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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 299 / 321
Tolrestat DB02383
small molecule | CAS: 82964-04-3

Tolrestat (INN) (AY-27773) is an aldose reductase inhibitor which was approved for the control of certain diabetic complications. While it was approved for marketed in several countries, it failed a Phase III trial in the U.S. due to toxicity and never receiv…

Kategori:
Aldehyde Reductase, antagonists & inhibitorsAldose Reductase InhibitorsAlimentary Tract and Metabolism +2
Target Protein:
Sigma non-opioid intracellular receptor 1Aldo-keto reductase family 1 member B1Aldo-keto reductase family 1 member A1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tolterodine Approved DB01036
small molecule | CAS: 124937-51-5

Tolterodine is an antimuscarinic drug that is used to treat urinary incontinence. Tolterodine acts on M2 and M3 subtypes of muscarinic receptors.

Kategori:
Agents producing tachycardiaAlcoholsAmines +26
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M5 +2
Waktu Paruh1.9-3.7 hours
Vol. Distribusi* 113 ± 26.7 L
Klirens-
Genetik -
Tolu balsam DB11223
small molecule | CAS: 9000-64-0

Deskripsi belum tersedia.

Kategori:
Biological ProductsBiopolymersComplex Mixtures +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Toluene DB11558
small molecule | CAS: 108-88-3

Toluene is a colorless, liquid that is immiscible in water. It is a mono-substituted benzene derivative used in veterinary medicine as a treatment for various parasites in dogs and cats.

Kategori:
Benzene DerivativesCompounds used in a research, industrial, or household settingSolvents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tolvaptan Approved DB06212
small molecule | CAS: 150683-30-0

Tolvaptan is used to treat low blood sodium levels (hyponatremia) associated with various conditions like congestive heart failure, cirrhosis, and syndrome of inappropriate antidiuretic hormones (SIADH). FDA approved on May 19, 2009.

Kategori:
Agents causing hyperkalemiaAntidiuretic Hormone Receptor AntagonistsBenzazepines +14
Target Protein:
Vasopressin V2 receptorVasopressin V1a receptor
Waktu ParuhTerminal half life,…
Vol. DistribusiHealthy subjects: 3…
Klirens4 mL/min/kg (post-o…
Genetik -
Tomaralimab DB15415
biotech | CAS: 1449294-76-1

Tomaralimab is under investigation in clinical trial NCT01794663 (Placebo-Controlled Study to Evaluate the Safety and Efficacy of OPN-305 in Preventing Delayed Renal Graft Function).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tominersen DB17924
biotech | CAS: 1709886-74-7

Deskripsi belum tersedia.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tomivosertib DB15219
small molecule | CAS: 1849590-01-7

Tomivosertib is under investigation in clinical trial NCT03318562 (A PD Study of Oral eFT508 in Subjects With Advanced TNBC and HCC).

Target Protein:
MAP kinase-interacting serine/threonine-protein kinase 1MAP kinase-interacting serine/threonine-protein kinase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tomligisiran DB19330
biotech | CAS: 2202789-48-6

Tomligisiran is under investigation in clinical trial NCT06537414 (A Study of Sequential Therapy With Daplusiran/tomligisiran (DAP/TOM) Followed by Bepirovirsen in Participants Living With Chronic Hepatitis B (CHB)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tomuzotuximab DB15178
biotech | CAS: 1646321-00-7

Tomuzotuximab is under investigation in clinical trial NCT02052960 (CetuGEX™ in Comparison to Cetuximab for the Treatment of Patients With Head and Neck Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tonabacase DB17964
biotech | CAS: 1788041-31-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tonabersat DB06578
small molecule | CAS: 175013-84-0

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +3
Target Protein:
5-hydroxytryptamine receptor 1D
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tonapofylline DB12569
small molecule | CAS: 340021-17-2

Tonapofylline has been used in trials studying the treatment of Heart Failure, Renal Insufficiency, and Congestive Heart Failure.

