Hasil Filter

1977

Total database: 17430
Struktur (SMILES)
1074 (54.3%)
Target
1046 (52.9%)
Genomik
39 (2.0%)
Referensi
1977 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (1977)

Halaman 30 / 40
Pyridoxine Approved DB00165
small molecule | CAS: 65-23-6

Pyridoxine is the 4-methanol form of vitamin B6, an important water-soluble vitamin that is naturally present in many foods. As its classification as a vitamin implies, Vitamin B6 (and pyridoxine) are essential nutrients required for normal functioning of man…

Kategori:
Alimentary Tract and MetabolismAnalogs/DerivativesAntiinfectives for Systemic Use +10
Target Protein:
Aromatic-L-amino-acid decarboxylasePyridoxal kinase
Waktu ParuhThe total adult bod…
Vol. DistribusiPyridoxine main act…
Klirens-
Genetik -
Pyroquilon DB02756
small molecule | CAS: 57369-32-1

Pyroquilon is a commercial blasticide which binds in the naphthol pocket of fungal trihydroxynaphthalene reductase active site.

Kategori:
Antifungal AgentsHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pyrotinib DB14993
small molecule | CAS: 1269662-73-8

Pyrotinib is under investigation in clinical trial NCT03756064 (Neoadjuvant Study of Pyrotinib in Patients With HER2 Positive Breast Cancer).

Kategori:
Acids, AcyclicAcrylatesAmides +2
Target Protein:
Epidermal growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pyrrolidone DB19152
small molecule | CAS: 616-45-5

Pyrrolidone is under investigation in clinical trial NCT05444998 (Neoadjuvant Inituomab, Pyrrolidone and Nab-paclitaxel for Her2+breast Cancer).

Kategori:
Pyrrolidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 72909-34-3

A pyrrolo-quinoline having two adjacent keto-groups at the 4 and 5 positions and three acidic carboxyl groups. It is a coenzyme of some DEHYDROGENASES. [PubChem]

Kategori:
CoenzymesEnzymes and CoenzymesHeterocyclic Compounds, Fused-Ring +3
Target Protein:
Quinohemoprotein ethanol dehydrogenase type-1Quinoprotein glucose dehydrogenase BPyrroloquinoline-quinone synthase +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PYX-201 DB18382
biotech

PYX-201 is an antibody-drug conjugate directed against the extra domain-B splice variant of fibronectin.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Q-Derp1 DB05857
biotech

Q-Derp1 is developed by Cytos Biotechnology as an immunodrug. It is an antigen for the prevention of various major chronic diseases. Derp1 is the dominant allergic protein found in dust mite feces.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
QS-21 DB05400
biotech

QS-21 is an investigational adjuvant, which is a substance added to vaccines and other immunotherapies that is designed to enhance the body’s immune response to the antigen contained within the treatment. It is the leading member of the Stimulon family of adj…

Kategori:
Adjuvants, ImmunologicCarbohydratesGlycosides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1396823-56-5

Quaratusugene ozeplasmid is under investigation in clinical trial NCT05062980 (Quaratusugene Ozeplasmid (Reqorsa) in Combination With Pembrolizumab in Previously Treated Non-small Lung Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quetiapine Approved DB01224
small molecule | CAS: 111974-69-7

Initially approved by the FDA in 1997, quetiapine is a second-generation atypical antipsychotic used in schizophrenia, major depression, and bipolar disorder.[L8546] Quetiapine demonstrates a high level of therapeutic efficacy and low risk of adverse effects …

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +44
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptor5-hydroxytryptamine receptor 1A +21
Waktu ParuhThe average termina…
Vol. DistribusiQuetiapine distribu…
KlirensThe clearance of qu…
Genetik -
small molecule | CAS: 8004-92-0

Deskripsi belum tersedia.

Kategori:
Agents causing angioedemaAgents that produce hypertensionHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quizartinib Approved DB12874
small molecule | CAS: 950769-58-1

Quizartinib is an oral and potent fms-like tyrosine kinase 3 (FLT3) inhibitor and it is the first drug developed specifically targeting FLT3, as other agents with FLT3 inhibition activities were investigated with other targets in mind.[A260641] Additionally, …

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +17
Target Protein:
Receptor-type tyrosine-protein kinase FLT3
Waktu ParuhThe mean (SD) effec…
Vol. DistribusiVolume of distribut…
KlirensTotal body clearanc…
Genetik -
R-30490 DB09179
small molecule | CAS: 60618-49-7

R-30490 is an opioid related to carfentanil used as an animal tranquilizer. It was first synthesized by Janssen Pharmaceutica as part of a structure-activity relationship study of fentanly and its derivatives. R-30490 was found to be the most selective agonis…

Kategori:
Piperidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

IMOGAM Rabies Pasteurized is indicated for post-exposure prophylaxis in persons suspected of exposure to rabies, who have not previously received a complete immunization regimen with a cell culture produced rabies vaccine. Persons previously vaccinated wit…

Kategori:
Human Rabies Immune GlobulinsSerumVaccines
Target Protein:
Rabies Virus Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Rabies virus inactivated antigen, A is an inactivated virus vacine for the intramuscular injection. It is an active immunization against rabies that can be administered pre- or post-exposure to the rabies virus.

