Hasil Filter

16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (16004)

Halaman 306 / 321
Ulixacaltamide DB18788
small molecule | CAS: 1199236-64-0

Deskripsi belum tersedia.

Kategori:
Antiarrhythmic agentsCalcium Channel BlockersCalcium-Regulating Hormones and Agents +2
Target Protein:
Voltage-dependent T-type calcium channel subunit alpha-1H
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ulixertinib DB13930
small molecule | CAS: 869886-67-9

Ulixertinib is a a novel, reversible, ATP-competitive ERK1/2 inhibitor with high potency and ERK1/2 selectivity [A31474]. It is currently in clinical trials for the treatment of a wide range of tumors.

Kategori:
AminesPyridines
Target Protein:
Ephrin type-B receptor 2Mitogen-activated protein kinase 3Mitogen-activated protein kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ulobetasol Approved DB00596
small molecule | CAS: 98651-66-2

Ulobetasol is a highly potent corticosteroid.[A215597] It is structurally related to [clobetasol].[A215597] Due to its high potency, it is mainly prescribed in the treatment of severe plaque psoriasis and corticosteroid responsive dermatoses.[L15047,L15052,L1…

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsAntipsoriatics +15
Target Protein:
Steroid hormone receptor ERR1Steroid hormone receptor ERR2Estrogen-related receptor gamma +1
Waktu Paruh_In vitro_ experime…
Vol. Distribusi-
Klirens-
Genetik -
Ulocuplumab DB12018
biotech | CAS: 1375830-34-4

Ulocuplumab is under investigation in Solid Tumor.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Target Protein:
C-X-C chemokine receptor type 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ulodesine DB12353
small molecule | CAS: 548486-59-5

Ulodesine has been used in trials studying the treatment of Gout, Arthritis, Hyperuricemia, and Joint Disease.

Kategori:
CarbohydratesIminesImino Sugars +3
Target Protein:
Purine nucleoside phosphorylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ulonivirine DB18787
small molecule | CAS: 1591823-76-5

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntiviral AgentsEnzyme Inhibitors +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ultevursen DB17835
biotech | CAS: 2642382-41-8

Ultevursen is a single-stranded RNA-based oligonucleotide targeting exon 13 of the USH2A gene that encodes usherin. It was developed by ProQR Therapeutics and is being investigated for the treatment of retinitis pigmentosa.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ulviprubart DB18281
biotech | CAS: 2569434-60-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

The use of umbilical cord blood (UCB) for therapies is advantageous because of its ease of access, non-invasive collection procedures, and more plasticity for multi-differentiation. UCB contains a large source of hematopoietic stem cells (HSCs) that are capab…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Umbralisib Approved DB14989
small molecule | CAS: 1532533-67-7

Marginal zone lymphoma is a rare, slowly progressing type of non-Hodgkin lymphoma initially treated with [rituximab] (an anti-CD20 drug), either alone or in combination with chemotherapy. Unfortunately, many patients experience a relapse or develop resistance…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP1A2 Substrates +9
Target Protein:
Casein kinase I isoform epsilonPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformTyrosine-protein kinase ABL1
Waktu ParuhThe effective half-…
Vol. DistribusiThe average apparen…
KlirensThe average apparen…
Genetik -
Umeclidinium Approved DB09076
small molecule | CAS: 869185-19-3

Umeclidinium is a long-acting muscarinic antagonist (LAMA) used as a maintenance treatment for symptoms of chronic obstructive pulmonary disease (COPD). COPD is a progressive obstructive lung disease characterized by shortness of breath, cough, sputum product…

Kategori:
Adrenergics, InhalantsAgents producing tachycardiaAgents to Treat Airway Disease +10
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M1 +2
Waktu ParuhThe effective half-…
Vol. DistribusiFollowing intraveno…
KlirensPlasma clearance fo…
Genetik -
Umifenovir DB13609
small molecule | CAS: 131707-25-0

