Hasil Filter

12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

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Hasil Pencarian (12560)

Halaman 34 / 252
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cap-specific mRNA (nucleoside-2'-O-)-methyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 104809-16-7

Deskripsi belum tersedia.

Target Protein:
m7GpppX diphosphataseCap-specific mRNA (nucleoside-2'-O-)-methyltransferaseEukaryotic translation initiation factor 4E
Waktu Paruh-
Vol. Distribusi-
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Genetik -
7-methyl-GpppA DB01649
small molecule

Deskripsi belum tersedia.

Target Protein:
m7GpppX diphosphataseEukaryotic translation initiation factor 4E
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Eukaryotic translation initiation factor 4E
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
m7GpppX diphosphataseRNA-directed RNA polymerase lambda-3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Nitric oxide synthase 3
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Focal adhesion kinase 1
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Monoamine Oxidase A Inhibitors for interaction with Monoamine Oxidase A substrates
Target Protein:
Amine oxidase [flavin-containing] AAmine oxidase [flavin-containing] B
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Amine oxidase [flavin-containing] B
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Bifunctional epoxide hydrolase 2
Waktu Paruh-
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Genetik -
small molecule | CAS: 141099-60-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Integrin alpha-L
Waktu Paruh-
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Genetik -
small molecule | CAS: 566-27-8

Deskripsi belum tersedia.

Kategori:
CholestanesCholestenesFused-Ring Compounds +5
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7MW3711 DB19298
biotech

Developed by Mabwell, 7MW3711 is an antibody-drug conjugate targeting B7-H3.[L50918,L50923]

Waktu Paruh-
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Genetik -
small molecule | CAS: 227458-60-8

Deskripsi belum tersedia.

Target Protein:
Glycogen phosphorylase, muscle form
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Glycogen phosphorylase, muscle form
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Phenylethanolamine N-methyltransferase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Heat shock protein HSP 90-alpha
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Heat shock protein HSP 90-alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Heat shock protein HSP 90-alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Heat shock protein HSP 90-alpha
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Heat shock protein HSP 90-betaHeat shock protein HSP 90-alpha
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Urokinase-type plasminogen activator
Waktu Paruh-
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Genetik -
small molecule | CAS: 19410-53-8

Deskripsi belum tersedia.

Target Protein:
Dihydroneopterin aldolase
Waktu Paruh-
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Genetik -
8-azaguanine DB01667
small molecule | CAS: 134-58-7

8-azaguanine is one of the early purine analogs showing antineoplastic activity. It functions as an antimetabolite and is easily incorporated into ribonucleic acids.

Kategori:
AntimetabolitesAntineoplastic AgentsAza Compounds +8
Target Protein:
Purine nucleoside phosphorylase
Waktu Paruh-
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Genetik -
8-azaxanthine DB01875
small molecule | CAS: 1468-26-4

Deskripsi belum tersedia.

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingPurines +1
Target Protein:
Uric acid degradation bifunctional protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Heat shock protein HSP 90-alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Heat shock protein HSP 90-alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Wee1-like protein kinase
Waktu Paruh-
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small molecule

Deskripsi belum tersedia.

Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4BAdenosine 5'-monophosphoramidase HINT1
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
S-adenosylmethionine synthase
Waktu Paruh-
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Genetik -
small molecule | CAS: 34408-14-5

8-Chloroadenosine is under investigation in clinical trial NCT02509546 (8-chloroadenosine in Treating Patients With Relapsed or Refractory Acute Myeloid Leukemia).

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
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Genetik -
small molecule | CAS: 85-18-7

8-Chlorotheophylline is a stimulant drug of the xanthine chemical class, with physiological effects similar to caffeine. Its main use is in combination with [Diphenhydramine] as the antiemetic drug [Dimenhydrinate]. The stimulant properties of 8-chlorotheophy…

Kategori:
AlkaloidsCytochrome P-450 CYP1A2 SubstratesCytochrome P-450 Substrates +4
Target Protein:
Adenosine receptor A2a
Waktu Paruh-
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Genetik -
small molecule | CAS: 41325-63-7

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
small molecule | CAS: 88847-89-6

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicDeoxyguanosineDeoxyribonucleosides +7
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small molecule

Deskripsi belum tersedia.

Target Protein:
P-proteinChorismate mutase AroHSecreted chorismate mutase
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Thiostrepton50S ribosomal protein L11
Waktu Paruh-
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8-iodo-guanine DB02985
small molecule

Deskripsi belum tersedia.

Target Protein:
Purine nucleoside phosphorylasePurine nucleoside phosphorylase
Waktu Paruh-
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Genetik -
8-oxo-dGMP DB02023
small molecule | CAS: 127027-50-3

Deskripsi belum tersedia.

Kategori:
Guanine NucleotidesHeterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
8-oxo-dGTP diphosphatase
Waktu Paruh-
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9(S)-HODE DB07302
small molecule | CAS: 73543-67-6

Deskripsi belum tersedia.

Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
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small molecule | CAS: 78111-17-8

A specific inhibitor of phosphoserine/threonine protein phosphatase 1 and 2a. It is also a potent tumor promoter. (Thromb Res 1992;67(4):345-54 & Cancer Res 1993;53(2):239-41)

Target Protein:
Dual specificity protein phosphatase 1Serine/threonine-protein phosphatase PP1-gamma catalytic subunit
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Histone deacetylase 8Histone deacetylase 4Histone deacetylase 1 +4
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Purine nucleoside phosphorylase DeoD-type
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small molecule

9-(4-hydroxybutyl)-N2-phenylguanine is a solid. This compound belongs to the hypoxanthines. These are compounds containing the purine derivative 1H-purin-6(9H)-one. 9-(4-hydroxybutyl)-n2-phenylguanine is known to target thymidine kinase.

Target Protein:
Thymidine kinase, cytosolicThymidine kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Purine nucleoside phosphorylase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Purine nucleoside phosphorylase DeoD-type
Waktu Paruh-
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Genetik -
small molecule | CAS: 143205-42-9

9-(N-methyl-L-isoleucine)-cyclosporin A (NIM811) has been used in trials studying the treatment of Chronic Hepatitis C Genotype-1 Relapse.

Kategori:
Amino Acids, Peptides, and ProteinsCyclosporinsImmunosuppressive Agents +2
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
CREB-binding protein
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Neuraminidase
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Genetik -
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