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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 309 / 321
Vatalanib DB04879
small molecule | CAS: 212141-54-3

Vatalanib (PTK787/ZK-222584) is a new oral antiangiogenic molecule that inhibits all known vascular endothelial growth factor receptors. Vatalanib is under investigation for the treatment of solid tumors.

Kategori:
Enzyme InhibitorsProtein Kinase InhibitorsPyridazines +1
Target Protein:
Epidermal growth factor receptorVascular endothelial growth factor receptor 3Vascular endothelial growth factor receptor 2 +1
Waktu ParuhApproximately 6 hou…
Vol. Distribusi-
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Vatelizumab DB12346
biotech | CAS: 1238217-55-4

Vatelizumab has been used in trials studying the treatment of Ulcerative Colitis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
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Vatiquinone DB11917
small molecule | CAS: 1213269-98-7

Vatiquinone has been investigated for the treatment and prevention of Retinopathy, Rett Syndrome, Genetic Disease, Noise-induced Hearing Loss, and Methylmalonic Aciduria and Homocystinuria,Cblc Type.

Kategori:
BenzoquinonesCoenzymesEnzymes and Coenzymes +1
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biotech | CAS: 897936-89-9

Vatreptacog Alfa (Activated) has been used in trials studying the treatment of Haemophilia B, Haemophilia A, Congenital Bleeding Disorder, Haemophilia A With Inhibitors, and Haemophilia B With Inhibitors.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +10
Waktu Paruh-
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VaxSyn DB17827
biotech

VaxSyn HIV-1 is a recombinant form of the HIV envelope protein gp 160 developed by MicroGeneSys and the National Institute of Allergy and Infectious Diseases (NIAID).

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Vayarin Approved DB09328
biotech

Vayarin is a prescription medical food for the clinical dietary management of certain lipid imbalances blamed to be associated with attention deficit hyperactivity disorder (ADHD) in children. Vayarin contains _Lipirinen_, a proprietary composition containing…

Kategori:
Cytochrome P-450 CYP2E1 InhibitorsCytochrome P-450 CYP2E1 Inhibitors (strength unknown)Cytochrome P-450 Enzyme Inhibitors
Waktu ParuhAbout 2h [L1507]
Vol. Distribusi-
KlirensMainly in the feces…
Genetik -
VB-201 DB15259
small molecule | CAS: 630112-41-3

VB-201 is under investigation in clinical trial NCT01001468 (Study to Assess VB-201 in Patients With Psoriasis).

Kategori:
AlcoholsCarbohydratesGlycerophosphates +10
Waktu Paruh-
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VB-309 DB18539
small molecule | CAS: 2699021-75-3

Deskripsi belum tersedia.

Kategori:
Cannabinoids and similars
Waktu Paruh-
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VB-310 DB18537
small molecule | CAS: 2699021-76-4

Deskripsi belum tersedia.

Kategori:
Cannabinoids and similars
Waktu Paruh-
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VB-311 DB18540
small molecule | CAS: 2699021-77-5

Deskripsi belum tersedia.

Kategori:
Cannabinoids and similars
Waktu Paruh-
Vol. Distribusi-
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VB-312 DB18542
small molecule | CAS: 2699021-78-6

Deskripsi belum tersedia.

Kategori:
Cannabinoids and similars
Waktu Paruh-
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VB-313 DB18541
small molecule | CAS: 2699021-79-7

Deskripsi belum tersedia.

Kategori:
Cannabinoids and similars
Waktu Paruh-
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VB10.16 DB17512
biotech

VB10.16 is a novel therapeutic antigen-presenting cell-targeting DNA vaccine developed to treat HPV16-positive cancers. It is composed of three parts, one encodes the E6/E7 fusion protein of human papillomavirus (HPV) type 16 (HPV16), a dimerization entity, a…

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VB2-011 DB05411
biotech

VB2-011 is an antibody developed as an anti-cancer treatment. According to some preclinical studies, it has a potential to inhibit tumour growth in various cancers including lymphoma and melanoma. This drug includes the parent IgM (H11 IgM) and a recombinant …

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VBI-1901 DB18476
biotech

VBI-1901 is a bivalent cytomeglaovirus gB/pp65 enveloped virus-like particles

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VCA-894A DB18609
biotech

VCA-894A is a synthetic 2'-O-methoxyethyl phosphorothioate oligoribonucleotide sodium salt consisting of 19 nucleotide residues with the sequence 5'-MeCMeUGMeUGGAAGMeUGAGGGMeCMeCAG-3'

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VCN-01 DB18193
biotech

VCN-01 is an investigational, genetically modified human adenovirus encoding human PH20.

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vCP2292 DB19292
biotech

vCP2292 is under investigation in clinical trial NCT01982487 (Vaccine Therapy and IDO1 Inhibitor INCB024360 in Treating Patients With Epithelial Ovarian, Fallopian Tube, or Primary Peritoneal Cancer Who Are in Remission).

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VE303 DB17794
biotech

VE303 is under clinical development by Vedanta Biosciences.

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Vebicorvir DB18784
small molecule | CAS: 2090064-66-5

Deskripsi belum tersedia.

