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3253

Total database: 17430
Struktur (SMILES)
2451 (75.3%)
Target
1833 (56.3%)
Genomik
35 (1.1%)
Referensi
3253 (100.0%)

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Hasil Pencarian (3253)

Halaman 34 / 66
biotech | CAS: 1469876-18-3

Labetuzumab govitecan has been used in trials studying the treatment of Colon Cancer, Rectal Cancer, and Metastatic Colorectal Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lacnotuzumab DB14928
biotech | CAS: 1831128-32-5

Lacnotuzumab is under investigation in clinical trial NCT01643850 (MCS110 in Patients With Pigmented Villonodular Synovitis (PVNS)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lactic acid Approved DB04398
small molecule | CAS: 50-21-5

A normal intermediate in the fermentation (oxidation, metabolism) of sugar. The concentrated form is used internally to prevent gastrointestinal fermentation. (From Stedman, 26th ed) Sodium lactate is the sodium salt of lactic acid, and has a mild saline tast…

Kategori:
Basic Ointments and ProtectantsGenito Urinary System and Sex HormonesGynecological Antiinfectives and Antiseptics +6
Target Protein:
Bifunctional protein PutANimA-related protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lactitol Approved DB12942
small molecule | CAS: 585-86-4

Lactitol, also known as 4-?-D-galactopyranosyl-D-glucitol, is a sugar alcohol synthesized from [lactose].[A190918] It is used in food manufacturing as a nutritive sweetener and is approximately 35% as sweet as table sugar (i.e. [sucrose]).[A190912] Clinically…

Kategori:
AlcoholsAlimentary Tract and MetabolismCarbohydrates +15
Waktu ParuhThe average half-li…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Ladarixin DB16212
small molecule | CAS: 849776-05-2

Ladarixin is under investigation in clinical trial NCT04628481 (A Study of Oral Ladarixin in New-onset Type 1 Diabetes and a Low Residual ?-Cell Function).

Kategori:
AmidesReceptors, Interleukin-8A, antagonists & inhibitorsSulfones +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Laevulinic Acid DB02239
small molecule | CAS: 123-76-2

Deskripsi belum tersedia.

Target Protein:
Delta-aminolevulinic acid dehydratase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lafutidine DB12770
small molecule | CAS: 118288-08-7

Lafutidine has been investigated in Peptic Ulcer, Community-acquired Pneumonia, and Gastroesophageal Reflux Disease (GERD).

Kategori:
AcetatesAcids, AcyclicAlimentary Tract and Metabolism +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lampalizumab DB11826
biotech | CAS: 1278466-20-8

Lampalizumab has been used in trials studying the treatment of Geographic Atrophy.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Landiolol Approved DB12212
small molecule | CAS: 133242-30-5

Landiolol is a rapid-acting beta-blocker used for rapid ventricular rate control.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Landipirdine DB16214
small molecule | CAS: 1000308-25-7

Landipirdine is under investigation in clinical trial NCT02258152 (SYN120 Study to Evaluate Its Safety, Tolerability and Efficacy in Parkinson's Disease Dementia (SYNAPSE)).

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsSerotonin 5-HT2 Receptor Antagonists +3
Target Protein:
5-hydroxytryptamine receptor 65-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Laninamivir DB12791
small molecule | CAS: 203120-17-6

Laninamivir has been used in trials studying the treatment of Influenza.

Kategori:
Acids, AcyclicAmidinesAmino Sugars +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 203120-46-1

Laninamivir octanoate has been used in trials studying the treatment of Asthma.

Kategori:
Acids, AcyclicAmidinesAmino Sugars +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Laniquidar DB12799
small molecule | CAS: 197509-46-9

Laniquidar has been used in trials studying the treatment of Breast Cancer.

