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17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
Referensi
17430 (100.0%)

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Halaman 324 / 349
Tivanisiran DB19105
biotech | CAS: 1848224-71-4

Tivanisiran is under investigation in clinical trial NCT03108664 (HELIX, a Double-masked Study of SYL1001 in Patients With Moderate to Severe Dry Eye Disease (DED)).

Waktu Paruh-
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Tivantinib DB12200
small molecule | CAS: 905854-02-6

Tivantinib has been investigated in Solid Tumors.

Kategori:
Heterocyclic Compounds, Fused-RingProto-Oncogene Proteins c-met, antagonists & inhibitorsPyrrolidines
Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
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biotech | CAS: 2641020-57-5

Tividenofusp alfa, also known as DNL-310, is a brain-penetrant enzyme replacement therapy being investigated for the treatment of Hunter syndrome.[L46802]

Waktu Paruh-
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Tivirapine DB08600
small molecule | CAS: 137332-54-8

Deskripsi belum tersedia.

Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
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Tivozanib Approved DB11800
small molecule | CAS: 475108-18-0

Renal cell carcinoma (RCC) is responsible for 3% of cancer cases[A231314] and is one of the 10 most common cancers in adults. The average age of diagnosis is between age 65 to 74.[L32529] Tivozanib, also known as FOTIVDA, is a kinase inhibitor developed to t…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +13
Target Protein:
Vascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 2Vascular endothelial growth factor receptor 3 +8
Waktu ParuhThe half-life of ti…
Vol. DistribusiTivozanib has an ap…
KlirensThe apparent cleara…
Genetik -
Tixagevimab Approved DB16394
biotech | CAS: 2420564-02-7

SARS-CoV-2, the causative agent of COVID-19, enters cells via the interaction between the trimeric spike (S) glycoprotein and host cell angiotensin-converting enzyme 2 (ACE2). Blocking the interaction between the receptor-binding domain (RBD) of the S1 subuni…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
Spike glycoprotein
Waktu ParuhTixagevimab has a h…
Vol. DistribusiTixagevimab has an …
KlirensTixagevimab has an …
Genetik -
Tixocortol Approved DB09091
small molecule | CAS: 61951-99-3

Tixocortol is a 21-thiol derivative of hydrocortisone classified as a class A corticosteroid. It is a synthetic steroid with topical anti-inflammatory properties without the systemic glucocorticoid and mineralocorticoid activities and toxicity.[L1078]

Kategori:
11-Hydroxycorticosteroids17-HydroxycorticosteroidsAdrenal Cortex Hormones +20
Target Protein:
Glucocorticoid receptorHistone deacetylase 2
Waktu ParuhTixocortol presents…
Vol. DistribusiStudies have shown …
KlirensStudies have shown …
Genetik -
Tizanidine Approved DB00697
small molecule | CAS: 51322-75-9

Tizanidine is a fast-acting drug used for the management of muscle spasm, which may result from the effects of multiple sclerosis, stroke, an acquired brain injury, or a spinal cord injury [T574]. It may also be caused by musculoskeletal injury [A177583]. R…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +24
Target Protein:
Alpha-1 adrenergic receptorsAlpha-2 adrenergic receptorsNischarin
Waktu ParuhApproximately 2.5 h…
Vol. DistribusiExtensively distrib…
Klirens**A note on renal i…
Genetik -
TJ003234 DB16470
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAnti-Inflammatory Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TK-112690 DB18822
small molecule | CAS: 22423-26-3

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
TK216 DB17414
small molecule | CAS: 1903783-48-1

Deskripsi belum tersedia.

Waktu Paruh-
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Tl-3-093 DB01891
small molecule

Deskripsi belum tersedia.

