:
Coagulation factor XCoagulation factor IXvon Willebrand factor +8
Waktu Paruh8.4-19.3 hrs
Vol. Distribusi-
Klirens* 4.1 mL/h•kg [Prev…
Genetik -
small molecule | CAS: 106900-12-3

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAntidiarrhealsAntidiarrheals, Intestinal Antiinflammatory/antiinfective Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lopinavir Approved DB01601
small molecule | CAS: 192725-17-0

Lopinavir is an antiretroviral protease inhibitor used in combination with other antiretrovirals in the treatment of HIV-1 infection.[L11163] Lopinavir is marketed and administered exclusively in combination with [ritonavir] - this combination, first marketed…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +42
Target Protein:
Pol polyprotein
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe estimated appar…
Genetik -
Lorlatinib Approved DB12130
small molecule | CAS: 1454846-35-5

Lorlatinib is a third-generation ALK tyrosine kinase inhibitor (TKI) for patients with ALK-positive metastatic non-small cell lung cancer[L39905] which was first approved by the US FDA in November of 2018. It was subsequently approved by the EMA in 2019 for t…

Kategori:
AmidesAminesAnaplastic lymphoma kinase (ALK) inhibitors +31
Target Protein:
Proto-oncogene tyrosine-protein kinase ROSALK tyrosine kinase receptor
Waktu ParuhThe mean plasma hal…
Vol. DistribusiThe mean (CV%) stea…
KlirensThe mean oral clear…
Genetik -
biotech | CAS: 1008106-64-6

Lorvotuzumab mertansine has been used in trials studying the treatment of SCLC, Leukemia, Ovarian Cancer, Multiple Myeloma, and Merkel Cell Carcinoma, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAntibodies +29
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Losmapimod DB12270
small molecule | CAS: 585543-15-3

Losmapimod has been investigated for the prevention of Chronic Obstructive Pulmonary Disease.

Kategori:
Cycloparaffinsp38 Mitogen-Activated Protein KinasesProtein Kinase Inhibitors
Target Protein:
Mitogen-activated protein kinase 14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Loteprednol Approved DB00873
small molecule | CAS: 129260-79-3

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesAndrostadienesAndrostanes +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lovotibeglogene autotemcel Approved DB18680
biotech

Lovotibeglogene autotemcel consists of autologous hematopoietic stem and progenitor cells transduced with the BB305 lentiviral vector encoding a modified ?-globin gene. Specifically, lovotibeglogene autotemcel provides a functional copy of a modified beta-glo…

Kategori:
Autologous Cultured CellAutologous Hematopoietic Stem Cell-Based Gene TherapyGenetic Therapy
Target Protein:
Hemoglobin subunit beta
Waktu ParuhLovotibeglogene aut…
Vol. DistribusiLovotibeglogene aut…
KlirensLovotibeglogene aut…
Genetik -
Loxicodegol DB14146
small molecule | CAS: 1211231-76-3

Loxicodegol was developed by Nektar Therapeutics as an opioid analgesic with low abuse potential for the treatment of chronic pain [L3263]. The lack of abuse potential is believed to be due to the drug's slow rate of entry into brain, a unique characteristic …

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingOpiate Alkaloids +1
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu ParuhLoxicodegol has a h…
Vol. DistribusiLoxicodegol has a s…
KlirensLoxicodegol has a c…
Genetik -
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