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11793

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8607 (73.0%)
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6418 (54.4%)
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11793 (100.0%)

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Halaman 34 / 236
Adrafinil DB08925
small molecule | CAS: 63547-13-7

Adrafinil is a mild central nervous system stimulating drug typically employed to relieve excessive sleepiness and inattention in geriatric patients. It is also been used off-label to prevent fatigue or falling asleep for extended periods of time. Adrafinil d…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-Agonists +10
Waktu Paruh-
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Adrenalone DB13394
small molecule | CAS: 99-45-6

Deskripsi belum tersedia.

Kategori:
AlcoholsAlimentary Tract and MetabolismAmines +16
Waktu Paruh-
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Adrenomedullin DB19102
biotech | CAS: 154835-90-2

Adrenomedullin is under investigation in clinical trial NCT06072118 (Adrenomedullin for CADASIL).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Asthmatic AgentsAntihypertensive Agents +13
Waktu Paruh-
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ADU-S100 DB14722
small molecule | CAS: 1638241-89-0

ADU-S100 (MIW815) is a synthetic cyclic dinucleotide (CDN) agonist (activator) of Stimulator of Interferon Genes (STING), a receptor crucial to activate the innate (endogenous) immune system. ADU-S100 (MIW815) activates all known human and mouse STINGs, and e…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotides
Target Protein:
Stimulator of interferon genes protein
Waktu Paruh-
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Aducanumab Approved DB12274
biotech | CAS: 1384260-65-4

Aducanumab, or BIIB037, is a monoclonal IgG1 antibody that targets extracellular amyloid-? plaques in the brain; similar to [gantenerumab], [bapineuzumab] and [solanezumab].[A235668,A235730] Aducanumab is a recombinant antibody derived from patients with slow…

Kategori:
Alzheimer Disease, drug therapyAmino Acids, Peptides, and ProteinsAmyloid Beta-directed Antibodies +11
Target Protein:
Amyloid-beta precursor protein
Waktu ParuhThe terminal half l…
Vol. DistribusiThe volume of distr…
KlirensA 10 mg/kg intraven…
Genetik -
ADVM-062 DB18341
biotech

ADVM-062 is an adeno-associated virus vector carrying complementary deoxyribonucleic acid encoding the human long-wave-sensitive opsin 1 (AAV.7m8-L-opsin)

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ADX-10061 DB05419
small molecule | CAS: 128022-68-4

ADX10061 is a potent, selective antagonist of the dopamine D1 receptor. It is developed by Addex Pharmaceuticals for the treatment of nicotine dependence.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Neuron-specific vesicular protein calcyon
Waktu Paruh-
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ADXS-31164 DB17325
biotech

Deskripsi belum tersedia.

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Aedes taeniorhynchus Approved DB10691
biotech

Aedes taeniorhynchus allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
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AEE-788 DB12558
small molecule | CAS: 497839-62-0

AEE788 has been used in trials studying the treatment of Cancer, Glioblastoma Multiforme, and Brain and Central Nervous System Tumors.

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, Vascular Endothelial Growth Factor, antagonists & inhibitors
Target Protein:
Fibroblast growth factor receptor 2Fibroblast growth factor receptor 3
Waktu Paruh-
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AEG35156 DB06184
small molecule

A second-generation synthetic antisense oligonucleotide with potential antineoplastic activity. AEG35156 selectively blocks the cellular expression of X-linked inhibitor of apoptosis protein (XIAP), a pivotal inhibitor of apoptosis that is overexpressed in ma…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
E3 ubiquitin-protein ligase XIAP
Waktu Paruh-
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AEM-28 DB17642
biotech

AEM-28 is a 28 amino acid mimetic of apolipoprotein E being investigated for lipid disorders, such as homozygous familial hypercholesterolemia. It possesses anti-inflammatory properties.[A258764]

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AEM-28-14 DB17643
biotech

AEM-28-14 is an analog of [AEM-28], an apolipoprotein E mimetic peptide, with a 400 percent greater cholesterol-lowering efficacy and a several-fold increase in drug tolerability.[L45909] It is being investigated for lipid disorders such as homozygous familia…

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AEOL-10150 DB05874
small molecule | CAS: 286475-30-7

AEOL 10150 is developed by Aeolus as a therapeutic agents based on its proprietary small molecule catalytic antioxidants.