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingPurines +2
Target Protein:
Adenosine receptor A1Adenosine receptor A2aAdenosine receptor A3 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TOP-1288 DB14839
small molecule | CAS: 1630202-02-6

TOP-1288 is under investigation in clinical trial NCT02888379 (Phase 2a Study to Evaluate the Safety/Tolerability and Efficacy of TOP1288 200 mg Rectal Solution Once Daily for 4 Weeks in Ulcerative Colitis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Topiramate Approved DB00273
small molecule | CAS: 97240-79-4

Topiramate is a anti-epileptic drug used to manage seizures and prevent migraines.[A175249] It was initially approved by the FDA in 1996. In 2004, topiramate was approved for the prevention of migraine in adults.[A188309,L10544,L43478] Since 2012, the extende…

Kategori:
Alimentary Tract and MetabolismAnti-Obesity AgentsAnticonvulsants +23
Target Protein:
Glutamate receptor ionotropic, kainate 1Gamma-aminobutyric acid receptor subunit alpha-1Voltage-gated sodium channel alpha subunit +7
Waktu ParuhThe elimination hal…
Vol. DistribusiThe mean apparent v…
KlirensThe mean oral plasm…
Genetik -
Topiroxostat DB01685
small molecule | CAS: 577778-58-6

Topiroxostat is a selective xanthine oxidase inhibitor developed for treatment and management of hyperuricemia and gout. Xanthine oxidase, or xanthine oxidoreductase (XOR), regulates purine metabolism, and inhibition of the enzyme results in efficacious reduc…

Kategori:
BCRP/ABCG2 InhibitorsCytochrome P-450 CYP2C19 InhibitorsCytochrome P-450 CYP2C19 inhibitors (strength unknown) +13
Target Protein:
Xanthine dehydrogenase/oxidase
Waktu ParuhThe mean half life …
Vol. DistribusiThe mean ± SD appar…
KlirensThe apparent total …
Genetik -
Topotecan Approved DB01030
small molecule | CAS: 123948-87-8

An antineoplastic agent used to treat ovarian cancer. It works by inhibiting DNA topoisomerases, type I.

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +21
Target Protein:
DNA topoisomerase 1DNADNA topoisomerase I, mitochondrial
Waktu Paruh2-3 hours
Vol. Distribusi-
Klirens-
Genetik -
Topramezone DB14826
small molecule | CAS: 210631-68-8

Topramezone is under investigation in clinical trial NCT00559520 (The Role of Preoperative Oral Immunonutrition in Major Vascular Surgery).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Topsalysin DB05160
small molecule | CAS: 917121-25-6

Topsalysin is being developed for the treatment of localized prostate cancer and also benign prostatic hyperplasia. Topsalysin is delivered locally to the prostate under ultrasound guidance.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsMembrane Proteins +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Toralizumab DB16384
biotech | CAS: 252662-47-8

Toralizumab is under investigation in clinical trial NCT03605927 (CD40-L Blockade for Prevention of Acute Graft-versus-host Disease).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Torapsel DB13057
biotech | CAS: 204658-47-9

Torapsel has been used in trials studying the prevention of Ischemia Reperfusion Injury.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Torasemide Approved DB00214
small molecule | CAS: 56211-40-6

Torasemide is a high-ceiling loop diuretic.[A174463] Structurally, it is a pyridine-sulfonylurea used as an antihypertensive agent.[A319] Torasemide was first approved for clinical use by the FDA in 1993.[L5257]

Kategori:
Antihypertensive AgentsAntihypertensive Agents Indicated for HypertensionCardiovascular Agents +21
Target Protein:
Solute carrier family 12 member 2Solute carrier family 12 member 1
Waktu ParuhThe average half-li…
Vol. DistribusiThe volume of distr…
KlirensThe clearance rate …
Genetik -
Torcetrapib DB06281
small molecule | CAS: 262352-17-0

Torcetrapib (CP-529414, Pfizer) was developed to treat hypercholesterolemia but its development was halted in 2006 when phase III studies showed excessive mortality in the treatment group receiving a combination of atorvastatin and the study drug.

Kategori:
Anticholesteremic AgentsBlood PressureCholesterol Ester Transfer Proteins +3
Target Protein:
Cholesteryl ester transfer protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Toreforant DB12522
small molecule | CAS: 952494-46-1

Toreforant has been used in trials studying the treatment of Asthma, Psoriasis, Hepatic Impairment, and Rheumatoid Arthritis.