Umifenovir is an indole-based, hydrophobic, dual-acting direct antiviral/host-targeting agent used for the treatment and prophylaxis of influenza and other respiratory infections.[A191475] It has been in use in Russia for approximately 25 years and in China s…

Kategori:
AnionsAntiinfectives for Systemic UseAntiviral Agents +19
Waktu ParuhThe half-life of um…
Vol. DistribusiData regarding the …
KlirensIn a study involvin…
Genetik -
Umirolimus DB15527
small molecule | CAS: 851536-75-9

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsAnti-Inflammatory AgentsImmunologic Factors +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Unasnemab DB18837
biotech | CAS: 2379805-59-9

Unasnemab is under investigation in clinical trial NCT04683848 (Study to Assess the Efficacy and Safety of MT-3921 in Subjects With Acute Traumatic Cervical Spinal Cord Injury).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Lysozyme C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Undecanal DB04093
small molecule | CAS: 112-44-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Undecanoic acid DB16857
small molecule | CAS: 112-37-8

Deskripsi belum tersedia.

Kategori:
Lipids
Target Protein:
G-protein coupled receptor 84
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1338-54-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
V-type sodium ATPase subunit K
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Gastric triacylglycerol lipase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrialLight-harvesting protein B-800/850 beta 1 chainLight-harvesting protein B-800/850 alpha chain +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Undecylenic acid Approved DB11117
small molecule | CAS: 112-38-9

Undecylenate, or undecylenic acid, is an unsaturated fatty acid with a terminal double bond that is derived from castor oil. Undecylenic acid is also found naturally in the human sweat. It is used as a precursor in the manufacture of aromatic chemicals, polym…

Kategori:
Antifungals for Dermatological UseAntifungals for Topical UseDermatologicals +4
Target Protein:
Calpain-1 catalytic subunit
Waktu ParuhNo information rega…
Vol. DistribusiNo information rega…
KlirensNo information rega…
Genetik -
Unesbulin DB18080
small molecule | CAS: 1610964-64-1

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Polycomb complex protein BMI-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Unoprostone Approved DB06826
small molecule | CAS: 120373-36-6

Unoprostone isopropyl is a prostaglandin analogue. Ophthalmic Solution 0.15% is a synthetic docosanoid. Unoprostone isopropyl has the chemical name isopropyl (+)-(Z)-7-[(1R,2R,3R,5S)-3,5 dihydroxy-2-(3-oxodecyl)cyclopentyl]-5-heptenoate. The main indication …

Kategori:
Antiglaucoma Preparations and MioticsAntihypertensive AgentsAutacoids +12
Waktu ParuhHalf-life of Unopr…
Vol. DistribusiIntended for local …
KlirensIntended for local …
Genetik -
Upadacitinib Approved DB15091
small molecule | CAS: 1310726-60-3

Upadacitinib is an oral Janus kinase (JAK)1-selective inhibitor and a disease-modifying antirheumatic drug (DMARD) used in the treatment of rheumatoid arthritis to slow down disease progression. Rheumatoid arthritis is a chronic autoimmune inflammatory diseas…

Kategori:
Antineoplastic and Immunomodulating AgentsAntirheumatic AgentsBCRP/ABCG2 Inhibitors +16
Target Protein:
Tyrosine-protein kinase JAK1
Waktu ParuhThe mean terminal e…
Vol. DistribusiThe volume of distr…
KlirensThe apparent oral c…
Genetik -
Upamostat DB13052
small molecule | CAS: 1191101-18-4

Upamostat has been used in trials studying the treatment of Pancreatic Cancer.

