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2279

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866 (38.0%)
Target
1100 (48.3%)
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Halaman 32 / 46
Oxycodone Approved DB00497
small molecule | CAS: 76-42-6

Oxycodone is a semisynthetic opioid analgesic derived from thebaine in Germany in 1917.[A178696] It is currently indicated as an immediate release product for moderate to severe pain and as an extended release product for chronic moderate to severe pain requi…

Kategori:
AlkaloidsAnalgesicsCentral Nervous System Agents +21
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor
Waktu ParuhThe apparent elimin…
Vol. Distribusi2.6L/kg.[Label]
KlirensTotal plasma cleara…
Genetik -
Oxygen Approved DB09140
small molecule | CAS: 7782-44-7

Oxygen is an element displayed by the symbol O, and atomic number 8. It is an essential element for human survival. Decreased oxygen levels may be treated with medical oxygen therapy. Treatment with oxygen serves to increase blood oxygen levels and also exer…

Kategori:
ChalcogensElementsGases +3
Target Protein:
Cytochrome c oxidase subunit 1NADPH oxidase 1
Waktu ParuhApproximately 122.2…
Vol. Distribusi-
Klirens-
Genetik -
Oxymetholone Approved DB06412
small molecule | CAS: 434-07-1

Oxymetholone is a synthetic anabolic steroid marketed under the brand name Anapolon by Hoffmann La Roche Limitedand used in the treatment of osteoporosis, anaemia, and as an agent to stimulate muscle growth in malnourished or underdeveloped patients. Anabolic…

Kategori:
Alimentary Tract and MetabolismAnabolic AgentsAnabolic Agents for Systemic Use +20
Target Protein:
Androgen receptorNatriuretic peptides B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxytocin Approved DB00107
biotech | CAS: 50-56-6

Sir Henry H. Dale first identified oxytocin and its uterine contractile properties in 1906.[A229008,A228593,A229108] Like all other neurohypophysial hormones, oxytocin is composed of nine amino acids with a disulfide bridge between the Cys 1 and 6 residues.[A…

Kategori:
Amino Acids, Peptides, and ProteinsGenito Urinary System and Sex HormonesHormones +15
Target Protein:
Oxytocin receptorVasopressin V1b receptorVasopressin V2 receptor +1
Waktu ParuhThe plasma half-lif…
Vol. Distribusi-
KlirensIn a study that obs…
Genetik -
Ozanezumab DB12891
biotech | CAS: 1310680-64-8

Ozanezumab has been used in trials studying the treatment of Multiple Sclerosis, Amyotrophic Lateral Sclerosis, and Multiple Sclerosis, Relapsing-Remitting.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ozekibart DB18675
biotech | CAS: 2539847-03-3

Ozekibart is a tetravalent recombinant humanized IgG1 agonist antibody targeting the human TRAIL death receptor 5 (DR5). It is being investigated for the treatment of chondrosarcoma.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
P-113D DB04987
biotech | CAS: 190673-60-0

P-113D is a novel 12 amino-acid antimicrobial peptide drug derived from histatins, which are compounds found naturally in human saliva. It is being pursued as a potential treatment for cystic fibrosis by Demegen, Inc.

Kategori:
Amino Acids, Peptides, and ProteinsAntimicrobial Cationic PeptidesAntimicrobial Peptides +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pabinafusp alfa DB15633
biotech | CAS: 2140211-48-7

Pabinafusp alfa is under investigation in clinical trial NCT03568175 (A Study of JR-141 in Patients With Mucopolysaccharidosis II).