Waktu Paruh-
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Vebreltinib DB16823
small molecule | CAS: 1440964-89-5

Deskripsi belum tersedia.

Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
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Vecabrutinib DB16657
small molecule | CAS: 1510829-06-7

Vecabrutinib is under investigation in clinical trial NCT03037645 (Safety, PK, PD, and Antitumor Activity of Vecabrutinib (SNS-062) in B Lymphoid Cancers).

Kategori:
Amines
Target Protein:
Tyrosine-protein kinase BTK
Waktu Paruh-
Vol. Distribusi-
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Vecuronium Approved DB01339
small molecule | CAS: 86029-43-8

Monoquaternary homolog of pancuronium. A non-depolarizing neuromuscular blocking agent with shorter duration of action than pancuronium. Its lack of significant cardiovascular effects and lack of dependence on good kidney function for elimination as well as i…

Kategori:
AndrostanesAndrostanolsAnticholinergic Agents +15
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2
Waktu Paruh51–80 minutes
Vol. Distribusi-
Klirens-
Genetik -
Vedolizumab Approved DB09033
biotech | CAS: 943609-66-3

Vedolizumab is a recombinant humanized IgG1 monoclonal antibody directed against the human lymphocyte ?4?7 integrin, a key mediator of gastrointestinal inflammation implicated in diseases like ulcerative colitis or Crohn's disease.[L48216] ?4?7 integrin facil…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
Integrin alpha-4Integrin beta-7
Waktu ParuhVedolizumab has a l…
Vol. DistribusiSerum apparent volu…
KlirensVedolizumab clearan…
Genetik -
Vedroprevir DB12037
small molecule | CAS: 1098189-15-1

Vedroprevir has been investigated for the treatment of Hepatitis C, Chronic.

Kategori:
Antiviral AgentsHeterocyclic Compounds, Fused-Ring
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 15966-93-5

Deskripsi belum tersedia.

Target Protein:
Vascular endothelial growth factor receptor 2
Waktu Paruh-
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VEGFR2-169 DB16152
small molecule | CAS: 673478-49-4

VEGFR2-169 is under investigation in clinical trial NCT00655785 (Antiangiogenic Peptide Vaccine Therapy With Gemcitabine in Treating Patient With Pancreatic Cancer (Phase1/2)).

Kategori:
Amino Acids, Peptides, and ProteinsCancer VaccinesEnzymes +15
Waktu Paruh-
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Veglin DB05890
small molecule | CAS: 1220118-27-3

VEGF-AS (Veglin) is an anti-angiogenesis non-chemotherapy drug (angiogenesis inhibitor) that was developed by VasGene Therapeutics, Inc. for the treatment of a variety of malignancies including mesothelioma. Veglin is one of several newly developed non-chemot…

Target Protein:
Vascular endothelial growth factor A, long form
Waktu Paruh-
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Velafermin DB06493
small molecule | CAS: 697766-75-9

Velafermin was a novel investigational protein therapeutic, also known as fibroblast growth factor-20 (FGF-20), which promotes both epithelial and mesenchymal cell proliferation in vitro and has demonstrated activity in multiple animal models. Velafermin was …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +2
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Velaglucerase alfa Approved DB06720
biotech | CAS: 884604-91-5

Velaglucerase alfa is a gene-activated human recombinant glucocerebrosidase used for the treatment of Type 1 Gaucher disease, caused by a deficiency of the lysosomal enzyme glucocerebrosidase. Additionally, Velaglucerase alfa has also been investigated for us…

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes +1
Target Protein:
Lysosomal acid glucosylceramidase
Waktu Paruh11-12 minutes.
Vol. DistribusiThe mean volume of …
KlirensMean clearance rang…
Genetik -
Veldoreotide DB12777
biotech | CAS: 252845-37-7

Somatoprim is under investigation for the treatment of Acromegaly.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +8
Waktu Paruh-
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Veledimex DB12170
small molecule | CAS: 1093130-72-3

Veledimex has been used in trials studying the treatment of Glioblastoma Multiforme, Metastatic Breast Cancer, and Anaplastic Oligoastrocytoma.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
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Veliflapon DB16346
small molecule | CAS: 128253-31-6

Veliflapon is under investigation in clinical trial NCT00353067 (Veliflapon (Dg-031)to Prevent Heart Attacks or Stroke in Patients With a History of Heart Attack or Unstable Angina).

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +7
Target Protein:
Arachidonate 5-lipoxygenase-activating protein
Waktu Paruh-
Vol. Distribusi-
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Veligrotug DB18976
biotech | CAS: 2728655-31-8

Veligrotug is under investigation in clinical trial NCT00791544 (Dose Finding Study of AVE1642 in Patients With Advanced or Metastatic Liver Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
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Klirens-
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Veliparib DB07232
small molecule | CAS: 912444-00-9

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsEnzyme Inhibitors +3
Target Protein:
Poly [ADP-ribose] polymerase 1Poly [ADP-ribose] polymerase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Velmanase alfa Approved DB12374
biotech | CAS: 1492823-75-2

Velmanase alfa is a recombinant human lysosomal alpha-mannosidase developed for enzyme replacement therapy to treat alpha-mannosidosis. Alpha-mannosidosis is a rare autosomal recessive lysosomal storage disorder. Patients with alpha-mannosidosis have a geneti…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +2
Waktu ParuhAt the end of intra…
Vol. DistribusiThe steady-state vo…
KlirensThe mean clearance …
Genetik -
Velmupressin DB18783
small molecule | CAS: 1647119-61-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
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Velneperit DB12889
small molecule | CAS: 342577-38-2

Velneperit has been used in trials studying the treatment of Obesity.