Kategori:
Heterocyclic Compounds, Fused-RingHistamine AgentsHistamine Antagonists +1
Target Protein:
Histamine H4 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Toremifene Approved DB00539
small molecule | CAS: 89778-26-7

Toremifene is a selective estrogen receptor modulator (SERM) and a nonsteroidal antiestrogen used to treat estrogen receptor positive breast cancer.[A256923] Like [tamoxifen], toremifene is part of the first-generation triphenylethylene derivative chemical cl…

Kategori:
Anti-EstrogensAntineoplastic AgentsAntineoplastic Agents, Hormonal +23
Target Protein:
Estrogen receptorSex hormone-binding globulin
Waktu Paruh5 days
Vol. Distribusi* 580 L
Klirens* 5 L/h
Genetik -
Toripalimab Approved DB15043
biotech | CAS: 1924598-82-2

The proliferation of some cancers can be attributed, at least in part, to the suppression of host tumor surveillance. One mechanism by which this occurs is through the overexpression of programmed cell death ligand (PD-L1)[A261506] - the binding of PD-L1 (and…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +13
Target Protein:
Programmed cell death protein 1
Waktu ParuhThe mean terminal e…
Vol. DistribusiAt steady-state, th…
KlirensThe mean clearance …
Genetik -
TORL-2-307 DB18376
biotech

TORL-2307 is a humanized immunoglobulin G1 (IgG1) monoclonal antibody (mAb) directed against claudin 18.2 (CLDN18.2) being investigated for the treatment of gastric and pancreatic cancer.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Torudokimab DB16671
biotech | CAS: 2241728-76-5

Torudokimab is under investigation in clinical trial NCT03831191 (A Study of LY3375880 in Adults With Moderate-to-severe Atopic Dermatitis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tosatoxumab DB16557
biotech | CAS: 1374419-41-6

Tosatoxumab is a fully-human monoclonal antibody (IgG1?) targeting the Staphylococcus aureus alpha-toxin or the S. aureus alpha-hemolysin[A191829, L31568, L31573] and thereby preserving human immune cells by protecting against destruction of host cells mediat…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tosedostat DB11781
small molecule | CAS: 238750-77-1

Tosedostat has been used in trials studying the treatment and supportive care of AML, Leukemia, Pancreas Cancer, Multiple Myeloma, and Pancreatic Cancer, among others. Tosedostat is an inhibitor of the M1 family of aminopeptidases, in particular PuSA, and …

Kategori:
AminesAmino AcidsAmino Acids, Peptides, and Proteins +3
Target Protein:
Puromycin-sensitive aminopeptidaseLeukotriene A-4 hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tositumomab Approved DB00081
biotech | CAS: 208921-02-2

Murine IgG2a lambda monoclonal antibody against CD20 antigen (2 heavy chains of 451 residues, 2 lambda chains of 220 residues). It is produced in an antibiotic-free culture of mammalian cells. It can be covalently linked to Iodine 131 (a radioactive isotope o…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntigens, CD20 +16
Target Protein:
B-lymphocyte antigen CD20Low affinity immunoglobulin gamma Fc region receptor II-b
Waktu Paruh0.8 hours (mammalia…
Vol. Distribusi-
Klirens* 68.2 mg/hr [patie…
Genetik -
biotech | CAS: 192391-48-3

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntigens, CD20 +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tosufloxacin DB16850
small molecule | CAS: 100490-36-6

Deskripsi belum tersedia.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tosyl-D-Proline DB02752
small molecule

Deskripsi belum tersedia.

Target Protein:
Thymidylate synthaseThymidylate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tosylchloramide DB14708
small molecule | CAS: 144-86-5

Tosylchloramide, also known as chloramine-T, is a chlorinated and deprotonated sulfonamide used as a mild disinfectant. It is not stable in the water dissolved form.

Kategori:
AminesAnti-Infective AgentsAnti-Infective Agents, Local +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tovetumab DB12609
biotech | CAS: 1243266-04-7

Tovetumab has been used in trials studying the treatment of Cancer, Glioblastoma Multiforme, and Advanced Solid Malignancies.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tovinontrine DB16193
small molecule | CAS: 2062661-53-2

Tovinontrine is an orally administered, highly selective phosphodiesterase 9 (PDE9) small molecule inhibitor. Tovinontrine is under investigation in clinical trial NCT04474314 (A Study of IMR-687 in Subjects With Sickle Cell Disease).