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pacmilimab DB18873
biotech | CAS: 2145091-51-4

Pacmilimab is under investigation in clinical trial NCT04596150 (Study to Evaluate the Safety and Antitumor Activity of CX-2009 Monotherapy and in Combination With CX-072 in Advanced Breast Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Padimate O Approved DB11570
small molecule | CAS: 21245-02-3

Padimate O is an active sunscreen agent in cosmetics and over-the-counter sunscreen drug products in concentrations up to 8%, as regulated by the FDA [L2153]. It is a structurally-related compound to [DB02362] that absorbs UV-B rays to prevent photodamage. It…

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +7
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Pagibaximab DB17786
biotech | CAS: 595566-61-3

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Palifermin Approved DB00039
biotech | CAS: 162394-19-6

Palifermin is a recombinant human keratinocyte growth factor (KGF). It is 140 residues long, and is produced using E. coli. Palifermin was granted FDA approval on 15 December 2004.[L17933]

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsDetoxifying Agents for Antineoplastic Treatment +6
Target Protein:
Fibroblast growth factor receptor 2Fibroblast growth factor receptor 1Basement membrane-specific heparan sulfate proteoglycan core protein
Waktu ParuhElimination half-li…
Vol. Distribusi-
Klirens-
Genetik -
Palivizumab Approved DB00110
biotech | CAS: 188039-54-5

Humanized monoclonal antibody (IgG1k) produced by recombinant DNA technology, directed to an epitope in the A antigenic site of the F protein of respiratory syncytial virus (RSV). Synagis is a composite of human (95%) and murine (5%) antibody sequences. The h…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +15
Target Protein:
Fusion glycoprotein F0Low affinity immunoglobulin gamma Fc region receptor III-BComplement C1r subcomponent +6
Waktu Paruh18-20 days (in adul…
Vol. Distribusi-
Klirens-
Genetik -
Palmidrol DB14043
small molecule | CAS: 544-31-0

A cannabinoid receptor-inactive eCB-related molecule used as prophylactic in helping to prevent respiratory viral infection. Palmidrol is available for human use as a supplement (400 mg capsules) and as food for medical purposes In Italy and Spain (300 mg and…

Kategori:
Agents producing tachycardiaAlcoholsAmines +15
Target Protein:
Cannabinoid receptor 2Glucose-dependent insulinotropic receptorG-protein coupled receptor 55
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Palopegteriparatide Approved DB18676
biotech | CAS: 2222514-07-8

Palopegteriparatide is a parathyroid hormone (PTH) analog. Palopegteriparatide is a prodrug consisting of PTH(1-34) conjugated to a methoxy polyethylene glycol carrier (mPEG) via a proprietary TransCon Linker.[L51134] PTH(1-34) contains the N-terminal part of…

Kategori:
Calcium HomeostasisParathyroid Hormones and AnaloguesSystemic Hormonal Preparations, Excl. Sex Hormones and Insulins +1
Target Protein:
Parathyroid hormone/parathyroid hormone-related peptide receptor
Waktu ParuhThe apparent half-l…
Vol. DistribusiThe estimated appar…
KlirensThe estimated clear…
Genetik -
Palovarotene Approved DB05467
small molecule | CAS: 410528-02-8

Fibrodysplasia Ossificans Progressiva (FOP), with an estimated worldwide prevalence of one in 2 million individuals, is an exceptionally rare genetic disorder.[A244920] FOP is caused by a gain-of-function mutation in the ACVR1/ALK2 gene which results in progr…

Kategori:
BCRP/ABCG2 InhibitorsBenzene DerivativesBenzylidene Compounds +17
Target Protein:
Retinoic acid receptor gamma
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean (SD) appar…
KlirensThe apparent total …
Genetik -
Palucorcel DB17955
biotech

Palucorcel is an investigational stem cell therapy consisting of human umbilical tissue-derived cells. Developed by Janssen Biotech, it is being investigated for the treatment of various conditions such as amyotrophic lateral sclerosis (ALS) and macular degen…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Panax ginseng whole is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsAraliaceaeBiological Products +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pancrelipase lipase Approved DB13147
biotech | CAS: 9001-62-1

