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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 315 / 321
XL820 DB05146
small molecule | CAS: 1123889-88-2

XL820 is investigated for use/treatment in solid tumors. XL820 is a solid. The proteins that XL820 inhibit include platelet-derived growth factor receptor beta (PDGFR), mast/stem cell growth factor receptor KIT, vascular endothelial growth factor receptor 2, …

Target Protein:
Vascular endothelial growth factor receptor 2Mast/stem cell growth factor receptor KitPlatelet-derived growth factor receptor alpha +1
Waktu Paruh-
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Genetik -
XL844 DB05149
small molecule

XL844 is investigated for the use and treatment solid tumors. XL844 is a solid. XL844 is a potent inhibitor of the checkpoint kinases CHK1 and CHK2, which induce cell cycle arrest in response to a variety of DNA damaging agents. Known drug targets of XL844 in…

Target Protein:
Serine/threonine-protein kinase Chk2Serine/threonine-protein kinase Chk1
Waktu Paruh-
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XL999 DB05014
small molecule | CAS: 921206-68-0

XL999 has the potential to provide benefit to patients with lung cancer and acute myelogenous leukemia. XL999 is a new chemical entity that inhibits a spectrum of receptor tyrosine kinases (RTKs) with growth promoting and angiogenic properties, including FGFR…

Target Protein:
Fibroblast growth factor receptor 3Fibroblast growth factor receptor 1Vascular endothelial growth factor receptor 2 +3
Waktu Paruh-
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XmAb24306 DB17526
biotech

XmAb24306 is an investigational cancer immunotherapy. It is a heterodimeric interleukin (IL)-15/IL-15-receptor alpha (IL-15Ra) complex fused to a bispecific Fc domain.

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biotech

Deskripsi belum tersedia.

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XMMME-001-RTA DB17203
biotech

Deskripsi belum tersedia.

Kategori:
AlbuminsAmino Acids, Peptides, and ProteinsAntibodies +17
Waktu Paruh-
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XMT-1001 DB06069
small molecule

XMT-1001 is a polymer-based prodrug of camptothecin (CPT), a well-characterized topoisomerase I inhibitor with potent anti-tumor activity. It is a water-soluble macromolecular conjugate of camptothecin (CPT). In this novel CPT pro-drug, CPT is conjugated with…

Kategori:
AcetalsAlkaloidsCompounds used in a research, industrial, or household setting +1
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
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XMT-2056 DB18230
biotech

XMT-2056 is a HER2-targeted antibody-drug conjugate (ADC) consisting of a HER2-targeted antibody conjugated with a stimulator of interferon genes (STING) agonist payload.

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XomaZyme-791 DB17216
biotech

Deskripsi belum tersedia.

Kategori:
AlbuminsAmino Acids, Peptides, and ProteinsAntibodies +17
Waktu Paruh-
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XP-102 DB18780
small molecule | CAS: 1392429-79-6

Deskripsi belum tersedia.

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XPro1595 DB16454
biotech | CAS: 2489785-77-3

XPro1595 is an investigational dominant-negative protein that neutralizes soluble TNF.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Proteins +10
Target Protein:
Tumor necrosis factor
Waktu Paruh-
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XR5944 DB06364
small molecule | CAS: 343247-32-5

XR5944 is a DNA bis-intercalating anticancer drug. It has both intercalating and antineoplastic activities.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
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XTL-001 DB05405
biotech | CAS: 339991-45-6

XTL001 is an investigational monoclonal antibody (MAb) product developed by XTL Biopharmaceuticals to evaluate the safety profile and antiviral activity of the compound in patients chronically infected with hepatitis B virus (HBV).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
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XTL-6865 DB06058
small molecule

XTL-6865 is a combination of two fully human monoclonal antibodies (Ab68 and Ab65) against the hepatitis C virus E2 envelope protein. It is being developed to prevent HCV re-infection following a liver transplant and for the treatment of chronic HCV disease.

Target Protein:
Genome polyprotein
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XTMAB-16 DB18380
biotech

XTMAB-16 is a monoclonal antibody directed against tumour necrosis factor-alpha (TNF?).

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XV638 DB02702
small molecule | CAS: 183854-11-7

Deskripsi belum tersedia.

Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
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Xylazine DB11477
small molecule | CAS: 7361-61-7

Xylazine is a clonidine analog used as a non-opioid tranquilizer in veterinary medicine and as an emetic, especially in cats.[A9095,L42675,A251420] It acts as an agonist at ?2 adrenoceptors; however, its affinity is lower than the one reported for other ?2 ad…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +15
Target Protein:
Alpha-2B adrenergic receptorAlpha-2C adrenergic receptorAlpha-2 adrenergic receptors
Waktu Paruh-
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Xylitol DB11195
small molecule | CAS: 87-99-0

Xylitol is a naturally occurring five-carbon sugar alcohol found in most plant material, including many fruits and vegetables. Xylitol-rich plant materials include birch and beechwood [A22081]. It is widely used as a sugar substitute and in "sugar-free" food …

Kategori:
AlcoholsCarbohydratesCompounds used in a research, industrial, or household setting +8
Target Protein:
Xylose isomeraseXylose isomeraseXylose isomerase +2
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Xylometazoline Approved DB06694
small molecule | CAS: 526-36-3

Xylometazoline is an imidazoline derivative [A228523] with sympathomimetic and nasal decongestant activity. Xylometazoline works by binding to alpha (?)-adrenergic receptors to cause vasoconstriction of nasal blood vessels.[A228508] Xylometazoline is avail…

Kategori:
Adrenergic AgonistsAdrenergic alpha-1 Receptor AgonistsAdrenergic alpha-2 Receptor Agonists +17
Target Protein:
Alpha-2A adrenergic receptorAlpha-2B adrenergic receptorAlpha-1A adrenergic receptor +3
Waktu ParuhNo information is a…
Vol. DistribusiNo information is a…
KlirensNo information is a…
Genetik -
Xylose Approved DB09419
small molecule | CAS: 58-86-6

Xylose is a monosaccharide of the aldopentose type consisted of five carbon atoms and an aldehyde functional group. Xylose is a sugar isolated from wood. D-Xylose is a sugar widely used as a diabetic sweetener in food and beverage. Xylose has also been used a…

Kategori:
CarbohydratesMonosaccharidesPentoses
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe renal clearance…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Exoglucanase/xylanase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Exoglucanase/xylanase
Waktu Paruh-
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Y-27632 DB08756
small molecule | CAS: 146986-50-7

Y-27632 is an inhibitor of Rho-associated protein kinase. It inhibits calcium sensitization to affect smooth muscle relaxation.

Kategori:
Antihypertensive AgentsCardiovascular AgentsCentral Nervous System Agents +6
Target Protein:
ProthrombincAMP-dependent protein kinase catalytic subunit alphacAMP-dependent protein kinase inhibitor alpha +2
Waktu Paruh-
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YA-101 DB18121
small molecule | CAS: 151602-49-2

Deskripsi belum tersedia.

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small molecule | CAS: 9041-22-9

Yeast beta-D-glucan is under investigation in clinical trial NCT00632008 (Soluble Beta-glucan (SBG) as Treatment for Diabetic Foot Ulcers).

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Yellow fever vaccine Approved DB10805
biotech

Yellow fever vaccine prevents against Yellow Fever, a viral hemorrhagic disease caused by the transmission of a _flavivirus_ through the bite of an infected mosquito. Symptoms of Yellow fever can range from asymptomatic, to mild flu-like illness, to more seve…

Kategori:
Actively Acquired ImmunityAntiinfectives for Systemic UseBiological Products +6
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Yellowfin tuna Approved DB15541
biotech

Yellowfin tuna allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
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Yimitasvir DB18768
small molecule | CAS: 1959593-23-7

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntiviral Agents
Waktu Paruh-
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YK-4-279 DB17428
small molecule | CAS: 1037184-44-3

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
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YKP-1358 DB06109
small molecule

YKP1358 is a novel serotonin (5-HT2A) and dopamine (D2) antagonist that has demonstrated potent activity in animals that relates to both positive and negative symptoms of schizophrenia. In addition, the YKP1358 pharmacological profile suggests a very low pote…

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsDopamine Agents +7
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptor
Waktu Paruh-
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Yohimbine Approved DB01392
small molecule | CAS: 146-48-5

A plant alkaloid with alpha-2-adrenergic blocking activity. Yohimbine has been used as a mydriatic and in the treatment of impotence. It is also alleged to be an aphrodisiac.

Kategori:
Adrenergic AgentsAdrenergic alpha-2 Receptor AntagonistsAdrenergic alpha-Antagonists +35
Target Protein:
Alpha-2A adrenergic receptorAlpha-2B adrenergic receptorAlpha-2C adrenergic receptor +9
Waktu ParuhElimination half-li…
Vol. Distribusi-
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YS-ON-001 DB17291
biotech

YS-ON-001 is a combination of an inactivated purified rabies virus (IPRV) and the PIKA adjuvant (Poly I:C, kanamycin and calcium).