Kategori:
Carbon RadioisotopesDrug Resistance, MultipleHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Phosphatidylcholine translocator ABCB4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lanolin Approved DB11112
small molecule | CAS: 8006-54-0

Lanolin is a yellow fat obtained from sheep's wool. It is used as an emollient, cosmetic, and pharmaceutic aid [L2580]. The US federal code of regulations states that lanolin in the concentration range of 12-50% may be included in over the counter skin ointme…

Kategori:
Basic Ointments and ProtectantsCompounds used in a research, industrial, or household settingCosmetics +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lanopepden DB11912
small molecule | CAS: 1152107-25-9

Lanopepden has been used in trials studying the treatment of Pneumonia, Infections, Bacterial, Skin Diseases, Infectious, and Skin Infections, Bacterial.

Kategori:
AminesAnti-Bacterial AgentsEnzyme Inhibitors +2
Target Protein:
Peptide deformylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lapatinib Approved DB01259
small molecule | CAS: 231277-92-2

Lapatinib is an anti-cancer drug developed by GlaxoSmithKline (GSK) as a treatment for solid tumours such as breast and lung cancer. It was approved by the FDA on March 13, 2007, for use in patients with advanced metastatic breast cancer in conjunction with t…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP2C19 Substrates +22
Target Protein:
Epidermal growth factor receptorEukaryotic elongation factor 2 kinaseReceptor tyrosine-protein kinase erbB-2
Gen Terkait:
HLA-DQA1 HLA-DRB1 HLA-DQB1 +1
Waktu ParuhSingle-dose termina…
Vol. Distribusi-
Klirens-
Genetik 4 Varian
Larotaxel DB12984
small molecule | CAS: 156294-36-9

Larotaxel has been used in trials studying the treatment of Cancer, Metastases, Breast Cancer, Breast Neoplasms, and Pancreatic Neoplasms, among others.

Kategori:
CyclodecanesCycloparaffinsDiterpenes +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Larotrectinib Approved DB14723
small molecule | CAS: 1223403-58-4

Larotrectinib is an orally administered inhibitor of tropomyosin receptor kinase (Trk), a receptor tyrosine kinase activated by neurotrophins which is mutated in a variety of cancer cell types and plays an important role in tumor cell growth and survival.[L49…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +8
Target Protein:
High affinity nerve growth factor receptorBDNF/NT-3 growth factors receptorNT-3 growth factor receptor
Waktu ParuhIn healthy subjects…
Vol. DistribusiFollowing intraveno…
KlirensThe mean clearance …
Genetik -
Latrunculin A DB02621
small molecule | CAS: 76343-93-6

Latrunculin A is an actin binding macrolide purified from the red sea sponge Latrunculia magnifica. It is under investigation for the treatment of cancer. It disrupts actin polymerization, prevents mitotic spindle formation and thus cell replication.

Kategori:
PoriferaSulfur CompoundsThiazoles
Target Protein:
Actin, alpha skeletal muscleGelsolinIota toxin component Ia
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lauric acid Approved DB03017
small molecule | CAS: 143-07-7

Lauric acid is an inexpensive, non-toxic and safe to handle compound often used in laboratory investigations of melting-point depression. Lauric acid is a solid at room temperature but melts easily in boiling water, so liquid lauric acid can be treated with v…

Kategori:
Fatty AcidsLipids
Target Protein:
Toll-like receptor 4LactotransferrinPhospholipase A2, membrane associated +18
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 112-16-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lavendustin A DB16768
small molecule | CAS: 125697-92-9

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesEnzyme InhibitorsTyrosine Kinase Inhibitors
Target Protein:
Epidermal growth factor receptorTyrosine-protein kinase Lck
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lavendustin b DB16760
small molecule | CAS: 125697-91-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lavoltidine DB12884
small molecule | CAS: 76956-02-0

Lavoltidine has been used in trials studying the diagnostic of Reflux, Gastroesophageal and Gastroesophageal Reflux Disease.

