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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 314 / 321
WP-1122 DB17192
small molecule

WP-1122 is a prodrug of 2-deoxy-D-glucose (2-DG). It was granted FDA orphan designation for the treatment of glioblastoma multiforme.[L47361]

Kategori:
CarbohydratesDeoxy Sugars
Waktu Paruh-
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WP-1301 DB17702
biotech | CAS: 1609460-62-9

WP1301 is a synthetic peptide derived from hFVIII. It binds to an MHC class II molecule and is recognized by a Factor VIII-specific T cell.[L46138]

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WRR-112 DB03691
small molecule

Deskripsi belum tersedia.

Target Protein:
CruzipainCathepsin F
Waktu Paruh-
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WRR-204 DB04502
small molecule

Deskripsi belum tersedia.

Target Protein:
Cruzipain
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WRR-99 DB03573
small molecule

Deskripsi belum tersedia.

Target Protein:
Cathepsin FCruzipain
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WSD-0922 DB17170
small molecule | CAS: 2226552-64-1

Deskripsi belum tersedia.

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WT-1 122 long DB17353
biotech | CAS: 952720-86-4

Deskripsi belum tersedia.

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WT-1 331 long DB17355
biotech | CAS: 935395-34-9

Deskripsi belum tersedia.

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WT-1 427 long DB17354
biotech | CAS: 935395-33-8

Deskripsi belum tersedia.

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WT-1 A1 DB17352
small molecule | CAS: 852243-39-1

Deskripsi belum tersedia.

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WTx-Bortezomib DB17389
biotech

Deskripsi belum tersedia.

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WU-CART-007 DB18617
biotech

WU-CART-007 consists of allogeneic, fratricide-resistant genetically modified T cells transduced with a 2nd generation 4-1BB-CD3z chimeric antigen receptor targeting human CD7.

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WU-NK-101 DB18350
biotech

WU-NK-101 is an allogeneic CD3-depleted, CD56-enriched activated natural killer-cell product

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WVE-003 DB17870
biotech

WVE-003 is an allele-selective antisense oligonucleotide that works to selectively reduce the toxic mutant huntingtin (mHTT) protein.[L46787]

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WVE-N531 DB17848
biotech

Deskripsi belum tersedia.

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WX-UK1 DB05476
small molecule | CAS: 255374-84-6

WX-UK1 is a 3-amidinophenylalanine-based non-cytotoxic small molecule that belongs to a new class of drugs. In animal models, WX-UK1 blocks tumor cell invasion, metastasis and primary tumor growth by inhibiting serine proteases and the urokinase Plasminogen A…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +1
Target Protein:
Urokinase plasminogen activator surface receptor
Waktu Paruh-
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WZB-117 DB16764
small molecule | CAS: 1223397-11-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +3
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X-165 DB18053
small molecule | CAS: 1815589-34-4

Deskripsi belum tersedia.

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X-396 DB13104
small molecule | CAS: 1365267-27-1

X-396 has been used in trials studying the treatment of Advanced Solid Tumors and Non-small Cell Lung Cancer.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsProtein Kinase Inhibitors
Target Protein:
ALK tyrosine kinase receptor
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Xaliproden DB06393
small molecule | CAS: 135354-02-8

Deskripsi belum tersedia.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsNervous System +5
Target Protein:
5-hydroxytryptamine receptor 1A
Waktu Paruh-
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Xaluritamig DB18137
biotech

Xaluritamig is a novel humanized bispecific T cell recruiting antibody cross-reactive to human and nonhuman primate STEAP1 and CD3.

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Xamoterol Approved DB13781
small molecule | CAS: 81801-12-9

Xamoterol is a ?1-adrenoceptor partial agonist that has shown to improve systolic and diastolic function in studies with heart failure patients. It modulates the sympathetic control of the heart but has no agonist action on ?2-adrenoceptors.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-1 Receptor Agonists +14
Target Protein:
Beta-3 adrenergic receptorBeta-1 adrenergic receptor
Waktu Paruh-
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Xanomeline Approved DB15357
small molecule | CAS: 131986-45-3

Schizophrenia is a complex disease involving a number of different neurotransmitters, including serotonin, dopamine, and acetylcholine.[A264509] Positive symptoms (e.g. hallucinations, delusions) have traditionally been attributed to increased dopaminergic ac…

Kategori:
Autonomic AgentsCentral Nervous System AgentsCholinergic Agents +18
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M4Muscarinic acetylcholine receptor M2 +2
Waktu ParuhThe half-life of xa…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
Xanthan gum Approved DB11253
small molecule | CAS: 11138-66-2