Pancrelipase, in general, is composed of a mixture of pancreatic enzymes which include amylases, lipases, and proteases. These enzymes are extracted from porcine pancreatic glands.[L2509] The pancrelipase lipase is an enzyme secreted by the pancreas that is r…

Kategori:
Carboxylic Ester HydrolasesEnzymesEnzymes and Coenzymes +4
Target Protein:
Dietary fat
Waktu ParuhPlease refer to [DB…
Vol. DistribusiPlease refer to [DB…
KlirensPlease refer to [DB…
Genetik -
Panitumumab Approved DB01269
biotech | CAS: 339177-26-3

Panitumumab (ABX-EGF) is a recombinant human IgG2 monoclonal antibody that binds specifically to the human epidermal growth factor receptor (EGFR). This drug is an antineoplastic agent. Panitumumab was granted FDA approval on 27 September 2006.[L17663]

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +16
Target Protein:
Epidermal growth factor receptor
Waktu Paruh7.5 days (range: 4-…
Vol. Distribusi-
Klirens* 4.9+/- 1.4 mL/kg/…
Genetik -
Panobacumab DB15342
biotech | CAS: 885053-97-4

Panobacumab is under investigation in clinical trial NCT00851435 (Safety and Pharmacokinetics of KBPA-101 in Hospital Acquired Pneumonia Caused by O11 Pseudomonas Aeruginosa).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Panthenol Approved DB11204
small molecule | CAS: 16485-10-2

Panthenol is an alcohol derivative of pantothenic acid, a component of the B complex vitamins and an essential component of a normally functioning epithelium. Panthenol exists as a racemic mixture containing both the dextrorotatory form (dexpanthenol) and the…

Kategori:
AlanineAmino AcidsAmino Acids, Peptides, and Proteins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pantoprazole Approved DB00213
small molecule | CAS: 102625-70-7

Pantoprazole is a first-generation proton pump inhibitor (PPI) used for the management of gastroesophageal reflux disease (GERD), for gastric protection to prevent recurrence of stomach ulcers or gastric damage from chronic use of NSAIDs, and for the treatmen…

Kategori:
2-PyridinylmethylsulfinylbenzimidazolesAcid ReducersAlimentary Tract and Metabolism +27
Target Protein:
Potassium-transporting ATPase alpha chain 1Potassium-transporting ATPase subunit betaN(G),N(G)-dimethylarginine dimethylaminohydrolase 1
Waktu ParuhAbout 1 hour[F3202]
Vol. DistribusiThe apparent volume…
Klirens**Adults**: With in…
Genetik -
Pantothenic acid Approved DB01783
small molecule | CAS: 79-83-4

Pantothenic acid, also called pantothenate or vitamin B5 (a B vitamin), is a water-soluble vitamin discovered by Roger J. Williams in 1919. For many animals, pantothenic acid is an essential nutrient as it is required to synthesize coenzyme-A (CoA), as well a…

Kategori:
AlanineAlimentary Tract and MetabolismAmino Acids +9
Target Protein:
Pantothenate kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Paquinimod DB13118
small molecule | CAS: 248282-01-1

Paquinimod is developed for the treatment of SLE (Systemic Lupus Erythematosus), which is an autoimmune disease. The disease affects mainly women of fertile age and progresses in flares with relatively symptom free periods in between. Current treatments of SL…

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Protein S100-A9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Parathyroid hormone Approved DB05829
biotech | CAS: 9002-64-6

Parathyroid hormone (PTH) is a single-chain polypeptide composed of 84 amino acids. Available as Preotact, it is an identical form of human recombinant hormome which produced as a fusion protein undergoeing post-translational processing involving the cleava…

Kategori:
Amino Acids, Peptides, and ProteinsCalcium HomeostasisCalcium-Regulating Hormones and Agents +7
Target Protein:
Parathyroid hormone 2 receptorParathyroid hormone/parathyroid hormone-related peptide receptor
Waktu Paruh1.5 hours.
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
biotech | CAS: 172867-62-8