Kategori:
Actively Acquired ImmunityAntiinfectives for Systemic UseBiological Products +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Radafaxine DB11790
small molecule | CAS: 192374-14-4

Radafaxine has been used in trials studying the treatment of Depressive Disorder, Major.

Kategori:
KetonesPropiophenones
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ragweed pollen extract Approved DB05368
biotech

Ragweed pollen extract has been developed by Curalogic. The company has initiated a phase III trial with its product for oral immunotherapy of ragweed allergy. While traditional disease-modifying immunotherapeutics are administered by subcutaneous injection, …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rainbow trout Approved DB15540
biotech

Rainbow trout allergenic extract is used in allergenic testing.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2610074-57-0

Raludotatug deruxtecan is under investigation in clinical trial NCT06660654 (A Study of Raludotatug Deruxtecan in Participants With Advanced/metastatic Solid Tumors (Rejoice-pantumor01)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ramosetron DB09290
small molecule | CAS: 132036-88-5

Ramosetron is a _serotonin 5-HT3 receptor antagonist_ commonly employed to treat nausea and vomiting, in addition to certain diarrheal conditions. It is believed to have higher potency and longer antiemetic action than other 1st generation 5-HT3 antagonists s…

Kategori:
Antidepressive AgentsAntiemeticsAutonomic Agents +10
Target Protein:
5-hydroxytryptamine receptor 3A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ramucirumab Approved DB05578
biotech | CAS: 947687-13-0

Ramucirumab is a human monoclonal antibody (IgG1) against vascular endothelial growth factor receptor 2 (VEGFR2), a type II trans-membrane tyrosine kinase receptor expressed on endothelial cells. By binding to VEGFR2, ramucirumab prevents binding of its ligan…

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +20
Target Protein:
Vascular endothelial growth factor receptor 2
Waktu Paruh15 days
Vol. Distribusi5.5 L
Klirens0.014 L/hour
Genetik -
Ranibizumab Approved DB01270
biotech | CAS: 347396-82-1

Ranibizumab is a recombinant humanized IgG1 kappa isotype monoclonal antibody fragment directed against human vascular endothelial growth factor A (VEGF-A), which is a glycoprotein implicated in the pathophysiology of age-related macular degeneration.[A2301, …

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +19
Target Protein:
Vascular endothelial growth factor A, long form
Waktu ParuhThe estimated avera…
Vol. DistribusiThe apparent volume…
KlirensIn patients with re…
Genetik -
Ranitidine Approved DB00863
small molecule | CAS: 66357-35-5

Ranitidine is a commonly used drug, classified as a histamine H2-receptor antagonist, and belongs to the same drug class as [cimetidine] and [famotidine]. This drug helps to prevent and treat gastric-acid associated conditions, including ulcers, because of it…

Kategori:
Acid ReducersAgents Causing Muscle ToxicityAlimentary Tract and Metabolism +29
Target Protein:
Histamine H2 receptorAcetylcholinesterase
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensRenal clearance is …
Genetik -
Rapastinel DB11801
small molecule | CAS: 117928-94-6

Rapastinel has been used in trials studying the treatment of Depressive Disorder, Major and Obsessive-Compulsive Disorder (OCD).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rasagiline Approved DB01367
small molecule | CAS: 136236-51-6

Rasagiline is an irreversible inhibitor of monoamine oxidase and is used as a monotherapy in early Parkinson's disease or as an adjunct therapy in more advanced cases.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAnti-Parkinson Drugs +19
Target Protein:
Amine oxidase [flavin-containing] BApoptosis regulator Bcl-2
Waktu ParuhRasagiline has a me…
Vol. Distribusi* 87 L
Klirens-
Genetik -
Raubasine DB15949
small molecule | CAS: 483-04-5

Deskripsi belum tersedia.