Xanthan gum is a polysaccharide gum derived from* Xanthomonas campestris* by a pure-culture fermentation process and purified by recovery with isopropyl alcohol. The major constituents include D-glucose, D-mannose, and D-glucuronic acid. Xanthan gum is a dire…

Kategori:
AntigensAntigens, BacterialBiological Factors +9
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Xanthine DB02134
small molecule | CAS: 69-89-6

A purine base found in most body tissues and fluids, certain plants, and some urinary calculi. It is an intermediate in the degradation of adenosine monophosphate to uric acid, being formed by oxidation of hypoxanthine. The methylated xanthine compounds caffe…

Kategori:
AlkaloidsCytochrome P-450 CYP1A2 SubstratesCytochrome P-450 Substrates +4
Target Protein:
Adenosine receptor A2bPurine nucleoside phosphorylase 2Xanthine phosphoribosyltransferase
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Xanthinol Approved DB09092
small molecule | CAS: 2530-97-4

Xanthinol is a very potent water-soluble derivative of niacin that can be found in diet supplements. It is also known as xanthinol nicotinate. [L1079] Xaninthol is known to be a potent vasodilator that can easily pass through the cell membrane and once inside…

Kategori:
Cardiovascular AgentsHeterocyclic Compounds, Fused-RingNicotinic Acids +6
Target Protein:
NAD(P) transhydrogenase, mitochondrialGlyceraldehyde-3-phosphate dehydrogenaseIsocitrate dehydrogenase [NAD] subunit alpha, mitochondrial +3
Waktu ParuhThe reported elimin…
Vol. DistribusiThe volume of distr…
KlirensThe total body clea…
Genetik -
Xanthohumol DB15359
small molecule | CAS: 6754-58-1

Xanthohumol is under investigation in clinical trial NCT01367431 (Xanthohumol and Metabolic Syndrome).

Kategori:
Angiogenesis InhibitorsAngiogenesis Modulating AgentsAntineoplastic Agents +7
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XAV-19 DB15895
biotech

XAV-19 is an intravenous antibody-based treatment targeted towards SARS-CoV-2 and other coronaviruses[L16553,L16558]. The therapy concept is based on [COVID-19 convalescent plasma]. However, rather than using human plasma, XAV-19 is a heterologous swine glyco…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
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XC221 DB16503
small molecule

XC221 was investigated in clinical trials to treat patients with respiratory infections, including influenza, COVID-19, and other acute viral upper respiratory infections.

Kategori:
Experimental Unapproved Treatments for COVID-19
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Xeligekimab DB18869
biotech | CAS: 2382921-73-3

Xeligekimab is under investigation in clinical trial NCT06028490 (A Study of Il4r? Monoclonal Antibody in Patients With Uncontrolled Seasonal Allergic Rhinitis.).

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Xempritolimod DB19412
biotech | CAS: 2639319-18-7

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
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XEN-2174 DB05012
small molecule | CAS: 701909-57-1

XEN-2174 is a synthetic drug modeled on a peptide from the venom of a cone shell found on Australia's Great Barrier Reef. XEN-2174 represents a new class of molecules, called the chi conopeptides that selectively inhibit the Norepinephrine Transporter (NET). …

Kategori:
Amino Acids, Peptides, and Proteins
Target Protein:
Sodium-dependent noradrenaline transporter
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XEN-D0101 DB06020
small molecule

XEN-D0101 is an investigational drug developed by Xention Inc. for the treatment of Atrial Fibrillation. XEN-D0101 works by being a selective antagonist of the voltage-gated potassium channel Kv1.5.

Kategori:
Kv1.5 Potassium Channel, antagonists & inhibitorsSulfur Compounds
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XEN-D0501 DB18673
small molecule

XEN-D0501 is a tetrahydronaphthyl urea-based selective TRPV1 antagonist being investigated for the treatment of erythromelalgia.

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Xenon DB13453
small molecule | CAS: 7440-63-3

Deskripsi belum tersedia.

Kategori:
Agents that produce hypertensionAnestheticsAnesthetics, General +7
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Xenon Xe-127 Approved DB09461
small molecule | CAS: 13994-19-9

Deskripsi belum tersedia.

