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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
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16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 313 / 321
biotech | CAS: 1165741-01-4

Vorsetuzumab mafodotin is under investigation in clinical trial NCT01677390 (A Phase 1b Study of SGN-75 in Combination With Everolimus in Patients With Renal Cell Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
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Vortioxetine Approved DB09068
small molecule | CAS: 508233-74-7

Vortioxetine is an antidepressant medication indicated for the treatment of major depressive disorder (MDD). It is classified as a serotonin modulator and stimulator (SMS) as it has a multimodal mechanism of action towards the serotonin neurotransmitter syste…

Kategori:
Agents that produce hypertensionAnti-Anxiety AgentsAntidepressive Agents +30
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 3A5-hydroxytryptamine receptor 7 +4
Waktu ParuhMean terminal half­…
Vol. DistribusiThe apparent volume…
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Voruciclib DB15157
small molecule | CAS: 1000023-04-0

Voruciclib is under investigation in clinical trial NCT03547115 (A Phase 1 Study of Voruciclib in Subjects With B-Cell Malignancies or AML).

Kategori:
Antineoplastic AgentsCarbohydratesEnzyme Inhibitors +6
Target Protein:
Cyclin-dependent kinase 4
Waktu Paruh-
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Vosaroxin DB11999
small molecule | CAS: 175414-77-4

Vosaroxin is under investigation for the treatment of Leukemia, Myeloid, Acute.

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsHeterocyclic Compounds, Fused-Ring +1
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
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Vosoritide Approved DB11928
biotech | CAS: 1480724-61-5

Achondroplasia is an autosomal dominant genetic disease and the most common cause of dwarfism in humans.[A242277] It results from a gain-of-function missense mutation in _FGFR3_ that results in a dramatic suppression of bone growth, both in volume and in leng…

Kategori:
Amino Acids, Peptides, and ProteinsC-type Natriuretic Peptide AnalogDrugs Affecting Bone Structure and Mineralization +7
Target Protein:
Atrial natriuretic peptide receptor 2
Waktu ParuhThe mean half-life …
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent c…
Genetik -
Voxelotor Approved DB14975
small molecule | CAS: 1446321-46-5

Voxelotor is a novel hemoglobin S polymerization inhibitor for the treatment of sickle cell disease. This is a genetically inherited condition most prevalent in the Middle East, Africa, and certain parts of India. Sickle cell disease can lead to excruciating …

Kategori:
AldehydesBlood and Blood Forming OrgansCytochrome P-450 CYP2B6 Substrates +7
Target Protein:
Hemoglobin subunit alpha
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe apparent volume…
KlirensThe apparent oral c…
Genetik -
Voxilaprevir Approved DB12026
small molecule | CAS: 1535212-07-7

Voxilaprevir is a Direct-Acting Antiviral (DAA) medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized i…

Kategori:
Acids, AcyclicAmidesAmino Acids +36
Target Protein:
Genome polyproteinGenome polyprotein
Waktu Paruh33 hr [FDA Label]
Vol. Distribusi-
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Voxtalisib DB12400
small molecule | CAS: 934493-76-2

Voxtalisib has been used in trials studying the treatment of Cancer, Melanoma, Lymphoma, Glioblastoma, and Breast Cancer, among others.

Kategori:
AmidesHeterocyclic Compounds, Fused-RingPhosphatidylinositol 3-Kinases, antagonists & inhibitors +2
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformSerine/threonine-protein kinase mTOR
Waktu Paruh-
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VP-14637 DB12195
small molecule | CAS: 235106-62-4

MDT-637 has been investigated for the treatment of Drug Safety.

