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17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
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17430 (100.0%)

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Halaman 325 / 349
TOL-101 DB16980
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TOL2 DB17918
biotech

TOL2 is a modified form of the acetylcholine receptor being investigated for the treatment of myasthenia gravis.[A260117]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tolazamide Approved DB00839
small molecule | CAS: 1156-19-0

A sulphonylurea hypoglycemic agent with actions and uses similar to those of chlorpropamide.

Kategori:
Alimentary Tract and MetabolismAmidesBenzene Derivatives +15
Target Protein:
Sulfonylurea receptor 1, Kir6.2ATP-sensitive inward rectifier potassium channel 10
Waktu ParuhThe average biologi…
Vol. Distribusi-
Klirens-
Genetik -
Tolazoline Approved DB00797
small molecule | CAS: 59-98-3

A vasodilator that apparently has direct actions on blood vessels and also increases cardiac output. Tolazoline can interact to some degree with histamine, adrenergic, and cholinergic receptors, but the mechanisms of its therapeutic effects are not clear. It …

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +14
Target Protein:
Alpha-1A adrenergic receptorD(2) dopamine receptorAlpha-2A adrenergic receptor +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tolbutamide Approved DB01124
small molecule | CAS: 64-77-7

Tolbutamide is an oral antihyperglycemic agent used for the treatment of non-insulin-dependent diabetes mellitus (NIDDM). It is structurally similar to acetohexamide, chlorpropamide and tolazamide and belongs to the sulfonylurea class of insulin secretagogues…

Kategori:
Alimentary Tract and MetabolismAmidesBenzene Derivatives +25
Target Protein:
ATP-binding cassette sub-family C member 9ATP-binding cassette sub-family C member 8ATP-sensitive inward rectifier potassium channel 1
Gen Terkait:
CYP2C9
Waktu ParuhApproximately 7 hou…
Vol. Distribusi-
Klirens-
Genetik 1 Varian
Tolcapone Approved DB00323
small molecule | CAS: 134308-13-7

Tolcapone is a drug that inhibits the enzyme catechol-O-methyl transferase (COMT). It is used in the treatment of Parkinson's disease as an adjunct to levodopa/carbidopa medication. It is a yellow, odorless, non-hygroscopic, crystalline compound. Tolcapone is…

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson DrugsBenzene Derivatives +16
Target Protein:
Catechol O-methyltransferase
Waktu Paruh2-3.5 hours
Vol. Distribusi* 9 L
Klirens* 7 L/h
Genetik -
Tolciclate DB13360
small molecule | CAS: 50838-36-3

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAnti-Infective AgentsAntifungal Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tolebrutinib DB18715
small molecule | CAS: 1971920-73-6

Deskripsi belum tersedia.

Target Protein:
Tyrosine-protein kinase BTK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tolevamer Approved DB01344
small molecule | CAS: 28210-41-5

Sodium polystyrene sulfonate is a medication used to treat abnormally high potassium levels. It may be taken orally or by rectum, as an enema, and functions as a potassium-binding resin in the intestines. It is also an effective topical microbicide and spermi…

Kategori:
AcidsAcids, NoncarboxylicBenzene Derivatives +19
Target Protein:
Potassium
Waktu Paruhnone
Vol. Distribusi-
Klirens-
Genetik -
Tolfenamic acid Approved DB09216
small molecule | CAS: 13710-19-5

Tolfenamic acid, with the formula N-(2-methyl-3-chlorphenyl)-anthranilic acid, is a nonsteroidal anti-inflammatory agent.[A31824] It was discovered by scientists at Medica Pharmaceutical Company in Finland. It is used in the UK as a treatment for migraine und…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +29
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu ParuhThe estimated half-…
Vol. DistribusiThe volume of distr…
KlirensThe estimated clear…
Genetik -
Tolimidone DB16841
small molecule | CAS: 41964-07-2

Deskripsi belum tersedia.

Kategori:
Pyrimidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tolinapant DB16160
small molecule | CAS: 1799328-86-1

ASTX660 is under investigation in clinical trial NCT02503423 (Phase 1-2 Study of ASTX660 in Subjects With Advanced Solid Tumors and Lymphomas).

Kategori:
Oxazines
Target Protein:
E3 ubiquitin-protein ligase XIAP
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Toll-like receptor 9 is under investigation in clinical trial NCT03007732 (Pembrolizumab in Combination With Intratumoral SD-101 Therapy).

