Hasil Filter

2279

Total database: 17430
Struktur (SMILES)
866 (38.0%)
Target
1100 (48.3%)
Genomik
31 (1.4%)
Referensi
2279 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (2279)

Halaman 30 / 46
NGN-101 DB18335
biotech

NGN-101 is an adeno-associated virus serotype 9 vector with engineered transgene encoding the human CLN5 gene

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NGN-401 DB18594
biotech

NGN-401 is a recombinant serotype 9 adeno-associated virus (AAV) encoding an intron encoding a miRNA generating sequence, complementary miRNA binding sites and a full-length human methyl cytosine binding protein 2 (MECP2). Developed by Neurogene Inc., it is b…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Niclosamide Approved DB06803
small molecule | CAS: 50-65-7

Niclosamide is an antihelminthic used for the treatment of tapeworm infections. Helminths (worms) are multicellular organisms that infect very large numbers of humans and cause a broad range of diseases. Over 1 billion people are infected with intestinal nema…

Kategori:
AgrochemicalsAmidesAmines +22
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nicoboxil Approved DB12911
small molecule | CAS: 13912-80-6

Nicoboxil has been investigated for the treatment of Acute Low Back Pain, where it is typically considered an effective and safe therapeutic option. Nevertheless, it is predominantly found paired with nonivamide as a combination topical analgesic product wher…

Kategori:
Drugs that are Mainly Renally ExcretedPyridines
Waktu ParuhThe half-life of es…
Vol. DistribusiDespite the fact th…
KlirensThe elimination of …
Genetik -
Nicotinamide Approved DB02701
small molecule | CAS: 98-92-0

An important compound functioning as a component of the coenzyme NAD. Its primary significance is in the prevention and/or cure of blacktongue and pellagra. Most animals cannot manufacture this compound in amounts sufficient to prevent nutritional deficiency …

Kategori:
Alimentary Tract and MetabolismCytochrome P-450 CYP2D6 InhibitorsCytochrome P-450 CYP2D6 Inhibitors (strength unknown) +13
Target Protein:
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 2Exotoxin APoly [ADP-ribose] polymerase 1 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nifurtimox Approved DB11820
small molecule | CAS: 23256-30-6

Chagas disease, caused by a parasite known as Trypanosoma cruzi (T.cruzi), is a vector-transmitted disease affecting animals and humans in the Americas. It is commonly known as American Trypanosomiasis.[L15366] The CDC estimates that approximately 8 millio…

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAnti-Infective AgentsAntiparasitic Agents +11
Target Protein:
NitroreductasesGlyceraldehyde-3-phosphate dehydrogenase, glycosomal
Waktu ParuhThe elimination hal…
Vol. DistribusiNifurtimox crosses …
KlirensOne pharmacokinetic…
Genetik -
Nimesulide Approved DB04743
small molecule | CAS: 51803-78-2

Nimesulide is a relatively COX-2 selective, non-steroidal anti-inflammatory drug (NSAID) with analgesic and antipyretic properties. Its approved indications are the treatment of acute pain, the symptomatic treatment of osteoarthritis and primary dysmenorrhoea…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +25
Target Protein:
Prostaglandin G/H synthase 2Tumor necrosis factor ligand superfamily member 10Lactotransferrin +1
Waktu Paruh1.8–4.7 hours
Vol. Distribusi-
Klirens-
Genetik -
Nipocalimab DB16257
biotech | CAS: 2211985-36-1

Nipocalimab is under investigation in clinical trial NCT04119050 (Efficacy and Safety of M281 in Adults With Warm Autoimmune Hemolytic Anemia).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nirsevimab Approved DB16258
biotech | CAS: 1989556-22-0

