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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 316 / 321
Zaleplon Approved DB00962
small molecule | CAS: 151319-34-5

Zaleplon is a sedative/hypnotic, mainly used for insomnia. It is known as a nonbenzodiazepine hypnotic. Zaleplon interacts with the GABA receptor complex and shares some of the pharmacological properties of the benzodiazepines. Zaleplon is a schedule IV drug …

Kategori:
AcetatesAcids, AcyclicAmides +22
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1
Waktu ParuhApproximately 1 hour
Vol. Distribusi* 1.4 L/kg
Klirens* 1 L/h/kg
Genetik -
Zalifrelimab DB15632
biotech | CAS: 2148321-69-9

Zalifrelimab is under investigation in clinical trial NCT03894215 (Phase 2 Study of Anti-pd-1 Independently or in Combination With Anti-ctla-4 in Second-line Cervical Cancer).

Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

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Zaltoprofen DB06737
small molecule | CAS: 74711-43-6

A non-steroidal anti-inflammatory drug approved for use in Japan in 1993.

Kategori:
Acids, AcyclicAgents causing hyperkalemiaAgents that produce hypertension +19
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Zalunfiban DB18766
small molecule | CAS: 1448313-27-6

Deskripsi belum tersedia.

Waktu Paruh-
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Zalutumumab DB12202
biotech | CAS: 667901-13-5

Zalutumumab is a fully human IgG1 monoclonal antibody designed to bind with selectivity to the epidermal growth factor receptor (EGFR). Zalutumumab has been investigated for the treatment of Squamous Cell Cancer and Head and Neck Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Target Protein:
Epidermal growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zalypsis DB12454
small molecule | CAS: 308359-57-1

Zalypsis has been used in trials studying the treatment of Lymphoma, Solid Tumors, Ewing's Sarcoma, Endometrial Cancer, and Uterine Cervical Cancer, among others.

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingIsoquinolines
Waktu Paruh-
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Genetik -
Zamaporvint DB18765
small molecule | CAS: 1900754-56-4

Deskripsi belum tersedia.

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Zamerovimab DB17766
biotech | CAS: 2419087-87-7

Deskripsi belum tersedia.

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Zamicastat DB12389
small molecule | CAS: 1080028-80-3

Zamicastat has been used in trials studying the treatment of Hypertension and Chronic Heart Failure.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingPyrans
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zampilimab DB16381
biotech | CAS: 2098280-42-1

Zampilimab is under investigation in clinical trial NCT04335578 (A Study to Evaluate Safety, Tolerability, Pharmacokinetics, and Efficacy of UCB7858 in Adult Kidney Transplant Recipients With Chronic Allograft Injury).

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biotech

Deskripsi belum tersedia.

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Zanamivir Approved DB00558
small molecule | CAS: 139110-80-8

A guanido-neuraminic acid that is used to inhibit neuraminidase.

Kategori:
Acids, AcyclicAmidinesAmino Sugars +15
Target Protein:
NeuraminidaseNeuraminidaseSialidase-2
Waktu Paruh2.5-5.1 hours
Vol. Distribusi-
Klirens* 2.5 - 10.9 L/h [F…
Genetik -
Zanapezil DB04859
small molecule | CAS: 142852-50-4

Zanapezil (TAK-147) is a selective acetylcholine (ACh) esterase inhibitor under investigation as a drug for Alzheimer's disease (AD) treatment.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Acetylcholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zandatrigine DB19051
small molecule | CAS: 2154406-04-7

Zandatrigine is under investigation in clinical trial NCT05226780 (Extension Study to Evaluate How Safe and Tolerable NBI-921352 Is as an Adjunctive Therapy for Participants With SCN8A-DEE).

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Zandelisib DB18245
small molecule | CAS: 1401436-95-0

Deskripsi belum tersedia.

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Zanidatamab Approved DB15471
biotech | CAS: 2169946-15-8

Zanidatamab is a bispecific antibody that binds two non-overlapping sites of HER2 (ERBB2).[A264718] It has been investigated for the treatment of HER2-positive solid tumors, including gastroesophageal, colorectal, and biliary tract cancers.[A264718] In No…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Target Protein:
Receptor tyrosine-protein kinase erbB-2
Waktu ParuhBased on population…
Vol. DistribusiBased on population…
KlirensBased on population…
Genetik -
biotech | CAS: 2329698-82-8

According to Zymeworks, "ZW49 (zanidatamab zovodotin) is a bispecific anti-HER2 ADC that is based on the same antibody framework as [ZW25] but armed with a cytotoxic payload."[L8234] It is being investigated for several indications characterized by HER2 expre…