Kategori:
AlkaloidsCardiovascular AgentsHeterocyclic Compounds, Fused-Ring +5
Target Protein:
Beta-1 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 8063-17-0

Rauwolfia (Rauwolfia serpentina), also spelled _ravolphia_, is a medicinal plant in the milkweed family. The root of the plant is ground into a powder or sold in tablets or capsules. It is a compound commonly used in Asian medicine, which includes traditional…

Kategori:
AlkaloidsAntiadrenergic Agents, Centrally ActingAntihypertensive Agents +6
Target Protein:
Synaptic vesicular amine transporter
Waktu ParuhAfter oral ingestio…
Vol. Distribusi-
KlirensHepatically and ren…
Genetik -
Ravulizumab Approved DB11580
biotech | CAS: 1803171-55-2

Ravulizumab is a potent and selective complement 5 (C5) inhibitor. It is a humanized monoclonal IgG2/4 kappa antibody produced in Chinese hamster ovary (CHO) cells.[L39690] Ravulizumab was engineered from [eculizumab], another complement inhibitor, to increas…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
Complement C5
Waktu ParuhThe mean (%CV) term…
Vol. DistribusiThe mean (%CV) volu…
KlirensThe mean (%CV) clea…
Genetik -
Razuprotafib DB16353
small molecule | CAS: 1008510-37-9

Razuprotafib, also known as AKB-9778, is a small-molecule inhibitor restoring Tie2 activation by inhibiting VE-PTP.[L27171,L27176] In investigations against diabetes and COVID-19, razuprotafib is self-administered by patients through subcutaneous injection.

Kategori:
AcidsAcids, NoncarboxylicAmines +2
Target Protein:
Receptor-type tyrosine-protein phosphatase betaAngiopoietin-1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RC118 DB18428
biotech

RC118 is an antibody-drug conjugate that consists of a recombinant humanized IgG1 anti-Claudin18.2 monoclonal antibody conjugated to MMAE.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RC88 DB18697
biotech

RC88 is an antibody-drug conjugate comprising a humanized anti-mesothelin monoclonal antibody conjugated to monomethyl auristatin E (MMAE).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rebamipide Approved DB11656
small molecule | CAS: 90098-04-7

Rebamipide has been investigated for the treatment of Stomach Ulcer, Keratoconjunctivitis Sicca, and Gastric Adenoma and Early Gastric Cancer.

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids, Peptides, and Proteins +11
Target Protein:
fMet-Leu-Phe receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
REC-994 DB15616
small molecule

REC-994 was cleared by the FDA in July, 2018 for a phase I trial for the treatment of cerebral cavernous malformation (CCM).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Receptor binding domain SARS-CoV-2 Hepatitis B surface antigen virus-like particle vaccine (RBD SARS-CoV-2 HBsAg VLP vaccine), is a virus-like particle vaccine candidate where the RBD antigen is conjugated to the hepatitis B surface antigen[A226593]. Virus-li…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 389069-73-2

Recombinant human kallikrein-1 is under investigation in clinical trial NCT01845064 (A Study to Evaluate the Safety and Effectiveness of DM199 in Healthy Subjects and Type 2 Diabetes Patients).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

The Recombinant SARS-CoV-2 Vaccine was created by inserting genes of the SARS-CoV-2 spike protein’s receptor-binding domain into a baculovirus expression system[F4738, A226853]. In pre-clinical trial testing on mice, rabbits, and non-human primates, the candi…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Recombinant stabilized RSV B prefusion F antigen is one component of a bivalent respiratory syncytial virus (RSV) vaccine called Abrysvo. The vaccine comprises two antigens - the other being [recombinant stabilized RSV A prefusion F antigen] - which have been…

Kategori:
Respiratory syncytial virus (RSV) vaccinesVaccinesViral Vaccines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Recombinant stabilized RSV B prefusion F antigen is one component of a bivalent respiratory syncytial virus (RSV) vaccine called Abrysvo. The vaccine comprises two antigens - the other being [recombinant stabilized RSV A prefusion F antigen] - which have been…

Kategori:
Respiratory syncytial virus (RSV) vaccinesVaccinesViral Vaccines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Relatlimab Approved DB14851
biotech | CAS: 1673516-98-7

Relatlimab is a human IgG4 monoclonal antibody and novel immune checkpoint inhibitor that targets lymphocyte activation gene-3 (LAG-3).[A246165,L41265] It was the first commercially developed anti-LAG-3 antibody, entering clinical trials in 2013,[A246155] and…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
Lymphocyte activation gene 3 protein
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
KlirensAt steady-state, th…
Genetik -
Relebactam Approved DB12377
small molecule | CAS: 1174018-99-5

Relebactam is a diazabicyclooctane beta-lactamase inhibitor, similar in structure to [avibactam].[A181195,A181207] It includes a piperidine ring which reduces export from bacterial cells by producing a positive charge.[A181207] It is currently available in a …

Kategori:
Antibacterials for Systemic UseAntiinfectives for Systemic UseAza Compounds +6
Target Protein:
Beta-lactamaseBeta-lactamase TEMBeta-lactamase SHV-1 +3
Waktu ParuhRelebactam has a ha…
Vol. DistribusiRelebactam has a vo…
KlirensRelebactam has a re…
Genetik -
Relmapirazin DB19130
small molecule | CAS: 1313706-17-0

Relmapirazin is under investigation in clinical trial NCT05425719 (Pharmacokinetics and Safety of MB-102 (Relmapirazin) and the Medibeacon Transdermal GFR Measurement System in Evaluation of Kidney Function in Normal and Renal Compromised Subjects).