Kategori:
AntioxidantsBiological FactorsCoordination Complexes +3
Target Protein:
Superoxide dismutase [Cu-Zn]
Waktu Paruh-
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AF-710B DB16911
small molecule | CAS: 1235733-73-9

Deskripsi belum tersedia.

Kategori:
Sulfur CompoundsThiazoles
Target Protein:
Muscarinic acetylcholine receptor M1Sigma non-opioid intracellular receptor 1
Waktu Paruh-
Vol. Distribusi-
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Afabicin DB15268
small molecule | CAS: 1518800-35-5

Afabicin is under investigation in clinical trial NCT03723551 (Study to Assess Safety, Tolerability and Efficacy of Afabicin in The Treatment of Participants With Bone or Joint Infection Due to Staphylococcus).

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
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Afamelanotide Approved DB04931
small molecule | CAS: 75921-69-6

Afamelanotide is a first-in-class, synthetic, 13-amino acid peptide analogue of the endogenous alpha melanocyte-stimulating hormone (?-MSH).[L9086] It differs structurally from its endogenous counterpart by only two amino acids - these structural differences …

Kategori:
Amino Acids, Peptides, and ProteinsCompounds used in a research, industrial, or household settingDermatologicals +11
Target Protein:
Melanocortin receptor 4Melanocyte-stimulating hormone receptor
Waktu ParuhThe half-life of af…
Vol. DistribusiThe apparent volume…
KlirensData regarding plas…
Genetik -
Afatinib Approved DB08916
small molecule | CAS: 850140-72-6

Afatinib is a 4-anilinoquinazoline tyrosine kinase inhibitor in the form of a dimaleate salt available as Boehringer Ingelheim's brand name Gilotrif [FDA Label]. For oral use, afatinib tablets are a first-line (initial) treatment for patients with metastatic …

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +11
Target Protein:
Epidermal growth factor receptorReceptor tyrosine-protein kinase erbB-2Receptor tyrosine-protein kinase erbB-4
Gen Terkait:
EGFR EGFR EGFR
Waktu ParuhAfatinib is elimina…
Vol. DistribusiThe volume of distr…
KlirensThe apparent total …
Genetik 3 Varian
Afegostat DB04545
small molecule | CAS: 169105-89-9

Deskripsi belum tersedia.

Kategori:
CarbohydratesGlycoside Hydrolases, antagonists & inhibitorsImines +2
Target Protein:
Lysosomal acid glucosylceramidaseEndoglucanase 5ABeta-glucosidase A +1
Waktu Paruh-
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Genetik -
Afelimomab DB04956
biotech | CAS: 156227-98-4

Afelimomab (also known as Fab 2 or MAK 195F) is an anti-TNF-? monoclonal antibody. Administration of 195F reduces the concentration of interleukin-6 in patients with sepsis.

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntibodies +11
Target Protein:
Tumor necrosis factor
Waktu Paruh44.7 hours
Vol. Distribusi-
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Affitope AD01 DB06086
biotech

Affitope AD01 is an investigational drug developed for immunization to treat Alzheimer's Disease. AD01 is a short peptide (7 amino acids in length) that induces Aß-targeting antibodies, therefore lowering Aß aggregates.

Target Protein:
Amyloid-beta precursor protein
Waktu Paruh-
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Aficamten DB18490
small molecule | CAS: 2364554-48-1

Deskripsi belum tersedia.

Target Protein:
Myosin-binding protein C, cardiac-type
Waktu Paruh-
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Afimetoran DB16580
small molecule | CAS: 2171019-55-7

Afimetoran is an immunomodulator and an antagonist of toll-like receptors 7 and 8.[L32018, L32023] It is also is under investigation in clinical trial NCT04269356 (Study to Assess the Way the Body Absorbs, Distributes, Breaks Down and Eliminates Radioactive B…

Target Protein:
Toll-like receptor 7Toll-like receptor 8
Waktu Paruh-
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Afimoxifene DB04468
small molecule | CAS: 68392-35-8

Afimoxifene (4-Hydroxytamoxifen, trade name TamoGel) is a new estrogen inhibitor under investigation for a variety of estrogen-dependent conditions, including cyclic breast pain and gynecomastia. TamoGel is formulated using Enhanced Hydroalcoholic Gel (EHG) T…