Waktu Paruh-
Vol. Distribusi-
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Zanolimumab DB17376
biotech | CAS: 652153-01-0

Zanolimumab is a fully human monoclonal antibody directed against CD4.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zansecimab DB16389
biotech | CAS: 2415205-37-5

Zansecimab is under investigation in clinical trial NCT04342897 (A Study of LY3127804 in Participants With COVID-19).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Zanthoxylum clava-herculis bark is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
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biotech

Zanthoxylum clava-herculis whole is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Zanubrutinib Approved DB15035
small molecule | CAS: 1691249-45-2

Zanubrutinib is a novel Bruton's tyrosine kinase (BTK) inhibitor used for the treatment of adult patients with mantle cell lymphoma (MCL) who have received at least one prior therapy.[L10163] Mantle cell lymphoma is an aggressive mature B-cell non-Hodgkin lym…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBruton's tyrosine kinase (BTK) inhibitors +19
Target Protein:
Tyrosine-protein kinase BTKEpidermal growth factor receptorReceptor tyrosine-protein kinase erbB-2 +12
Waktu ParuhFollowing administr…
Vol. DistribusiThe geometric mean …
KlirensThe mean (%CV) appa…
Genetik -
Zanzalintinib DB17525
small molecule | CAS: 2367004-54-2

Deskripsi belum tersedia.

Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zapnometinib DB18244
small molecule | CAS: 303175-44-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAminesAminobenzoates +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zardaverine DB02918
small molecule | CAS: 101975-10-4

Deskripsi belum tersedia.

Kategori:
Anti-Asthmatic AgentsAutonomic AgentsBronchodilator Agents +4
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4D
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zasocitinib DB19278
small molecule | CAS: 2272904-53-5

Deskripsi belum tersedia.

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Zastumotide DB14926
biotech | CAS: 949885-73-8

Zastumotide is a recombinant MAGE-A3 Antigen-Specific Cancer Immunotherapeutic (MAGE-A3 ASCI) also known as astuprotimut-R. It is under investigation in clinical trial NCT00257738 (0804 GCC: MAGE-A3/HPV 16 Vaccine for Squamous Cell Carcinoma of the Head and N…

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Zatolmilast DB14790
small molecule | CAS: 1606974-33-7

BPN-14770 is under investigation in clinical trial NCT02840279 (A Multiple Ascending Dose Study of BPN14770 in Healthy Young and Elderly Male or Female Subjects).

Kategori:
Acids, AcyclicEnzyme InhibitorsFatty Acids +5
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4D
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zavegepant Approved DB15688
small molecule | CAS: 1337918-83-8

Zavegepant (BHV-3500) is a calcitonin gene-related peptide (CGRP) receptor antagonist.[L45505] CGRP is released from sensory nerves and acts as a strong vasodilator, and thanks to these properties, it is involved in pain pathways. CGRP receptors are expressed…

Kategori:
Antimigraine PreparationsCalcitonin Gene-Related Peptide (CGRP) AntagonistsCalcitonin Gene-Related Peptide Receptor Antagonists +14
Target Protein:
Calcitonin gene-related peptide type 1 receptor
Waktu ParuhFollowing a 10 mg d…
Vol. DistribusiIntranasal zavegepa…
KlirensIntranasal zavegepa…
Genetik -
ZB131 DB17164
biotech

ZB131 is a monoclonal antibody with a high affinity and specificity for cancer-specific plectin (CSP), a cell surface protein identified in a wide range of cancers that correlates with poor prognosis and aggressive tumors.[L44081]

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ZD-6126 DB11872
small molecule | CAS: 219923-05-4

ZD6126 has been used in trials studying the treatment of Kidney Neoplasms, Colorectal Neoplasms, Metastases, Neoplasm, and Carcinoma, Renal Cell.