Kategori:
Benzene DerivativesHydrazines
Waktu Paruh-
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VP025 DB05133
small molecule

VP025, a novel drug formulation based on phospholipid microparticles incorporating phosphatidylglycerol, can inhibit neuroinflammation. VP025 may inhibit immune system activation and protect motoneurons from injury. It also shows the ability to reduce inflamm…

Target Protein:
Interleukin-1 beta
Waktu Paruh-
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VPM1002 DB15801
biotech

The bacille Calmette-Guérin (BCG) vaccine protects against severe extrapulmonary forms of tuberculosis (TB) but does not adequately protect against pulmonary TB -- the most prevalent form of TB. This recombinant BCG, VPM1002, has been created in response and …

Kategori:
Bacterial VaccinesBiological ProductsComplex Mixtures +2
Waktu Paruh-
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VPM4001 DB05089
biotech

VPM4001 is an allogeneic vaccine for treatment of prostate carcinoma. It consists of irradiated human LNCaP cells that have been genetically modified to permanently secrete interferon-? and interleukin-2 (LNCaP/IL-2/IFN-?). Interferon-? enhances presentation …

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VPO-227 DB18004
small molecule | CAS: 1314873-02-3

Deskripsi belum tersedia.

Waktu Paruh-
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VS-4718 DB15273
small molecule | CAS: 1061353-68-1

VS-4718 is under investigation in clinical trial NCT02215629 (Dose Escalation Study in Acute Myeloid or B-Cell Acute Lymphoblastic Leukemia).

Kategori:
AminesFocal Adhesion Protein-Tyrosine Kinases, antagonists & inhibitorsPyridines
Target Protein:
Focal adhesion kinase 1
Waktu Paruh-
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VS-5584 DB12986
small molecule | CAS: 1246560-33-7

VS-5584 has been used in trials studying the treatment of Lymphoma, Metastatic Cancer, and Non Hematologic Cancers.

Kategori:
Heterocyclic Compounds, Fused-RingOxazines
Target Protein:
Target of rapamycin complex 2 subunit MAPKAP1Serine/threonine-protein kinase mTORPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
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VSF-173 DB05753
small molecule

VSF-173 is an oral small molecule. It is an oral compound that has demonstrated effects on animal sleep/wake patterns and gene expression patterns suggestive of a stimulant effect. It is developed for the treatment of excessive sleepiness. Study shows that VS…

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VT-111 DB05646
biotech

VT-111 is a 55 kDa secreted glycoprotein belonging to a superfamily of proteins called SERPINS, which share a general structure and mechanism for proteinase inhibition.

Target Protein:
Tissue-type plasminogen activator
Waktu Paruh-
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VT-1598 DB17757
small molecule | CAS: 2089320-99-8

Deskripsi belum tersedia.

Target Protein:
Lanosterol 14-alpha demethylase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
VTP-194204 DB11806
small molecule | CAS: 220619-73-8

Nrx194204 has been used in trials studying the treatment of Parkinson's Disease and Non-small Cell Lung Cancer.

Kategori:
Fatty AcidsLigandsLipids +1
Target Protein:
Retinoic acid receptor RXR-gamma
Waktu Paruh-
Vol. Distribusi-
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VTP-201227 DB05652
small molecule

VTP-201227 has a novel mechanism of action and is being developed as a topical agent for the treatment of psoriasis with potential extensions into other dermatological indications. It is being developed by Vitae Pharmaceuticals.

Waktu Paruh-
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VTP-27999 DB12416
small molecule | CAS: 942142-51-0

VTP-27999 has been used in trials studying the basic science of Renal Function.

Kategori:
Acids, AcyclicAgents Acting on the Renin-Angiotensin SystemRenin Inhibitors
Target Protein:
Renin
Waktu Paruh-
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VTX-801 DB17646
biotech

VTX-801 is a replication-deficient recombinant adeno-associated viral vector (rAAV) consisting of an AAV liver tropic capsid containing a single-stranded DNA genome carrying a shortened version of the ATP7B gene (ATP7B-minigene). It is being investigated in W…

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VTX-803 DB18271
biotech

Deskripsi belum tersedia.

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Vudalimab DB18833
biotech | CAS: 2329669-72-7

Vudalimab is under investigation in clinical trial NCT05005728 (Xmab®20717 (Vudalimab) Alone or in Combination With Chemotherapy or Targeted Therapy in Patients With Metastatic Castration-resistant Prostate Cancer).

