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17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
Referensi
17430 (100.0%)

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Halaman 283 / 349
Ramelteon Approved DB00980
small molecule | CAS: 196597-26-9

Ramelteon is the first in a new class of sleep agents that selectively binds to the melatonin receptors in the suprachiasmatic nucleus (SCN). It is used for insomnia, particularly delayed sleep onset. Ramelteon has not been shown to produce dependence and has…

Kategori:
Central Nervous System DepressantsCytochrome P-450 CYP1A2 SubstratesCytochrome P-450 CYP2C19 Substrates +9
Target Protein:
Melatonin receptor type 1BMelatonin receptor type 1A
Waktu Paruh~1-2.6 hours
Vol. Distribusi* 73.6 L
Klirens-
Genetik -
Ramipril Approved DB00178
small molecule | CAS: 87333-19-5

Ramipril is a prodrug belonging to the angiotensin-converting enzyme (ACE) inhibitor class of medications. It is metabolized to ramiprilat in the liver and, to a lesser extent, kidneys. Ramiprilat is a potent, competitive inhibitor of ACE, the enzyme responsi…

Kategori:
ACE Inhibitors and Calcium Channel BlockersACE Inhibitors and DiureticsAgents Acting on the Renin-Angiotensin System +14
Target Protein:
Angiotensin-converting enzymeB1 bradykinin receptor
Gen Terkait:
ACE
Waktu ParuhPlasma concentratio…
Vol. Distribusi-
KlirensThe renal clearance…
Genetik 1 Varian
Ramiprilat DB14208
small molecule | CAS: 87269-97-4

The active metabolite of the prodrug [Ramipril].

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ramoplanin DB04952
biotech | CAS: 76168-82-6

Ramoplanin is a novel glycolipodepsipeptide antibiotic under development for the treatment of CDAD.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ramosetron DB09290
small molecule | CAS: 132036-88-5

Ramosetron is a _serotonin 5-HT3 receptor antagonist_ commonly employed to treat nausea and vomiting, in addition to certain diarrheal conditions. It is believed to have higher potency and longer antiemetic action than other 1st generation 5-HT3 antagonists s…

Kategori:
Antidepressive AgentsAntiemeticsAutonomic Agents +10
Target Protein:
5-hydroxytryptamine receptor 3A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ramucirumab Approved DB05578
biotech | CAS: 947687-13-0

Ramucirumab is a human monoclonal antibody (IgG1) against vascular endothelial growth factor receptor 2 (VEGFR2), a type II trans-membrane tyrosine kinase receptor expressed on endothelial cells. By binding to VEGFR2, ramucirumab prevents binding of its ligan…

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +20
Target Protein:
Vascular endothelial growth factor receptor 2
Waktu Paruh15 days
Vol. Distribusi5.5 L
Klirens0.014 L/hour
Genetik -
Ranibizumab Approved DB01270
biotech | CAS: 347396-82-1

Ranibizumab is a recombinant humanized IgG1 kappa isotype monoclonal antibody fragment directed against human vascular endothelial growth factor A (VEGF-A), which is a glycoprotein implicated in the pathophysiology of age-related macular degeneration.[A2301, …

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +19
Target Protein:
Vascular endothelial growth factor A, long form
Waktu ParuhThe estimated avera…
Vol. DistribusiThe apparent volume…
KlirensIn patients with re…
Genetik -
Ranimustine DB13832
small molecule | CAS: 58994-96-0

Deskripsi belum tersedia.

Kategori:
Alkylating DrugsAmidesAntineoplastic Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ranirestat DB05327
small molecule | CAS: 147254-64-6

Ranirestat is a structurally novel and stereospecifically potent aldose reductase (AKR1B; EC 1.1.1.21) inhibitor, which contains a succinimide ring that undergoes ring-opening at physiological pH levels. It has been used in trials studying the treatment of M…

Kategori:
Aldehyde Reductase, antagonists & inhibitorsEnzyme Inhibitors
Target Protein:
Aldo-keto reductase family 1 member B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ranitidine Approved DB00863
small molecule | CAS: 66357-35-5

Ranitidine is a commonly used drug, classified as a histamine H2-receptor antagonist, and belongs to the same drug class as [cimetidine] and [famotidine]. This drug helps to prevent and treat gastric-acid associated conditions, including ulcers, because of it…

Kategori:
Acid ReducersAgents Causing Muscle ToxicityAlimentary Tract and Metabolism +29
Target Protein:
Histamine H2 receptorAcetylcholinesterase
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensRenal clearance is …
Genetik -
Ranolazine Approved DB00243
small molecule | CAS: 95635-55-5

Chronic angina is a common cardiovascular condition affecting millions worldwide and causes significant disability while interfering with daily activities.[A189234] Ranolazine is a well-tolerated piperazine derivative used for the management of this condition…

Kategori:
AcetamidesAntianginal AgentsBSEP/ABCB11 Substrates +26
Target Protein:
PlasminogenSodium channel proteinInward rectifier potassium channel +4
Waktu ParuhThe apparent termin…
Vol. DistribusiThe mean apparent v…
KlirensThe reported cleara…
Genetik -
Ranpirnase DB04950
biotech | CAS: 196488-72-9

Ranpirnase is a ribonuclease enzyme found in <i>Rana pipiens</i> oocytes. It is being studied in the treatment of cancer. It is manufactured by Alfacell Corporation. It is the first ribonuclease to enter cancer clinical trials.