Kategori:
Gastric Acid Lowering AgentsHistamine AgentsHistamine Antagonists +2
Target Protein:
Histamine H2 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LAX-101 DB05301
small molecule | CAS: 909712-41-0

LAX-101 treats hungtington’s disease, not just the symptoms but the disease itself. The active molecule in LAX-101 is Eicosapentaenoic Acid (EPA). All molecules of EPA are identical. The molecules of EPA found in LAX-101 are identical to the molecules of EPA …

Target Protein:
Phospholipase D1Caspase-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LB-100 DB15412
small molecule | CAS: 1632032-53-1

LB-100 is under investigation in clinical trial NCT03886662 (A Study of LB-100 in Patients With Low or Intermediate-1 Risk Myelodysplastic Syndromes (MDS)).

Kategori:
Antineoplastic AgentsEnzyme Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LCL-161 DB12085
small molecule | CAS: 1005342-46-0

LCL161 has been used in trials studying the treatment of Leukemia, Neoplasms, Solid Tumors, Breast Cancer, and Ovarian Cancer, among others.

Kategori:
Antineoplastic AgentsProto-Oncogene Proteins c-bcl-2, antagonists & inhibitorsSulfur Compounds
Target Protein:
E3 ubiquitin-protein ligase XIAPBaculoviral IAP repeat-containing protein 2Baculoviral IAP repeat-containing protein 3 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lebrikizumab Approved DB11914
biotech | CAS: 953400-68-5

Lebrikizumab is a monoclonal antibody that binds to IL-13 with high affinity and slow off-rate.[L51374] It binds to a different epitope compared [tralokinumab].[A262874,A262879] On November 17, 2023, lebrikizumab was approved by the EMA under the brand nam…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAmino Acids, Peptides, and ProteinsAntibodies +10
Target Protein:
Interleukin-13
Waktu ParuhThe mean eliminatio…
Vol. DistribusiBased on a populati…
KlirensIn the population P…
Genetik -
Lecanemab Approved DB14580
biotech | CAS: 1260393-98-3

Lecanemab is a recombinant humanized immunoglobulin gamma 1 (IgG1) monoclonal antibody directed against aggregated soluble and insoluble forms of amyloid beta (A?), which are implicated in the pathophysiology of Alzheimer’s disease.[L44537] Lecanemab works to…

Kategori:
Alzheimer DiseaseAlzheimer Disease, drug therapyAmino Acids, Peptides, and Proteins +12
Target Protein:
Amyloid-beta precursor protein
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe mean value (95%…
KlirensThe clearance of le…
Genetik -
Lecozotan DB12540
small molecule | CAS: 434283-16-6

Lecozotan has been used in trials studying the treatment of Alzheimer Disease.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsSerotonin 5-HT1 Receptor Antagonists +3
Target Protein:
5-hydroxytryptamine receptor 15-hydroxytryptamine receptor 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ledipasvir Approved DB09027
small molecule | CAS: 1256388-51-8

Ledipasvir is a direct acting antiviral (DAA) medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized int…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +10
Target Protein:
Genome polyproteinNonstructural protein 5A
Waktu ParuhThe median terminal…
Vol. Distribusi-
Klirens-
Genetik -
Lefamulin Approved DB12825
small molecule | CAS: 1061337-51-6

Lefamulin is a pleuromutilin antibiotic used for the treatment of bacterial community-acquired pneumonia. A pleuromotilin is a more recently developed type of antibiotic that is derived from the fungus, Pleurotus mutilus.[A183206] Lefamulin is available in in…

Kategori:
AcetatesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
50S ribosomal protein L22
Waktu ParuhThe average elimina…
Vol. DistribusiThe average volume …
KlirensThe total body clea…
Genetik -
Leflunomide Approved DB01097
small molecule | CAS: 75706-12-6

Leflunomide is a pyrimidine synthesis inhibitor belonging to the DMARD (disease-modifying antirheumatic drug) class of drugs, which are chemically and pharmacologically very heterogeneous. Leflunomide was approved by FDA and in many other countries (e.g., Can…