Parathyroid Hormone-Related Protein 1-36 is under investigation in clinical trial NCT00853723 (Comparison Study of Pthrp and PTH to Treat Osteoporosis).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsHormones +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2259927-72-3

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PARPI F-18 DB18657
small molecule | CAS: 1883580-48-0

PARPI F-18 is a diagnostic agent under investigation for use in the management of glioblastoma multiforme.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pascolizumab DB06560
biotech | CAS: 331243-22-2

Pascolizumab (SB 240683) is a humanized anti-interleukin-4 antibody with therapeutic potential in asthma.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Target Protein:
Interleukin-4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PAT-SM6 DB17406
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PBFT02 DB18580
biotech

PBFT02 is a non-replicating recombinant adeno-associated virus serotype 1 vector delivering human GRN gene encoding the protein progranulin.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PBGM01 DB18581
biotech

PBGM01 is a non-replicating recombinant adeno-associated virus serotype hu68 vector, which contains human GLB1 transgene encoding the galactosidase beta 1 enzyme.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PBKR03 DB18138
biotech

PBKR03 is a non-replicating recombinant adeno-associated virus serotype hu68 vector, containing a transgene encoding the human galactosylceramidase (GALC) enzyme.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegaspargase Approved DB00059
biotech | CAS: 130167-69-0

Pegaspargase is a conjugate of monomethoxypolyethylene glycol (mPEG) and L-asparaginase (L-asparagine amidohydrolase), an asparagine-specific enzyme that converts L-asparagine into aspartic acid and ammonia.[L44667] Asparagine is an amino acid that is vital f…

Kategori:
AlcoholsAmidohydrolasesAntineoplastic Agents +15
Target Protein:
L-asparagine
Waktu ParuhThe mean eliminatio…
Vol. DistribusiBased on a non-comp…
KlirensFor a single intram…
Genetik -
Pegfilgrastim Approved DB00019
biotech | CAS: 208265-92-3

Pegfilgrastim is a PEGylated form of the recombinant human granulocyte colony-stimulating factor (G-CSF) analogue, [filgrastim].[A187601] The drug is approved for use to decrease the incidence of infection, as manifested by febrile neutropenia, in susceptible…

Kategori:
Adjuvants, ImmunologicAlcoholsAmino Acids, Peptides, and Proteins +21
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhThe serum half-life…
Vol. DistribusiPegfilgrastim appea…
KlirensPegfilgrastim has a…
Genetik -
Pegilodecakin DB15162
biotech | CAS: 1966111-35-2

Pegilodecakin is under investigation in clinical trial NCT03382912 (Study of Pegilodecakin (LY3500518) With Nivolumab Compared to Nivolumab Alone Second-line Tx in Participants With Metastatic Non-Small Cell Lung Cancer).

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Peginterferon alfa-2a Approved DB00008
biotech | CAS: 198153-51-4

Peginterferon alfa-2a is a form of recombinant interferon used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized in…

Kategori:
Adjuvants, ImmunologicAlcoholsAlfa Interferons +29
Target Protein:
Interferon alpha/beta receptor 2Interferon alpha/beta receptor 1
Gen Terkait:
IFNL3
Waktu ParuhThe mean terminal h…
Vol. Distribusi-
KlirensThe mean systemic c…
Genetik 1 Varian
Peginterferon alfa-2b Approved DB00022
biotech | CAS: 215647-85-1

Peginterferon alfa-2b is a form of recombinant interferon used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized in…

Kategori:
Adjuvants, ImmunologicAlcoholsAlfa Interferons +34
Target Protein:
Interferon alpha/beta receptor 1Interferon alpha/beta receptor 2
Gen Terkait:
IFNL3
Waktu ParuhThe mean half-life …
Vol. Distribusi-
KlirensThe estimated appar…
Genetik 1 Varian
Peginterferon beta-1a Approved DB09122
biotech | CAS: 1211327-92-2