Kategori:
AmidesAminesHydroxylamines +3
Target Protein:
Urokinase-type plasminogen activator
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Upanovimab DB16505
biotech | CAS: 2500633-46-3

Upanovimab (SCTA01) was under investigation in clinical trials (NCT04683328, NCT04644185, NCT04709328 and NCT05156645) to evaluate its safety and efficacy in patients with severe COVID-19

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2254119-00-9

Upinitatug rilsodotin is under investigation in clinical trial NCT05329545 (Upifitamab Rilsodotin Maintenance in Platinum-sensitive Recurrent Ovarian Cancer (UP-NEXT)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Uprifosbuvir DB15206
small molecule | CAS: 1496551-77-9

Uprifosbuvir is under investigation in clinical trial NCT02332707 (Efficacy and Safety of Grazoprevir (MK-5172) and Uprifosbuvir (MK-3682) With Elbasvir (MK-8742) or Ruzasvir (MK-8408) for Chronic Hepatitis C Genotype (GT)1 and GT2 Infection (MK-3682-011)).

Kategori:
Anti-Infective AgentsAntiviral AgentsNucleic Acids, Nucleotides, and Nucleosides +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Uproleselan DB14829
small molecule | CAS: 1983970-12-2

Uproleselan is a novel, specific E-Selectin antagonist under investigation in clinical trial NCT02306291 (Study to Determine Safety, Pharmacokinetics and Efficacy of GMI-1271 in Combination With Chemotherapy in AML).

Kategori:
CarbohydratesE-Selectin, antagonists & inhibitorsGlycoconjugates +1
Target Protein:
E-selectin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Uprosertib DB11969
small molecule | CAS: 1047634-65-0

Uprosertib has been used in trials studying the treatment of Cancer, Melanoma, Solid Tumours, Cervical Cancer, and HER2/Neu Negative, among others.

Kategori:
AminesPolyamines
Target Protein:
RAC-gamma serine/threonine-protein kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Urabrelimab DB17209
biotech | CAS: 2249722-58-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Uracil DB03419
small molecule | CAS: 66-22-8

Deskripsi belum tersedia.

Kategori:
Fluorouracil and prodrugsPyrimidinesPyrimidinones
Target Protein:
Dihydropyrimidine dehydrogenase [NADP(+)]Uridine-cytidine kinase-like 1Uracil-DNA glycosylase +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Uracil C-13 DB16345
small molecule | CAS: 35803-45-3

Uracil C-13 is under investigation in clinical trial NCT01677338 (Phase 2 Study to Evaluate the Preliminary Performance of the C13-URA Breath Test Kit in Dyspeptic Subjects).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Uracil mustard Approved DB00791
small molecule | CAS: 66-75-1

Nitrogen mustard derivative of uracil. It is a alkylating antineoplastic agent that is used in lymphatic malignancies, and causes mainly gastrointestinal and bone marrow damage.

Kategori:
Alkylating DrugsAntineoplastic AgentsAntineoplastic Agents, Alkylating +10
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Urapidil DB12661
small molecule | CAS: 34661-75-1

Urapidil has been investigated for the treatment of Hypertension During Pre-Eclampsia.

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +12
Target Protein:
5-hydroxytryptamine receptor 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Urea Approved DB03904
small molecule | CAS: 57-13-6

A compound formed in the liver from ammonia produced by the deamination of amino acids. It is the principal end product of protein catabolism and constitutes about one half of the total urinary solids.

Kategori:
AmidesBlood and Blood Forming OrgansBlood Substitutes and Perfusion Solutions +7
Target Protein:
Dihydrofolate reductaseArginase-1Carbonic anhydrase 2 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Urea C-13 Approved DB09510
small molecule | CAS: 58069-82-2

Urea 13C is a urea molecule radiolabelled with the non-radioactive element carbon-13. It is currently used for the Urea Breath Test (UBT) and is available as a rapid diagnostic test (marketed as Pranactin-Citric) for the detection of Helicobacter pylori infec…

Kategori:
Diagnostic AgentsHelicobacter pylori Diagnostic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Urea C-14 Approved DB09513
small molecule | CAS: 594-05-8

Urea 14C is a urea molecule radiolabelled with a radioactive carbon-14. It is currently used for the Urea Breath Test (UBT) and is available as a rapid diagnostic test (marketed as PyTest) for the detection of Helicobacter pylori infections. H pylori is a com…