Nirsevimab (MEDI8897) is a recombinant human immunoglobulin G1 kappa (IgG1?) monoclonal antibody used to prevent respiratory syncytial virus (RSV) lower respiratory tract disease in neonates and infants.[L44146] It binds to the prefusion conformation of the R…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Fusion glycoprotein F0Fusion glycoprotein F0Fusion glycoprotein F0
Waktu ParuhThe terminal half-l…
Vol. DistribusiFor an infant weigh…
KlirensFor an infant weigh…
Genetik -
Nisoldipine Approved DB00401
small molecule | CAS: 63675-72-9

Nisoldipine is a 1,4-dihydropyridine calcium channel blocker. It acts primarily on vascular smooth muscle cells by stabilizing voltage-gated L-type calcium channels in their inactive conformation. By inhibiting the influx of calcium in smooth muscle cells, ni…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntihypertensive Agents +23
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent calcium channel subunit alpha-2/delta-1Voltage-dependent L-type calcium channel subunit beta-2 +2
Waktu Paruh7-12 hours
Vol. Distribusi-
Klirens-
Genetik -
Nitric Oxide Approved DB00435
small molecule | CAS: 10102-43-9

Nitric oxide or Nitrogen monoxide is a chemical compound with chemical formula NO. This gas is an important signaling molecule in the body of mammals including humans and is an extremely important intermediate in the chemical industry. It is also a toxic air …

Kategori:
Anti-Asthmatic AgentsAntioxidantsAutonomic Agents +30
Target Protein:
Guanylate cyclase soluble subunit alpha-1Guanylate cyclase soluble subunit beta-1Guanylate cyclase soluble subunit alpha-2 +3
Waktu Paruh2–6 seconds
Vol. Distribusi-
Klirens-
Genetik -
Nitrofurantoin Approved DB00698
small molecule | CAS: 67-20-9

Nitrofurantoin is a nitrofuran antibiotic used to treat uncomplicated urinary tract infections.[L6856,L6859,L6862] Nitrofurantoin is converted by bacterial nitroreductases to electrophilic intermediates which inhibit the citric acid cycle as well as synthesis…

Kategori:
Agents causing hyperkalemiaAnti-Bacterial AgentsAnti-Infective Agents +15
Target Protein:
Probable pyruvate-flavodoxin oxidoreductaseOxygen-insensitive NADPH nitroreductase30S ribosomal protein S10
Waktu ParuhThe half life of ni…
Vol. DistribusiData regarding the …
KlirensThe clearance of ni…
Genetik -
Nivatrotamab DB16654
biotech | CAS: 2278244-14-5

Nivatrotamab is under investigation in clinical trial NCT03860207 (Study of the Safety and Efficacy of Humanized 3F8 Bispecific Antibody (Hu3f8-bsab) in Patients With Relapsed/refractory Neuroblastoma, Osteosarcoma and Other Solid Tumor Cancers).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nivolumab Approved DB09035
biotech | CAS: 946414-94-4

Nivolumab is a fully human IgG4 antibody targeting the immune checkpoint programmed death receptor-1 (PD-1).[L12129] This antibody was produced entirely in mice and grafted onto human kappa and IgG4 Fc region with the mutation _S228P_ for additional stability…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntibodies +20
Target Protein:
Programmed cell death protein 1Programmed cell death 1 ligand 1
Waktu ParuhThe serum half life…
Vol. DistribusiThe volume of distr…
KlirensThe estimated clear…
Genetik -
biotech

These cells are prepared as universal off-the-shelf CAR-NK cells from cord blood with NKG2D-ACE2 proteins engineered as part of the CARs; the cell secretes IL-15 and GM-CSF. Chimeric antigen receptors (CARs) are artificial receptors consisting of an antibody-…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NKTT-120 DB17730
biotech

NKTT-120 is a recombinant humanized IgG1k monoclonal antibody to human invariant T cell receptor (iTCR).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NM-702 DB05505
small molecule

Nissan Chemical and Taisho have been jointly developing NM-702, a drug for the treatment of arteriosclerosis obliterans. M-702 is an orally active inhibitor of phosphodiesterase and thromboxane synthetase. In Japan, Phase 2 studies are being conducted for …

