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17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
Referensi
17430 (100.0%)

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Hasil Pencarian (17430)

Halaman 323 / 349
Timdarpacept DB17544
biotech | CAS: 2749520-17-8

IMM01 is a recombinant human signal regulatory protein ? (SIRP?) IgG 1 fusion protein.[A257261] IMM01 is under investigation in clinical trial NCT05140811 (A Study of IMM01 Combined With Azacitidine in Patients With Acute Myeloid Leukemia and Myelodysplastic …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Timepidium DB13850
small molecule | CAS: 97094-64-9

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnticholinergic Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Timolol Approved DB00373
small molecule | CAS: 26839-75-8

Timolol is a nonselective beta-adrenergic antagonist given in an eye drop solution to reduce intraocular pressure, or pressure in the eyes.[L6724] It is also used in tablet form as a drug to treat hypertension.[L6727] Timolol was first approved by the FDA in …

Kategori:
Adrenergic AntagonistsAdrenergic beta-AntagonistsAgents causing hyperkalemia +28
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorEndolysin
Waktu ParuhTimolol half-life w…
Vol. Distribusi1.3 - 1.7 L/kg [L6]…
KlirensOne pharmacokinetic…
Genetik -
Timolumab DB18597
biotech | CAS: 1073538-99-4

Timolumab is a recombinant, fully-human, IgG4 immunoglobulin with antigen-binding specificity for human vascular adhesion protein-1 (VAP-1).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Timonacic DB12856
small molecule | CAS: 444-27-9

Timonacic has been used in trials studying the treatment of HIV Infections.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1905415-02-2

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 14325-05-4

Deskripsi belum tersedia.

Kategori:
Biological FactorsCoordination ComplexesEnzyme Inhibitors +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tinengotinib DB17384
small molecule | CAS: 2230490-29-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tinidazole Approved DB00911
small molecule | CAS: 19387-91-8

A nitroimidazole antitrichomonal agent effective against _Trichomonas vaginalis_, _Entamoeba histolytica_, and _Giardia lamblia_ infections.

Kategori:
Alimentary Tract and MetabolismAlkylating DrugsAnti-Bacterial Agents +24
Target Protein:
DNA
Waktu ParuhThe elimination hal…
Vol. Distribusi* 50 L
Klirens-
Genetik -
Tinlarebant DB17832
small molecule | CAS: 1821327-95-0

Deskripsi belum tersedia.

Target Protein:
Retinol-binding protein 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tinlorafenib DB17082
small molecule | CAS: 2573781-75-4

Tinlorafenib (PF-07284890) is a potent, selective, highly brain-penetrant, small-molecule inhibitor of BRAF V600 mutations.[A253992]

Kategori:
Heterocyclic Compounds, Fused-RingSulfonamides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tinodasertib DB18796
small molecule | CAS: 1464151-33-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tinoridine DB13001
small molecule | CAS: 24237-54-5

Tinoridine is under investigation in clinical trial NCT01224756 (Efficacy of Tinoridine in Treating Pain and Inflammation in Adults).

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tinostamustine DB15147
small molecule | CAS: 1236199-60-2

Tinostamustine is under investigation in clinical trial NCT03452930 (Tinostamustine With or Without Radiation Therapy in Treating Patients With Newly Diagnosed MGMT-Unmethylated Glioblastoma).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tinzaparin Approved DB06822
small molecule | CAS: 9041-08-1

Tinzaparin is a low molecular weight heparin (LMWH), produced by enzymatic depolymerization of unfractionated heparin from porcine intestinal mucosa. It is a heterogeneous mixture of with an average molecular weight between 5500 and 7500 daltons. Tinzaparin i…

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +8
Target Protein:
Antithrombin-IIIIntegrin alpha-4Stromal cell-derived factor 1
Waktu ParuhAnti-Xa activity is…
Vol. DistribusiAnti-Xa activity is…
KlirensClearance is dose-d…
Genetik -
Tiocarlide DB13608
small molecule | CAS: 910-86-1

Deskripsi belum tersedia.

Kategori:
Antiinfectives for Systemic UseAntimycobacterialsDrugs for Treatment of Tuberculosis +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tioclomarol DB13451
small molecule | CAS: 22619-35-8

Deskripsi belum tersedia.