Target Protein:
Pol polyproteinGag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TL-895 DB16471
small molecule | CAS: 1415823-49-2

TL-895 is a potent, orally active, ATP-competitive, and highly selective irreversible BTK inhibitor with an IC50 and a Ki of 1.5 nM and 11.9 nM, respectively. TL-895 is under investigation in several clinical trials for its safety and efficacy in various cond…

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TLR-AD1 DB18241
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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TLY-012 DB18336
biotech

TLY-012 is a PEGylated recombinant human tumor necrosis factor-related apoptosis-inducing ligand (PEGylated TRAIL).[L48166]

Waktu Paruh-
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TM30339 DB05085
small molecule

TM30339 is an analogue of the natural hormone Pancreatic Polypeptide (PP), which is released in connection with meals. TM30339 works through the same receptor as the natural satiety hormone, Pancreatic Polypeptide (PP), but TM30339 has improved properties com…

Target Protein:
Neuropeptide Y receptor type 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TM5614 DB16516
small molecule

TM5614 is a novel, orally active, plasminogen activator inhibitor 1 (PAI-1) inhibitor[A228788,A228793,]. PAI-1 is a marker of obesity, type 2 diabetes, and metabolic syndrome[L31673,A228793,A228798], and current studies are exploring downstream effects of its…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
Plasminogen activator inhibitor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TMC-310911 DB15623
small molecule | CAS: 1000287-05-7

TMC-310911 (also known as ASC-09) is a novel investigational protease inhibitor (PI) that is structurally similar to the currently available [darunavir].[L12045] It is being investigated for use in HIV-1 infections. TMC-310911 has shown marked activity agains…

Kategori:
Acids, AcyclicAmidesAnti-HIV Agents +10
Target Protein:
Gag-Pol polyproteinHIV-1 protease
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TMC-647055 DB11822
small molecule | CAS: 1204416-97-6

TMC647055 has been used in trials studying the treatment of Hepatitis C, Chronic Hepatitis C, Hepatitis C, Chronic, and Chronic Hepatitis C Virus.

Kategori:
AmidesHeterocyclic Compounds, Fused-RingSulfones +1
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TMC-649128 DB15152
small molecule | CAS: 1019639-33-8

TMC-649128 is under investigation in clinical trial NCT01391117 (TMC649128HPC1002 - a Trial inGenotype 1 Hepatitis C Virus (HCV) - Infected Participants to Determine the Safety, Tolerability, Pharmacokinetics and Antiviral Activity of TMC649128, Alone and Com…

Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TMP DB04243
small molecule

Deskripsi belum tersedia.

Kategori:
DeoxyribonucleotidesNucleic Acids, Nucleotides, and NucleosidesNucleotides +3
Target Protein:
Single-stranded DNA-binding protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tmr DB03903
small molecule

Deskripsi belum tersedia.

Target Protein:
Actin, alpha skeletal muscle
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TMV-083 DB16430
biotech

TMV-083 is an attenuated live virus COVID-19 vaccine candidate which employs the measles vaccine as a vector[L30433]. It expresses a spike protein antigen from SARS-CoV-2[L30433].

Waktu Paruh-
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TN-201 DB18700
biotech

TN-201 is a gene therapy comprising a native AAV9 capsid with a genomic cassette containing a cardiomyocyte-specific promoter and the wild-type human MYBPC3 gene.

Waktu Paruh-
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Genetik -
TN-401 DB18140
biotech

TN-401 is a native AAV9 capsid with a genomic cassette containing a cardiomyocyte-specific promoter and the wild-type human PKP2 gene.

Waktu Paruh-
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TNB-383B DB17268
biotech

TNB-383B is a CD3 and B-cell maturation antigen T-cell engaging bispecific antibody.

Waktu Paruh-
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TNB-486 DB19420
biotech

TNB-486 is under investigation in clinical trial NCT06564038 (A Study of AZD0486 Monotherapy or in Combination With Other Anti-cancer Agents for Mature B-cell Malignancies).

Waktu Paruh-
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TNG908 DB17411
small molecule

TNG908 is a small molecule inhibitor of protein arginine methyl transferase 5 (PRMT5).

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TNP-2092 DB16312
small molecule | CAS: 922717-97-3

TNP-2092 is under investigation in clinical trial NCT03964493 (TNP-2092 to Treat Acute Bacterial Skin and Skin Structure Infection).