Target Protein:
Thromboxane-A synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NM3086 DB17719
biotech

NM3086 is a recombinant, humanized, aglycosylated, IgG1-kappa anti-properdin monoclonal antibody being developed by Novelmed Therapeutics Inc.[L46193]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NN344 DB05115
small molecule

NN344 is a neutral, soluble long-acting human insulin analogue with 24 hour coverage by once daily injection. NN344 has a very flat and predictable action profile. The product is intended for basal insulin treatment of diabetes mellitus.

Kategori:
Amino Acids, Peptides, and ProteinsBlood Glucose Lowering AgentsCytochrome P-450 CYP1A2 Inducers +9
Target Protein:
Insulin receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NNZ-2591 DB15601
small molecule | CAS: 847952-38-9

NNZ-2591 (cyclo-L-glycyl-L-2-allylproline)[A189390] is an investigational synthetic analog of cyclic glycine-proline (cGP), a breakdown product of human insulin-like growth factor 1 (IGF-1), that has been chemically modified to increase its half-life, stabili…

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesPiperazines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nofazinlimab DB18852
biotech | CAS: 2377845-98-0

Nofazinlimab is under investigation in clinical trial NCT04194775 (A Study of Nofazinlimab (CS1003) in Subjects With Advanced Hepatocellular Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nogapendekin alfa Approved DB18740
biotech | CAS: 1622189-43-8

Nogapendekin alfa is a human IL-15N72D variant. It is one of the active ingredients in Anktiva, a combination product also containing [inbakicept], where a single inbakicept is complexed with two nogapendekin alfa components.[L50592] This combination product …

Kategori:
Amino Acids, Peptides, and ProteinsInterleukin-15Proteins +2
Target Protein:
Interleukin-2 receptor subunit betaCytokine receptor common subunit gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nonivamide DB11324
small molecule | CAS: 2444-46-4

Nonivamide is found in herbs and spices. It is an alkaloid from the Capsicum species. The structures of [DB06774] and nonivamide differ only slightly with respect to the fatty acid moiety of the side chain (8-methyl nonenoic acid versus nonanoic acid) [F31]. …

Kategori:
Acids, CarbocyclicAlkaloidsAlkenes +20
Target Protein:
Transient receptor potential cation channel subfamily V member 1
Waktu ParuhAbout 7 minutes [F3…
Vol. Distribusi-
Klirens-
Genetik -
NP2 DB06308
small molecule

NP2 is a replication defective HSV-1 based gene transfer vector engineered to express human preproenkephalin. It was under investigation in clinical trial NCT01291901 (NP2 Enkephalin For Treatment of Intractable Cancer Pain).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NSI-566 DB17954
biotech

NSI-566 is a stem cell therapy consisting of human spinal cord-derived neural stem cells. Developed by Seneca Biopharma, it is being investigated for the treatment of amyotrophic lateral sclerosis (ALS), stroke, and chronic spinal cord injury (cSCI).[L47097]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NTLA-2001 DB18525
biotech

NTLA-2001 is a clustered regularly interspaced short palindromic repeats CRISPR/ Cas9-based gene therapy consisting of a single guide RNA targeting the human TTR gene and a messenger RNA encoding Cas9.

