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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 300 / 321
TPIV 200 DB17318
biotech

TPIV 200 is a vaccine consisting of proteins from the folate receptor alpha mixed with Granulocyte-macrophage colony-stimulating factor (GM-CSF).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
TPMPA DB16754
small molecule | CAS: 182485-36-5

TPMPA ((1,2,5,6-tetrahydropyridine-4-yl)methylphosphinic acid) is a selective antagonist of GABA<sub>C</sub> receptors (also known as GABA-? or GABA<sub>A-?</sub> receptors).[A245303] GABA<sub>C</sub> receptors are found primarily in the retina, although they…

Target Protein:
Gamma-aminobutyric acid receptor subunit rho-1Gamma-aminobutyric acid receptor subunit rho-2Gamma-aminobutyric acid receptor subunit rho-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TPX-4589 DB18604
biotech

TPX-4589 is an antibody-drug conjugate composed of a humanized monoclonal antibody targeting CLDN18.2 and linker-payload MC-VC-PAB-MMAE.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TQS-168 DB18108
small molecule | CAS: 49671-76-3

Deskripsi belum tersedia.

Kategori:
Blood Glucose Lowering AgentsHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trabectedin Approved DB05109
small molecule | CAS: 114899-77-3

Trabectedin, also referred as ET-743 during its development, is a marine-derived antitumor agent discovered in the Carribean tunicate _Ecteinascidia turbinata_ and now produced synthetically. Trabectedin has a unique mechanism of action. It binds to the minor…

Kategori:
Agents Causing Muscle ToxicityAlkylating ActivityAlkylating Drugs +24
Target Protein:
DNA
Waktu Paruh33-50 hours
Vol. Distribusi-
Klirens-
Genetik -
Trabedersen DB05697
biotech | CAS: 925681-61-4

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsNucleic Acids, Nucleotides, and NucleosidesNucleotides +3
Target Protein:
Transforming growth factor beta-2 proprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trabodenoson DB13122
small molecule | CAS: 871108-05-3

Trabodenoson has been used in trials studying the treatment of Ocular Hypertension (OHT) and Primary Open-Angle Glaucoma (POAG).

Kategori:
Adenosine A receptor agonistsAdenosine A1 Receptor AgonistsAnions +9
Target Protein:
Adenosine receptor A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tradipitant DB12580
small molecule | CAS: 622370-35-8

Tradipitant has been used in trials studying the treatment and prevention of Eczema, Pruritus, Gastroparesis, Chronic Pruritus, and Atopic Dermatitis, among others.

Target Protein:
Substance-P receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trafermin DB06244
biotech | CAS: 131094-16-1

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCardiovascular Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tragacanth Approved DB10667
biotech | CAS: 9000-65-1

Tragacanth allergenic extract is used in allergenic testing.

Kategori:
Biological ProductsBiopolymersCarbohydrates +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1808916-28-0

Tralesinidase alfa is a chimeric fusion protein comprised of recombinant human NAGLU and a modified human insulin-like growth factor 2. It is being investigated for the treatment of mucopolysaccharidosis type IIIB (MPS IIIB), also known as Sanfilippo syndrome…

Kategori:
Amino Acids, Peptides, and Proteinsbeta-N-AcetylhexosaminidasesBiological Factors +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tralokinumab Approved DB12169
biotech | CAS: 1044515-88-9

Atopic dermatitis (AD) is an inflammatory skin disorder that causes skin inflammation, skin barrier dysfunction, and chronic pruritus.[A242432] It is estimated to affect up to 20% of adults and children worldwide, and is frequently associated with other atopi…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAmino Acids, Peptides, and ProteinsAntibodies +9
Target Protein:
Interleukin-13
Waktu ParuhThe half-life of tr…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of tr…
Genetik -
Tramadol Approved DB00193
small molecule | CAS: 27203-92-5

Tramadol is a centrally acting synthetic opioid analgesic and SNRI (serotonin/norepinephrine reuptake-inhibitor) that is structurally related to [codeine] and [morphine]. Due to its good tolerability profile and multimodal mechanism of action, tramadol is gen…

