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2279

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Halaman 29 / 46
Mubodina DB17616
biotech

Mubodina is an investigational drug developed by Adienne Pharma & Biotech. It is a recombinant human minibody directed against complement component C5. It was investigated in various conditions including primary membranoproliferative glomerulonephritis and ty…

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Genetik -
biotech

Mucor circinelloides f. circinelloides allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Muparfostat DB05808
small molecule | CAS: 1020105-89-8

Muparfostat (PI-88) is a mixture of highly sulfated, monophosphorylated mannose oligosaccharides, derived from the extracellular phosphomannan of the yeast Pichia (Hansenula) holstii, with potential antiangiogenic activity.

Kategori:
CarbohydratesPolysaccharides
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Mupirocin Approved DB00410
small molecule | CAS: 12650-69-0

Mupirocin, formerly termed pseudomonic acid A,[A178531] is a novel antibacterial agent with a unique chemical structure and mode of action apart from other antibiotic agents. Produced by fermentation using the organism _Pseudomonas fluorescens_, mupirocin is …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibiotics for Topical Use +12
Target Protein:
Isoleucine--tRNA ligase
Waktu ParuhIn healthy male vol…
Vol. DistribusiNo information avai…
KlirensNo information avai…
Genetik -
Muplestim DB12431
biotech | CAS: 148641-02-5

Muplestim is under investigation in clinical trial NCT00002258 (A Phase I, Open Label Trial to Evaluate the Safety, Tolerance and Biological Effects of SDZ ILE-964 (Recombinant Human Interleukin-3, RhIL-3) in HIV Infected Patients With Cytopenia).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCarbohydrates +10
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Muromonab Approved DB00075
biotech | CAS: 140608-64-6

Murine monoclonal antibody specific to CD3 T-cell lymphocyte antigens. More specifically it is a purified murine (mouse) monoclonal antibody, directed against the CD3 (T3) receptor on the surface of human T-cells (T-lymphocytes) cultured using the murine asci…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
T-cell surface glycoprotein CD3 delta chainT-cell surface glycoprotein CD3 epsilon chainT-cell surface glycoprotein CD3 gamma chain +2
Waktu Paruh0.8 hours (mammalia…
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Genetik -
biotech

MVA-BN-brachyury-TRICOM vaccine is an investigational cancer vaccine. It is composed of recombinant vaccinia viral vector, modified vaccinia Ankara-Bavarian Nordic (MVA-BN), encoding the human transcription factor and tumour-associated antigen (TAA) brachyury…

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MVR-T3011 DB17378
biotech

MVR-T3011 is a genetically modified oncolytic Herpes Simplex Virus (HSV-1) with 2 exogenous genes encoding the active heterodimer human interleukin 12 (IL-12) and the Fab fragment of an anti-human PD-1 antibody.

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MW33 DB16358
biotech

MW33 is a recombinant fully human antibody to SARS-CoV-2.[L27411] This antibody injection is currently being investigated against COVID-19 in the clinical trial NCT04533048 (A Clinical Study to Evaluate MW33 Injection).

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MX6 DB05789
small molecule

MX6 is adamantyl group derivatives containing retinoid-related compounds induce apoptosis of cancer cells and therefore may be used for the treatment of cancer, including advanced cancer. More specifically, it has been shown that such adamantyl compounds, e.g…

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Genetik -
biotech

The Mycobacterium w (M.w) vaccine is a heat-killed suspension derived from a non-pathogenic mycobacterium: mycobacterium indicus pranii. As an immunotherapy, M.w is used against leprosy; the compound also shares antigens with M. tuberculosis. Its use has show…

Kategori:
Biological ProductsComplex MixturesMycobacterium +1
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small molecule | CAS: 30315-93-6

Asymmetric dimethylarginine (ADMA) is a naturally occurring chemical found in blood plasma. It is a metabolic by-product of continual protein modification processes in the cytoplasm of all human cells which is closely related to L-arginine, a conditionally-es…

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +3
Target Protein:
Nitric oxide synthase, inducibleNitric oxide synthase 3
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Urokinase-type plasminogen activator
Waktu Paruh-
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Genetik -
small molecule | CAS: 21646-00-4

An N-acyl derivative of neuraminic acid. N-acetylneuraminic acid occurs in many polysaccharides, glycoproteins, and glycolipids in animals and bacteria. (From Dorland, 28th ed, p1518)

Target Protein:
P-selectinE-selectinLiver carboxylesterase 1 +15
Waktu Paruh-
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Genetik -
small molecule | CAS: 19342-33-7

An N-acyl derivative of neuraminic acid. N-acetylneuraminic acid occurs in many polysaccharides, glycoproteins, and glycolipids in animals and bacteria. (From Dorland, 28th ed, p1518)

Target Protein:
Tetanus toxinSialidaseEndo-N-acetylneuraminidase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 3615-17-6

N-acetylmannosamine is under investigation for the other of GNE Myopathy.