Kategori:
Biomimetic MaterialsDrug CarriersMembranes, Artificial +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NTLA-2002 DB17597
biotech

NTLA-2002 is a lipid nanoparticle encapsulating single guide RNA (G012267) targeting the human KLKB1 gene and messenger RNA (mRNA000042) encoding Cas9. It is an investigational therapy designed to knock out the target gene kallikrein B1 (KLKB1) to reduce plas…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NUC B1000 DB05242
biotech

NUC B1000 is an expressed interfering RNA (eiRNA)- based product consisting of a plasmid DNA construct designed to produce four short interfering RNA (siRNA) molecules, formulated with a proprietary cationic-lipid delivery system. [F3910] eiRNA is an approach…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nuvaxovid Approved DB15810
biotech

SARS-CoV-2, the causative agent of COVID-19, relies on the interaction between its trimeric spike (S) glycoprotein and angiotensin-converting enzyme 2 (hACE2) expressed on host cells in order to establish a productive infection in humans.[A243789] Antibodies …

Kategori:
Biological ProductsComplex MixturesCOVID-19 Vaccines +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NV-18 DB05886
small molecule

NV-18 is a product of the Novogen diphenolic synthetic analogue program that is creating drugs with diverse activities against specific types of cancer. Like phenoxodiol, NV-18 is broadly effective in the laboratory against almost all human cancer types, but …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NVS antibody DB05312
small molecule

This drug has been developed using Medarex's UltiMAb Human Antibody Development System to treat autoimmune diseases.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NZ-1002 DB17688
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cyanovirin-N
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OAV201 DB17842
biotech

OAV201 is a non-replicating, recombinant adeno-associated virus serotype 9 (AAV9) containing the human Methyl CpG Binding Protein 2B (MECP2B) cDNA under the control of a segment of the murine MECP2 promoter. It was first developed by Novartis and investigated…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Obatoclax DB12191
small molecule | CAS: 803712-67-6

Obatoclax has been used in trials studying the treatment of AML, Leukemia, Myelofibrosis, Hodgkin's Lymphoma, and Mantle-Cell Lymphoma, among others.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-Ring
Target Protein:
Apoptosis regulator Bcl-2Induced myeloid leukemia cell differentiation protein Mcl-1Bcl-2-like protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OBE101 DB05080
small molecule

OBE101 is a new weight loss drug developed by Obecure Ltd. It is a new formulation that is based on the vertigo medication, Betahistine. Obecure is repurposing betahistine, which is an H1 receptor agonist and partial H3 receptor antagonist for the treatment o…

Target Protein:
Histamine H1 receptorHistamine H3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Obexelimab DB15032
biotech | CAS: 1690307-05-1

Obexelimab is under investigation in clinical trial NCT02725515 (A Study of the Effect of XmAb®5871 in Patients With Systemic Lupus Erythematosus).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OBI-999 DB17356
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Obinepitide DB05045
small molecule | CAS: 348119-84-6

Obinepitide is a synthetic analogue of two natural human hormones, PYY and Pancreatic Polypeptide, which normally are released during a meal. These hormones are known to play a role in the regulation of food intake and appetite in man as satiety signal from t…

Target Protein:
Neuropeptide Y receptor type 4Neuropeptide Y receptor type 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Obinutuzumab Approved DB08935
biotech | CAS: 949142-50-1

Obinutuzumab is a humanized monoclonal antibody used as a combination treatment with chlorambucil to treat patients with untreated chronic lymphocytic leukemia. It was approved by the FDA in November 2013 and is marketed under the brand name Gazyva. There is …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +20
Target Protein:
B-lymphocyte antigen CD20
Waktu ParuhThe half life of ob…
Vol. DistribusiObinutuzumab has a …
KlirensThe clearance of ob…
Genetik -
Ocaratuzumab DB17359
biotech | CAS: 1169956-08-4

Ocaratuzumab is a humanized monoclonal antibody directed against CD20. It is being investigated for cancers and autoimmune disorders.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ociperlimab DB18947
biotech | CAS: 2342597-93-5

Ociperlimab is under investigation in clinical trial NCT04866017 (A Study to Compare Ociperlimab Plus Tislelizumab Versus Durvalumab Following Concurrent Chemoradiotherapy (Ccrt) in Patients With Stage III Unresectable Non-small Cell Lung Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ocrelizumab Approved DB11988
biotech | CAS: 637334-45-3

