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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 311 / 321
Vilastobart DB19327
biotech | CAS: 2760549-50-4

Vilastobart is under investigation in clinical trial NCT04896697 (Vilastobart (XTX101) Monotherapy and Vilastobart and Atezolizumab Combination Therapy in Advanced Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Vilazodone Approved DB06684
small molecule | CAS: 163521-12-8

Vilazodone is a novel compound with combined high affinity and selectivity for the 5-hydroxytryptamine (5-HT) transporter and 5-HT(1A) receptors[Label,A177622]. Vilazodone may also be associated with less sexual dysfunction and weight gain[A6947]. Vilazodone …

Kategori:
Agents that produce hypertensionAntidepressive AgentsAntidepressive Agents Indicated for Depression +26
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 1A
Waktu Paruh25 hours[Label,A384…
Vol. DistribusiVilazodone's volume…
KlirensClearance of vilazo…
Genetik -
Vildagliptin Approved DB04876
small molecule | CAS: 274901-16-5

Vildagliptin (LAF237) is an orally active antihyperglycemic agent that selectively inhibits the dipeptidyl peptidase-4 (DPP-4) enzyme. It is used to manage type II diabetes mellitus, where GLP-1 secretion and insulinotropic effects are impaired.[A232488] By i…

Kategori:
Agents causing angioedemaAlimentary Tract and MetabolismBlood Glucose Lowering Agents +11
Target Protein:
Dipeptidyl peptidase 4
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean volume of …
KlirensAfter intravenous a…
Genetik -
Vilobelimab DB16416
biotech | CAS: 2250440-41-4

Vilobelimab is a chimeric monoclonal immunoglobulin G4 (IgG4) antibody that binds to the soluble form of human C5a with high affinity. It consists of mouse anti-human complement factor 5a (C5a) monoclonal binding sites (variable regions of heavy and light cha…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Complement C5
Waktu ParuhThe elimination hal…
Vol. DistribusiNo information is a…
KlirensNo information is a…
Genetik -
Viloxazine Approved DB09185
small molecule | CAS: 46817-91-8

Viloxazine is a selective norepinephrine reuptake inhibitor.[L41685] For decades, an immediate-release formulation of viloxazine has been used in Europe as an antidepressant. It was first approved in the UK in 1974; however, the immediate-release formulation …

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +46
Target Protein:
Sodium-dependent noradrenaline transporter5-hydroxytryptamine receptor 2B5-hydroxytryptamine receptor 2C +10
Waktu ParuhThe mean (± SD) hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance rate …
Genetik -
Viltolarsen Approved DB15005
biotech | CAS: 2055732-84-6

Duchenne muscular dystrophy (DMD) is an X-linked recessive allelic disorder characterized by a lack of functional dystrophin protein, which leads to progressive ambulatory, pulmonary, and cardiac function and is invariably fatal. A related, albeit a less seve…

Kategori:
Antisense OligonucleotidesMorpholinesMusculo-Skeletal System +5
Target Protein:
DMD gene (exon 53 viltolarsen target site)
Waktu ParuhViltolarsen has a r…
Vol. DistribusiViltolarsen has a s…
KlirensViltolarsen has a r…
Genetik -
Viminol DB13353
small molecule | CAS: 21363-18-8

Deskripsi belum tersedia.

Kategori:
AlcoholsAminesAmino Alcohols +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vimseltinib DB17520
small molecule | CAS: 1628606-05-2

Deskripsi belum tersedia.

Target Protein:
Macrophage colony-stimulating factor 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vinbarbital DB13377
small molecule | CAS: 125-42-8

Deskripsi belum tersedia.

Kategori:
Barbiturates, PlainCentral Nervous System DepressantsHypnotics and Sedatives +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vinblastine Approved DB00570
small molecule | CAS: 865-21-4

Antitumor alkaloid isolated from Vinca rosea. (Merck, 11th ed.)