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Vunakizumab DB15154
biotech | CAS: 1792181-33-9

Vunakizumab is under investigation in clinical trial NCT03463187 (Multi-Dose Study of SHR-1314 in Subjects With Moderate-to-severe Plaque Psoriasis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
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Genetik -
Vurolenatide DB18440
biotech | CAS: 2434640-83-0

Vurolenatide is a recombinant fusion protein comprising exenatide and XTEN.

Waktu Paruh-
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Vutiglabridin DB18781
small molecule | CAS: 1800188-47-9

Deskripsi belum tersedia.

Waktu Paruh-
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Vutrisiran Approved DB16699
biotech | CAS: 1867157-35-4

Vutrisiran is a double-stranded small interfering ribonucleic acid (siRNA) that targets wild-type and mutant transthyretin (TTR) messenger RNA (mRNA).[L42065] This siRNA therapeutic is indicated for the treatment of neuropathies associated with hereditary tra…

Kategori:
Antisense OligonucleotidesNervous SystemNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
Transthyretin mRNA
Waktu ParuhThe median half-lif…
Vol. DistribusiBased on a populati…
KlirensThe apparent cleara…
Genetik -
VX-148 DB06103
small molecule

VX-148 is a second-generation, orally administered inhibitor of inosine monophosphate dehydrogenase (IMPDH). The IMPDH enzyme plays a key role in regulating immune response and proliferation of specific cell types, including lymphocytes. VX-148 is a developed…

Kategori:
AmidesBenzene Derivatives
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1Inosine-5'-monophosphate dehydrogenase 2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
VX-702 DB05470
small molecule | CAS: 745833-23-2

VX-702 is a small molecule investigational oral anti-cytokine therapy for treatment of inflammatory diseases, specifically rheumatoid arthritis (RA). It acts as a p38 MAP kinase inhibitor. In the future, VX-702 may be investigated for combination with methotr…

Kategori:
AmidesBenzene Derivatives
Target Protein:
Mitogen-activated protein kinase 14Tumor necrosis factorInterleukin-1 beta +1
Waktu Paruh-
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Genetik -
VX-765 DB05507
small molecule

VX-765 is the orally available prodrug of a potent and selective competitive inhibitor of ICE/caspase-1 (VRT-043198). VX-765 is currently under clinical development for the treatment of inflammatory and autoimmune conditions, as it blocks the hypersensitive r…

Kategori:
Acids, CarbocyclicAmino Acids, Peptides, and ProteinsAminobenzoates +4
Target Protein:
Caspase-1Interleukin-1 beta
Waktu Paruh-
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VXA-CoV2-1 DB16433
biotech

VXA-CoV2-1 is a non-replicating adenoviral vector-based oral tableted vaccine candidate that expresses a SARS-CoV-2 antigen and dsRNA adjuvant[L30493]. This oral vaccine aims to induce immunogenicity through induction of potent serum neutralizing antibodies t…

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VXM01 DB17420
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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VY-HTT01 DB16999
biotech

VY-HTT01 is a gene therapy designed to reduce the expression of huntingtin, thereby altering disease progression. VY-HTT01 is comprised of an adeno-associated virus capsid (AAV1) and a proprietary transgene that harnesses the canonical RNA interference pathwa…

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Warfarin Approved DB00682
small molecule | CAS: 81-81-2

Warfarin is an anticoagulant drug normally used to prevent blood clot formation as well as migration. Although originally marketed as a pesticide (d-Con, Rodex, among others), Warfarin has since become the most frequently prescribed oral anticoagulant in Nort…

Kategori:
4-HydroxycoumarinsAgrochemicalsAnticoagulants +38
Target Protein:
Vitamin K epoxide reductase complex subunit 1Nuclear receptor subfamily 1 group I member 2
Gen Terkait:
CYP2C9 VKORC1 CYP4F2 +2
Waktu ParuhR-warfarin is clear…
Vol. DistribusiVd of 0.14 L/kg.[la…
KlirensClearance of warfar…
Genetik 5 Varian
biotech

Fecal microbiota transplantation (FMT) is effective in enhancing the gut microbiota of patients experiencing a high range of disease states, including Clostridioides difficile (C. diff) infection, Crohn’s disease, and ulcerative colitis. Washed microbiota pre…

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Water Approved DB09145
small molecule | CAS: 7732-18-5

Water (chemical formula: H2O) is a transparent fluid which forms the world's streams, lakes, oceans and rain, and is the major constituent of the fluids of organisms. As a chemical compound, a water molecule contains one oxygen and two hydrogen atoms that are…

Kategori:
DiluentsEENT Drugs, MiscellaneousIrrigating Solutions +2
Waktu Paruh-
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WAY-151693 DB02071
small molecule

Deskripsi belum tersedia.

