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17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
Referensi
17430 (100.0%)

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Hasil Pencarian (17430)

Halaman 298 / 349
small molecule | CAS: 63795-61-9

Deskripsi belum tersedia.

Kategori:
Diagnostic RadiopharmaceuticalsSelenium CompoundsVarious Diagnostic Radiopharmaceuticals
Waktu Paruh-
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Genetik -
Selenium Sulfide Approved DB00971
small molecule | CAS: 7488-56-4

Selenium Sulfide is an antifungal agent as well as a cytostatic agent, slowing the growth of hyperproliferative cells in seborrhea. Selenium Sulfide is the active ingredient often used in shampoos for the treatment of dandruff, seborrheic dermatitis and tinea…

Kategori:
Antifungals for Dermatological UseAntifungals for Topical UseDermatologicals +1
Waktu Paruh-
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Genetik -
Selenocysteine DB02345
small molecule | CAS: 10236-58-5

A naturally occurring amino acid in both eukaryotic and prokaryotic organisms. It is found in tRNAs and in the catalytic site of some enzymes. The genes for glutathione peroxidase and formate dehydrogenase contain the TGA codon, which codes for this amino aci…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAmino Acids, Sulfur +5
Target Protein:
Cathelicidin antimicrobial peptideNucleoside diphosphate kinase AFormate dehydrogenase H +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Selenoinosine DB02753
small molecule | CAS: 40093-99-0

Deskripsi belum tersedia.

Kategori:
Selenium Compounds
Target Protein:
Nucleoside 2-deoxyribosyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Selenomethionine Approved DB11142
small molecule | CAS: 3211-76-5

Selenomethionine is a naturally occuring amino acid in some plant materials such as cereal grains, soybeans and enriched yeast but it cannot be synthesized from animals or humans. It can be produced from post-structural modifications. *In vivo*, selenomethion…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsOrganoselenium Compounds +1
Waktu Paruh-
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Genetik -
Selenomethionine Se-75 Approved DB09400
small molecule | CAS: 1187-56-0

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsOrganoselenium Compounds +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Selenium Compounds
Waktu Paruh-
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Selepressin DB12495
small molecule | CAS: 876296-47-8

Selepressin has been used in trials studying the treatment of Septic Shock.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +11
Target Protein:
Vasopressin V1a receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seletalisib DB12706
small molecule | CAS: 1362850-20-1

Seletalisib has been used in trials studying the treatment and basic science of Primary Sjogren's Syndrome.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seletracetam DB05885
small molecule | CAS: 357336-74-4

Seletracetam is a pyrrolidone derivative and with a structural similarity to newer generation antiepileptic drug levetiracetam. It binds to the same target as levetiracetam but with higher affinity and has shown potent seizure suppression in models of acquire…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +6
Target Protein:
Synaptic vesicle glycoprotein 2AVoltage-dependent N-type calcium channel subunit alpha-1BGlycine receptor (alpha-1/beta)
Waktu ParuhApproximately 8 hou…
Vol. DistribusiThe volume of distr…
KlirensThe total apparent …
Genetik -
Selexipag Approved DB11362
small molecule | CAS: 475086-01-2

Selexipag was approved by the United States FDA on December 22, 2015 for the treatment of pulmonary arterial hypertension (PAH) to delay disease progression and reduce risk of hospitalization. PAH is a relatively rare disease with usually a poor prognosis req…

Kategori:
AcetatesAcids, AcyclicAmides +19
Target Protein:
Prostacyclin receptor
Waktu ParuhSelexipag's termina…
Vol. Distribusi-
KlirensOn average, 35 L/ho…
Genetik -
Selgantolimod DB16324
small molecule | CAS: 2004677-13-6

Selgantolimod is under investigation in clinical trial NCT03491553 (Safety, Tolerability and Antiviral Activity of Selgantolimod in Virally-suppressed Adults With Chronic Hepatitis B).