Kategori:
AnticoagulantsBenzopyransBlood and Blood Forming Organs +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tioconazole Approved DB01007
small molecule | CAS: 65899-73-2

Tioconazole is an imidazole antifungal used to treat fungal and yeast infections. Topical formulations are used for ringworm, jock itch, athlete's foot, and tinea versicolor or "sun fungus". Tioconazole interacts with 14-alpha demethylase, a cytochrome P-450 …

Kategori:
14-alpha Demethylase InhibitorsAnti-Infective AgentsAntifungal Agents +21
Target Protein:
Lanosterol 14-alpha demethylaseLanosterol 14-alpha demethylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tioguanine Approved DB00352
small molecule | CAS: 154-42-7

An antineoplastic compound which also has antimetabolite action. The drug is used in the therapy of acute leukemia.

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +9
Target Protein:
DNA
Gen Terkait:
TPMT TPMT TPMT +1
Waktu ParuhWhen the compound w…
Vol. Distribusi-
Klirens-
Genetik 4 Varian
Tiopronin Approved DB06823
small molecule | CAS: 1953-02-2

Tiopronin is a prescription thiol drug used primarily in the treatment of severe homozygous cystinuria. Patients with cystinuria excrete high levels of cystine in their urine and are at risk for kidney stone formation. Tiopronin is used as a second-line thera…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAmino Acids, Sulfur +7
Waktu ParuhTiopronin has a lon…
Vol. DistribusiThe volume of distr…
KlirensTotal renal clearan…
Genetik -
Tiotropium Approved DB01409
small molecule | CAS: 186691-13-4

Tiotropium is a long-acting, antimuscarinic bronchodilator used in the management of chronic obstructive pulmonary disease (COPD) and asthma.[A180163,L7084,L7087,L7090,L7093] Tiotropium acts mainly on M3 muscarinic receptors located in the airways to produce …

Kategori:
Adrenergics, InhalantsAgents producing tachycardiaAgents to Treat Airway Disease +22
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2 +2
Waktu ParuhThe terminal half l…
Vol. DistribusiThe volume of distr…
KlirensThe total clearance…
Genetik -
Tioxidazole DB11472
small molecule | CAS: 61570-90-9

Deskripsi belum tersedia.

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tioxolone DB13343
small molecule | CAS: 4991-65-5

Deskripsi belum tersedia.

Kategori:
Anti-Acne PreparationsAnti-Acne Preparations for Topical UseDermatologicals +1
Target Protein:
Carbonic anhydrase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1052105-48-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tipelukast DB12435
small molecule | CAS: 125961-82-2

Tipelukast is under investigation for the treatment of IPF and Idiopathic pulmonary fibrosis.

Target Protein:
Polyunsaturated fatty acid 5-lipoxygenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tipepidine DB13474
small molecule | CAS: 5169-78-8

Deskripsi belum tersedia.

Kategori:
Cough and Cold Preparations
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tiphenamil DB19367
small molecule | CAS: 82-99-5

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicPhenylacetates
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tipifarnib DB04960
small molecule | CAS: 192185-72-1

Tipifarnib (R-115777) is a substance that is being studied in the treatment of acute myeloid leukemia (AML) and other types of cancer. It belongs to the family of drugs called farnesyltransferase inhibitors. It is also called Zarnestra. In June 2005, the FDA …

Kategori:
Antineoplastic AgentsHeterocyclic Compounds, Fused-RingP-glycoprotein inhibitors +1
Target Protein:
Farnesyl pyrophosphate synthaseProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alphaProtein farnesyltransferase subunit beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tipiracil Approved DB09343
small molecule | CAS: 183204-74-2

Tipiracil is a thymidine phosphorylase inhibitor. It is used in combination with trifluridine, in a ratio of 1:0.5, to form TAS-102. The main function of Tipiracil in TAS-102 is to increase trifluridine bioavailability by inhibiting its catabolism.[A31255] TA…

Kategori:
MATE 1 SubstratesMATE 1 Substrates with a Narrow Therapeutic IndexMATE substrates +6
Target Protein:
Thymidine phosphorylase
Waktu ParuhAfter administratio…
Vol. DistribusiFollowing a single …
KlirensFollowing a single …
Genetik -
Tiplimotide DB12738
biotech | CAS: 178823-49-9

Tiplimotide has been used in trials studying the treatment of Multiple Sclerosis.