Kategori:
Amino SugarsCarbohydrates
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Capsule biosynthesis protein
Waktu Paruh-
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small molecule | CAS: 3258-02-4

N4-Hydroxyctidine, or EIDD-1931, is a ribonucleoside analog which induces mutations in RNA virions.[A193008,A193011] N4-hydroxycytidine was first described in the literature in 1980 as a potent mutagen of bacteria and phage.[A193023] It has shown antiviral ac…

Kategori:
CarbohydratesCytosine NucleotidesExperimental Unapproved Treatments for COVID-19 +6
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Nabilone Approved DB00486
small molecule | CAS: 51022-71-0

Nabilone (marketed as Cesamet) is a synthetic form of delta-9-tetrahydrocannabinol (??-THC), the primary psychoactive component of cannabis (marijuana). Although structurally distinct from THC, nabilone mimics THC's structure and pharmacological activity thro…

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAntiemetics +30
Target Protein:
Cannabinoid receptor 2Cannabinoid receptor 1
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe apparent volume…
Klirens-
Genetik -
Nabiximols DB14011
small molecule | CAS: 56575-23-6

Nabiximols (tradename Sativex®) is a whole plant extract from the Cannabis species _Cannabis sativa L._ that has been purified into the active components CBD (cannabidiol) and THC (delta-9-tetrahydrocannabinol). For trademark purposes, purified CBD is branded…

Kategori:
Agents producing tachycardiaAnalgesicsBCRP/ABCG2 Inhibitors +24
Target Protein:
Cannabinoid receptor 1Cannabinoid receptor 2G-protein coupled receptor 12 +41
Waktu ParuhElimination from pl…
Vol. DistribusiCannabinoids are di…
Klirens-
Genetik -
Nadofaragene firadenovec Approved DB17381
biotech | CAS: 1823059-12-6

Nadofaragene firadenovec (nadofaragene firadenovec-vncg) is a recombinant non-replicating adenovirus serotype 5 vector containing a transgene encoding human interferon alfa-2b (IFN?2b).[L44381] It was approved by the FDA on December 2022 for the treatment of …

Kategori:
Adeno-associated Viral Vector TherapiesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +4
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Nalmefene Approved DB06230
small molecule | CAS: 55096-26-9

Nalmefene, a 6-methylene analogue of [naltrexone], is an opioid receptor antagonist.[L40684] It acts as an antagonist at the mu (?)-opioid and delta (?)-opioid receptors and a partial agonist at the kappa (?)-opioid receptor.[L1024] In Europe, nalmefene or…

Kategori:
AlkaloidsAntidotesAntipruritics +18
Target Protein:
Kappa-type opioid receptorDelta-type opioid receptorMu-type opioid receptor
Waktu ParuhThe terminal half-l…
Vol. DistribusiFollowing a 1 mg pa…
KlirensThe oral clearance …
Genetik -
biotech

Deskripsi belum tersedia.

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Nandrolone decanoate Approved DB08804
small molecule | CAS: 360-70-3

Nandrolone decanoate, also known as nandrolone caprinate, is an alkylated anabolic steroid indicated in the management of anemia of renal insufficiency and as an adjunct therapy in the treatment of senile and postmenopausal osteoporosis.[A233789,A233849,L3256…

Kategori:
Anabolic AgentsAndrogensBone Density Conservation Agents +16
Target Protein:
Androgen receptorProtein c-Fos5-hydroxytryptamine 2 receptor +3
Waktu ParuhNandrolone decanoat…
Vol. Distribusi-
Klirens50 mg, 100 mg, and …
Genetik -
biotech

Nanrilkefusp alfa is a human fusion protein consisting of the cytokine interleukin (IL)-15 and the high-affinity binding sushi+ domain of IL-15 receptor alpha (IL-15Ra).

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Naphazoline Approved DB06711
small molecule | CAS: 835-31-4

Naphazoline is a rapid acting imidazoline sympathomimetic vasoconstrictor of ocular or nasal artierioles[L5804,L5807]. It acts to decrease congestion and is found in many over the counter (OTC) eye drops and nasal preparations[L5804,L5807]. Naphazoline was…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +17
Target Protein:
D(2) dopamine receptorAlpha-2A adrenergic receptorAlpha-1A adrenergic receptor
Waktu ParuhHalf life has not b…
Vol. DistribusiDistribution data f…
KlirensClearance data for …
Genetik -
Naproxen Approved DB00788
small molecule | CAS: 22204-53-1

Naproxen is classified as a nonsteroidal anti-inflammatory dug (NSAID) and was initially approved for prescription use in 1976 and then for over-the-counter (OTC) use in 1994.[A178975] It can effectively manage acute pain as well as pain related to rheumatic …

