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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 308 / 321
Valganciclovir Approved DB01610
small molecule | CAS: 175865-60-8

Valganciclovir hydrochloride (Valcyte, manufactured by Roche) is an antiviral medication used to treat cytomegalovirus infections. As the L-valyl ester of ganciclovir, it is actually a prodrug for ganciclovir. After oral administration, it is rapidly converte…

Kategori:
Agents that reduce seizure thresholdAnti-Infective AgentsAntiinfectives for Systemic Use +13
Target Protein:
DNA polymerase catalytic subunitDNA
Waktu ParuhApproximately 4.08 …
Vol. Distribusi* 0.703 ± 0.134 L/kg
Klirens* 3.07+/- 0.64 mL/m…
Genetik -
small molecule | CAS: 238401-16-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1034190-08-3

Valiltramiprosate is under investigation in clinical trial NCT06304883 (Long-term Extension of Phase 3 Study of ALZ- 801 in APOE4/4 Early AD Subjects).

Kategori:
AlkanesAlkanesulfonic AcidsAmino Acids +7
Target Protein:
Amyloid-beta precursor protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valine Approved DB00161
small molecule | CAS: 72-18-4

Valine is a branched-chain essential amino acid that has stimulant activity. It promotes muscle growth and tissue repair. It is a precursor in the penicillin biosynthetic pathway.

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Essential +4
Target Protein:
Propionyl-CoA carboxylase beta chain, mitochondrialBranched-chain-amino-acid aminotransferase, cytosolicValine--tRNA ligase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 897937-73-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valinomycin DB14057
small molecule | CAS: 2001-95-8

A cyclododecadepsipeptide ionophore antibiotic produced by Streptomyces fulvissimus and related to the enniatins. It is composed of 3 moles each of L-valine, D-alpha-hydroxyisovaleric acid, D-valine, and L-lactic acid linked alternately to form a 36-membered …

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valnoctamide DB13099
small molecule | CAS: 4171-13-5

Valnoctamide has been used in trials studying the treatment of Mania and Schizoaffective Disorder, Manic Type.

Kategori:
Central Nervous System DepressantsHypnotics and SedativesNervous System +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valoctocogene roxaparvovec Approved DB15561
biotech | CAS: 1819334-78-5

Valoctocogene roxaparvovec is an adeno-associated virus serotype 5 (AAV5) based gene therapy vector that expresses the B-domain deleted SQ form of human coagulation factor VIII (hFVIII-SQ).[L43282] The expression of hFVIII-SQ is driven by a liver-specific pro…

Kategori:
Adeno-associated Viral Vector TherapiesAmino Acids, Peptides, and ProteinsBiological Factors +9
Target Protein:
Coagulation factor VIII (F8)
Waktu Paruh-
Vol. Distribusi-
KlirensThe maximum time to…
Genetik -
Valomaciclovir DB06575
small molecule | CAS: 195157-34-7

Deskripsi belum tersedia.

Kategori:
Antiviral AgentsHerpes ZosterHeterocyclic Compounds, Fused-Ring +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 195156-77-5

Valomaciclovir stearate is under investigation in clinical trial NCT00831103 (A Phase 2b Trial of EPB-348 for the Treatment of Herpes Zoster).

Kategori:
Antiviral AgentsHerpes ZosterHeterocyclic Compounds, Fused-Ring +4
Target Protein:
DNA polymerase catalytic subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valopicitabine DB13920
small molecule | CAS: 640281-90-9

The 3-O-valine ester prodrug of the nucleoside analog 2'-C-methylcytidine with anti-hepatitis C virus (HCV) activity. Upon administration, valopicitabine is converted into 2'-C-methylcytidine; upon phosphorylation into its 5-triphosphate form, this metabolite…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosidesPyrimidines
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valproate bismuth Approved DB13910
small molecule | CAS: 60364-28-5

Valproate bismuth is available in Canada in the over-the-counter medication Neo-Laryngobis.