Kategori:
Amino Acids, Peptides, and ProteinsMembrane ProteinsMyelin Proteins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tipranavir Approved DB00932
small molecule | CAS: 174484-41-4

Tipranavir is a sulfonamide-containing dyhydropyrone and a nonpeptidic protease inhibitor that targets the HIV protease. Tipranavir and ritonavir are coadministered to treat HIV.

Kategori:
AmidesAnti-HIV AgentsAnti-Infective Agents +37
Target Protein:
Gag-Pol polyproteinPol polyprotein
Waktu Paruh5-6 hours
Vol. Distribusi-
Klirens-
Genetik -
Tipranavir C-14 DB15108
small molecule | CAS: 1141509-98-9

Tipranavir C-14 is under investigation in clinical trial NCT02253797 (Pharmacokinetics of Tipranavir/Ritonavir and Its Metabolites in Healthy Male Subjects).

Kategori:
AmidesAnti-HIV AgentsAnti-Infective Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tiprelestat DB18368
biotech | CAS: 820211-82-3

Deskripsi belum tersedia.

Target Protein:
MyeloblastinNeutrophil elastase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tirabrutinib DB15227
small molecule | CAS: 1351636-18-4

Tirabrutinib is under investigation in clinical trial NCT02626026 (Safety and Pharmacokinetics of GS-4059 in Healthy Volunteers and Subjects With Rheumatoid Arthritis (RA)).

Target Protein:
Tyrosine-protein kinase BTK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tiracizine DB13635
small molecule | CAS: 83275-56-3

Deskripsi belum tersedia.

Kategori:
Antiarrhythmic agentsCardiac TherapyCardiovascular Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tiragolumab DB16409
biotech | CAS: 1918185-84-8

Tiragolumab is under investigation in clinical trial NCT04513925 (A Study of Atezolizumab and Tiragolumab Compared With Durvalumab in Participants With Locally Advanced, Unresectable Stage III Non-small Cell Lung Cancer (NSCLC)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tirapazamine DB04858
small molecule | CAS: 27314-97-2

Tirapazamine, also known as SR-4233, is an experimental anticancer drug that is activated in hypoxic conditions. This activation is very useful as this hypoxic state is found in human solid tumors in a common phenomenon known as tumor hypoxia. Hence, tirapaza…

Kategori:
Antineoplastic AgentsCytochrome P-450 CYP2E1 SubstratesCytochrome P-450 Substrates +2
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-betaDNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tirasemtiv DB12209
small molecule | CAS: 1005491-05-3

Tirasemtiv has been used in trials studying the treatment of Myasthenia Gravis, Intermittent Claudication, and Amyotrophic Lateral Sclerosis.

Target Protein:
Troponin C, skeletal muscle
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tiratricol DB03604
small molecule | CAS: 51-24-1

A metabolite of T3 and T4 thyroid hormones; promoted for hyperlipidemia, localized lipodystrophy, and obesity. Tiratricol has been used in trials studying the treatment of Allan-Herndon-Dudley Syndrome.

Kategori:
Agents used to treat hypothyroidismAmino AcidsAmino Acids, Aromatic +9
Target Protein:
Thyroid hormone receptor alphaThyroid hormone receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tirbanibulin Approved DB06137
small molecule | CAS: 897016-82-9

Tirbanibulin (KX-O1 or KX2–391) is a dual inhibitor of Src Kinase and tubulin.[A225726] On December 14, 2020, tirbanibulin was approved by the FDA for the topical treatment of actinic keratosis on the face or scalp. It is marketed under the brand name Klisyri…

Kategori:
AcetatesAcids, AcyclicAmides +39
Target Protein:
Tubulin beta chainProto-oncogene tyrosine-protein kinase Src
Waktu ParuhThe half-life is ab…
Vol. DistribusiThere is limited in…
KlirensThere is limited in…
Genetik -
Tirilazad DB13050
small molecule | CAS: 110101-66-1

Tirilazad has been used in trials studying the treatment of Spinal Cord Injury.

