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124

Total database: 17430
Struktur (SMILES)
63 (50.8%)
Target
70 (56.5%)
Genomik
6 (4.8%)
Referensi
124 (100.0%)

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Halaman 3 / 3
Rotigotine Approved DB05271
small molecule | CAS: 99755-59-6

Rotigotine (Neupro) is a non-ergoline dopamine agonist indicated for the treatment of Parkinson's disease (PD) and restless legs syndrome (RLS) in Europe and the United States. It is formulated as a once-daily transdermal patch which provides a slow and const…

Kategori:
Agents that produce hypertensionAnti-Parkinson Agents (Dopamine Agonist)Anti-Parkinson Drugs +23
Target Protein:
D(3) dopamine receptorD(4) dopamine receptorD(2) dopamine receptor +4
Waktu ParuhAfter removal of th…
Vol. DistribusiThe weight normaliz…
Klirens-
Genetik -
Rozanolixizumab Approved DB14919
biotech | CAS: 1584645-37-3

Rozanolixizumab is a humanized high-affinity anti-human neonatal Fc receptor (FcRn) monoclonal antibody (IgG4P) targeting the immunoglobulin G (IgG). Rozonolixizumab itself is an IgG4P, an inactive isotype, to reduce the likelihood of unwanted chain exchange.…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
IgG receptor FcRn large subunit p51
Waktu Paruh-
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
RP-L201 DB17595
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Satralizumab Approved DB15762
biotech | CAS: 1535963-91-7

Satralizumab is a recombinant humanized monoclonal antibody targeted against human interleukin-6 (IL-6) receptors, similar to [tocilizumab], which is produced in Chinese hamster ovary cells and based on an IgG2 framework.[L15536] Satralizumab is used in the t…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Interleukin-6 receptor subunit alpha
Waktu ParuhThe terminal half-l…
Vol. DistribusiSatralizumab is sub…
KlirensThe total clearance…
Genetik -
SBT-100 DB17215
biotech

SBT-100 is an anti-signal transducer and activator of transcription 3 (STAT3) B VHH13 single-domain antibody (sdAb). It was granted orphan drug designation by the FDA for the treatment of pancreatic cancer and osteosarcoma.[L44131,L44136]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Scopolamine Approved DB00747
small molecule | CAS: 51-34-3

Scopolamine is a tropane alkaloid isolated from members of the _Solanaceae_ family of plants, similar to [atropine] and [hyoscyamine], all of which structurally mimic the natural neurotransmitter [acetylcholine].[A228423, A228763] Scopolamine was first synthe…

Kategori:
AdjuvantsAdjuvants, AnesthesiaAgents producing tachycardia +30
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +5
Waktu ParuhThe half-life of sc…
Vol. DistribusiThe volume of distr…
KlirensIV infusion of 0.5 …
Genetik -
scyllo-inositol DB03106
small molecule | CAS: 488-59-5

An isomer of glucose that has traditionally been considered to be a B vitamin although it has an uncertain status as a vitamin and a deficiency syndrome has not been identified in man. (From Martindale, The Extra Pharmacopoeia, 30th ed, p1379) Inositol phosph…

Kategori:
AlcoholsCarbohydratesStereoisomerism +1
Target Protein:
Lysosomal acid glucosylceramidase1-phosphatidylinositol phosphodiesteraseCDP-diacylglycerol--inositol 3-phosphatidyltransferase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SD-0006 DB07943
small molecule | CAS: 271576-80-8

Deskripsi belum tersedia.

Target Protein:
Mitogen-activated protein kinase 14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SD118 DB05207
small molecule

SD118 was previously under investigation in Japan for a different indication and now, following re-profiling and evaluation in experimental animal models, has demonstrated its potential as a new oral therapy for neuropathic pain.

Target Protein:
Tumor necrosis factorInterleukin-1 receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SD146 DB02729
small molecule | CAS: 183854-21-9

Deskripsi belum tersedia.

Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sevirumab DB17771
biotech | CAS: 138660-96-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 151-21-3

Sodium Lauryl Sulfate (SLS) is an anionic surfactant naturally derived from coconut and/or palm kernel oil. It usually consists of a mixture of sodium alkyl sulfates, mainly the lauryl. SLS lowers surface tension of aqueous solutions and is used as fat emulsi…

Kategori:
AlcoholsAlkanesulfonatesAlkanesulfonic Acids +9
Target Protein:
Albumin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sotatercept Approved DB12118
biotech | CAS: 1001080-50-7

Sotatercept is an activin signalling inhibitor. It is a homodimeric recombinant fusion protein consisting of the extracellular domain of the human activin receptor type IIA (ActRIIA) linked to the human IgG1 Fc domain.[L50351] On March 26, 2024, sotatercep…

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsImmunoglobulin G +5
Target Protein:
Activin receptor type-2AActivin receptor type-1BGrowth/differentiation factor 8 +1
Waktu ParuhThe effective half-…
Vol. DistribusiThe population PK m…
KlirensClearance is approx…
Genetik -
Strimvelis DB17594
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 30344-00-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +1
Target Protein:
Haloalkane dehalogenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tacrolimus Approved DB00864
small molecule | CAS: 104987-11-3

Tacrolimus (also FK-506 or Fujimycin) is an immunosuppressive drug whose main use is after organ transplant to reduce the activity of the patient's immune system and so the risk of organ rejection. It is also used in a topical preparation in the treatment of …

Kategori:
Agents causing hyperkalemiaAgents Causing Muscle ToxicityAgents for Dermatitis, Excluding Corticosteroids +33
Target Protein:
Protein phosphatase 3 catalytic subunit alphaPeptidyl-prolyl cis-trans isomerase FKBP1A
Gen Terkait:
CYP3A5 ABCB1
Waktu ParuhThe elimination hal…
Vol. Distribusi* 2.6 ± 2.1 L/kg [p…
Klirens* 0.040 L/hr/kg [he…
Genetik 2 Varian
Thalagen DB17714
biotech

Thalagen is a branded product developed by San Rocco Therapeutics. It consists of autologous CD34-positive hematopoietic progenitor cells transduced with TNS9.3.55, a lentiviral vector encoding the normal human beta-globin gene. It is being investigated for t…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tocofersolan Approved DB11635
small molecule | CAS: 9002-96-4

D-Alpha-tocopheryl polyethylene glycol 1000 succinate (Tocofersolan, Vedrop), has been developed in Europe as an orally bioavailable source of vitamin E in children suffering from cholestasis [L2371]. Cholestasis is the reduction or stoppage of bile flow, eit…

Kategori:
Alimentary Tract and MetabolismBenzopyransCompounds used in a research, industrial, or household setting +9
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh29.7 h [L2371]
Vol. DistribusiLocated principally…
Klirens-
Genetik -
biotech

Toll-like receptor 9 is under investigation in clinical trial NCT03007732 (Pembrolizumab in Combination With Intratumoral SD-101 Therapy).

Kategori:
Amino Acids, Peptides, and ProteinsDNA-Binding ProteinsMembrane Proteins +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Virginiamycin DB11476
small molecule | CAS: 11006-76-1

Virginiamycin is a streptogramin antibiotic similar to pristinamycin and quinupristin/dalfopristin. It is a combination of pristinamycin IIA and virginiamycin S1. Virginiamycin is used in the fuel ethanol industry to prevent microbial contamination and in liv…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vofopitant DB12436
small molecule | CAS: 168266-90-8

Vofopitant has been used in trials studying the treatment of PTSD, Primary Insomnia, and Sleep Initiation and Maintenance Disorders.

Kategori:
AntiemeticsAutonomic AgentsCentral Nervous System Agents +4
Target Protein:
Substance-P receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
WSD-0922 DB17170
small molecule | CAS: 2226552-64-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
WU-CART-007 DB18617
biotech

WU-CART-007 consists of allogeneic, fratricide-resistant genetically modified T cells transduced with a 2nd generation 4-1BB-CD3z chimeric antigen receptor targeting human CD7.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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