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +41
Target Protein:
Pancreatic triacylglycerol lipaseProstaglandin G/H synthase 1Prostaglandin G/H synthase 2 +1
Waktu ParuhThe elimination hal…
Vol. DistribusiNaproxen has a volu…
KlirensNaproxen is cleared…
Genetik -
Narsoplimab DB16418
biotech | CAS: 2108782-45-0

Thrombotic microangiopathies (TMA), including thrombotic thrombocytopenic purpura and atypical hemolytic uremic syndrome, are associated with injury and dysregulation of microvascular endothelium and platelets.[A241030] Evidence increasingly points to a role …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Mannan-binding lectin serine protease 2
Waktu Paruh-
Vol. Distribusi-
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Natalizumab Approved DB00108
biotech | CAS: 189261-10-7

Natalizumab is a recombinant humanized IgG4? monoclonal antibody that binds to ?4-integrin.[L48041] While natalizumab was originally approved by the FDA to treat multiple sclerosis in 2004, it was withdrawn from the market following multiple reports of fatal …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +14
Target Protein:
Integrin alpha-4Low affinity immunoglobulin gamma Fc region receptor III-BHigh affinity immunoglobulin gamma Fc receptor I +1
Waktu ParuhFollowing the repea…
Vol. DistribusiFollowing the repea…
KlirensFollowing the repea…
Genetik -
biotech

Natural Killer (NK) cells originate and differentiate from hematopoietic stem cells through various signalling pathways involving cytokines and interleukins. These cells arise from CD34+ lymphoid progenitors and comprise 10-15% of all lymphocytes in human per…

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Naxitamab Approved DB15965
biotech | CAS: 1879925-92-4

Naxitamab (humanized 3F8, hu3F8) is an IgG1 monoclonal antibody directed against the oncofetal differentiation antigen GD2 disialoganglioside.[L24454,A224604] Normally expressed during fetal development and in mature neurons, pain fibers, and skin cells, GD2 …

Kategori:
Agents that produce hypertensionAmino Acids, Peptides, and ProteinsAntibodies +18
Target Protein:
GD2 disialoganglioside
Waktu ParuhThe mean terminal h…
Vol. Distribusi-
KlirensThe clearance of na…
Genetik -
NBL-015 DB18183
biotech

Deskripsi belum tersedia.

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NDX-3315 DB18671
small molecule

NDX-3315 is an investigational radiopharmaceutical agent for the diagnosis, treatment monitoring, and management of eosinophilic esophagitis. It is a technetium-99m radiolabeled [heparin].

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Nebivolol Approved DB04861
small molecule | CAS: 118457-14-0

Nebivolol is a racemic mixture of 2 enantiomers where one is a beta adrenergic antagonist and the other acts as a cardiac stimulant without beta adrenergic activity.[A182579] Treatment with nebivolol leads to a greater decrease in systolic and diastolic blood…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic Antagonists +29
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorBeta-3 adrenergic receptor
Waktu Paruhd-nebivolol has a h…
Vol. DistribusiFor a 20mg dose, d-…
KlirensFor a 20mg dose, th…
Genetik -
Necitumumab Approved DB09559
biotech | CAS: 906805-06-9

Necitumumab is an intravenously administered recombinant monoclonal IgG1 antibody used in the treatment of non-small cell lung cancer (NSCLC) as an EGFR antagonist. It functions by binding to epidermal growth factor receptor (EGFR) and prevents binding of its…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
Epidermal growth factor receptor
Waktu ParuhElimination half li…
Vol. DistribusiSteady state volume…
Klirens14.1 mL/h
Genetik -
Neihulizumab DB16698
biotech

Neihulizumab is a novel immune checkpoint agonistic antibody that binds to human CD162 (PSGL-1), thereby preferentially inducing apoptosis in late stage activated T cells.[L34450]

Target Protein:
P-selectin glycoprotein ligand 1
Waktu Paruh-
Vol. Distribusi-
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Nelarabine Approved DB01280
small molecule | CAS: 121032-29-9

Nelarabine is an antineoplastic agent that is typically used to treat acute T-cell lymphoblastic leukemia, particularly T-cell acute lymphoblastic leukemia (T-ALL) and T-cell lymphoblastic lymphoma (T-LBL), in both adult and pediatric patients whose disease h…

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +8
Target Protein:
DNADNA polymerase alpha catalytic subunitDNA ligase 1 +2
Waktu ParuhNelarabine and ara-…
Vol. DistribusiNelarabine and ara-…
KlirensRenal clearance ave…
Genetik -
Nelipepimut-S DB06226
biotech | CAS: 160212-35-1

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Surface +25
Target Protein:
Receptor tyrosine-protein kinase erbB-2HLA class I histocompatibility antigen, A-3 alpha chain
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Nelistotug DB19334
biotech | CAS: 2645437-82-5

Nelistotug is under investigation in clinical trial NCT06062420 (A Platform Study of Novel Immunotherapy Combinations as First-line Treatment in Participants With PD-L1 Positive Recurrent/metastatic Squamous Cell Carcinoma of the Head and Neck- GALAXIES H&N-2…

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Nelonicline DB19040
small molecule | CAS: 1026134-63-3

Nelonicline is under investigation in clinical trial NCT01678755 (A Phase 2 Study to Evaluate ABT-126 for the Treatment of Cognitive Deficits in Schizophrenia).