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YSIL6 DB05017
small molecule

YSIL6 is a small-molecule drug in development for the treatment of inflammatory diseases, including rheumatoid arthritis and psoriasis. The molecule works by inhibiting TNF-alpha and IL-6 production in T-cells and macrophages, and by inhibiting T-cell prolife…

Target Protein:
Tumor necrosis factorInterleukin-6
Waktu Paruh-
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YT-001 DB18564
small molecule | CAS: 1072301-78-0

Deskripsi belum tersedia.

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Yttrium Y-90 Approved DB13076
small molecule | CAS: 10098-91-6

Yttrium 90 has been investigated for the treatment of Colon Cancer and Colorectal Cancer.

Kategori:
Acids, AcyclicAnti-Inflammatory AgentsElements +11
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biotech | CAS: 943976-23-6

Yttrium Y-90 clivatuzumab tetraxetan is under investigation in clinical trial NCT00603863 (Safety and Efficacy Study of Different Doses of 90Y-hPAM4 Combined With Gemcitabine in Pancreatic Cancer).

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biotech | CAS: 501423-25-2

Deskripsi belum tersedia.

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Genetik -
biotech | CAS: 501423-27-4

Deskripsi belum tersedia.

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Z-160 DB12743
small molecule | CAS: 41332-24-5

Z160 has been used in trials studying the treatment of Postherpetic Neuralgia and Lumbosacral Radiculopathy.

Kategori:
Antiarrhythmic agentsBenzene DerivativesCalcium Channel Blockers +3
Target Protein:
Voltage-dependent calcium channel subunit alpha-2/delta-1
Waktu Paruh-
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Genetik -
Z-Ala Prolinal DB04033
small molecule

Deskripsi belum tersedia.

Target Protein:
Prolyl endopeptidase Pep
Waktu Paruh-
Vol. Distribusi-
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Z-Pro-Prolinal DB03535
small molecule

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Target Protein:
Prolyl endopeptidaseProlyl endopeptidase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 161401-82-7

Non-methylated, competitive, and irreversible inhibitor of caspase 1, as well as other caspases,1 which can be used directly with purified enzymes. It does not require an esterase to hydrolyze the O-methyl ester like the cell-permeable form, Z-Val-Ala-Asp(O-M…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsCaspase Inhibitors +7
Target Protein:
Caspase-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zabedosertib DB18767
small molecule | CAS: 1931994-81-8

Deskripsi belum tersedia.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors +1
Target Protein:
Interleukin-1 receptor-associated kinase 4
Waktu Paruh-
Vol. Distribusi-
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Zabofloxacin DB12479
small molecule | CAS: 219680-11-2

Zabofloxacin has been used in trials studying the treatment of Community Acquired Pneumonia and Chronic Obstructive Pulmonary Disease.

Kategori:
4-QuinolonesHeterocyclic Compounds, Fused-RingQuinolines +1
Waktu Paruh-
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Zafiride DB18371
biotech

Zafiride is a human tumor necrosis factor coupled to the C terminus of CNGRCG peptide.

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Zafirlukast Approved DB00549
small molecule | CAS: 107753-78-6

Zafirlukast is an oral leukotriene receptor antagonist (LTRA) for the maintenance treatment of asthma, often used in conjunction with an inhaled steroid and/or long-acting bronchodilator. It is available as a tablet and is usually dosed twice daily. Another l…

Kategori:
Acids, AcyclicAgents to Treat Airway DiseaseAmides +37
Target Protein:
Cysteinyl leukotriene receptor 1
Waktu Paruh10 hours
Vol. Distribusi* 70 L
Klirens* apparent oral CL=…
Genetik -
biotech | CAS: 2567881-78-9

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
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Zagociguat DB18315
small molecule | CAS: 2201048-82-8

Deskripsi belum tersedia.

Target Protein:
Guanylate cyclase soluble subunit alpha-1Guanylate cyclase soluble subunit beta-1
Waktu Paruh-
Vol. Distribusi-
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Zagotenemab DB16674
biotech | CAS: 2019133-28-7

Zagotenemab is under investigation in clinical trial NCT03518073 (A Study of LY3303560 in Participants With Early Symptomatic Alzheimer's Disease).

Waktu Paruh-
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Zalcitabine Approved DB00943
small molecule | CAS: 7481-89-2

A dideoxynucleoside compound in which the 3'-hydroxyl group on the sugar moiety has been replaced by a hydrogen. This modification prevents the formation of 5' to 3' phosphodiester linkages, which are needed for the elongation of DNA chains, thus resulting in…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +20
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Waktu Paruh2 hours
Vol. Distribusi* 0.304 to 0.734 L/…
Klirens* 285 mL/min [HIV-i…
Genetik -
Menampilkan 15701–15750 dari 16004
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