Kategori:
Antineoplastic AgentsEgg ProteinsEnzyme Inhibitors +6
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2143578-32-7

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RAPA-201 DB18446
biotech

RAPA-201 is an autologous rapamycin-resistant T-cell therapy.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RAPA-501-Allo DB15890
biotech

RAPA-501-ALLO is composed of T-cells extracted from healthy volunteers; these cells are then reprogrammed _ex vivo_ in a process that involves de-differentiation and re-differentiation.[L16483]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rapacuronium Approved DB04834
small molecule | CAS: 465499-11-0

Rapacuronium was withdrawn in 2001 in many countries due to risk of fatal bronchospasm.

Kategori:
Agents producing tachycardiaAndrostanesAndrostanols +9
Target Protein:
Muscarinic acetylcholine receptor M2
Waktu Paruh141 minutes (mean)
Vol. Distribusi-
Klirens-
Genetik -
Rapastinel DB11801
small molecule | CAS: 117928-94-6

Rapastinel has been used in trials studying the treatment of Depressive Disorder, Major and Obsessive-Compulsive Disorder (OCD).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Raphanus sativus Approved DB10650
biotech

Radish allergenic extract is used in allergenic testing.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rasagiline Approved DB01367
small molecule | CAS: 136236-51-6

Rasagiline is an irreversible inhibitor of monoamine oxidase and is used as a monotherapy in early Parkinson's disease or as an adjunct therapy in more advanced cases.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAnti-Parkinson Drugs +19
Target Protein:
Amine oxidase [flavin-containing] BApoptosis regulator Bcl-2
Waktu ParuhRasagiline has a me…
Vol. Distribusi* 87 L
Klirens-
Genetik -
Rasburicase Approved DB00049
biotech | CAS: 134774-45-1

Rasburicase is a recombinant urate-oxidase enzyme produced by a genetically modified <i>Saccharomyces cerevisiae</i> strain. The cDNA coding for rasburicase was cloned from a strain of _Aspergillus flavus_.

Kategori:
Antigout PreparationsDetoxifying Agents for Antineoplastic TreatmentEnzymes +7
Target Protein:
Uric acid
Waktu Paruh18 hours
Vol. Distribusi* 110 to 127 mL/kg …
Klirens-
Genetik -
biotech | CAS: 1587257-96-2

Rasdegafusp alfa is under investigation in clinical trial NCT03206047 (Atezolizumab, Guadecitabine, and CDX-1401 Vaccine in Treating Patients With Recurrent Ovarian, Fallopian Tube, or Primary Peritoneal Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Raspberry Approved DB10636
biotech

Raspberry allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rattus norvegicus skin Approved DB10608
biotech

Rattus norvegicus skin or pelt is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Raubasine DB15949
small molecule | CAS: 483-04-5

Deskripsi belum tersedia.

Kategori:
AlkaloidsCardiovascular AgentsHeterocyclic Compounds, Fused-Ring +5
Target Protein:
Beta-1 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 8063-17-0

Rauwolfia (Rauwolfia serpentina), also spelled _ravolphia_, is a medicinal plant in the milkweed family. The root of the plant is ground into a powder or sold in tablets or capsules. It is a compound commonly used in Asian medicine, which includes traditional…

Kategori:
AlkaloidsAntiadrenergic Agents, Centrally ActingAntihypertensive Agents +6
Target Protein:
Synaptic vesicular amine transporter
Waktu ParuhAfter oral ingestio…
Vol. Distribusi-
KlirensHepatically and ren…
Genetik -
RAV12 DB05140
biotech

RAV12 is investigated for use/treatment in solid tumors. RAV12 is a solid. RAV12 is a chimeric antibody that recognizes RAAG12, an N-linked carbohydrate antigen found on gastric, colon, pancreatic, prostate, ovarian, breast, and kidney cancer cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ravagalimab DB16676
biotech | CAS: 2050816-56-1

Ravagalimab is under investigation in clinical trial NCT03695185 (A Study to Investigate How Well Ravagalimab (ABBV-323) Works and How Safe It Is in Participants With Moderate to Severe Ulcerative Colitis Who Failed Prior Therapy).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ravidasvir DB15652
small molecule | CAS: 1242087-93-9

Ravidasvir is under investigation in clinical trial NCT02961426 (Sofosbuvir Plus Ravidasvir for the Treatment of HCV Chronic Infection).

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Peptides, and Proteins +6
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ravoxertinib DB15281
small molecule | CAS: 1453848-26-4

Ravoxertinib is under investigation in clinical trial NCT01875705 (A Dose-Escalation Study of GDC-0994 in Patients With Locally Advanced or Metastatic Solid Tumors).