Kategori:
Heterocyclic Compounds, Fused-RingLactams, MacrocyclicQuinolines
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA topoisomerase 4 subunit A
Waktu Paruh-
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TNP-470 DB08633
small molecule | CAS: 129298-91-5

O-(chloroacetylcarbamoyl)fumagillol (TNP-470) has been used in trials studying the treatment of HIV Infections, Sarcoma, Kaposi, and Pancreatic Neoplasms.

Kategori:
Angiogenesis InhibitorsAngiogenesis Modulating AgentsAntibiotics, Antineoplastic +7
Target Protein:
Methionine aminopeptidase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TNT-1 DB17348
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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TNX-901 DB05797
biotech

TNX-901 is a therapeutic monoclonal antibodies designed to address significant unmet medical needs in the areas of asthma, allergy, inflammation and other diseases affecting the human immune system.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
High affinity immunoglobulin epsilon receptor subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TO-901317 DB07080
small molecule | CAS: 293754-55-9

TO-901317 is an LXRalpha and LXRbeta agonist.

Kategori:
AmidesBenzene DerivativesHydrocarbons, Fluorinated +4
Target Protein:
Oxysterols receptor LXR-betaNuclear receptor coactivator 2Retinoic acid receptor RXR-beta +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tobacco leaf Approved DB10710
biotech | CAS: 8037-19-2

Tobacco leaf allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
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Tobemstomig DB18987
biotech | CAS: 2648839-43-2

Tobemstomig is under investigation in clinical trial NCT05908786 (A Study Evaluating the Efficacy and Safety of Neoadjuvant Immunotherapy Combinations in Patients With Surgically Resectable Hepatocellular Carcinoma).

Waktu Paruh-
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Tobevibart DB18986
biotech | CAS: 2645440-65-7

Tobevibart is under investigation in clinical trial NCT05612581 (A Platform Study to Evaluate Investigational Therapies in Chronic Hepatitis B Infection).

Waktu Paruh-
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Tobramycin Approved DB00684
small molecule | CAS: 32986-56-4

Aminoglycosides, many of which are derived directly from _Streptomyces_ spp., are concentration-dependent bactericidal antibiotics with a broad spectrum of activity against Gram-positive and Gram-negative organisms.[A232294] Inhaled tobramycin is notable for …

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +13
Target Protein:
16S ribosomal RNA23S ribosomal RNABacterial outer membrane +1
Waktu ParuhTobramycin has an a…
Vol. DistribusiInhalation tobramyc…
KlirensInhaled tobramycin …
Genetik -
Tocainide Approved DB01056
small molecule | CAS: 41708-72-9

An antiarrhythmic agent which exerts a potential- and frequency-dependent block of sodium channels.

Kategori:
AmidesAminesAnilides +14
Target Protein:
Sodium channel protein type 5 subunit alpha
Waktu ParuhThe average plasma …
Vol. Distribusi-
Klirens-
Genetik -
Tocilizumab Approved DB06273
biotech | CAS: 375823-41-9

Tocilizumab is a recombinant humanized monoclonal antibody IL-6 receptor inhibitor used to treat inflammatory and autoimmune conditions.[L12789] It was first described in the literature in 2003 when Chugai, a subsidiary of Roche began developing IL-6 inhibiti…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntibodies +21
Target Protein:
Interleukin-6 receptor subunit alpha
Waktu ParuhThe half life of to…
Vol. DistribusiIn rheumatoid arthr…
KlirensThe linear clearanc…
Genetik -
Tocladesine DB13046
small molecule | CAS: 41941-56-4

Tocladesine has been used in trials studying the treatment of Colorectal Cancer and Multiple Myeloma and Plasma Cell Neoplasm.

