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2279

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1100 (48.3%)
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Halaman 3 / 46
AGT-182 DB17630
biotech

AGT-182 is an investigational enzyme replacement therapy engineered by the fusion of the iduronate-2-sulfatase (IDS) enzyme and a human insulin receptor monoclonal antibody.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AI-128 DB05841
small molecule

AI-128 is the first human demonstration of sustained release drug administration in the lung. AI-128 consists of slowly dissolving microspheres designed to control where drug particles go in the lung and how quickly they release their drug.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Ajmaline Approved DB01426
small molecule | CAS: 4360-12-7

An alkaloid found in the root of Rauwolfia serpentina, among other plant sources. It is a class Ia antiarrhythmic agent that apparently acts by changing the shape and threshold of cardiac action potentials. Ajmaline produces potent sodium channel blocking eff…

Kategori:
Ajmaline and derivativesAlkaloidsAntiarrhythmic agents +16
Target Protein:
Sodium channel protein type 5 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AK119 DB16423
biotech

AK119 is a humanized anti-CD73 monoclonal antibody being investigated in the clinical trial NCT04516564 (A Study of AK119 (Anti-CD73 Antibody), a Treatment for COVID-19, in Healthy Subjects).[L28315]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Albendazole Approved DB00518
small molecule | CAS: 54965-21-8

A benzimidazole broad-spectrum anthelmintic structurally related to mebendazole that is effective against many diseases. (From Martindale, The Extra Pharmacopoeia, 30th ed, p38)

Kategori:
Acids, AcyclicAnthelminticsAnti-Infective Agents +23
Target Protein:
Tubulin beta-2 chainTubulin alpha-1A chainTubulin beta-4B chain +1
Waktu ParuhTerminal eliminatio…
Vol. Distribusi-
Klirens-
Genetik -
Albiglutide Approved DB09043
biotech | CAS: 782500-75-8

Albiglutide is a glucagon-like peptide-1 agonist (GLP-1) biologic drug indicated in the treatment of type 2 diabetes. It is marketed under the brands Eperzan and Tanzeum by GSK (GlaxoSmithKline). It is a dipeptidyl peptidase-4-resistant glucagon-like peptide-…

Kategori:
Alimentary Tract and MetabolismBlood Glucose Lowering AgentsDrugs Used in Diabetes +10
Target Protein:
Glucagon-like peptide 1 receptor
Waktu Paruh4-7 days.
Vol. Distribusi11 L.
Klirens67 mL/h.
Genetik -
biotech | CAS: 472960-22-8

Albumin-interferon alpha (Albuferon) is a novel, long-acting form of interferon alpha. Recombinant interferon alpha is approved for the treatment of hepatitis C, hepatitis B, and a broad range of cancers. Human Genome Sciences modified interferon alpha to imp…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Albumin human Approved DB00062
biotech | CAS: 9048-46-8

Human serum albumin is the primary protein present in human blood plasma. The main function of albumin is to maintain the oncotic pressure of blood [A33706]. It binds to water, cations (such as Ca2+, Na+ and K+), fatty acids, hormones, bilirubin, thyroxine (T…

Kategori:
AlbuminsAmino Acids, Peptides, and ProteinsBlood and Blood Forming Organs +13
Target Protein:
Nitric oxide
Waktu Paruh-
Vol. DistribusiAlbumin is distribu…
Klirens-
Genetik -
biotech

I-125 iodinated albumin is a radiolabeled albumin-based diagnostic agent used in the determination of total blood and plasma volume.[L12780]

Kategori:
Radioactive Diagnostic AgentRadiopharmaceutical Activity
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Iodinated I-131 serum albumin is a radiopharmaceutical agent used for several diagnostic purposes, including the determination of body fluid volumes and the imaging of certain tissues.[L12783]

Kategori:
Radiopharmaceutical Activity
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Albusomatropin DB12950
biotech | CAS: 1613273-96-3

Albusomatropin has been used in trials studying the treatment of Growth Hormone-Deficiency and Growth Hormone Deficiency.