Kategori:
ElementsGasesInhalation Diagnostic Agent +6
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Xenon Xe-129 Approved DB17386
small molecule | CAS: 13965-99-6

Hyperpolarized Xenon-129 (Xe-129) is a contrast agent used in the lung's clinical magnetic resonance imaging (MRI). Lung MRIs are challenging due to the low proton density of this tissue, as well as the presence of artifacts due to respiration and cardiovascu…

Kategori:
Contrast MediaDiagnostic Uses of ChemicalsHyperpolarized Contrast Agent +3
Waktu ParuhXenon-129 in a 75% …
Vol. DistribusiXenon is readily di…
KlirensNot available.
Genetik -
Xenon-133 Approved DB09315
small molecule | CAS: 14932-42-4

Xenon-133 is an inhaled radionuclide used for lung imaging, imaging blood flow in the brain, and to assess pulmonary function.

Kategori:
Diagnostic RadiopharmaceuticalsElementsGases +6
Waktu ParuhHalf Life 5.245 days
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Xentuzumab DB14871
biotech | CAS: 1417158-65-6

Xentuzumab is under investigation in clinical trial NCT02191891 (Xentuzumab (BI 836845) Plus Afatinib in Patients With Epidermal Growth Factor Receptor (EGFR) Mutant Non-small Cell Lung Cancer (NSCLC)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Xenysalate DB13815
small molecule | CAS: 3572-52-9

Deskripsi belum tersedia.

Kategori:
DermatologicalsMedicated Shampoos
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Xevinapant DB16305
small molecule | CAS: 1071992-99-8

Deskripsi belum tersedia.

Kategori:
Benzene Derivatives
Target Protein:
E3 ubiquitin-protein ligase XIAPBaculoviral IAP repeat-containing protein 2Baculoviral IAP repeat-containing protein 3 +3
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Xibornol DB13714
small molecule | CAS: 13741-18-9

Deskripsi belum tersedia.

Kategori:
Antibacterials for Systemic UseAntiinfectives for Systemic UseBicyclic Monoterpenes +4
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Ximelagatran Approved DB04898
small molecule | CAS: 192939-46-1

Ximelagatran is an anticoagulant intended to become a replacement for warfarin by overcoming the dietary restrictions, drug interaction, and monitoring issues associated with the former. In 2006, its manufacturer AstraZeneca announced that it would not attemp…

Kategori:
AminesAnticoagulantsAntithrombins +10
Target Protein:
Prothrombin
Waktu Paruh3-5 hours
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Xipamide DB13803
small molecule | CAS: 14293-44-8

Deskripsi belum tersedia.

Kategori:
AmidesAntihypertensive AgentsCardiovascular Agents +6
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small molecule | CAS: 157435-10-4

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
DNA topoisomerase 2-beta
Waktu Paruh-
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XL-888 DB12981
small molecule | CAS: 1149705-71-4

XL888 has been used in trials studying the treatment of Cancer and Melanoma.

Kategori:
Acids, CarbocyclicAza CompoundsHSP90 Heat-Shock Proteins, antagonists & inhibitors
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XL228 DB05184
small molecule

XL228 is a novel anticancer compound designed to inhibit the insulin-like growth factor type-1 receptor (IGF1R), Src and Abl tyrosine kinases – targets that play crucial roles in cancer cell proliferation, survival and metastasis.

Target Protein:
Insulin-like growth factor 1 receptorProto-oncogene tyrosine-protein kinase SrcTyrosine-protein kinase ABL1 +1
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XL281 DB05190
small molecule

XL281 is a novel anticancer compound designed to potently inhibit the RAS/RAF/MEK/ERK signaling pathway. Mutational activation of RAS occurs in about 30 percent of all human tumors, including non-small cell lung, pancreatic, and colon cancer. XL281 is a speci…

Target Protein:
Serine/threonine-protein kinase B-rafRAF proto-oncogene serine/threonine-protein kinase
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XL765 DB05241
small molecule

XL765 is an orally available small molecule that has been shown in preclinical studies to selectively inhibit the activity of phosphoinositide-3 kinase (PI3K) and mammalian target of rapamycin (mTOR). It is being developed by Exelixis, Inc.

Kategori:
AmidesHeterocyclic Compounds, Fused-RingPhosphatidylinositol 3-Kinases, antagonists & inhibitors +2
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform +2
Waktu Paruh-
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XL784 DB04991
small molecule

XL784 is a potent inhibitor of the ADAM-10 metalloprotease enzyme, a target of significant interest because of its important role in blood vessel formation and cell proliferation. XL784 was specifically optimized to be MMP-1 sparing, thus potentially enhancin…

Target Protein:
Disintegrin and metalloproteinase domain-containing protein 10
Waktu ParuhApproximately 8 hou…
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Menampilkan 15651–15700 dari 16004
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