Kategori:
AndrostanesAndrostenesAndrostenols +12
Target Protein:
Estrogen receptorTrefoil factor 1Steroid hormone receptor ERR1 +4
Waktu Paruh-
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Aflibercept Approved DB08885
biotech | CAS: 862111-32-8

Aflibercept is a recombinant protein composed of the binding domains of two human vascular endothelial growth factor (VEGF) receptors, VEGFR1 and VEGFR2, fused with the Fc region of human immunoglobulin gamma 1 (IgG1).[A261130] Structurally, Aflibercept is a …

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +16
Target Protein:
Vascular endothelial growth factor A, long formPlacenta growth factorVascular endothelial growth factor B
Waktu ParuhFor the intravitrea…
Vol. DistribusiThe volume of distr…
KlirensFollowing an hour o…
Genetik -
AFM-13 DB17404
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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AFN-1252 DB12658
small molecule | CAS: 620175-39-5

AFN-1252 has been used in trials studying the treatment of Cellulitis, Burn Infection, Wound Infection, Cutaneous Abscess, and Skin and Subcutaneous Tissue Bacterial Infections.

Kategori:
Heterocyclic Compounds, Fused-RingPyrans
Waktu Paruh-
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Genetik -
Afoxolaner DB11369
small molecule | CAS: 1093861-60-9

Deskripsi belum tersedia.

Waktu Paruh-
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Afuresertib DB11648
small molecule | CAS: 1047644-62-1

Afuresertib has been used in trials studying the treatment of Cancer and Neoplasms, Haematologic.

Kategori:
AminesPolyaminesSulfur Compounds
Target Protein:
RAC-alpha serine/threonine-protein kinase
Waktu Paruh-
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AG-24322 DB13035
small molecule | CAS: 837364-57-5

AG-024322 has been used in trials studying the treatment of Neoplasms and Lymphoma, Non-Hodgkin.

Kategori:
CDC2 Protein Kinase, antagonists & inhibitorsCyclin-Dependent Kinase 2, antagonists & inhibitorsHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Cyclin-dependent kinase 2Cyclin-dependent kinase 4Cyclin-dependent kinase 1
Waktu Paruh-
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AG-702 DB05836
biotech

AG-702 is a recombinant human heat shock protein also known as stress protein. It is also known as HSPs, which are a group of proteins that are induced when a cell undergoes various types of environmental stresses like heat, cold and oxygen deprivation. HSPs …

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AG0301-COVID19 DB15856
biotech

AG0301-COVID19 is a vaccine candidate developed by AnGes Inc. and Osaka University. The candidate is a plasmid DNA vaccine developed using an intradermal gene transfer method targeting the SARS-CoV-2 spike protein. The gene transfer method increases the effic…

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AG0302-COVID19 DB16435
biotech

Sponsored by Anges, Inc. in Japan, the AG0302-COVID19 is a DNA-based vaccine that recently completed Phase I/II trials (NCT04527081)[A226813, L30548].

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AGA2115 DB17840
biotech

AGA2115 is a humanized bispecific antibody neutralizing both sclerostin and Dickkopf-1. Developed by Angitia Biopharmaceuticals, AGA2115 is being investigated for the treatment of osteogenesis imperfect.[L46646]

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Agalsidase alfa Approved DB15874
biotech

Agalsidase alfa is a recombinant human ?-galactosidase A similar to [agalsidase beta]. While patients generally do not experience a clinically significant difference in outcomes between the two drugs, some patients may experience greater benefit with agalsida…

Kategori:
Alimentary Tract and Metabolismalpha-Galactosidase, antagonists & inhibitorsAmino Acids, Peptides, and Proteins +9
Target Protein:
Globotriaosylceramide
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance for d…
Genetik -
Agalsidase beta Approved DB00103
biotech

Agalsidase beta is a recombinant human ?-galactosidase A similar to [agalsidase alfa]. While patients generally do not experience a clinically significant difference in outcomes between the two drugs, some patients may experience greater benefit with agalsida…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsEnzymes +7
Target Protein:
Globotriaosylceramide
Waktu Paruhagalsidase beta has…
Vol. DistribusiA 1 mg/kg dose of a…
KlirensA 1 mg/kg dose of a…
Genetik -
small molecule | CAS: 910562-20-8

Aganepag isopropyl is under investigation in clinical trial NCT01110499 (Safety and Efficacy of AGN-210961 Ophthalmic Solution Compared With Bimatoprost Ophthalmic Solution in Patients With Glaucoma or Ocular Hypertension).