Kategori:
Bismuth containing drugsEENT Drugs, MiscellaneousNeurotoxic agents +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valproic acid Approved DB00313
small molecule | CAS: 99-66-1

Valproic acid, or valproate, is an fatty acid derivative and anticonvulsant originally synthesized in 1881 by Beverly S. Burton.[A178051] It enjoyed use as a popular organic solvent in industry and pharmaceutical manufacturing for nearly a century. In 1963, a…

Kategori:
Acids, AcyclicAnti-epileptic AgentAnticonvulsants +68
Target Protein:
4-aminobutyrate aminotransferase, mitochondrialGlycogen synthase kinase-3 alphaHistone deacetylase 9 +13
Gen Terkait:
POLG POLG
Waktu Paruh13-19 hours.[label]…
Vol. Distribusi11 L/1.73m<sup>2</s…
Klirens0.56 L/hr/m<sup>2</…
Genetik 2 Varian
Valrocemide DB06657
small molecule | CAS: 92262-58-3

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, Peptides, and Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valrubicin Approved DB00385
small molecule | CAS: 56124-62-0

Valrubicin (N-trifluoroacetyladriamycin-14-valerate) is a chemotherapy drug commonly marketed under the trade name VALSTAR. It is a semisynthetic analog of the [doxorubicin], which is an anthracycline drug. Used in the treatment of the bladder cancer, valrub…

Kategori:
Anthracycline Topoisomerase InhibitorAnthracyclinesAnthracyclines and Related Substances +9
Target Protein:
DNADNA topoisomerase 2-betaDNA topoisomerase 2-alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valsartan Approved DB00177
small molecule | CAS: 137862-53-4

Valsartan belongs to the angiotensin II receptor blocker (ARB) family of drugs, which also includes [telmisartan], [candesartan], [losartan], [olmesartan], and [irbesartan]. ARBs selectively bind to angiotensin receptor 1 (AT1) and prevent the protein angiote…

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +22
Target Protein:
Type-1 angiotensin II receptor
Waktu ParuhAfter intravenous (…
Vol. DistribusiThe steady-state vo…
KlirensFollowing intraveno…
Genetik -
Valspodar DB11869
small molecule | CAS: 121584-18-7

Valspodar has been used in trials studying the treatment of Cancer, Sarcoma, Leukemia, Lymphoma, and Breast Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsATP Binding Cassette Transporter, Subfamily B, Member 1Drug Resistance, Multiple +6
Target Protein:
Coagulation factor X
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valtorcitabine DB06187
small molecule | CAS: 380886-95-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Valziflocept DB17728
biotech | CAS: 1804910-11-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vamifeport DB17692
small molecule | CAS: 2095668-10-1

Vamifeport is being investigated for the treatment of beta-thalassemia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vamikibart DB18896
biotech | CAS: 2744320-12-3

Vamikibart is under investigation in clinical trial NCT05642312 (A Study to Investigate Vamikibart in Participants With Uveitic Macular Edema).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Vamorolone Approved DB15114
small molecule | CAS: 13209-41-1

Vamorolone is a novel and fully synthetic glucocorticoid developed by Santhera Pharmaceuticals. It is used to manage inflammation and immune dysregulation in patients with Duchenne muscular dystrophy (DMD), a neuromuscular disorder characterized by the insidi…

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroids +20
Target Protein:
Glucocorticoid receptorMineralocorticoid receptor
Waktu ParuhThe terminal elimin…
Vol. DistribusiBased on population…
KlirensBased on population…
Genetik -
Vamotinib DB15396
small molecule | CAS: 1416241-23-0

Vamotinib (PF-114) is under investigation in clinical trial NCT02885766 (Study to Evaluate Tolerability, Safety, Pharmacokinetics and Preliminary Efficacy of PF-114 for Oral Administration in Adults With Ph+ Chronic Myeloid Leukemia, Which is Resistant to the…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vanadium Approved DB13971
small molecule | CAS: 7440-62-2

Deskripsi belum tersedia.

Kategori:
Diet, Food, and NutritionElementsFood +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vancomycin Approved DB00512
small molecule | CAS: 1404-90-6

Antibacterial obtained from Streptomyces orientalis. It is a glycopeptide related to ristocetin that inhibits bacterial cell wall assembly and is toxic to kidneys and the inner ear. As of January 29 2018, CutisPharma's Firvanq is the only FDA approved vanc…

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAmino Acids, Peptides, and Proteins +17
Target Protein:
D-Ala-D-Ala moiety of NAM/NAG peptide subunits of peptidoglycan
Waktu ParuhHalf-life in normal…
Vol. DistribusiThe volume of distr…
KlirensThe mean plasma cle…
Genetik -
Vandetanib Approved DB05294
small molecule | CAS: 443913-73-3