Kategori:
AlcoholsFatty AlcoholsLipids
Target Protein:
Toll-like receptor 8
Waktu Paruh-
Vol. Distribusi-
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Seliciclib DB06195
small molecule | CAS: 186692-46-6

R-roscovitine (Seliciclib or CYC202) is a cyclin-dependent kinase (CDK) inhibitor that preferentially inhibits multiple enzyme targets including CDK2, CDK7 and CDK9, which alter the growth phase of treated cells. Developed by Cyclacel, seliciclib is being res…

Kategori:
Anti-Infective AgentsAntineoplastic AgentsEnzyme Inhibitors +3
Target Protein:
Cyclin-dependent kinase 2Cyclin-dependent kinase 7Cyclin-dependent kinase 1 +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Selicrelumab DB14958
biotech | CAS: 1622140-49-1

Selicrelumab is under investigation in clinical trial NCT01008527 (Phase I Oncovir Poly IC:LC and NY-ESO-1/gp100).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seliforant DB15220
small molecule | CAS: 1164115-89-2

Seliforant is under investigation in clinical trial NCT01260753 (Proof of Activity Study of UR-63325 in Allergic Rhinitis Induced by Nasal Challenge).

Kategori:
Azetines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Selinexor Approved DB11942
small molecule | CAS: 1393477-72-9

Selinexor is a first-in-class selective inhibitor of nuclear transport (SINE) compound. Selinexor, in combination with [bortezomib] and [dexamethasone], is currently approved for the treatment of multiple myeloma, a type of cancer formed from antibody-produci…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP3A Substrates +4
Target Protein:
Exportin-1
Waktu ParuhSelinexor has a mea…
Vol. DistribusiThe mean apparent v…
KlirensSelinexor has a mea…
Genetik -
Selisistat DB13978
small molecule | CAS: 49843-98-3

Selective inhibitor of SIRT1 that does not inhibit histone deacetylase (HDAC) or other sirtuin deacetylase family members (IC50 values are 98, 19600, 48700, > 100000 and > 100000 nM for SIRT1, SIRT2, SIRT3, HDAC and NADase respectively). Enhances p53 acetylat…

Kategori:
Heterocyclic Compounds, Fused-RingIndolesSirtuin 1, antagonists & inhibitors
Target Protein:
NAD-dependent protein deacetylase sirtuin-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Selitrectinib DB14896
small molecule | CAS: 2097002-61-2

Selitrectinib is under investigation in clinical trial NCT03215511 (Phase 1/2 Study of LOXO-195 in Patients With Previously Treated NTRK Fusion Cancers).

Kategori:
Enzyme Inhibitors
Target Protein:
High affinity nerve growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Selodenoson DB16325
small molecule | CAS: 110299-05-3

Selodenoson is under investigation in clinical trial NCT00040001 (Safety and Efficacy Study of an A1-adenosine Receptor Agonist to Slow Heart Rate in Atrial Fibrillation).

Kategori:
CycloparaffinsHeterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
Adenosine receptor A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Selonsertib DB14916
small molecule | CAS: 1448428-04-3

Selonsertib is under investigation in clinical trial NCT03053050 (Safety and Efficacy of Selonsertib in Adults With Nonalcoholic Steatohepatitis (NASH) and Bridging (F3) Fibrosis).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +3
Target Protein:
Mitogen-activated protein kinase kinase kinase 5
Waktu Paruh-
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Genetik -
Selpercatinib Approved DB15685
small molecule | CAS: 2152628-33-4

Selpercatinib is a kinase inhibitor with enhanced specificity for RET tyrosine kinase receptors (RTKs) over other RTK classes.[A202055, A202052, L13604] Enhanced RET (Rearranged during transfection) oncogene expression is a hallmark of many cancers. Although …

Kategori:
Agents that produce hypertensionAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +19
Target Protein:
Proto-oncogene tyrosine-protein kinase receptor RetVascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 3 +3
Waktu ParuhSelpercatinib has a…
Vol. DistribusiSelpercatinib has a…
KlirensSelpercatinib has a…
Genetik -
Seltorexant DB14961
small molecule | CAS: 1452539-75-1