Kategori:
Adenine NucleotidesAntineoplastic AgentsCyclic AMP +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tocofersolan Approved DB11635
small molecule | CAS: 9002-96-4

D-Alpha-tocopheryl polyethylene glycol 1000 succinate (Tocofersolan, Vedrop), has been developed in Europe as an orally bioavailable source of vitamin E in children suffering from cholestasis [L2371]. Cholestasis is the reduction or stoppage of bile flow, eit…

Kategori:
Alimentary Tract and MetabolismBenzopyransCompounds used in a research, industrial, or household setting +9
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh29.7 h [L2371]
Vol. DistribusiLocated principally…
Klirens-
Genetik -
Tocopherol Approved DB11251
small molecule | CAS: 1406-66-2

Tocopherol exists in four different forms designated as ?, ?, ?, and ?. They present strong antioxidant activities, and it is determined as the major form of vitamin E. Tocopherol, as a group, is composed of soluble phenolic compounds that consist of a chroma…

Kategori:
Alimentary Tract and MetabolismAntioxidantsBenzopyrans +16
Target Protein:
Free radicals
Waktu ParuhThe elimination hal…
Vol. DistribusiThe apparent volume…
KlirensClearance ranged fr…
Genetik -
small molecule | CAS: 43119-47-7

Deskripsi belum tersedia.

Kategori:
BenzopyransHeterocyclic Compounds, Fused-RingPyrans +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 7559-04-8

Deskripsi belum tersedia.

Kategori:
AnticoagulantsAntihypertensive AgentsAntioxidants +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tocotrienol DB12647
small molecule | CAS: 6829-55-6

Tocotrienol has been investigated for the treatment of Cholesterol Lowering.

Kategori:
AntioxidantsBenzopyransBiological Factors +11
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tofacitinib Approved DB08895
small molecule | CAS: 477600-75-2

Tofacitinib is an inhibitor of Janus kinases, a group of intracellular enzymes involved in signalling pathways that affect hematopoiesis and immune cell function. It is approved by the FDA for treatment of moderate to severe rheumatoid arthritis that responds…

Kategori:
Antineoplastic and Immunomodulating AgentsAntirheumatic AgentsBiologics for Rheumatoid Arthritis Treatment +14
Target Protein:
Tyrosine-protein kinase JAK1Tyrosine-protein kinase JAK2Tyrosine-protein kinase JAK3 +1
Waktu Paruh~3 hours
Vol. DistribusiVd= 87L after intra…
Klirens-
Genetik -
Tofersen Approved DB14782
biotech | CAS: 2088232-70-4

Tofersen is under an intrathecally administered antisense oligonucleotide targeting the mutated SOD1 gene that causes amyotrophic lateral sclerosis (ALS).[L46108] Although there were various causes of ALS, 2% of ALS cases are due to SOD1 mutations, with more …

Kategori:
Antisense OligonucleotidesNervous SystemNucleic Acids, Nucleotides, and Nucleosides +2
Target Protein:
Superoxide dismutase 1 (SOD1)
Waktu ParuhThe effective half-…
Vol. Distribusi-
Klirens-
Genetik -
Tofimilast DB11681
small molecule | CAS: 185954-27-2

Tofimilast has been used in trials studying the treatment of Asthma and Pulmonary Disease, Chronic Obstructive.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4B3',5'-cyclic-AMP phosphodiesterase 4D3',5'-cyclic-AMP phosphodiesterase 4A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tofisopam DB08811
small molecule | CAS: 22345-47-7

Tofisopam (marketed under brand names Emandaxin and Grandaxin) is a 2,3-benzodiazepine drug which is a benzodiazepine derivative. In contrast to classical 1,4-benzodiazepines, the compound does not bind to the benzodiazepine binding site of the gamma-aminobut…

Kategori:
Anti-Anxiety AgentsAntidepressive AgentsBenzazepines +12
Target Protein:
cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A3',5'-cyclic-AMP phosphodiesterase 4AcGMP-dependent 3',5'-cyclic phosphodiesterase +1
Waktu Paruh6-8 hours
Vol. Distribusi-
Klirens-
Genetik -
Tofogliflozin DB11824
small molecule | CAS: 903565-83-3

Tofogliflozin has been used in trials studying the treatment and prevention of Diabetes Mellitus Type 2.

Kategori:
Benzene DerivativesBlood Glucose Lowering AgentsCarbohydrates +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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