Kategori:
AlbuminsAmino Acids, Peptides, and ProteinsBlood Proteins +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Albutrepenonacog alfa Approved DB13884
biotech | CAS: 1357448-54-4

Albutrepenonacog alfa (rIX-RFP) is a recombinant fusion protein that links a recombinant coagulation factor IX (rFIX) with a recombinant human albumin (rAlbumin).[A32547] It was developed by CSL Behring Canada, Inc and approved by Health Canada on April 26, 2…

Kategori:
AlbuminsAmino Acids, Peptides, and ProteinsBiological Factors +9
Target Protein:
Coagulation factor X
Waktu ParuhThe fusion of the r…
Vol. DistribusiThe reported volume…
KlirensIn clinical trials,…
Genetik -
Aldafermin DB16086
biotech | CAS: 1616639-03-2

Aldafermin is under investigation in clinical trial NCT03912532 (Evaluation of Efficacy, Safety and Tolerability of Aldafermin in a Phase 2b, Randomized, Double-blind, Placebo-controlled, Multi-center Study in Subjects With Nonalcoholic Steatohepatitis and St…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aldesleukin Approved DB00041
biotech | CAS: 110942-02-4

Aldesleukin, a lymphokine, is produced by recombinant DNA technology using a genetically engineered E. coli strain containing an analog of the human interleukin-2 gene. Genetic engineering techniques were used to modify the human IL-2 gene, and the resulting …

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAnti-HIV Agents +26
Target Protein:
Interleukin-2 receptor subunit betaInterleukin-2 receptor subunit alphaCytokine receptor common subunit gamma
Waktu Paruh13 min-85 min
Vol. Distribusi0.18 l/kg
Klirens-
Genetik -
Alefacept Approved DB00092
biotech | CAS: 222535-22-0

Immunosuppressive dimeric fusion protein that consists of the extracellular CD2-binding portion of the human leukocyte function antigen-3 (LFA-3) linked to the Fc (hinge, CH2 and CH3 domains) portion of human IgG1. Produced by CHO cells, mW is 91.4 kD.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntineoplastic and Immunomodulating Agents +20
Target Protein:
T-cell surface antigen CD2Low affinity immunoglobulin gamma Fc region receptor III-ALow affinity immunoglobulin gamma Fc region receptor III-B
Waktu Paruh~270 hours
Vol. Distribusi-
Klirens-
Genetik -
Aleglitazar DB08915
small molecule | CAS: 475479-34-6

Aleglitazar is an investigational drug from the company Hoffmann–La Roche and is currently in a phase III clinical trial called ALECARDIO. It is being investigated for use in patients with type II diabetes to reduce their risks of cardiovascular mortality and…

Kategori:
Sulfur Compounds
Target Protein:
Peroxisome proliferator-activated receptor alphaPeroxisome proliferator-activated receptor gammaNuclear receptor coactivator 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alemtuzumab Approved DB00087
biotech | CAS: 216503-57-0

Alemtuzumab is a humanized monoclonal antibody specific to lymphocyte antigens. It is a recombinant DNA-derived humanized monoclonal antibody (Campath-1H) that is directed against the 21-28 kD cell surface glycoprotein, CD52. The Campath-1H antibody is an IgG…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
CAMPATH-1 antigenLow affinity immunoglobulin gamma Fc region receptor III-BLow affinity immunoglobulin gamma Fc region receptor III-A +4
Waktu ParuhThe elimination hal…
Vol. DistribusiAlemtuzumab is larg…
KlirensClearance of alemtu…
Genetik -
Alfacalcidol Approved DB01436
small molecule | CAS: 41294-56-8

Alfacalcidol, or 1-alpha-hydroxycholecalciferol or 1-alpha-hydroxyvitamin D3, is a non-endogenous analogue of [vitamin D].[A234044] It plays an essential function in calcium homeostasis and bone metabolism. Alfacaldisol is activated by the enzyme 25-hydroxyla…