Kategori:
AlkaloidsAntimitotic AgentsAntineoplastic Agents +37
Target Protein:
Tubulin beta-2A chainTubulin alpha-1A chainTubulin beta chain +4
Waktu ParuhTriphasic: 35 min, …
Vol. Distribusi-
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Genetik -
small molecule | CAS: 61936-68-3

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsVinca Alkaloids
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Vinburnine DB13793
small molecule | CAS: 4880-88-0

Deskripsi belum tersedia.

Kategori:
AlkaloidsCardiovascular AgentsHeterocyclic Compounds, Fused-Ring +7
Target Protein:
Muscarinic acetylcholine receptor M3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vincamine DB13374
small molecule | CAS: 1617-90-9

Vincamine is a monoterpenoid indole alkaloid obtained from the leaves of *Vinca minor* with a vasodilatory property. Studies indicate that vincamine increases the regional cerebral blood flow.

Kategori:
AlkaloidsAntihypertensive AgentsAntineoplastic Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vincristine Approved DB00541
small molecule | CAS: 57-22-7

Vincristine is an antitumor vinca alkaloid isolated from Vinca Rosea. It is marketed under several brand names, many of which have different formulations such as Marqibo (liposomal injection) and Vincasar. Vincristine is indicated for the treatment of acute l…

Kategori:
Agents Causing Muscle ToxicityAlkaloidsAntimitotic Agents +33
Target Protein:
Tubulin beta chainTubulin alpha-4A chain
Waktu ParuhWhen intravenously …
Vol. DistribusiWithin 15 to 30 min…
Klirens-
Genetik -
Vindesine Approved DB00309
small molecule | CAS: 53643-48-4

Vinblastine derivative with antineoplastic activity against cancer. Major side effects are myelosuppression and neurotoxicity. Vindesine is used extensively in chemotherapy protocols (antineoplastic combined chemotherapy protocols).

Kategori:
AlkaloidsAntimitotic AgentsAntineoplastic Agents +19
Target Protein:
Tubulin beta-1 chain
Waktu Paruh24 hours.
Vol. Distribusi-
Klirens-
Genetik -
Vinflunine Approved DB11641
small molecule | CAS: 162652-95-1

Vinflunine is a third-generation member of the vinca alkaloid family with anti-tumour actions. It was first described in 1998 at the Pierre Fabre research center in France. Like other vinca agents, vinflunine is an anti-mitotic agent that induces a cell cycle…

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +14
Target Protein:
Tubulin beta chain
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe terminal volume…
KlirensThe total blood cle…
Genetik -
Vinorelbine Approved DB00361
small molecule | CAS: 71486-22-1

Vinorelbine is an anti-mitotic chemotherapy drug that is used in the treatment of several types of malignancies, including breast cancer and non-small cell lung cancer (NSCLC) [L1998]. It was initially approved in the USA in 1990's for the treatment of NSCLC…

Kategori:
AlkaloidsAntimitotic AgentsAntineoplastic Agents +23
Target Protein:
Tubulin beta chain
Waktu ParuhThe terminal phase …
Vol. DistribusiThe volume of distr…
KlirensThe plasma clearanc…
Genetik -
Vinpocetine DB12131
small molecule | CAS: 42971-09-5

Vinpocetine has been investigated for the treatment of Epilepsy.

Kategori:
Agents causing hyperkalemiaAlkaloidsAntiarrhythmic agents +25
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vintafolide DB05168
small molecule | CAS: 742092-03-1

Vintafolide is a folate-targeted chemotherapeutic conjugate (folate vitamin + vinca alkaloid) in clinical stage development as a treatment for folate-receptor positive cancers.

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +9
Target Protein:
Folate receptor alphaFolate receptor betaFolate receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vinyl ether DB13690
small molecule | CAS: 109-93-3

Deskripsi belum tersedia.

Kategori:
AlkenesAnestheticsAnesthetics, General +5
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Vinylbital DB13770
small molecule | CAS: 2430-49-1

Deskripsi belum tersedia.

Kategori:
Barbiturates, PlainCentral Nervous System DepressantsHypnotics and Sedatives +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vinylglycine DB03214
small molecule | CAS: 70982-53-5

Vinylglycine is an irreversible inhibitor of aspartate aminotransferase.