Kategori:
AmidesAminesHydroxy Acids +3
Target Protein:
Collagenase 3
Waktu Paruh-
Vol. Distribusi-
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Wheat germ oil DB16570
biotech | CAS: 313258-61-6

Deskripsi belum tersedia.

Kategori:
Biological ProductsComplex MixturesLipids +4
Waktu Paruh-
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Whey DB18685
biotech

Whey allergenic extract is used in allergenic testing.

Kategori:
Amino Acids, Peptides, and ProteinsAnimal Proteins, DietaryDairy Products +10
Waktu Paruh-
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White mustard seed Approved DB15606
biotech

White mustard seed allergenic extract is used in allergenic testing.

Waktu Paruh-
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Willardiine DB04129
small molecule | CAS: 21416-43-3

Willardiine is a compound isolated from seeds of _Acacia willariana_.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsPyrimidines +1
Target Protein:
Glutamate receptor 1Glutamate receptor 2
Waktu Paruh-
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WIN 55212-2 DB13950
small molecule | CAS: 131543-22-1

WIN 55,212-2 is a chemical described as an aminoalkylindole derivative, which produces effects similar to those of cannabinoids such as tetrahydrocannabinol (THC) but has an entirely different chemical structure. It is a potent cannabinoid receptor agonist th…

Kategori:
Agents causing hyperkalemiaAgents producing tachycardiaAnalgesics +21
Target Protein:
Cannabinoid receptor 1Cannabinoid receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
WIN-54954 DB08723
small molecule | CAS: 107355-45-3

WIN-54954 is a broad-spectrum antipicornavirus drug.

Target Protein:
Genome polyproteinGenome polyprotein
Waktu Paruh-
Vol. Distribusi-
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Genetik -
WL-1002 DB05346
small molecule

WL-1002 is developed by Winston Laboratories which is a topical cream formulation of 075% zucapaicin (also known as civamide), for the treatment of pain due to osteoarthritis.

Waktu Paruh-
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WNT-974 DB12561
small molecule | CAS: 1243244-14-5

WNT974 has been used in trials studying the treatment of Metastatic Colorectal Cancer and Squamous Cell Carcinoma, Head And Neck.

Kategori:
Enzyme Inhibitors
Target Protein:
Protein-serine O-palmitoleoyltransferase porcupine
Waktu Paruh-
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Wood creosote DB13271
small molecule | CAS: 8021-39-4

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesCough and Cold PreparationsCresols +2
Waktu Paruh-
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Wormwood Approved DB14291
biotech

Wormwood is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
LipidsOils
Waktu Paruh-
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Wortmannin DB08059
small molecule | CAS: 19545-26-7

Wortmannin is a steroid metabolite of _Penicillium funiculosum_ and _Talaromyces wortmannii_ fungi. This drug acts as a nonspecific, covalent inhibitor of phosphoinositide 3-kinase enzymes (PI3Ks).

Kategori:
AndrostadienesAndrostanesAndrostenes +16
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformSerine/threonine-protein kinase PLK1 +2
Waktu Paruh-
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WP-1066 DB12679
small molecule | CAS: 857064-38-1

WP1066 has been used in trials studying the treatment of Melanoma, Brain Cancer, Solid Tumors, and Central Nervous System Neoplasms.

Kategori:
Benzene DerivativesBenzylidene CompoundsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Signal transducer and activator of transcription 3
Waktu Paruh-
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Menampilkan 15601–15650 dari 16004
Sebelumnya Halaman 313 / 321 Berikutnya