Ocrelizumab is a CD20-directed cytolytic antibody indicated for the treatment of patients with primary progressive or relapsing forms of multiple sclerosis (MS).[L42895] It is a second-generation recombinant humanized monoclonal IgG1 antibody that selectively…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +14
Target Protein:
B-lymphocyte antigen CD20
Waktu ParuhThe terminal elimin…
Vol. DistribusiIn a population pha…
KlirensThe constant cleara…
Genetik -
Ocriplasmin Approved DB08888
biotech | CAS: 1048016-09-6

Ocriplasmin is a recombinant truncated form of human plasmin with a molecular weight of 27.2 kDa produced by recombinant DNA technology in a Pichia pastoris expression system. Ocriplasmin is a protein made up of 249 amino acids and has two peptide chains. Ag…

Kategori:
Amino Acids, Peptides, and ProteinsEENT Drugs, MiscellaneousEndopeptidases +10
Target Protein:
FibronectinAlpha-2-macroglobulinAlpha-2-antiplasmin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Octasulfur Approved DB09353
small molecule | CAS: 10544-50-0

Sulfur is a chemical element that is present in all living tissues. The most commonly used form of pharmaceutical sulfur is Octasulfur (S8). After calcium and phosphorus, it is the third most abundant mineral in the human body. Sulfur is also found in garlic,…

Kategori:
ChalcogensElementsKeratolytic Agents
Waktu ParuhIntended for local …
Vol. DistribusiIntended for local …
KlirensIntended for local …
Genetik -
Octreotide Approved DB00104
biotech | CAS: 83150-76-9

Acromegaly is a disorder caused by excess growth hormone (GH), increasing the growth of body tissues and causing metabolic dysfunction.[L14501] In most cases, it results from an anterior pituitary growth hormone-releasing tumor. Typically, the feet, hands, an…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic Agents, Hormonal +19
Target Protein:
Somatostatin receptor type 2Somatostatin receptor
Waktu ParuhAfter a subcutaneou…
Vol. DistribusiIn a pharmacokineti…
KlirensThe total body clea…
Genetik -
OCU400 DB18277
biotech

OCU400 is a novel gene therapy comprising an adeno-associated viral vector expressing human nuclear hormone receptor subfamily 2 group E member 3 (hNR2E3).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Odesivimab Approved DB15900
biotech | CAS: 2135632-30-1

Ebola virus (EBOV) remains an important human pathogen within the _Ebolavirus_ genus, having been responsible for at least 17 known outbreaks with an average case fatality rate of 43.92%.[A221825] Immune therapy using monoclonal antibodies (mAbs) is becoming …

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +10
Target Protein:
Envelope glycoprotein
Waktu ParuhOdesivimab administ…
Vol. DistribusiOdesivimab administ…
KlirensOdesivimab administ…
Genetik -
Odronextamab DB16684
biotech | CAS: 1801338-64-6

Odronextamab is a hinge-stabilized, fully human immunoglobulin G4 (IgG4)-based CD20×CD3 bispecific antibody currently evaluated for the treatment of relapsed/refractory (R/R) B-Cell non-Hodgkin lymphoma (NHL).[A254187,A254197] Preliminary studies have shown t…

Target Protein:
B-lymphocyte antigen CD20T-cell surface glycoprotein CD3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ofatumumab Approved DB06650
biotech | CAS: 679818-59-8

Ofatumumab is a novel anti-CD20 monoclonal antibody that targets B-cells. It is an IgG1? human monoclonal antibody produced from a recombinant murine cell line (NS0) via transgenic mouse and hybridoma technology.[L12612] Ofatumumab works by recognizing antige…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
B-lymphocyte antigen CD20
Waktu ParuhIn patients with CL…
Vol. DistribusiIn patients with CL…
KlirensIn patients with CL…
Genetik -
Menampilkan 1451–1500 dari 2279
Sebelumnya Halaman 30 / 46 Berikutnya