Kategori:
AntioxidantsBiological FactorsCentral Nervous System Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tirofiban Approved DB00775
small molecule | CAS: 144494-65-5

Tirofiban prevents the blood from clotting during episodes of chest pain or a heart attack, or while the patient is undergoing a procedure to treat a blocked coronary artery. It is a non-peptide reversible antagonist of the platelet glycoprotein (GP) IIb/IIIa…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +9
Target Protein:
Integrin alpha-IIbIntegrin beta-3
Waktu Paruh2 hours
Vol. Distribusi* 22 to 42 L
Klirens* 213 - 314 mL/min …
Genetik -
Tiropramide DB13091
small molecule | CAS: 55837-29-1

Tiropramide is under investigation in clinical trial NCT01629212 (Comparison of the Efficacy and Safety of Tiropramide and Octylonium in the Treatment of Irritable Bowel Syndrome).

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids, Aromatic +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tirzepatide Approved DB15171
biotech | CAS: 2023788-19-2

Tirzepatide is a novel dual glucose-dependent insulinotropic polypeptide (GIP) and glucagon-like peptide-1 (GLP-1) receptor agonist. Dual GIP/GLP-1 agonists gained increasing attention as new therapeutic agents for glycemic and weight control as they demonstr…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +17
Target Protein:
Glucagon-like peptide 1 receptorGastric inhibitory polypeptide receptor
Waktu ParuhThe half-life is ap…
Vol. DistribusiFollowing subcutane…
KlirensThe apparent popula…
Genetik -
Tisagenlecleucel Approved DB13881
biotech | CAS: 1823078-37-0

Tisagenlecleucel is a CD19-directed genetically modified autologous T cell immunotherapy, or a CAR-T cell therapy for B-cell acute lymphoblastic leukemia. It was granted approval by FDA in August 2017 under the market name Kymriah. Tisagenlecleucel is an immu…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic Agents, Immunological +10
Target Protein:
B-lymphocyte antigen CD19
Waktu ParuhThe mean half life …
Vol. DistribusiThe drug is found t…
Klirens-
Genetik -
Tislelizumab Approved DB14922
biotech | CAS: 1858168-59-8

Tislelizumab is a humanized monoclonal IgG4 antibody against programmed death receptor-1 (PD-1). It was engineered to have a nullified Fc portion, thus minimizing binding to Fc?R on macrophages and limiting treatment resistance via antibody-dependent phagocyt…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
Programmed cell death protein 1
Waktu ParuhBased on population…
Vol. DistribusiA population pharma…
KlirensBased on population…
Genetik -
Tisopurine DB13807
small molecule | CAS: 5334-23-6

Deskripsi belum tersedia.

Kategori:
Antigout PreparationsAntirheumatic AgentsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tisotumab vedotin Approved DB16732
biotech | CAS: 1418731-10-8

Tisotumab vedotin is a tissue factor-directed antibody-drug conjugate (ADC) comprised of an anti-tissue factor (TF) human IgG1-kappa antibody conjugated to monomethyl auristatin E (MMAE), a microtubule-disrupting agent, via a protease-cleavable valine-citrull…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
Tissue factor
Waktu ParuhThe median terminal…
Vol. DistribusiThe tisotumab vedot…
KlirensThe linear clearanc…
Genetik -
Titanium DB14160
small molecule | CAS: 7440-32-6

Deskripsi belum tersedia.

Kategori:
ElementsMetalsMetals, Light +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Titanium dioxide Approved DB09536
small molecule | CAS: 13463-67-7

Titanium dioxide, also known as titanium(IV) oxide or titania, is the naturally occurring oxide of titanium. It is used as a pigment under the names titanium white, Pigment White 6 (PW6), or CI 77891. It is typically extracted from ilmenite, rutile and anatas…

Kategori:
Astringents and DeodorantsBiocompatible MaterialsColoring Agents +13
Target Protein:
Macrophage receptor MARCO
Waktu ParuhThe kinetics of TiO…
Vol. DistribusiSix hours after tit…
KlirensThe clearance of ti…
Genetik -
Menampilkan 16101–16150 dari 17430
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