Seltorexant is under investigation in clinical trial NCT03494907 (A Study to Evaluate the Effects of Single-dose Seltorexant on Electrocardiogram Intervals in Healthy Adult Participants).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Selumetinib Approved DB11689
small molecule | CAS: 606143-52-6

Activation of the Raf-MEK-ERK signalling pathway is known to be implemented in several types of malignancies; thus, mitogen-activated protein kinase kinase (MEK) inhibitors such as selumetinib are important tools that can target the problematic overactivity o…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +18
Target Protein:
Dual specificity mitogen-activated protein kinase kinase 1Dual specificity mitogen-activated protein kinase kinase 2
Waktu ParuhSelumetinib is char…
Vol. DistribusiThe mean apparent v…
KlirensThe clearance of se…
Genetik -
Selurampanel DB12367
small molecule | CAS: 912574-69-7

Selurampanel has been investigated in Adrenocortical Adenoma and Sarcoma, Endometrial Stromal.

Kategori:
Heterocyclic Compounds, Fused-RingQuinazolines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Semagacestat DB12463
small molecule | CAS: 425386-60-3

Semagacestat has been used in trials studying the treatment of Alzheimer Disease.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAmyloid Precursor Protein Secretases, antagonists & inhibitors +2
Target Protein:
Gamma-secretase subunit APH-1BNicastrinGamma-secretase subunit APH-1A +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Semaglutide Approved DB13928
small molecule | CAS: 910463-68-2

Semaglutide is a glucagon-like peptide 1 (GLP-1) analog used to manage type 2 diabetes along with lifestyle changes, such as dietary restrictions and increased physical activity.[A31421,L8681] Other members of this drug class include [Exenatide] and [Liraglut…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +11
Target Protein:
Glucagon-like peptide 1 receptor
Waktu ParuhOne of the major pr…
Vol. DistribusiThe volume of distr…
KlirensThe clearance rate …
Genetik -
Semapimod DB12094
small molecule | CAS: 352513-83-8

Semapimod has been used in trials studying the treatment of Crohn Disease.

Kategori:
AmidesAmidinesAmines +9
Target Protein:
RAF proto-oncogene serine/threonine-protein kinase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Semaxanib DB06436
small molecule | CAS: 194413-58-6

Deskripsi belum tersedia.

Kategori:
Angiogenesis InhibitorsAngiogenesis Modulating AgentsAntineoplastic Agents +5
Target Protein:
Aryl hydrocarbon receptorPlatelet-derived growth factor receptor betaVascular endothelial growth factor receptor 1 +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Semduramicin DB11545
small molecule | CAS: 113378-31-7

Deskripsi belum tersedia.

Kategori:
EthersEthers, CyclicFurans +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Semorinemab DB15234
biotech | CAS: 2159141-27-0

Semorinemab is under investigation in clinical trial NCT03289143 (A Study to Evaluate the Efficacy and Safety of RO7105705 in Patients With Prodromal to Mild Alzheimer's Disease).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Semuloparin DB06294
small molecule

Deskripsi belum tersedia.

Kategori:
AnticoagulantsCarbohydratesCardiovascular Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Semustine DB13647
small molecule | CAS: 13909-09-6

Deskripsi belum tersedia.

Kategori:
Alkylating DrugsAmidesAntineoplastic Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Semzuvolimab DB18920
biotech | CAS: 2409099-32-5

Semzuvolimab is under investigation in clinical trial NCT03149211 (To Investigate the Efficacy and Safety of UB-421 Monotherapy in HIV-1 Infected Adults).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAnti-Retroviral Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Senaparib DB17163
small molecule | CAS: 1401682-78-7

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Senicapoc DB06280
small molecule | CAS: 289656-45-7

Senicapoc (ICA-17043) is a novel Gardos channel blocker.[A259068] It is being investigated for the treatment of sickle cell disease.

Kategori:
AcetatesAcids, AcyclicAmides +1
Target Protein:
Intermediate conductance calcium-activated potassium channel protein 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Senlizumab DB17894
biotech | CAS: 336128-48-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAnalgesics, Non-Narcotic +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Senna leaf Approved DB15889
biotech

Deskripsi belum tersedia.