Kategori:
Amino Acids, Peptides, and ProteinsDNA-Binding ProteinsMembrane Proteins +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tolmetin Approved DB00500
small molecule | CAS: 26171-23-3

A non-steroidal anti-inflammatory agent (anti-inflammatory agents, NON-steroidal) similar in mode of action to indomethacin.

Kategori:
Acetic Acid Derivatives and Related SubstancesAgents causing hyperkalemiaAgents that produce hypertension +18
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhBiphasic eliminatio…
Vol. Distribusi-
Klirens-
Genetik -
Tolnaftate Approved DB00525
small molecule | CAS: 2398-96-1

Tolnaftate is a synthetic over-the-counter anti-fungal agent. It may come as a cream, powder, spray, or liquid aerosol, and is used to treat jock itch, athlete's foot and ringworm. It is sold under several brand names, most notably Tinactin and Odor Eaters.

Kategori:
Acids, AcyclicAnti-Infective AgentsAntifungal Agents +7
Target Protein:
Squalene monooxygenaseSqualene monooxygenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tolonidine DB13429
small molecule | CAS: 4201-22-3

Deskripsi belum tersedia.

Kategori:
Antiadrenergic Agents, Centrally ActingAntihypertensive AgentsImidazoles +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Toloxatone DB09245
small molecule | CAS: 29218-27-7

Toloxatone is an antidepressant agent, the first ever use of which was in France, 1984. It acts as a selective and reversible inhibitor of monoamine oxidase-A (MOA) [L1388].

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +12
Target Protein:
Amine oxidase [flavin-containing] BAmine oxidase [flavin-containing] A
Waktu Paruh1-3 h [A31957]
Vol. Distribusi-
KlirensHigh hepatic excret…
Genetik -
Tolperisone DB06264
small molecule | CAS: 728-88-1

Tolperisone is an oral, centrally acting muscle relaxant. Its precise mechanism is not completely understood, though it blocks sodium and calcium channels. It possesses a high affinity for nervous system tissue, reaching highest concentrations in brain stem, …

Kategori:
Central Nervous System AgentsCentral Nervous System DepressantsCytochrome P-450 CYP1A2 Substrates +10
Target Protein:
Sodium channel protein type 11 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tolpropamine DB13305
small molecule | CAS: 5632-44-0

Deskripsi belum tersedia.

Kategori:
AminesAntihistamines for Topical UseAntipruritics, Incl. Antihistamines, Anesthetics, Etc. +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tolrestat DB02383
small molecule | CAS: 82964-04-3

Tolrestat (INN) (AY-27773) is an aldose reductase inhibitor which was approved for the control of certain diabetic complications. While it was approved for marketed in several countries, it failed a Phase III trial in the U.S. due to toxicity and never receiv…

Kategori:
Aldehyde Reductase, antagonists & inhibitorsAldose Reductase InhibitorsAlimentary Tract and Metabolism +2
Target Protein:
Sigma non-opioid intracellular receptor 1Aldo-keto reductase family 1 member B1Aldo-keto reductase family 1 member A1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tolterodine Approved DB01036
small molecule | CAS: 124937-51-5

Tolterodine is an antimuscarinic drug that is used to treat urinary incontinence. Tolterodine acts on M2 and M3 subtypes of muscarinic receptors.

Kategori:
Agents producing tachycardiaAlcoholsAmines +26
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M5 +2
Waktu Paruh1.9-3.7 hours
Vol. Distribusi* 113 ± 26.7 L
Klirens-
Genetik -
Tolu balsam DB11223
small molecule | CAS: 9000-64-0

Deskripsi belum tersedia.

Kategori:
Biological ProductsBiopolymersComplex Mixtures +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Toluene DB11558
small molecule | CAS: 108-88-3

Toluene is a colorless, liquid that is immiscible in water. It is a mono-substituted benzene derivative used in veterinary medicine as a treatment for various parasites in dogs and cats.

Kategori:
Benzene DerivativesCompounds used in a research, industrial, or household settingSolvents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tolvaptan Approved DB06212
small molecule | CAS: 150683-30-0

Tolvaptan is used to treat low blood sodium levels (hyponatremia) associated with various conditions like congestive heart failure, cirrhosis, and syndrome of inappropriate antidiuretic hormones (SIADH). FDA approved on May 19, 2009.