Kategori:
AdjuvantsAgents Causing Muscle ToxicityAntineoplastic and Immunomodulating Agents +16
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrialDihydroorotate dehydrogenase (quinone), mitochondrialAryl hydrocarbon receptor +1
Gen Terkait:
CYP1A2
Waktu Paruh2 weeks
Vol. Distribusi* 0.13 L/kg
Klirens-
Genetik 1 Varian
Lemzoparlimab DB17572
biotech | CAS: 2377483-71-9

Lemzoparlimab is under investigation in clinical trial NCT04912063 (Study to Evaluate Adverse Events and Movement of Lemzoparlimab in Body When Used Intravenously (IV) With Azacitidine Subcutaneously or IV and Venetoclax Orally in Participants With Acute Myel…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lenabasum DB12193
small molecule | CAS: 137945-48-3

Ajulemic acid has been used in trials studying the treatment of Cystic Fibrosis, Dermatomyositis, and Diffuse Cutaneous Systemic Sclerosis.

Kategori:
Agents producing tachycardiaCannabinoid Receptor AgonistsCannabinoids and similars +5
Target Protein:
Tumor necrosis factor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lenzilumab DB15148
biotech | CAS: 1229575-09-0

Lenzilumab is under investigation in clinical trial NCT02546284 (Study of Lenzilumab in Previously Treated Patients With Chronic Myelomonocytic Leukemia (CMML)).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Inflammatory AgentsAntibodies +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lepirudin Approved DB00001
biotech | CAS: 138068-37-8

Lepirudin is a recombinant hirudin formed by 65 amino acids that acts as a highly specific and direct thrombin inhibitor.[L41539,L41569] Natural hirudin is an endogenous anticoagulant found in _Hirudo medicinalis_ leeches.[L41539] Lepirudin is produced in yea…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsAntithrombin Proteins +12
Target Protein:
Prothrombin
Waktu ParuhLepirudin has an in…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of le…
Genetik -
Lerisetron DB12964
small molecule | CAS: 143257-98-1

Lerisetron has been used in trials studying the supportive care of Nausea and Vomiting and Testicular Germ Cell Tumor.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leronlimab DB05941
biotech | CAS: 674782-26-4

Leronlimab, or PRO-140, is a human monoclonal antibody developed by CytoDyn.[L12684] It was first described in the literature in 2001.[A3922] This antibody binds to CCR5, which may be useful in treating HIV, cancers, and severely ill COVID-19 patients.[A19284…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-HIV AgentsAnti-Infective Agents +17
Target Protein:
C-C chemokine receptor type 5
Waktu ParuhThe half life of a …
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Lersivirine DB11649
small molecule | CAS: 473921-12-9

Lersivirine has been used in trials studying the treatment of HIV-1.

Kategori:
RNA-Directed DNA Polymerase
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Letermovir Approved DB12070
small molecule | CAS: 917389-32-3

Letermovir recieved approval from the FDA on November 8th, 2017 for use in prophylaxis of cytomegalovirus (CMV) infection in allogeneic hematopoietic stem cell transplant patients.[L1021] It is the first of a new class of CMV anti-infectives called DNA termin…

Kategori:
Acids, AcyclicAnti-Infective AgentsAntiinfectives for Systemic Use +44
Target Protein:
CMV DNA Terminase Complex
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe mean steady sta…
KlirensThe mean clearance …
Genetik -
Letrazuril DB12663
small molecule | CAS: 103337-74-2

Letrazuril has been used in trials studying the treatment of HIV Infections and Cryptosporidiosis.

Kategori:
Nitriles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Letrozole Approved DB01006
small molecule | CAS: 112809-51-5

Letrozole, or CGS 20267, is an oral non-steroidal type II aromatase inhibitor first described in the literature in 1990.[A190543,A1559,L11623,L11626] It is a third generation aromatase inhibitor like [exemestane] and [anastrozole], meaning it does not signifi…

Kategori:
Agents Causing Muscle ToxicityAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +21
Target Protein:
Aromatase
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensThe average clearan…
Genetik -
Leukotriene B4 DB12961
small molecule | CAS: 71160-24-2

Leukotriene B4 has been used in trials studying the treatment of HIV Infections.