Kategori:
Alimentary Tract and MetabolismBone Density Conservation AgentsCholestanes +13
Target Protein:
Vitamin D3 receptor25-hydroxyvitamin D-1 alpha hydroxylase, mitochondrialRetinoic acid receptor RXR-alpha
Waktu ParuhThe half-life of al…
Vol. Distribusi-
Klirens-
Genetik -
Alginic acid Approved DB13518
small molecule | CAS: 9005-32-7

Alginic acid, also referred to as algin or alginate, is a hydrophilic or anionic polysaccharide isolated from certain brown seaweed (_Phacophycae_) via alkaline extraction. It is present in cell walls of brown algae where it forms a viscous gel when binding w…

Kategori:
Acids, AcyclicAcids, AldehydicAlginates +11
Waktu ParuhThis pharmacokineti…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Alglucerase Approved DB00088
biotech | CAS: 143003-46-7

Human Beta-glucocerebrosidase or Beta-D-glucosyl-N-acylsphingosine glucohydrolase E.C. 3.2.1.45. 497 residue protein with N-linked carbohydrates, MW=59.3 kD. Alglucerase is prepared by modification of the oligosaccharide chains of human Beta-glucocerebrosidas…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +6
Target Protein:
Glucocerebroside
Waktu Paruh3.6-10.4 min
Vol. Distribusi* 49.4 to 282.1 mL/…
Klirens-
Genetik -
Alglucosidase alfa Approved DB01272
biotech | CAS: 420784-05-0

Aglucosidase alfa consists of the human enzyme acid alpha-glucosidase (GAA) which is essential for the degradation of glygogen to glucose in lysosomes. It is encoded by the most predominant of nine observed haplotypes of this gene. Aglucosidase alfa is produc…

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes +5
Target Protein:
Cation-dependent mannose-6-phosphate receptorGlycogen
Waktu Paruh2.3 ± 0.4 ho…
Vol. Distribusi* 96 ± 16 mL/kg [20…
Klirens* 25+/- 4 mL/hr/kg …
Genetik -
Alidornase alfa DB18144
biotech | CAS: 1788036-49-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alipogene tiparvovec Approved DB13521
biotech | CAS: 929881-05-0

Alipogene tiparvovec is an adeno-associated viral vector of serotype 1-based gene therapy that delivers the Ser(447)X variant of the human lipoprotein lipase (LPL) gene. It is being investigated for the treatment of lipoprotein lipase (LPL) deficiency.[A25979…

Kategori:
Adeno-associated Viral Vector TherapiesLipid Modifying AgentsLipid Modifying Agents, Plain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alirocumab Approved DB09302
biotech | CAS: 1245916-14-6

Alirocumab is a biopharmaceutical that obtained FDA approval in July 2015 as a second line treatment for high cholesterol in adults whose LDL-cholesterol (LDL-C) is not controlled by the combination of diet and statin treatment. It is a human monoclonal antib…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +20
Target Protein:
Proprotein convertase subtilisin/kexin type 9
Waktu ParuhIn monotherapy, the…
Vol. DistribusiAlirocumab is mainl…
Klirens-
Genetik -
Allantoin Approved DB11100
small molecule | CAS: 97-59-6

Allantoin is a substance that is endogenous to the human body and also found as a normal component of human diets [FDA Label]. In healthy human volunteers, the mean plasma concentration of allantoin is about 2-3 mg/l. During exercise, the plasma allantoin con…

Kategori:
AmidesBasic Ointments and ProtectantsDermatologicals +5
Waktu ParuhWhen studied in cat…
Vol. Distribusi-
KlirensSome studies sugges…
Genetik -
biotech

Cardiosphere-derived cells (CDCs) are derived from human neonatal heart tissue with a distinct antigenic profile (CD105+, CD45-, and CD90low). They exert their effects by secreting exosomes: nanometer-sized, membrane-bound vesicles used for the purpose of cel…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Stratagraft (allogeneic cultured keratinocytes and dermal fibroblasts in murine collagen-dsat) is an allogeneic cellularized scaffold product used for the treatment of adults with thermal burns containing intact dermal elements for which surgical intervention…