Kategori:
AnthracenesAnthraquinonesBiological Products +6
Waktu Paruh-
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Klirens-
Genetik -
Sennosides DB11365
small molecule | CAS: 517-43-1

Sennosides (also known as senna glycoside or senna) is a medication used to treat constipation[FDA Label][L771] and empty the large intestine before surgery. The medication is taken by mouth or via the rectum[FDA Label]. It typically begins working in minutes…

Kategori:
Alimentary Tract and MetabolismAnthracenesAnthraquinones +13
Target Protein:
Aquaporin-3Reverse transcriptase/RNaseH
Waktu ParuhThe half life of ra…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ra…
Genetik -
Senrebotase DB12626
biotech | CAS: 1290102-81-6

Senrebotase has been used in trials studying the treatment of Neuralgia, Postherpetic and Urinary Bladder, Overactive.

Waktu Paruh-
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Genetik -
Seocalcitol DB04258
small molecule | CAS: 134404-52-7

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsCholestanesCholestenes +11
Target Protein:
Vitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SEP-363856 DB15665
small molecule | CAS: 1310426-33-5

SEP-363856 is a novel psychotropic drug being investigated for the treatment of schizophrenia. Unlike other drugs used for this condition, SEP-363856 does not bind to the dopamine D2 receptors, but exerts actions on the trace amine–associated receptor 1 (TAA…

Target Protein:
5-hydroxytryptamine receptor 1ATrace amine-associated receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sepantronium DB17062
small molecule | CAS: 753440-91-4

Sepantronium is a compound that suppresses survivin expression in a dose and time-dependent manner, and causes broad-range apoptosis.[A253167]

Kategori:
NaphthalenesQuinones
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Sepetaprost DB12043
small molecule | CAS: 1262873-06-2

Sepetaprost has been used in trials studying the treatment of Open Angle-glaucoma, Ocular Hypertension, and Mild Open Angle-glaucoma (OAG).

Kategori:
EthersEthers, Cyclic
Waktu Paruh-
Vol. Distribusi-
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Genetik -
SEphB4-HSA DB14797
biotech

SEphB4-HSA is under investigation in clinical trial NCT02495896 (Recombinant EphB4-HSA Fusion Protein With Standard Chemotherapy Regimens in Treating Patients With Advanced or Metastatic Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Deskripsi belum tersedia.

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Genetik -
Sepiapterin DB16326
small molecule | CAS: 17094-01-8

Sepiapterin is under investigation in clinical trial NCT03519711 (A Study of CNSA-001 in Primary Tetrahydrobiopterin (BH4) Deficient Participants With Hyperphenylalaninemia).

Kategori:
Biological FactorsHeterocyclic Compounds, Fused-RingPigments, Biological +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sepofarsen DB16327
biotech | CAS: 2227173-68-2

Sepofarsen is under investigation in clinical trial NCT03913143 (A Study to Evaluate Efficacy, Safety, Tolerability and Exposure After a Repeat-dose of Sepofarsen (QR-110) in LCA10 (ILLUMINATE)).

Kategori:
OphthalmologicalsSensory Organs
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sepranolone DB12972
small molecule | CAS: 516-55-2

Sepranolone has been investigated for the treatment of Premenstrual Dysphoric Disorder.

Kategori:
AnestheticsCentral Nervous System AgentsCentral Nervous System Depressants +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seproxetine DB06731
small molecule | CAS: 126924-38-7

Seproxetine is also known as (S)-norfluoxetine. It is a selective serotonin reuptake inhibitor (SSRI). It is an active metabolite of fluoxetine. Seproxetine was being investigated by Eli Lilly as an antidepressant but development was never completed and the d…

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsCytochrome P-450 CYP2C19 Inhibitors +14
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporterSodium-dependent dopamine transporter
Waktu Paruh4-16 days
Vol. Distribusi-
Klirens-
Genetik -
Sequifenadine DB13566
small molecule | CAS: 57734-69-7

Deskripsi belum tersedia.

Kategori:
Antihistamines for Systemic Use
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Menampilkan 14851–14900 dari 17430
Sebelumnya Halaman 298 / 349 Berikutnya