Kategori:
Arachidonic AcidsAutacoidsBiological Factors +7
Target Protein:
Leukotriene B4 receptor 1Leukotriene B4 receptor 2Peroxisome proliferator-activated receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leupeptin DB16961
small molecule | CAS: 55123-66-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsCathepsins, antagonists & inhibitorsCysteine Proteinase Inhibitors +4
Target Protein:
Plasmepsin-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leuprolide Approved DB00007
biotech | CAS: 53714-56-0

Leuprolide is a synthetic 9-residue peptide analogue of gonadotropin-releasing hormone (GnRH). Unlike the endogenous decapeptide GnRH, leuprolide contains a single D-amino acid (D-leucyl) residue, which helps to increase its circulating half-life from three t…

Kategori:
Adrenal Cortex HormonesAgents Causing Muscle ToxicityAmino Acids, Peptides, and Proteins +25
Target Protein:
Gonadotropin-releasing hormone receptorProgonadoliberin-1
Waktu ParuhLeuprolide has a te…
Vol. DistribusiLeuprolide has an a…
KlirensLeuprolide administ…
Genetik -
Levacetylmethadol Approved DB01227
small molecule | CAS: 1477-40-3

Levacetylmethadol is a narcotic analgesic with a long onset and duration of action. It is used mainly in the treatment of narcotic dependence. Levacetylmethadol was withdrawn from use in the European Union due to its high risk of QT interval prolongation.…

Kategori:
AnalgesicsAnticholinergic AgentsCentral Nervous System Agents +20
Target Protein:
Mu-type opioid receptorNeuronal acetylcholine receptor subunit beta-4Neuronal acetylcholine receptor subunit alpha-3
Waktu Paruh2.6 days
Vol. Distribusi-
Klirens-
Genetik -
Levamisole Approved DB00848
small molecule | CAS: 14769-73-4

Levamisole is an antihelminthic drug that was commonly used for the treatment of parasitic, viral, and bacterial infections. [A178117] It was manufactured by _Janssen_ and first used in 1969 as an agent to treat worm infestations[A178123] Levamisole was appro…

Kategori:
Adjuvants, ImmunologicAnthelminticsAnti-Infective Agents +10
Target Protein:
Neuronal acetylcholine receptor subunit alpha-3Alkaline phosphatase, tissue-nonspecific isozymeAlkaline phosphatase, germ cell type +4
Waktu Paruh4.4-5.6 hours (biph…
Vol. Distribusi-
Klirens-
Genetik -
Levamlodipine Approved DB09237
small molecule | CAS: 103129-82-4

Levamlodipine, also known as S-amlodipine, is a pharmacologically active enantiomer of [amlodipine], an antihypertensive medication.[L10833] Levamlodipine belongs to the dihydropyridine group of calcium channel blockers.[L10833] This medication was first mark…

Kategori:
Antiarrhythmic agentsAntihypertensive AgentsAntihypertensive Agents Indicated for Hypertension +11
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent L-type calcium channel subunit alpha-1DNitric oxide synthase 3 +1
Waktu ParuhLevamlodipine has a…
Vol. DistribusiThe volume of distr…
KlirensThe oral clearance …
Genetik -
Levetiracetam Approved DB01202
small molecule | CAS: 102767-28-2

Levetiracetam is a drug within the pyrrolidine class that is used to treat various types of seizures stemming from epileptic disorders. It was first approved for use in the United States in 1999 and is structurally and mechanistically unrelated to other anti-…

Kategori:
AcetamidesAmidesAnticonvulsants +8
Target Protein:
5-hydroxytryptamine receptor 3AVoltage-dependent N-type calcium channel subunit alpha-1BSynaptic vesicle glycoprotein 2A
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe volume of distr…
KlirensThe total plasma cl…
Genetik -
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