Kategori:
FibroblastsKeratinocytes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

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Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

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Vol. Distribusi-
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Genetik -
biotech

ORBCEL-C™ is the trade name of a product composed of highly purified stromal cells derived from the human umbilical cord. The isolated cells are expanded in culture and are able to be used allogenically -- meaning that one donor’s cells can be given to other …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Umbilical-cord derived MSCs are currently being tested for numerous clinical applications due to their immunosuppressive and anti-inflammatory properties. In comparison to bone-marrow derived MSCs, these cells are more resilient, easier to extract, and genera…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Human olfactory mucosa-derived mesenchymal stem cells (OM-MSCs) reside in an accessible location of the nasal cavity and have properties of multipotency and high proliferation, which contributes to high potential for regenerative medicine. In humans, OM-MSCs …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Allopurinol Approved DB00437
small molecule | CAS: 315-30-0

Gout is a disease that occurs by the deposition of monosodium urate crystals (MSU) in body tissues, especially around joints [A175942]. This disease has been well-documented in historical medical records and appears in the biographies of several prominent, h…

Kategori:
Antigout PreparationsAntimetabolitesAntioxidants +12
Target Protein:
Xanthine dehydrogenase/oxidase
Gen Terkait:
HCP5
Waktu ParuhThe plasma half-lif…
Vol. DistribusiAllopurinol and oxy…
KlirensSince allopurinol a…
Genetik 1 Varian
Allylestrenol DB01431
small molecule | CAS: 432-60-0

A synthetic steroid with progestational activity. It is widely marketed throughout Europe, including Russia and many other European countries, and is also available in Japan, Hong Kong, India, Bangladesh, Indonesia, and much of Southeast Asia, though notably …

Kategori:
Adrenal Cortex HormonesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +13
Target Protein:
Progesterone receptorSodium- and chloride-dependent glycine transporter 1Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ALM201 DB17206
biotech

ALM201 is an anti-angiogenic synthetic peptide identified from the endogenous human protein, FKBPL. It is being investigated in the treatment of various cancers.[A254556]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ALMB-0166 DB17937
biotech

ALMB-0166 is a umanized connexin 43 (Cx43) monoclonal antibody being investigated for the treatment of acute spinal cord injury. It was granted FDA orphan designation in November 2018.[L47067]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ALMB-0168 DB16926
biotech

ALMB-0168 is a humanized connexin 43 (Cx43) monoclonal antibody being investigated for osteosarcoma.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aloe vera leaf DB13906
biotech | CAS: 8001-97-6

Aloe describes a genus including over 500 species of flowering succulent plants that grow in the Southern peninsula and various islands. Aloe vera, or _Aloe barbadensis miller_, is the most common species of Aloe that is cultivated for agricultural and medica…

Target Protein:
Free radicals
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Alosetron Approved DB00969
small molecule | CAS: 122852-42-0

Alosetron is a 5-HT3 antagonist used only for the management of severe diarrhoea-predominant irritable bowel syndrome (IBS) in women. Alosetron has an antagonist action on the 5-HT3 receptors and thus may modulate serotonin-sensitive gastrointestinal (GI) pro…

Kategori:
Alimentary Tract and MetabolismAntidepressive AgentsAntiemetic Serotonin 5-HT3 Receptor Antagonists +23
Target Protein:
5-hydroxytryptamine receptor 3A
Waktu Paruh1.5 hours
Vol. Distribusi* 65 to 95 L
Klirens* 600 mL/min
Genetik -
Alpelisib Approved DB12015
small molecule | CAS: 1217486-61-7

Alpelisib is a phosphatidylinositol 3-kinase (PI3K) inhibitor with potent antitumor activity. It works by selectively inhibiting class I PI3K p110? [A179203], which is the catalytic subunit of PI3K, a lipid kinase that plays a role in various biological proce…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +32
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
Waktu ParuhThe mean half life …
Vol. DistribusiThe apparent volume…
KlirensThe mean apparent o…
Genetik -
Alpha-1-proteinase inhibitor Approved DB00058
biotech | CAS: 9041-92-3

Human alpha-1 proteinase inhibitor or alpha-1-antitrypsin, prepared from human plasma via Cohn alcohol fractionation followed by PEG and zinc chloride fractionation.