Kategori:
Agents producing tachycardiaAgents that reduce seizure thresholdAlcohols +33
Target Protein:
Mu-type opioid receptorSodium-dependent noradrenaline transporterSodium-dependent serotonin transporter +12
Waktu ParuhTramadol reported a…
Vol. DistribusiThe volume of distr…
KlirensIn clinical trials,…
Genetik -
Tramazoline DB13064
small molecule | CAS: 1082-57-1

Tramazoline is under investigation in clinical trial NCT01601509 (Nasal Tramazoline and Dexamethazone in Obstructive Sleep Apnea (OSA) Patients Tramazoline and).

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAutonomic Agents +4
Target Protein:
Alpha-2A adrenergic receptorAlpha-2B adrenergic receptorAlpha-2C adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Trametes versicolor fruiting body is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trametinib Approved DB08911
small molecule | CAS: 871700-17-3

Trametinib is an orally bioavailable mitogen-activated extracellular signal-regulated kinase 1 (MEK1) and MEK2 inhibitor.[A258298,A258293] It was first approved by the FDA in May 2013 for the treatment of melanoma.[A258298] It was later approved by Health Can…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP2C8 Inhibitors +20
Target Protein:
Dual specificity mitogen-activated protein kinase kinase 1Dual specificity mitogen-activated protein kinase kinase 2
Waktu ParuhThe estimated elimi…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
Tramiprosate DB06527
small molecule | CAS: 3687-18-1

Deskripsi belum tersedia.

Kategori:
AlkanesAlkanesulfonic AcidsAnticonvulsants +10
Target Protein:
Amyloid-beta precursor protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trandolapril Approved DB00519
small molecule | CAS: 87679-37-6

Trandolapril is a non-sulhydryl prodrug that belongs to the angiotensin-converting enzyme (ACE) inhibitor class of medications. It is metabolized to its biologically active diacid form, trandolaprilat, in the liver. Trandolaprilat inhibits ACE, the enzyme res…

Kategori:
ACE Inhibitors and Calcium Channel BlockersAgents Acting on the Renin-Angiotensin SystemAgents causing angioedema +9
Target Protein:
Angiotensin-converting enzyme
Waktu ParuhThe elimination hal…
Vol. Distribusi* 18 L
Klirens* 52 L/h [After app…
Genetik -
Trandolaprilat DB14209
small molecule | CAS: 87679-71-8

The active metabolite of the prodrug [Trandolapril].

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAngiotensin-Converting Enzyme Inhibitors +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tranexamic acid Approved DB00302
small molecule | CAS: 1197-18-8

Tranexamic acid is a synthetic derivative of [lysine] used as an antifibrinolytic in the treatment and prevention of major bleeding. It possesses a similar mechanism of action to [aminocaproic acid] but is approximately 10-fold more potent.[L31883] It was …

Kategori:
Acids, CarbocyclicAmino AcidsAmino Acids, Peptides, and Proteins +10
Target Protein:
Plasminogen
Waktu ParuhFollowing intraveno…
Vol. DistribusiThe initial volume …
KlirensThe plasma clearanc…
Genetik -
Tranilast DB07615
small molecule | CAS: 53902-12-8

Tranilast is an antiallergic drug developed by Kissei Pharmaceuticals. In 1982, it was approved in Japan and South Korea for the management of bronchial asthma. Indications for keloid and hypertrophic scar were added in 1993. It has been used for the treatmen…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAminobenzoates +23
Target Protein:
Steryl-sulfataseHistamine H1 receptorHematopoietic prostaglandin D synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
trans NV-04 DB05843
small molecule

trans NV-04 is a cardiovascular drug which shows a significant reduction in blood pressure and arterial stiffness.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Phenylethanolamine N-methyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Immunoglobulin heavy constant gamma 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 614-60-8

Deskripsi belum tersedia.