Target Protein:
Interleukin-3 receptor subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Relugolix Approved DB11853
small molecule | CAS: 737789-87-6

Relugolix is a gonadotropin-releasing hormone (GnRH) receptor antagonist used in the treatment of several hormone-responsive conditions. It was first approved in Japan in 2019, under the brand name Relumina, for the symptomatic treatment of uterine fibroids,[…

Kategori:
AmidesAnti-Gonadotropin-Releasing HormonesAntiandrogens +30
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu ParuhThe average effecti…
Vol. Distribusi-
KlirensThe average renal c…
Genetik -
Remdesivir Approved DB14761
small molecule | CAS: 1809249-37-3

Severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) is the causative agent of coronavirus disease 2019 (COVID-19), which is a respiratory disease that is capable of progressing to viral pneumonia and acute respiratory distress syndrome (ARDS); COVID-…

Kategori:
Adenine NucleotidesAmino AcidsAmino Acids, Peptides, and Proteins +37
Target Protein:
Replicase polyprotein 1abReplicase polyprotein 1abReplicase polyprotein 1ab +1
Waktu ParuhRemdesivir has an e…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Remifentanil Approved DB00899
small molecule | CAS: 132875-61-7

Remifentanil (marketed by Abbott as Ultiva) is a potent ultra short-acting synthetic opioid given to patients during surgery for pain relief and adjunctive to an anaesthetic. Remifentanil is a specific mu-type-opioid receptor agonist which means it reduces sy…

Kategori:
Acids, AcyclicAgents producing tachycardiaAgents that produce hypertension +24
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu Paruh1-20 minutes
Vol. Distribusi* 350 mL/kg * 452 …
Klirens* 40 mL/min/kg [you…
Genetik -
Remimazolam Approved DB12404
small molecule | CAS: 308242-62-8

Remimazolam is an ultra short-acting benzodiazepine used in the induction and maintenance of sedation during short (<30 minute) procedures.[L14647] Recent trends in anesthesia-related drug development have touted the benefits of so-called "soft drugs" - these…

Kategori:
BenzazepinesBenzodiazepine hypnotics and sedativesBenzodiazepines and benzodiazepine derivatives +8
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu ParuhFollowing intraveno…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of re…
Genetik -
Remlarsen DB19131
biotech | CAS: 1848266-71-6

Remlarsen is under investigation in clinical trial NCT03601052 (Efficacy, Safety, and Tolerability of Remlarsen (MRG-201) Following Intradermal Injection in Subjects With a History of Keloids).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Remtolumab DB15128
biotech | CAS: 1791410-27-9

Remtolumab is under investigation in clinical trial NCT02433340 (Phase 2, Multicenter, Open-Label Extension (OLE) Study With ABT-122 in Rheumatoid Arthritis Subjects Who Have Completed the Preceding M12-963 Study).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
REP8839 DB05224
small molecule

REP8839 is a novel methionyl-tRNA synthetase (MetS) inhibitor being developed by Replidyne (GlaxoSmithKline licensed REP8839 to Replidyne in June of 2003).

Kategori:
AminesPolyaminesSulfur Compounds
Target Protein:
Methionine--tRNA ligase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Repotrectinib Approved DB16826
small molecule | CAS: 1802220-02-5

Repotrectinib is a next-generation tyrosine kinase inhibitor (TKI) specifically designed to address resistance in the treatment of non-small cell lung cancer (NSCLC), specifically due to mutations in the ROS1 gene.[A262056] ROS1 mutations are one of the defin…

Kategori:
BCRP/ABCG2 InhibitorsCytochrome P-450 CYP2B6 InducersCytochrome P-450 CYP2B6 Inducers (strength unknown) +28
Target Protein:
Proto-oncogene tyrosine-protein kinase ROSHigh affinity nerve growth factor receptorBDNF/NT-3 growth factors receptor +1
Waktu ParuhThe repotrectinib m…
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Reproxalap DB16688
small molecule | CAS: 916056-79-6

Reproxalap (previously ADX 102 or NS-2) is a small molecule inhibitor being developed by Aldeyra Therapeutics investigated against dry eye disease, allergic conjunctivitis, noninfectious anterior uveitis, and Sjögren-Larsson syndrome.[L32990] NS-2 has orphan …

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 1451–1500 dari 1977
Sebelumnya Halaman 30 / 40 Berikutnya