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ZD4407 DB06539
small molecule | CAS: 166882-70-8

The drug ZD4407, an antiasthmatic developed by AstraZeneca, functions as a 5-lipoxygenase inhibitor. It entered Phase 1 clinical trials for chronic obstructive pulmonary disease (COPD) in the United Kingdom but was discontinued during this phase in March 2003

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Zeatin DB11337
small molecule | CAS: 1637-39-4

An aminopurine factor in plant extracts that induces cell division. (Grant & Hackh's Chemical Dict, 5th ed)

Kategori:
CytokininsGrowth SubstancesHeterocyclic Compounds, Fused-Ring +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Zeaxanthin Approved DB11176
small molecule | CAS: 144-68-3

Zeaxanthin is a most common carotenoid alcohols found in nature that is involved in the xanthophyll cycle. As a coexistent isomer of lutein, zeaxanthin is synthesized in plants and some micro-organisms. It gives the distinct yellow color to many vegetables an…

Kategori:
AlkenesBiological FactorsCarotenoids +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zebularine DB03068
small molecule | CAS: 3690-10-6

A chemically stable, cytidine analog that displays anti-tumor properties. It acts as a transition state analog inhibitor of cytidine deaminase by binding to the active site as covalent hydrates. Also shown to inhibit DNA methylation and tumor growth both in v…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosidesPyrimidine Nucleosides +2
Target Protein:
Cytidine deaminase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ZED-1227 DB19208
small molecule | CAS: 1542132-88-6

ZED-1227 is under investigation in clinical trial NCT05305599 (Different Doses of ZED1227 vs. Placebo in NAFLD).

Waktu Paruh-
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Zelasudil DB19315
small molecule | CAS: 2365193-22-0

Deskripsi belum tersedia.

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Zelavespib DB12638
small molecule | CAS: 873436-91-0

Zelavespib (PU-H71) has been used in trials studying the treatment of LYMPHOMA, Solid Tumors, Metastatic Solid Tumor, and Myeloproliferative Neoplasms (MPN).

Kategori:
Antineoplastic AgentsDioxolesHeterocyclic Compounds, Fused-Ring
Target Protein:
Heat shock protein HSP 90-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zelpultide alfa DB18587
biotech | CAS: 2245003-06-7

Zelpultide alfa is a recombinant human surfactant protein D.

Waktu Paruh-
Vol. Distribusi-
Klirens-
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Zelquistinel DB19336
small molecule | CAS: 2151842-64-5

Zelquistinel is under investigation in clinical trial NCT06547489 (GATE-251 or Placebo for the Reduction of Symptoms of Major Depressive Disorder).

Waktu Paruh-
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Zeluvalimab DB18868
biotech | CAS: 2315361-37-4

Zeluvalimab is under investigation in clinical trial NCT04631601 (Safety and Efficacy of Therapies for Metastatic Castration-resistant Prostate Cancer (Mcrpc)).

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Zemirciclib DB18823
small molecule | CAS: 2057509-72-3

Deskripsi belum tersedia.

Target Protein:
Cyclin-dependent kinase 9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ZEN-012 DB06042
small molecule

ZEN-012 is a novel small molecule and the first anti-cancer drug in development involving two mechanisms of action: tubulin and topoisomerase II inhibition. ZEN-012 also expresses additional modes of action such as pro-apoptotic and anti-angiogenic properties…

Target Protein:
Tubulin beta chainTubulin beta-1 chainTubulin beta-3 chain +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Zenarestat DB02132
small molecule | CAS: 112733-06-9

Deskripsi belum tersedia.

Kategori:
Aldehyde Reductase, antagonists & inhibitorsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring
Target Protein:
Aldo-keto reductase family 1 member B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Zenocutuzumab Approved DB15559
biotech | CAS: 1969309-56-5

Zenocutuzumab is under investigation in clinical trial NCT03321981 (MCLA-128 With Trastuzumab/chemotherapy in HER2+ and With Endocrine Therapy in ER+ and Low HER2 Breast Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
Vol. Distribusi-
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Zeranol DB11478
small molecule | CAS: 26538-44-3

Zeranol is a non-steroidal estrogen agonist. It is a mycotoxin, derived from fungi in the Fusarium family, and may be found as a contaminant in fungus-infected crops. It is 3-4x more potent as an estrogen agonist than the related compound zearalenone.

Kategori:
Benzene DerivativesEstrogensEstrogens, Non-Steroidal +6
Target Protein:
Estrogen receptorSex hormone-binding globulin
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Zetomipzomib DB16070
small molecule | CAS: 1629677-75-3

Zetomipzomib is under investigation in clinical trial NCT04033926 (A Phase 2 Study of KZR-616 to Evaluate Safety and Efficacy in Patients With Active Polymyositis or Dermatomyositis).

Kategori:
Oxazines
Waktu Paruh-
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biotech

Deskripsi belum tersedia.

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Zibotentan DB06629
small molecule | CAS: 186497-07-4

Deskripsi belum tersedia.

Target Protein:
Endothelin-1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 15751–15800 dari 16004
Sebelumnya Halaman 316 / 321 Berikutnya