Kategori:
Antineoplastic AgentsEnzyme InhibitorsProtein Kinase Inhibitors +1
Target Protein:
Mitogen-activated protein kinase 3Mitogen-activated protein kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ravuconazole DB06440
small molecule | CAS: 182760-06-1

Deskripsi belum tersedia.

Kategori:
Antifungal AgentsAzole AntifungalsSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ravulizumab Approved DB11580
biotech | CAS: 1803171-55-2

Ravulizumab is a potent and selective complement 5 (C5) inhibitor. It is a humanized monoclonal IgG2/4 kappa antibody produced in Chinese hamster ovary (CHO) cells.[L39690] Ravulizumab was engineered from [eculizumab], another complement inhibitor, to increas…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
Complement C5
Waktu ParuhThe mean (%CV) term…
Vol. DistribusiThe mean (%CV) volu…
KlirensThe mean (%CV) clea…
Genetik -
Raxibacumab Approved DB08902
biotech | CAS: 565451-13-0

Raxibacumab is a human IgG1? monoclonal antibody that binds the protective antigen (PA) component of B. anthracis toxin. Raxibacumab has a molecular weight of approximately 146 kilodaltons. Raxibacumab is produced by recombinant DNA technology in a murine cel…

Kategori:
Amino Acids, Peptides, and ProteinsAnthrax Protective Antigen-directed AntibodyAnthrax Protective Antigen-directed Antibody Interactions +12
Target Protein:
Protective antigen
Waktu ParuhMean terminal elimi…
Vol. DistribusiSteady state volume…
KlirensClearance values we…
Genetik -
Raxtozinameran Approved DB18228
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Razupenem DB12587
small molecule | CAS: 426253-04-5

Razupenem has been used in trials studying the treatment of Skin Infections.

Kategori:
Amidesbeta-LactamsHeterocyclic Compounds, Fused-Ring +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Razuprotafib DB16353
small molecule | CAS: 1008510-37-9

Razuprotafib, also known as AKB-9778, is a small-molecule inhibitor restoring Tie2 activation by inhibiting VE-PTP.[L27171,L27176] In investigations against diabetes and COVID-19, razuprotafib is self-administered by patients through subcutaneous injection.

Kategori:
AcidsAcids, NoncarboxylicAmines +2
Target Protein:
Receptor-type tyrosine-protein phosphatase betaAngiopoietin-1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RB106 DB02669
small molecule

Deskripsi belum tersedia.

Target Protein:
Poly [ADP-ribose] polymerase 1ThermolysinThermolysin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RBIO-101 DB18425
biotech

RBIO-101 is a recombinant adeno-associated virus vector encoding human CYP4V2 protein.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RC118 DB18428
biotech

RC118 is an antibody-drug conjugate that consists of a recombinant humanized IgG1 anti-Claudin18.2 monoclonal antibody conjugated to MMAE.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RC88 DB18697
biotech

RC88 is an antibody-drug conjugate comprising a humanized anti-mesothelin monoclonal antibody conjugated to monomethyl auristatin E (MMAE).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RCT1100 DB18830
biotech

RCT1100 is an investigational mRNA-based therapeutic that aims to treat primary ciliary dyskinesia caused by pathogenic mutations in DNAI1.[L50788]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RDEA806 DB05228
small molecule

RDEA806 is a new HIV non-nucleoside reverse transcriptase inhibitor (NNRTI) with a high genetic barrier to resistance and a broad spectrum of activity.

Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RDP58 DB06566
small molecule

RDP58 (NH2-arg-norleucine (nle)-nle-arg-nle-nle-nle-gly-tyr-CONH2) (Sangstat Corp., Fremont, California) is a novel synthetic peptide that inhibits early signal transduction pathways for the expression of inflammatory cytokines.

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rebamipide Approved DB11656
small molecule | CAS: 90098-04-7

Rebamipide has been investigated for the treatment of Stomach Ulcer, Keratoconjunctivitis Sicca, and Gastric Adenoma and Early Gastric Cancer.

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids, Peptides, and Proteins +11
Target Protein:
fMet-Leu-Phe receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rebastinib DB13005
small molecule | CAS: 1020172-07-9

Rebastinib has been used in trials studying the treatment of Chronic Myeloid Leukemia. It is an inhibitor of Tie2 tyrosine kinase receptor and an antineoplastic agent.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Tyrosine-protein kinase ABL1Angiopoietin-1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rebaudioside A DB15136
small molecule | CAS: 58543-16-1

Rebaudioside A is under investigation in clinical trial NCT03510624 (Acute Effect of Rebaudioside A on Glucose Excursion During an Oral Glucose Tolerance Test in Type 2 Diabetes Mellitus).

Kategori:
AlkaloidsDiterpene AlkaloidsDiterpenes +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rebeccamycin DB14729
small molecule | CAS: 93908-02-2

Rebeccamycin is a weak topoisomerase I inhibitor isolated from _Nocardia sp_.

Kategori:
Heterocyclic Compounds, Fused-RingIndoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rebimastat DB06573
small molecule | CAS: 259188-38-0

Deskripsi belum tersedia.

Kategori:
Matrix Metalloproteinases
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1966978-67-5

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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