Target Protein:
High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tovorafenib Approved DB15266
small molecule | CAS: 1096708-71-2

Tovorafenib is a selective type II RAF kinase inhibitor with anti-tumour activity.[A263597] It was granted accelerated approval by the FDA, making it the first FDA approval of a systemic therapy for the treatment of pediatric low-grade glioma, with BRAF rearr…

Kategori:
B-Raf serine-threonine kinase (BRAF) inhibitorsBCRP/ABCG2 InhibitorsCytochrome P-450 CYP1A2 Inducers +31
Target Protein:
RAF proto-oncogene serine/threonine-protein kinaseSerine/threonine-protein kinase A-RafSerine/threonine-protein kinase B-raf
Waktu ParuhTovorafenib termina…
Vol. DistribusiTovorafenib apparen…
KlirensThe apparent cleara…
Genetik -
Toyocamycin DB13916
small molecule | CAS: 606-58-6

4-Amino-5-cyano-7-(D-ribofuranosyl)-7H- pyrrolo(2,3-d)pyrimidine. Antibiotic antimetabolite isolated from Streptomyces toyocaensis cultures. It is an analog of adenosine, blocks RNA synthesis and ribosome function, and is used mainly as a tool in biochemistry.

Kategori:
Antibiotics, AntineoplasticAntimetabolitesAntineoplastic Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tozadenant DB12203
small molecule | CAS: 870070-55-6

Tozadenant has been investigated for the basic science of Cocaine Dependence.

Kategori:
Heterocyclic Compounds, Fused-RingThiazoles
Target Protein:
Adenosine receptor A2a
Waktu ParuhFollowing the oral …
Vol. Distribusi-
Klirens-
Genetik -
Tozinameran Approved DB15696
biotech | CAS: 2417899-77-3

The Pfizer-BioNTech COVID-19 vaccine (also known as BNT162b2, Tozinameran, and Comirnaty), is one of four advanced mRNA-based vaccines developed through "Project Lightspeed," a joint program between Pfizer and BioNTech.[L15002,L15007,L36025] Comirnaty is a nu…

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tozuleristide DB15375
biotech | CAS: 1673565-40-6

Tozuleristide is under investigation in clinical trial NCT02464332 (Safety Study of BLZ-100 in Adult Subjects With Sarcoma Undergoing Surgery).

Kategori:
Arthropod VenomsBiological FactorsComplex Mixtures +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TP-1287 DB18104
small molecule | CAS: 2044686-42-0

Deskripsi belum tersedia.

Target Protein:
Cyclin-dependent kinase 9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TP-252 DB17912
small molecule | CAS: 1841444-50-5

TP-252 consists of magnesium L-lysinate bis-eicosapentaenoate, an ionizable salt of eicosapentaenoic acid (EPA), currently being investigated to treat familial adenomatous polyposis.[A259956]

Kategori:
Dietary FatsDietary Fats, UnsaturatedEicosanoids +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TP-271 DB15040
small molecule | CAS: 1207284-17-0

TP-271 is under investigation in clinical trial NCT02724085 (A Phase 1 Study to Assess the Safety, Tolerability and PK of IV TP-271).

Kategori:
Naphthacenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TP-3654 DB18109
small molecule | CAS: 1361951-15-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsGastrointestinal HormonesHormones +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TP-508 DB05309
small molecule

TP508 is a non-proteolytic synthetic peptide representing the portion of human thrombin originally identified as the fibroblast high-affinity receptor binding domain.

Target Protein:
Fibroblast growth factor 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TPCA-1 DB17058
small molecule | CAS: 507475-17-4

TPCA-1 is a selective inhibitor of human I?B kinase 2 (IKK-2).[A253152]

Kategori:
Enzyme InhibitorsProtein Kinase InhibitorsSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TPI-287 DB17168
small molecule | CAS: 849213-15-6

Deskripsi belum tersedia.

Kategori:
CyclodecanesCycloparaffinsDiterpenes +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TPI-ASM8 DB05572
small molecule

TPI-ASM8 was under investigation in clinical trials NCT00822861, NCT01158898, NCT00402948, and NCT00550797, all for the treatment of Asthma.

Kategori:
Antisense OligonucleotidesNucleic Acids, Nucleotides, and NucleosidesNucleotides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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