Target Protein:
Neuropeptide Y receptor type 5
Waktu Paruh-
Vol. Distribusi-
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Velpatasvir Approved DB11613
small molecule | CAS: 1377049-84-7

Velpatasvir is a Direct-Acting Antiviral (DAA) medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized in…

Kategori:
Acids, AcyclicAnti-Infective AgentsAntiinfectives for Systemic Use +22
Target Protein:
Nonstructural protein 5A
Waktu Paruh15h [FDA Label].
Vol. Distribusi1.4-1.6 L/kg [A191…
KlirensEstimated 0.12 L/h/…
Genetik -
Velsecorat DB16347
small molecule | CAS: 1196509-60-0

Velsecorat is under investigation in clinical trial NCT02479412 (A Multiple Dosing (14 Days) Study to Assess Efficacy and Safety of Three Dose Levels of AZD7594, Given Once Daily by Inhalation, in Patients With Mild to Moderate Asthma).

Kategori:
Dioxins and Dioxin-like CompoundsHeterocyclic Compounds, Fused-RingPyrazoles
Waktu Paruh-
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Veltuzumab DB05656
biotech | CAS: 728917-18-8

Veltuzumab is a monoclonal antibody which, as of October 2009, is undergoing Phase I/II clinical trials for the treatment of non-Hodgkin's lymphoma.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Velusetrag DB12702
small molecule | CAS: 866933-46-2

Velusetrag has been used in trials studying the treatment of Gastroparesis and Alzheimer's Disease. It is a highly selective serotonin receptor agonist effective in patients with chronic constipation. It is being developed by Theravance. Velusetrag was discov…

Kategori:
Aza Compounds
Target Protein:
5-hydroxytryptamine receptor 4
Waktu Paruh-
Vol. Distribusi-
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Vemircopan DB18012
small molecule | CAS: 2086178-00-7

Deskripsi belum tersedia.

Target Protein:
Complement factor D
Waktu Paruh-
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Vemurafenib Approved DB08881
small molecule | CAS: 918504-65-1

Vemurafenib is a competitive kinase inhibitor with activity against BRAF kinase with mutations like V600E.[A31269] It exerts its function by binding to the ATP-binding domain of the mutant BRAF.[A31270] Vemurafenib was co-developed by Roche and Plexxikon and …

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +41
Target Protein:
Serine/threonine-protein kinase B-raf
Waktu ParuhThe elimination hal…
Vol. DistribusiThe estimation of t…
KlirensThe total body clea…
Genetik -
Venadaparib DB17105
small molecule | CAS: 1681017-83-3

Deskripsi belum tersedia.

Waktu Paruh-
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Venanprubart DB18891
biotech | CAS: 2635407-50-8

Venanprubart is under investigation in clinical trial NCT05781451 (Anti-btla Agonist Therapy in Subjects With Primary Sjogren's Syndrome).

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Venetoclax Approved DB11581
small molecule | CAS: 1257044-40-8

Venetoclax is a BCL-2 inhibitor that was initially approved by the FDA in April 2016 [FDA label]. Proteins in the B cell CLL/lymphoma 2 (BCL-2) family are important regulators of the apoptotic (programmed cell death) process [A18565], [A18566]. Venetoclax is…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +19
Target Protein:
Apoptosis regulator Bcl-2
Waktu ParuhThe half-life of ve…
Vol. DistribusiThe population esti…
KlirensMainly hepatic [FDA…
Genetik -
Venglustat DB14966
small molecule | CAS: 1401090-53-6

Venglustat is under investigation in clinical trial NCT01674036 (Safety, Tolerability and Pharmacokinetics of Genz-682452 in Healthy Men).

Kategori:
Acids, AcyclicEnzyme Inhibitors
Target Protein:
Ceramide glucosyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Venlafaxine Approved DB00285
small molecule | CAS: 93413-69-5

Venlafaxine is an antidepressant and a serotonin and norepinephrine reuptake inhibitor (SNRI). Its active metabolite, [desvenlafaxine], works by blocking the reuptake of serotonin and norepinephrine, which are key neurotransmitters in mood regulation. Venlafa…

Kategori:
Agents producing tachycardiaAgents that reduce seizure thresholdAmines +39
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporterSodium-dependent dopamine transporter
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +2
Waktu ParuhThe apparent elimin…
Vol. DistribusiThe apparent volume…
KlirensMean ± SD plasma ap…
Genetik 5 Varian
biotech | CAS: 2724922-85-2

Deskripsi belum tersedia.

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Menampilkan 15401–15450 dari 16004
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