Kategori:
OAT3/SLC22A8 Inhibitors
Target Protein:
Carbonic anhydrase 2Carbonic anhydrase 1Major NAD(P)H-flavin oxidoreductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Prothrombin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Urokinase-type plasminogen activator
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Chymotrypsinogen B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 3465-72-3

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAcrylatesImidazoles
Target Protein:
Urocanate hydratase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 27876-94-4

Vitamin A-analog that increases diffusivity of oxygen in aqueous solutions, including plasma.

Kategori:
AlkenesAnticarcinogenic AgentsAntineoplastic Agents +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 721946-42-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Transfluthrin DB15117
small molecule | CAS: 118712-89-3

Transfluthrin is under investigation in clinical trial NCT02394522 (Spatial Repellent Products for Control of Vector Borne Diseases - Malaria - Zambia (SR-M-ZM)).

Kategori:
AgrochemicalsBenzene DerivativesCompounds used in a research, industrial, or household setting +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tranylcypromine Approved DB00752
small molecule | CAS: 155-09-9

A propylamine formed from the cyclization of the side chain of amphetamine. This monoamine oxidase inhibitor is effective in the treatment of major depression, dysthymic disorder, and atypical depression. It also is useful in panic and phobic disorders (From …

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAmines +32
Target Protein:
Amine oxidase [flavin-containing] BAmine oxidase [flavin-containing] A
Waktu Paruh1.5-3.2 hours in pa…
Vol. Distribusi1.1-5.7 L/kg
Klirens-
Genetik -
Trapidil DB09283
small molecule | CAS: 15421-84-8

Trapidil, a platelet-derived growth factor antagonist, was originally developed as a vasodilator and anti-platelet agent and has been used to treat patients with ischemic coronary heart, liver, and kidney disease.

Kategori:
Antiplatelet agentsCardiac TherapyCardiovascular Agents +7
Target Protein:
Fibroblast growth factor receptor 3Cyclic nucleotide phosphodiesterasePlatelet-derived growth factor receptor beta
Waktu ParuhThe half life of el…
Vol. Distribusi-
KlirensThe apparent cleara…
Genetik -
Trastuzumab Approved DB00072
biotech | CAS: 180288-69-1

Produced in CHO cell cultures, trastuzumab is a recombinant IgG1 kappa, humanized monoclonal antibody [A40276] that selectively binds with high affinity in a cell-based assay (Kd = 5 nM) to the extracellular domain of the human epidermal growth factor recepto…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +21
Target Protein:
Receptor tyrosine-protein kinase erbB-2
Gen Terkait:
ERBB2
Waktu ParuhThe terminal half-l…
Vol. Distribusi-
KlirensThe predicted stead…
Genetik 1 Varian
Trastuzumab deruxtecan Approved DB14962
biotech | CAS: 1826843-81-5

Trastuzumab deruxtecan is a HER2-directed antibody attached to a topoisomerase inhibitor that is approved for use in certain types of treatment-resistant HER2-positive cancers.[L10842] It is classified as an antibody-drug conjugate. The cleavable peptide link…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +27
Target Protein:
High affinity immunoglobulin gamma Fc receptor IDNA topoisomerase 1
Waktu ParuhIn a pharmacokineti…
Vol. DistribusiThe estimated volum…
KlirensTrastuzumab deruxte…
Genetik -
biotech | CAS: 1642152-40-6

Trastuzumab duocarmazine is under investigation in clinical trial NCT03262935 (SYD985 vs. Physician's Choice in Participants With Her2-positive Locally Advanced or Metastatic Breast Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trastuzumab emtansine Approved DB05773
biotech | CAS: 1018448-65-1

Trastuzumab emtansine, formerly called Trastuzumab-DM1 (T-DM1) is a first-in-class HER2 antibody drug conjugate (ADC) comprised of Genentech's trastuzumab antibody linked to ImmunoGen's cell-killing agent, DM1. T-DM1 combines two strategies-- anti-HER2 activi…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +42
Target Protein:
Receptor tyrosine-protein kinase erbB-2
Waktu ParuhTrastuzumab emtansi…
Vol. DistribusiThe volume of distr…
KlirensAfter IV infusion, …
Genetik -
Travoprost Approved DB00287
small molecule | CAS: 157283-68-6