Kategori:
Amino AcidsAmino Acids, Peptides, and Proteins
Target Protein:
L-amino-acid oxidase1-aminocyclopropane-1-carboxylate synthase-like protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1184-84-5

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicAlkenes +4
Target Protein:
Phosphonoacetaldehyde hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Violaxanthin DB03460
small molecule | CAS: 126-29-4

Deskripsi belum tersedia.

Kategori:
AlkenesBiological FactorsCarotenoids +7
Waktu Paruh-
Vol. Distribusi-
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Viomycin Approved DB06827
small molecule | CAS: 32988-50-4

Viomycin is a tuberactinomycin antibiotic that was used to treat Mycobacterium tuberculosis until it was replaced by the less toxic capreomycin. These drugs bind RNA in bacterial ribosomes and inhibit protein synthesis. Viomycin was derived from the actinomyc…

Kategori:
Agents that produce neuromuscular block (indirect)Amino Acids, Peptides, and ProteinsAnti-Bacterial Agents +8
Target Protein:
16S/23S rRNA (cytidine-2'-O)-methyltransferase TlyA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vipadenant DB06625
small molecule | CAS: 442908-10-3

Deskripsi belum tersedia.

Kategori:
Adenosine A2 Receptor AntagonistsNeurotransmitter AgentsPurinergic Agents +2
Target Protein:
Adenosine receptor A2a
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Viper antivenom Approved DB14114
biotech

Viper antivenom consists of antibodies derived from horses immunized and subsequently developed antibodies against snake venoms. ANAVIP, an equine-derived antivenom made with venom from _Bothrops asper_ and _Crotalus durissus_, was first approved by the FDA o…

Kategori:
Antivenins
Waktu ParuhFollowing intraveno…
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
Genetik -
Vipoglanstat DB18126
small molecule | CAS: 1360622-01-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Viral macrophage inflammatory protein-II (vMIP) is a highly basic protein and human chemokine analog encoded by human herpesvirus-8. The structure of vMIP consists of 71 residues and is a monomer under most conditions. It helps its virus evade the host immune…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-HIV AgentsAnti-Infective Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Viralym-C DB17975
biotech

Viralym-C is an investigational T-cell immunotherapy developed by ViraCyte. It consists of Human Leukocyte Antigen (HLA)-matched cytomegalovirus (CMV)-specific T lymphocytes. It was granted FDA orphan designation in January 2017 and investigated for the treat…

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Virginiamycin DB11476
small molecule | CAS: 11006-76-1

Virginiamycin is a streptogramin antibiotic similar to pristinamycin and quinupristin/dalfopristin. It is a combination of pristinamycin IIA and virginiamycin S1. Virginiamycin is used in the fuel ethanol industry to prevent microbial contamination and in liv…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 21411-53-0

Pristinamycin IIA is a macrolide antibiotic, a member of the streptogramin A group of antibiotics, and one component of pristinamycin. It is produced by Streptomyces graminofaciens and other bacteria.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +4
Target Protein:
Streptogramin A acetyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 23152-29-6

One of the components of virginiamycin, a cyclic polypeptide antibiotic complex from streptomyces virginiae, s. Loidensis, s. Mitakaensis, s. Pristina-spiralis, s. Ostreogriseus, and others. It is used to treat infections with gram-positive organisms and as a…

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesPeptides, Cyclic +1
Target Protein:
Large ribosomal subunit protein eL37
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Virulizin DB17098
biotech | CAS: 216586-46-8

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicBodily SecretionsComplex Mixtures +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Virus Specific T-Cells (VSTs) are a target therapy that are generated for specific viral antigens. These products are generated from virus-naive or virus-experienced autologous or allogenic sources. Antigens identified as an immune target are presented by ant…

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VIS-410 DB19067
biotech | CAS: 2043950-09-8

VIS-410 is under investigation in clinical trial NCT03040141 (Study of Efficacy and Safety of IV VIS410 Plus Oseltamivir Versus Oseltamivir in Hospitalized Adults With Influenza A).