Vandetanib is an oral once-daily kinase inhibitor of tumour angiogenesis and tumour cell proliferation with the potential for use in a broad range of tumour types. On April 6 2011, vandetanib was approved by the FDA to treat nonresectable, locally advanced…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +15
Target Protein:
Vascular endothelial growth factor receptor 2Proto-oncogene tyrosine-protein kinase receptor RetEpidermal growth factor receptor +3
Waktu ParuhMedian half life of…
Vol. DistribusiVd of about 7450 L.
Klirens-
Genetik -
biotech | CAS: 2382896-00-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vanillic acid DB02130
small molecule | CAS: 121-34-6

A flavoring agent. It is the intermediate product in the two-step bioconversion of ferulic acid to vanillin. (J Biotechnol 1996;50(2-3):107-13).

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +5
Target Protein:
Chorismate pyruvate-lyase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 498-00-0

Vanillyl alcohol has been used in trials studying the treatment of Smoking.

Kategori:
AlcoholsBenzene DerivativesBenzyl Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vanillyl butyl ether Approved DB11299
small molecule | CAS: 82654-98-6

Vanillyl butyl ether is an ether of monohydroxybenzoic acid. It is added to food products as a flavoring agent. It is also present in cosmetics and personal care products as a fragrance ingredient, oral care agent, hair conditioning agent, and warming or cool…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vaniprevir DB11929
small molecule | CAS: 923590-37-8

Vaniprevir has been used in trials studying the treatment and diagnostic of Hepatitis C, Chronic Hepatitis C, Hepatitis C, Chronic, Chronic Hepatitis C Infection, and Chronic Genotype 1 Hepatitis C Virus Infection.

Kategori:
AmidesAmino AcidsAmino Acids, Branched-Chain +9
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vanoxerine DB03701
small molecule | CAS: 67469-69-6

Vanoxerine is a highly selective dopamine transporter antagonist. It was synthesized in the late 1970s and developed as a potential treatment for depression.[A19824] Vanoxerine was later evaluated as a potential treatment for cocaine addiction due to its abil…

Kategori:
Antiarrhythmic agentsCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +6
Target Protein:
Sodium-dependent dopamine transporterHERG human cardiac K+ channel
Waktu ParuhThe mean eliminatio…
Vol. DistribusiVanoxerine is capab…
KlirensAt 25, 75 and 125 m…
Genetik -
Vantictumab DB12956
biotech | CAS: 1345009-45-1

Vantictumab has been used in trials studying the treatment of Solid Tumors, Pancreatic Cancer, and Stage IV Pancreatic Cancer.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vanucizumab DB12317
biotech | CAS: 1448221-05-3

Vanucizumab has been used in trials studying the treatment of ColoRectal Cancer and Advanced/Metastatic Solid Tumors.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Angiopoietin-2Vascular endothelial growth factor A, long form
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 886584-10-7

Vanutide cridificar has been investigated for the treatment of Alzheimer Disease.

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vanzacaftor DB18373
small molecule | CAS: 2374124-49-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vapitadine DB05738
small molecule | CAS: 793655-64-8

Vapitadine is an antihistamine that Barrier Therapeutics is developing as a treatment for allergic reactions of the skin, such as those associated with hives and for the itch associated with atopic dermatitis. An advantage of vapitadine over other antihistami…

Target Protein:
Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vapreotide DB04894
biotech | CAS: 103222-11-3

Vapreotide is a synthetic octapeptide somatostatin analog. It was being studied for the treatment of cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAntineoplastic Agents +20
Target Protein:
Somatostatin receptor type 2Somatostatin receptor type 5Substance-P receptor
Waktu Paruh30 minutes
Vol. Distribusi-
Klirens-
Genetik -
Vardenafil Approved DB00862
small molecule | CAS: 224785-90-4

Vardenafil is a selective inhibitor of cyclic guanosine monophosphate (cGMP)-specific phosphodiesterase type 5 (PDE5) and an oral therapy for the treatment of erectile dysfunction.[L45563,L45568] During sexual stimulation, nitric oxide (NO) is released from n…