Multiple Sclerosis (MS) is a chronic and inflammatory autoimmune disease of the central nervous system, disrupting communication between the brain and other parts of the body. Most patients diagnosed with this illness experience their initial disease symptoms…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +13
Target Protein:
Interferon alpha/beta receptor 1
Waktu ParuhThe mean half life …
Vol. DistribusiThe volume of distr…
KlirensThe average steady …
Genetik -
Pegsitacianine DB19098
small molecule | CAS: 2396651-85-5

Pegsitacianine is under investigation in clinical trial NCT05576974 (A Phase 2a, Single-dose, Open-label Study to Evaluate Diagnostic Performance and Safety of Pegsitacianine, an Intraoperative Fluorescence Imaging Agent for the Detection of Cancer, in Patien…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegunigalsidase alfa Approved DB14992
biotech | CAS: 1644392-61-9

Pegunigalsidase alfa (PRX-102) is a recombinant form of human ?-galactosidase-A indicated for long-term enzyme replacement therapy in patients with Fabry disease, a rare genetic disorder characterized by the deficiency of alpha-galactosidase A.[A259352,L46342…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +6
Target Protein:
Alpha-galactosidase AGlobotriaosylceramide
Waktu ParuhPegunigalsidase alf…
Vol. DistribusiIn enzyme replaceme…
KlirensPatients treated wi…
Genetik -
Pegvaliase Approved DB12839
biotech | CAS: 1585984-95-7

Pegvaliase is a recombinant phenylalanine ammonia lyase (PAL) enzyme derived from _Anabaena variabilis_ that converts phenylalanine to ammonia and _trans_-cinnamic acid [A33284]. Both the U.S. Food and Drug Administration and European Medicines Agency approve…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAmmonia-Lyases +7
Target Protein:
Phenylalanine-4-hydroxylase
Waktu ParuhFollowing once-dail…
Vol. DistribusiThe mean ± SD (rang…
KlirensAt steady state fol…
Genetik -
Pegvisomant Approved DB00082
biotech | CAS: 218620-50-9

Pegvisomant is a highly selective growth hormone (GH) receptor antagonist. It is used to treat acromegaly. Unlike dopamine or somatostatin analogs (which inhibit growth hormone secretion), this drug actually blocks the hepatic (GH-mediated) production of ins…

Kategori:
AcromegalyAmino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and Analogues +17
Target Protein:
Growth hormone receptor
Waktu Paruh~6 days
Vol. Distribusi* 7 L
Klirens* 36 - 28 mL/h [SC …
Genetik -
biotech | CAS: 1620390-06-8

Pegvorhyaluronidase alfa is under investigation in clinical trial NCT02241187 (Two Stage Study Of Single Dose PEGPH20 And Cetuximab In Patients With Pancreatic Adenocarcinoma Prior To Surgical Resection).

Kategori:
Carbon-Oxygen LyasesEnzymesEnzymes and Coenzymes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1417412-83-9

PEGylated Recombinant Factor VIII is under investigation in clinical trial NCT02585960 (BAX 855 Pk-guided Dosing).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1433787-75-7

Pegylated Recombinant Human Arginase I is under investigation in clinical trial NCT03455140 (A Study Evaluating the Safety and Activity of Pegylated Recombinant Human Arginase (BCT-100)).

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsEnzymes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1350661-05-0

Deskripsi belum tersedia.

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegzilarginase Approved DB14780
biotech | CAS: 1659310-95-8

Pegzilarginase is under investigation in clinical trial NCT02488044 (A Phase 1/2 Study of AEB1102 in Patients With Arginase I Deficiency).

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pelacarsen DB16284
biotech | CAS: 1637637-70-7

Pelacarsen is under investigation in clinical trial NCT03070782 (Phase 2 Study of ISIS 681257 (Akcea-apo(a)-lrx) in Participants With Hyperlipoproteinemia(a) and Cardiovascular Disease).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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