Kategori:
Acute-Phase ProteinsAlpha-GlobulinsAmino Acids, Peptides, and Proteins +21
Target Protein:
Neutrophil elastase
Waktu Paruh-
Vol. Distribusi* 5632 ± 2006 mL [A…
Klirens* 940 +/- 275 mL/da…
Genetik -
small molecule | CAS: 15978-07-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 40436-60-0

Deskripsi belum tersedia.

Target Protein:
Cation-dependent mannose-6-phosphate receptorPhosphomannomutase/phosphoglucomutaseCation-independent mannose-6-phosphate receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
alpha-Linolenic acid Approved DB00132
small molecule | CAS: 463-40-1

Alpha-linolenic acid (ALA) is a polyunsaturated omega-3 fatty acid. It is a component of many common vegetable oils and is important to human nutrition.

Kategori:
Dietary FatsDietary Fats, UnsaturatedDietary Supplements +8
Target Protein:
Free fatty acid receptor 1Prostaglandin G/H synthase 2Acyl-CoA (8-3)-desaturase +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
alpha-Tocopherol acetate Approved DB14003
small molecule | CAS: 7695-91-2

Alpha-tocopherol is the primary form of vitamin E that is preferentially used by the human body to meet appropriate dietary requirements. In particular, the RRR-alpha-tocopherol (or sometimes called the d-alpha-tocopherol stereoisomer) stereoisomer is conside…

Kategori:
AntioxidantsBenzopyransBiological Factors +16
Target Protein:
Free radicals
Waktu ParuhThe apparent half-l…
Vol. DistribusiWhen three particul…
KlirensWhen three specific…
Genetik -
alpha-Tocopherol succinate Approved DB14001
small molecule | CAS: 4345-03-3

Alpha-tocopherol is the primary form of vitamin E that is preferentially used by the human body to meet appropriate dietary requirements. In particular, the RRR-alpha-tocopherol (or sometimes called the d-alpha-tocopherol stereoisomer) stereoisomer is conside…

Kategori:
AntioxidantsBenzopyransBiological Factors +12
Target Protein:
SEC14-like protein 3SEC14-like protein 2Nuclear receptor subfamily 1 group I member 2 +5
Waktu Paruh_In addition to any…
Vol. Distribusi_In addition to any…
Klirens_In addition to any…
Genetik -
ALT-P1 DB18485
biotech

ALT-P1 is a long-acting recombinant human growth hormone fused to an alpha1-antitrypsin variant. It is under investigation for the treatment of growth hormone deficiency.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alteplase Approved DB00009
biotech | CAS: 105857-23-6

Alteplase is a recombinant tissue plasminogen activator (rt-PA) used as a thrombolytic agent.[L43125] It cleaves plasminogen to form plasmin, an enzyme involved in the degradation of fibrin clots. In the absence of fibrin, the alteplase-mediated conversion of…

Kategori:
Agents causing angioedemaAmino Acids, Peptides, and ProteinsAnticoagulants +19
Target Protein:
PlasminogenFibrinogen alpha chainFibrinogen gamma chain +1
Waktu ParuhAlteplase has an in…
Vol. DistribusiThe initial volume …
KlirensAlteplase has a pla…
Genetik -
ALTU-135 DB05330
biotech

ALTU-135, the Company's orally administered enzyme replacement therapy for patients with pancreatic insufficiency, is manufactured by blending three drug substance enzymes: lipase, protease and amylase. This consistent and pure enzyme combination is designed …

Kategori:
Carboxylic Ester HydrolasesEnzymesEnzymes and Coenzymes +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 53026-85-0

Aluminum chlorohydrex propylene glycol is a complex consisting of Aluminum Chorohydrate and propylene glycol (PG). It is an antiperspirant active ingredient found in antiperspirant drug products for over-the-counter human use.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
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