Waktu Paruh-
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Aganirsen DB15369
biotech | CAS: 1146887-67-3

Aganirsen is under investigation in clinical trial NCT02947867 (Trial of Aganirsen in iCRVO Patients at Risk of Developing NVG).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
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Agatolimod DB15018
biotech | CAS: 207623-20-9

Agatolimod is under investigation in clinical trial NCT00471471 (Vaccine Therapy in Treating Patients With Recurrent Stage III or Stage IV Melanoma That Cannot Be Removed by Surgery).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Waktu Paruh-
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Agerafenib DB15068
small molecule | CAS: 1188910-76-0

Agerafenib is under investigation in clinical trial NCT03052569 (Expanded Access to RXDX-105 for Cancers With RET Alterations).

Kategori:
AmidesBenzene DerivativesEnzyme Inhibitors +3
Target Protein:
Proto-oncogene tyrosine-protein kinase receptor RetSerine/threonine-protein kinase B-raf
Waktu Paruh-
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Genetik -
AGF-94 DB18023
small molecule | CAS: 136784-51-5

Deskripsi belum tersedia.

Waktu Paruh-
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AGG-523 DB15460
small molecule | CAS: 920289-29-8

AGG-523 is under investigation in clinical trial NCT00380900 (Study Evaluating the Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of Multiple Ascending Doses in Healthy subjects and in subjects with osteoarthritis).

Target Protein:
A disintegrin and metalloproteinase with thrombospondin motifs 5
Waktu Paruh-
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AGI-1096 DB05840
small molecule

AGI-1096 is a novel oral antioxidant and selective anti-inflammatory agent that is being developed to address the accelerated inflammation of grafted blood vessels, known as transplant arteritis, common in chronic organ transplant rejection.

Kategori:
Acids, AcyclicBenzene DerivativesFatty Acids +2
Waktu Paruh-
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AGI-134 DB19005
small molecule | CAS: 1821461-84-0

AGI-134 is under investigation in clinical trial NCT03593226 (Study to Evaluate Safety & Tolerability of AGI-134 in Solid Tumour).

Waktu Paruh-
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AGIL-FA DB16973
biotech

Deskripsi belum tersedia.

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biotech | CAS: 1621271-62-2

Aglatimagene besadenovec is under investigation in clinical trial NCT00638612 (AdV-tk Therapy With Surgery and Chemoradiation for Pancreas Cancer (PaTK01)).

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Agmatine DB08838
small molecule | CAS: 306-60-5

Agmantine is a natural metabolite of the amino acid arginine. It is formed when arginine is decarboxylated by the enzyme arginine decarboxylase and is found naturally in ragweed pollen, ergot fungi, octopus muscle, herring sperm, sponges, and the mammalian br…

Kategori:
Agents causing hyperkalemiaAmidinesAntiarrhythmic agents +12
Target Protein:
Alpha-2C adrenergic receptorNischarinAcetylcholine receptor subunit alpha +4
Waktu Paruh-
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AGN-201904 DB13135
small molecule | CAS: 651729-53-2

Agn 201904 has been used in trials studying the prevention of Peptic Ulcer.

Kategori:
2-PyridinylmethylsulfinylbenzimidazolesBenzimidazolesHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
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Agomelatine Approved DB06594
small molecule | CAS: 138112-76-2

Agomelatine is structurally closely related to melatonin. Agomelatine is a potent agonist at melatonin receptors and an antagonist at serotonin-2C (5-HT2C) receptors, tested in an animal model of depression. Agomelatine was developed in Europe by Servier Labo…

Kategori:
AcetatesAcids, AcyclicAmides +15
Target Protein:
5-hydroxytryptamine receptor 2CMelatonin receptor type 1AMelatonin receptor type 1B
Waktu Paruh<2 hours
Vol. Distribusi-
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AGRO100 DB04998
biotech | CAS: 301636-59-9

AGRO100 is an oligonucleotide that functions as an aptamer and binds to nucleolin, a protein found intranuclear in all cells, but uniquely expressed on the surface of tumor cells. Such binding leads to internalization of the complex, and a strong anti-prolife…

Kategori:
Aptamers, NucleotideNucleic Acids, Nucleotides, and NucleosidesNucleotides +2
Target Protein:
NF-kappa-B essential modulator
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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