Travoprost is a synthetic isopropyl ester prodrug of a prostaglandin F2alpha (F2?) analogue and selective FP prostanoid receptor agonist. It is used to decrease intraocular pressure in open-angle glaucoma and ocular hypertension.[L49434] Unlike other prostagl…

Kategori:
Antiglaucoma Preparations and MioticsAntihypertensive AgentsEicosanoids +10
Target Protein:
Prostaglandin F2-alpha receptor
Waktu ParuhThe terminal elimin…
Vol. DistribusiNo information is a…
KlirensNo information is a…
Genetik -
Traxoprodil DB18795
small molecule | CAS: 134234-12-1

Deskripsi belum tersedia.

Target Protein:
Glutamate receptor ionotropic, NMDA 2B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trazodone Approved DB00656
small molecule | CAS: 19794-93-5

Trazodone is triazolopyridine derivative from the serotonin receptor antagonists and reuptake inhibitors (SARIs) class of antidepressants.[A181180] It is used in adults and has been shown to be comparable in efficacy to other drugs such as tricyclic antidepre…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +45
Target Protein:
5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2CSodium-dependent serotonin transporter +5
Waktu ParuhThe plasma eliminat…
Vol. DistribusiA single-dose pharm…
KlirensA decrease in total…
Genetik -
Trazpiroben DB18794
small molecule | CAS: 1352993-39-5

Deskripsi belum tersedia.

Target Protein:
D(3) dopamine receptorD(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRC150094 DB16046
small molecule | CAS: 1092551-88-6

TRC150094 is under investigation in clinical trial NCT03254446 (Safety and Efficacy Study of TRC150094 to Improve the CV Risk in Subjects With Diabetes, Dyslipidemia and Hypertension).

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Treamid DB16365
small molecule

Treamid, also known as bisamide derivative of dicarboxylic acid (BDDA), is a complexing agent that has been found to chelate metal ions, including calcium, copper, iron, magnesium, and zinc.[A225701] This drug has shown regenerative properties and restoration…

Kategori:
Acids, AcyclicDicarboxylic Acids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trebananib DB12056
biotech | CAS: 894356-79-7

Trebananib is under investigation for the treatment of Ovarian Cancer, Peritoneal Cancer, and Fallopian Tube Cancer. Trebananib has been investigated for the treatment of Cancer, Oncology, Carcinoma, Metastases, and Colon Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trefentanil DB09181
small molecule | CAS: 120656-74-8

Trefentanil (A-3665) is a fentanyl analogue opioid developed in 1992. It is more potent and shorter acting than alfentanil. Trefentanil is not used in clinics due to the severity of its respiratory depression, though it is still used in research.

Target Protein:
Mu-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

The trefoil factor 2 (TFF2) peptide is a low-molecular weight protein and one of the three trefoil-motif-containing proteins. They are expressed predominantly in gastric tissues with the source for them being predominantly stromal cells, although expression o…

Kategori:
Trefoil Factors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tregalizumab DB13073
biotech | CAS: 1207446-68-1

Tregalizumab has been used in trials studying the treatment of Rheumatoid Arthritis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trehalose DB12310
small molecule | CAS: 99-20-7

Cabaletta has been used in trials studying the treatment of Oculopharyngeal Muscular Dystrophy.

Kategori:
CarbohydratesCompounds used in a research, industrial, or household settingDisaccharides +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 4484-88-2

Deskripsi belum tersedia.

Kategori:
CarbohydratesCompounds used in a research, industrial, or household settingDisaccharides +5
Target Protein:
HTH-type transcriptional regulator TreR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 14951–15000 dari 16004
Sebelumnya Halaman 300 / 321 Berikutnya