Kategori:
Cardiovascular AgentsCytochrome P-450 CYP2C19 InhibitorsCytochrome P-450 CYP2C19 Inhibitors (weak) +30
Target Protein:
cGMP-specific 3',5'-cyclic phosphodiesteraseRetinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gammaRetinal cone rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma
Waktu ParuhVardenafil and its …
Vol. DistribusiVardenafil has a st…
KlirensVardenafil has a to…
Genetik -
Varenicline Approved DB01273
small molecule | CAS: 249296-44-4

Varenicline is a prescription medication used to treat smoking addiction. This medication is the first approved nicotinic receptor partial agonist. Specifically, varenicline is a partial agonist of the alpha4/beta2 subtype of the nicotinic acetylcholine recep…

Kategori:
BenzazepinesCholinergic AgentsCholinergic Agonists +17
Target Protein:
Neuronal acetylcholine receptor subunit alpha-4Neuronal acetylcholine receptor subunit alpha-7Neuronal acetylcholine receptor subunit alpha-3 +2
Waktu ParuhThe elimination hal…
Vol. Distribusi-
Klirens-
Genetik -
Varespladib DB11909
small molecule | CAS: 172732-68-2

Varespladib has been investigated for the treatment and prevention of Sickle Cell Disease, Vaso-occlusive Crisis, and Acute Coronary Syndrome.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +4
Target Protein:
Phospholipase A2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 172733-08-3

Varespladib methyl has been investigated for the treatment of Acute Coronary Syndrome. Studies showed that Varespladib methyl treatment resulted in significant positive changes on lipoproteins and inflammation.

Kategori:
Acids, AcyclicEnzyme InhibitorsFatty Acids +4
Target Protein:
Phospholipase A2, membrane associatedGroup 10 secretory phospholipase A2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Live attenuated zoster vaccine is available as two products: Zostavax for the prevention of shingles in immunocompetent people over the age of 50, and Varivax for the prevention of chickenpox in individuals 12 months of age and older. While the two vaccines c…

Kategori:
Actively Acquired ImmunityAntiinfectives for Systemic UseBiological Products +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Recombinant zoster vaccine, manufactured as the product Shingrix by GlaxoSmithKline, is an adjuvanted non-live recombinant vaccine indicated for prevention of shingles. First approved in October 2017 by the Food and Drug Administration, Shingrix is the prefer…

Kategori:
VaccinesVaricella Zoster Vaccines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Varlilumab DB11930
biotech | CAS: 1393344-72-3

Varlilumab has been used in trials studying the treatment of MELANOMA, Skin Ulcer, Burkett's Lymphoma, Mantle cell lymphoma, and Any T-cell Malignancy, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Varlitinib DB05944
small molecule | CAS: 845272-21-1

Varlitinib is an oral, selective, reversible, small molecule tyrosine kinase inhibitor of both ErbB-2 (Her-2/neu) and EGFR. Over-expression of ErbB-2 and EGFR receptors in tumors is predictive of poor prognosis in cancer patients. Varlitinib has shown signifi…

Kategori:
Heterocyclic Compounds, Fused-RingSulfur Compounds
Target Protein:
Epidermal growth factor receptorReceptor tyrosine-protein kinase erbB-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Varoglutamstat DB18785
small molecule | CAS: 1276021-65-8

Deskripsi belum tersedia.

Target Protein:
Glutaminyl-peptide cyclotransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 37221-79-7

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsCardiovascular AgentsCentral Nervous System Agents +13
Target Protein:
Vasoactive intestinal polypeptide receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vasomera DB16498
small molecule

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiopolymersCardiovascular Agents +26
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vasopressin Approved DB00067
biotech | CAS: 11000-17-2

Vasopressin (arginine-vasopressin or antidiuretic hormone) is a nonapeptide primarily produced in the hypothalamus that exhibits diverse physiological functions related to diuresis, hemodynamic modulation, and behaviour.[A110, A111, A112, A113, A228008] Vasop…

Kategori:
Amino Acids, Peptides, and ProteinsAntidiuretic AgentsArginine Vasopressin +22
Target Protein:
Vasopressin V2 receptorVasopressin V1a receptorVasopressin V1b receptor +1
Waktu ParuhVasopressin adminis…
Vol. Distribusi-
KlirensVasopressin has a c…
Genetik -
Menampilkan 15351–15400 dari 16004
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