Kategori:
Radioactive Diagnostic Agent
Waktu Paruh14C-urea that is no…
Vol. Distribusi-
Klirens-
Genetik -
Urelumab DB12077
biotech | CAS: 934823-49-1

Urelumab has been used in trials studying the treatment of Leukemia, Multiple Myeloma, Malignant Tumors, and Cancer - Solid Tumors and B-Cell Non-Hodgkin's Lymphoma. Urelumab is a fully human antibody that targets CD137. The antibody product was developed usi…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Tumor necrosis factor receptor superfamily member 9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Urethane Approved DB04827
small molecule | CAS: 51-79-6

Urethane, formerly marketed as an inactive ingredient in Profenil injection, was determined to be carcinogenic and was removed from the Canadian, US, and UK markets in 1963.

Kategori:
Acids, AcyclicAnestheticsAnesthetics, General +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Uric acid DB08844
small molecule | CAS: 69-93-2

Uric acid is the last product of purine metabolism in humans. The formation of uric acid is through the enzyme xanthine oxidase, which oxidizes oxypurines. Normally a small amount of uric acid is present in the body, but when there is an excess amount in the …

Kategori:
AlkaloidsAntioxidantsBiological Factors +6
Target Protein:
Glycogen phosphorylase, liver form
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Uridine DB02745
small molecule | CAS: 58-96-8

Deskripsi belum tersedia.

Kategori:
Analogs/DerivativesNucleic Acids, Nucleotides, and NucleosidesNucleosides +4
Target Protein:
Thymidine phosphorylaseU6 snRNA-associated Sm-like protein LSm6Nucleoside-specific channel-forming protein tsx
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 63-39-8

Uridine 5'-(tetrahydrogen triphosphate). A uracil nucleotide containing three phosphate groups esterified to the sugar moiety.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPyrimidine Nucleotides +3
Target Protein:
P2Y purinoceptor 2P2Y purinoceptor 6P2Y purinoceptor 4 +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 133-89-1

A key intermediate in carbohydrate metabolism. Serves as a precursor of glycogen, can be metabolized into UDPgalactose and UDPglucuronic acid which can then be incorporated into polysaccharides as galactose and glucuronic acid. Also serves as a precursor of s…

Kategori:
CarbohydratesGlycosidesNucleic Acids, Nucleotides, and Nucleosides +8
Target Protein:
Galactose-1-phosphate uridylyltransferaseUDP-glucose 4-epimeraseAlpha,alpha-trehalose-phosphate synthase [UDP-forming] +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 58-97-9

5'-Uridylic acid. A uracil nucleotide containing one phosphate group esterified to the sugar moiety in the 2', 3' or 5' position.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPyrimidine Nucleotides +3
Target Protein:
Thymidylate synthaseUridine-cytidine kinase-like 1Galactose-1-phosphate uridylyltransferase +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Uridine triacetate Approved DB09144
small molecule | CAS: 4105-38-8

Uridine triacetate, formerly known as vistonuridine, is an orally active prodrug of the naturally occurring nucleoside uridine. It is used for the treatment of hereditary orotic aciduria (Xuriden), or for the emergency treatment of fluorouracil or capecitabin…

Kategori:
Acids, AcyclicAlimentary Tract and MetabolismFatty Acids +9
Waktu Paruh2 to 2.5 hours
Vol. DistribusiCirculating uridine…
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Vanadates
Target Protein:
Ribonuclease pancreatic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 58-98-0

A uracil nucleotide containing a pyrophosphate group esterified to C5 of the sugar moiety. [PubChem]

Target Protein:
UDP-N-acetylglucosamine 2-epimeraseHisto-blood group ABO system transferaseGalactose-1-phosphate uridylyltransferase +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Alpha,alpha-trehalose-phosphate synthase [UDP-forming]
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 15251–15300 dari 16004
Sebelumnya Halaman 306 / 321 Berikutnya