Kategori:
Agents causing hyperkalemiaAntidiuretic Hormone Receptor AntagonistsBenzazepines +14
Target Protein:
Vasopressin V2 receptorVasopressin V1a receptor
Waktu ParuhTerminal half life,…
Vol. DistribusiHealthy subjects: 3…
Klirens4 mL/min/kg (post-o…
Genetik -
Tomaralimab DB15415
biotech | CAS: 1449294-76-1

Tomaralimab is under investigation in clinical trial NCT01794663 (Placebo-Controlled Study to Evaluate the Safety and Efficacy of OPN-305 in Preventing Delayed Renal Graft Function).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tomato Approved DB10573
biotech

Tomato allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tominersen DB17924
biotech | CAS: 1709886-74-7

Deskripsi belum tersedia.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tomivosertib DB15219
small molecule | CAS: 1849590-01-7

Tomivosertib is under investigation in clinical trial NCT03318562 (A PD Study of Oral eFT508 in Subjects With Advanced TNBC and HCC).

Target Protein:
MAP kinase-interacting serine/threonine-protein kinase 1MAP kinase-interacting serine/threonine-protein kinase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tomligisiran DB19330
biotech | CAS: 2202789-48-6

Tomligisiran is under investigation in clinical trial NCT06537414 (A Study of Sequential Therapy With Daplusiran/tomligisiran (DAP/TOM) Followed by Bepirovirsen in Participants Living With Chronic Hepatitis B (CHB)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tomuzotuximab DB15178
biotech | CAS: 1646321-00-7

Tomuzotuximab is under investigation in clinical trial NCT02052960 (CetuGEX™ in Comparison to Cetuximab for the Treatment of Patients With Head and Neck Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tonabacase DB17964
biotech | CAS: 1788041-31-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tonabersat DB06578
small molecule | CAS: 175013-84-0

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +3
Target Protein:
5-hydroxytryptamine receptor 1D
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tonapofylline DB12569
small molecule | CAS: 340021-17-2

Tonapofylline has been used in trials studying the treatment of Heart Failure, Renal Insufficiency, and Congestive Heart Failure.

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingPurines +2
Target Protein:
Adenosine receptor A1Adenosine receptor A2aAdenosine receptor A3 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TOP-1288 DB14839
small molecule | CAS: 1630202-02-6

TOP-1288 is under investigation in clinical trial NCT02888379 (Phase 2a Study to Evaluate the Safety/Tolerability and Efficacy of TOP1288 200 mg Rectal Solution Once Daily for 4 Weeks in Ulcerative Colitis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Topiramate Approved DB00273
small molecule | CAS: 97240-79-4

Topiramate is a anti-epileptic drug used to manage seizures and prevent migraines.[A175249] It was initially approved by the FDA in 1996. In 2004, topiramate was approved for the prevention of migraine in adults.[A188309,L10544,L43478] Since 2012, the extende…

Kategori:
Alimentary Tract and MetabolismAnti-Obesity AgentsAnticonvulsants +23
Target Protein:
Glutamate receptor ionotropic, kainate 1Gamma-aminobutyric acid receptor subunit alpha-1Voltage-gated sodium channel alpha subunit +7
Waktu ParuhThe elimination hal…
Vol. DistribusiThe mean apparent v…
KlirensThe mean oral plasm…
Genetik -
Topiroxostat DB01685
small molecule | CAS: 577778-58-6

Topiroxostat is a selective xanthine oxidase inhibitor developed for treatment and management of hyperuricemia and gout. Xanthine oxidase, or xanthine oxidoreductase (XOR), regulates purine metabolism, and inhibition of the enzyme results in efficacious reduc…

Kategori:
BCRP/ABCG2 InhibitorsCytochrome P-450 CYP2C19 InhibitorsCytochrome P-450 CYP2C19 inhibitors (strength unknown) +13
Target Protein:
Xanthine dehydrogenase/oxidase
Waktu ParuhThe mean half life …
Vol. DistribusiThe mean ± SD appar…
KlirensThe apparent total …
Genetik -
Topotecan Approved DB01030
small molecule | CAS: 123948-87-8

An antineoplastic agent used to treat ovarian cancer. It works by inhibiting DNA topoisomerases, type I.