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Visilizumab DB12053
biotech | CAS: 219716-33-3

Visilizumab has been investigated for the treatment of Ulcerative Colitis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vismodegib Approved DB08828
small molecule | CAS: 879085-55-9

Vismodegib is an orally active small molecule that inhibits the hedgehog signaling pathway by binding to and inhibiting the transmembrane protein smoothened homologue (SMO).[A258613,A258618,L45803] It was discovered by high-throughput screening of a library o…

Kategori:
AmidesAminesAniline Compounds +18
Target Protein:
Protein smoothened
Waktu ParuhThe half-life of vi…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Visnadine DB13355
small molecule | CAS: 477-32-7

Deskripsi belum tersedia.

Kategori:
BenzopyransHeterocyclic Compounds, Fused-RingPeripheral Vasodilators +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 934960-96-0

Deskripsi belum tersedia.

Kategori:
AminesBenzoquinonesBenzylammonium Compounds +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vistusertib DB11925
small molecule | CAS: 1009298-59-2

Vistusertib is under investigation for the treatment of Advanced Gastric Adenocarcinoma.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +3
Target Protein:
Target of rapamycin complex 2 subunit MAPKAP1Serine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Visugromab DB18894
biotech | CAS: 2556646-63-8

Visugromab is under investigation in clinical trial NCT06059547 (Neoadjuvant Immunotherapy in Combination With the Anti-gdf-15 Antibody Visugromab (CTL-002) for Treatment of Muscle Invasive Bladder Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VIT-100 DB05865
small molecule

VIT-100 was developed by ItherX Pharmaceuticals of San Diego. In preclinical studies, companyl has shown that VIT-100 inhibits the growth of cells taken from multiple keloid biopsies as compared to the same keloidal cells treated with a control. It is believe…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Vitamin A Approved DB00162
small molecule | CAS: 68-26-8

Retinol and derivatives of retinol that play an essential role in metabolic functioning of the retina, the growth of and differentiation of epithelial tissue, the growth of bone, reproduction, and the immune response. Dietary vitamin A is derived from a varie…

Kategori:
Adjuvants, ImmunologicAlimentary Tract and MetabolismAlkenes +33
Target Protein:
Retinoic acid receptor RXR-gammaApolipoprotein DProstaglandin-H2 D-isomerase +13
Waktu Paruh1.9 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 15713-12-9

Deskripsi belum tersedia.

Target Protein:
5-methyltetrahydrofolate--homocysteine S-methyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Aspartate aminotransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Aspartate aminotransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vitamin D Approved DB11094
small molecule | CAS: 1406-16-2

Vitamin D ultimately comprises a group of lipid-soluble secosteroids responsible for a variety of biological effects, some of which include increasing the intestinal absorption of calcium, magnesium, and phosphate. With reference to human use, there are 2 mai…

Kategori:
Bone Density Conservation AgentsCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +12
Target Protein:
Vitamin D3 receptorVitamin D-binding protein
Waktu ParuhAlthough certain st…
Vol. Distribusi-
KlirensSome studies propos…
Genetik -
Vitamin E Approved DB00163
small molecule | CAS: 59-02-9

In 1922, vitamin E was demonstrated to be an essential nutrient[A32448]. Vitamin E is a term used to describe 8 different fat soluble tocopherols and tocotrienols, alpha-tocopherol being the most biologically active[A176104]. Vitamin E acts as an antioxidant,…

Kategori:
AntioxidantsBasic Ointments and ProtectantsBenzopyrans +23
Target Protein:
SEC14-like protein 4SEC14-like protein 3SEC14-like protein 2 +7
Waktu Paruh44 hours in prematu…
Vol. Distribusi0.41L/kg in prematu…
Klirens6.5mL/hr/kg in prem…
Genetik -
Vitamin K7 DB15664
small molecule | CAS: 83-69-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Menampilkan 15501–15550 dari 16004
Sebelumnya Halaman 311 / 321 Berikutnya