Kategori:
Sulfur CompoundsThiazoles
Waktu Paruh-
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Nemolizumab Approved DB15252
biotech | CAS: 1476039-58-3

Nemolizumab is a humanized monoclonal modified immunoglobulin 2 (IgG2) antibody directed against interleukin-31 receptor alpha (IL-31RA),[L51159] which is an endogenous cytokine implicated in the pathophysiology of various skin inflammatory disorders.[A264254…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAmino Acids, Peptides, and ProteinsAntibodies +10
Target Protein:
Interleukin-31 receptor subunit alpha
Waktu ParuhThe estimated termi…
Vol. DistribusiThe estimated volum…
KlirensThe estimated syste…
Genetik -
biotech | CAS: 2315268-27-8

Deskripsi belum tersedia.

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Nepidermin DB14145
biotech | CAS: 62253-63-8

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsEGF Family of Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Neratinib Approved DB11828
small molecule | CAS: 698387-09-6

Neratinib was approved in July 2017 for use as an extended adjuvant therapy in Human Epidermal Growth Factor Receptor 2 (HER2) positive breast cancer. Approval was granted to Puma Biotechnology Inc. for the tradename Nerlynx. Neratinib is currently under inve…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP3A Substrates +11
Target Protein:
Vascular endothelial growth factor receptor 2Receptor tyrosine-protein kinase erbB-2Epidermal growth factor receptor
Waktu ParuhThe mean half life …
Vol. DistribusiThe apparent volume…
KlirensThe total clearance…
Genetik -
Nesiritide Approved DB04899
biotech | CAS: 124584-08-3

Nesiritide is a medication used to treat acutely decompensated congestive heart failure with dyspnea at rest or with minimal exertion (such as talk, eating or bathing). Nesiritide is a 32 amino acid recombinant human B-type natriuretic peptide.

Kategori:
Amino Acids, Peptides, and ProteinsCardiac TherapyCardiovascular Agents +11
Target Protein:
Atrial natriuretic peptide receptor 1Atrial natriuretic peptide receptor 2Atrial natriuretic peptide receptor 3
Waktu ParuhApproximately 18 mi…
Vol. Distribusi* 0.19 L/kg
Klirens* 9.2 mL/min/k [pat…
Genetik -
Netakimab DB18870
biotech | CAS: 1796570-08-5

Netakimab is under investigation in clinical trial NCT03447704 (International Multicenter Comparative Randomized Placebo-controlled Clinical Study of Efficacy and Safety of BCD-085 in Patients With Ankylosing Spondylitis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Netarsudil Approved DB13931
small molecule | CAS: 1254032-66-0

A Rho kinase inhibitor with norepinephrine transport inhibitory activity that reduces production of aqueous As of December 18, 2017 the FDA approved Aerie Pharmaceutical's Rhopressa (netarsudil ophthalmic solution) 0.02% for the indication of reducing elev…

Kategori:
Acids, CarbocyclicAlanineAmino Acids +8
Target Protein:
Rho-associated protein kinase 1Rho-associated protein kinase 2Sodium-dependent noradrenaline transporter
Waktu ParuhThe half-life of ne…
Vol. DistribusiAs netarsudil and i…
KlirensThe clearance of ne…
Genetik -
Nevirapine Approved DB00238
small molecule | CAS: 129618-40-2

A potent, non-nucleoside reverse transcriptase inhibitor (NNRTI) used in combination with nucleoside analogues for treatment of Human Immunodeficiency Virus Type 1 (HIV-1) infection and AIDS. Structurally, nevirapine belongs to the dipyridodiazepinone chemica…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +39
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Waktu Paruh45 hours
Vol. Distribusi* 1.21 ± 0.09 L/kg …
Klirens-
Genetik -
NFS-02 DB18422
biotech

NFS-02 is a recombinant adeno-associated virus serotype 2 containing human mitochondrial ND1 codon optimized gene (rAAV2-ND1).

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NGGT-002 DB17881
biotech

NGGT-002 is a recombinant adeno-associated virus serotype 8 vector encoding human phenylalanine hydroxylase (PAH).

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