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +21
Target Protein:
DNA topoisomerase 1DNADNA topoisomerase I, mitochondrial
Waktu Paruh2-3 hours
Vol. Distribusi-
Klirens-
Genetik -
Topramezone DB14826
small molecule | CAS: 210631-68-8

Topramezone is under investigation in clinical trial NCT00559520 (The Role of Preoperative Oral Immunonutrition in Major Vascular Surgery).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Topsalysin DB05160
small molecule | CAS: 917121-25-6

Topsalysin is being developed for the treatment of localized prostate cancer and also benign prostatic hyperplasia. Topsalysin is delivered locally to the prostate under ultrasound guidance.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsMembrane Proteins +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Toralizumab DB16384
biotech | CAS: 252662-47-8

Toralizumab is under investigation in clinical trial NCT03605927 (CD40-L Blockade for Prevention of Acute Graft-versus-host Disease).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Torapsel DB13057
biotech | CAS: 204658-47-9

Torapsel has been used in trials studying the prevention of Ischemia Reperfusion Injury.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Torasemide Approved DB00214
small molecule | CAS: 56211-40-6

Torasemide is a high-ceiling loop diuretic.[A174463] Structurally, it is a pyridine-sulfonylurea used as an antihypertensive agent.[A319] Torasemide was first approved for clinical use by the FDA in 1993.[L5257]

Kategori:
Antihypertensive AgentsAntihypertensive Agents Indicated for HypertensionCardiovascular Agents +21
Target Protein:
Solute carrier family 12 member 2Solute carrier family 12 member 1
Waktu ParuhThe average half-li…
Vol. DistribusiThe volume of distr…
KlirensThe clearance rate …
Genetik -
Torcetrapib DB06281
small molecule | CAS: 262352-17-0

Torcetrapib (CP-529414, Pfizer) was developed to treat hypercholesterolemia but its development was halted in 2006 when phase III studies showed excessive mortality in the treatment group receiving a combination of atorvastatin and the study drug.

Kategori:
Anticholesteremic AgentsBlood PressureCholesterol Ester Transfer Proteins +3
Target Protein:
Cholesteryl ester transfer protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Toreforant DB12522
small molecule | CAS: 952494-46-1

Toreforant has been used in trials studying the treatment of Asthma, Psoriasis, Hepatic Impairment, and Rheumatoid Arthritis.

Kategori:
Heterocyclic Compounds, Fused-RingHistamine AgentsHistamine Antagonists +1
Target Protein:
Histamine H4 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Toremifene Approved DB00539
small molecule | CAS: 89778-26-7

Toremifene is a selective estrogen receptor modulator (SERM) and a nonsteroidal antiestrogen used to treat estrogen receptor positive breast cancer.[A256923] Like [tamoxifen], toremifene is part of the first-generation triphenylethylene derivative chemical cl…

Kategori:
Anti-EstrogensAntineoplastic AgentsAntineoplastic Agents, Hormonal +23
Target Protein:
Estrogen receptorSex hormone-binding globulin
Waktu Paruh5 days
Vol. Distribusi* 580 L
Klirens* 5 L/h
Genetik -
Toripalimab Approved DB15043
biotech | CAS: 1924598-82-2

The proliferation of some cancers can be attributed, at least in part, to the suppression of host tumor surveillance. One mechanism by which this occurs is through the overexpression of programmed cell death ligand (PD-L1)[A261506] - the binding of PD-L1 (and…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +13
Target Protein:
Programmed cell death protein 1
Waktu ParuhThe mean terminal e…
Vol. DistribusiAt steady-state, th…
KlirensThe mean clearance …
Genetik -
TORL-2-307 DB18376
biotech

TORL-2307 is a humanized immunoglobulin G1 (IgG1) monoclonal antibody (mAb) directed against claudin 18.2 (CLDN18.2) being investigated for the treatment of gastric and pancreatic cancer.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Torudokimab DB16671
biotech | CAS: 2241728-76-5

Torudokimab is under investigation in clinical trial NCT03831191 (A Study of LY3375880 in Adults With Moderate-to-severe Atopic Dermatitis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tosatoxumab DB16557
biotech | CAS: 1374419-41-6

Tosatoxumab is a fully-human monoclonal antibody (IgG1?) targeting the Staphylococcus aureus alpha-toxin or the S. aureus alpha-hemolysin[A191829, L31568, L31573] and thereby preserving human immune cells by protecting against destruction of host cells mediat…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tosedostat DB11781
small molecule | CAS: 238750-77-1

Tosedostat has been used in trials studying the treatment and supportive care of AML, Leukemia, Pancreas Cancer, Multiple Myeloma, and Pancreatic Cancer, among others. Tosedostat is an inhibitor of the M1 family of aminopeptidases, in particular PuSA, and …

Kategori:
AminesAmino AcidsAmino Acids, Peptides, and Proteins +3
Target Protein:
Puromycin-sensitive aminopeptidaseLeukotriene A-4 hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 16201–16250 dari 17430
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