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17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
Referensi
17430 (100.0%)

Tipe Molekul

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Hasil Pencarian (17430)

Halaman 281 / 349
Quinbolone DB13484
small molecule | CAS: 2487-63-0

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAnabolic Agents for Systemic UseAnabolic Steroids +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quinestrol Approved DB04575
small molecule | CAS: 152-43-2

The 3-cyclopentyl ether of ethinyl estradiol.

Kategori:
Estradiol CongenersEstrogenic Steroids, AlkylatedEstrogens +11
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quinethazone Approved DB01325
small molecule | CAS: 73-49-4

Quinethazone, marketed as Hydromox, is a thiazide diuretic indicated for hypertension. Patients may experience adverse reactions such as dizziness, dry mouth, nausea, and hypokalemia.

Kategori:
AmidesCardiovascular AgentsDiuretics +10
Target Protein:
Solute carrier family 12 member 1Solute carrier family 12 member 2Solute carrier family 12 member 3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quinfamide DB12780
small molecule | CAS: 62265-68-3

Quinfamide has been used in trials studying the treatment of Amoebiasis and Helminthiasis.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quingestanol DB13685
small molecule | CAS: 10592-65-1

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 3000-39-3

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesFused-Ring CompoundsNorpregnanes +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quinidine Approved DB00908
small molecule | CAS: 56-54-2

Quinidine is a D-isomer of [quinine] present in the bark of the Cinchona tree and similar plant species. This alkaloid was first described in 1848 and has a long history as an antiarrhythmic medication.[A38016,A250050] Quinidine is considered the first antiar…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +81
Target Protein:
Sodium channel protein type 5 subunit alphaPotassium channel subfamily K member 1Potassium channel subfamily K member 6 +4
Waktu ParuhThe elimination hal…
Vol. DistribusiQuinidine has a vol…
KlirensThe clearance of qu…
Genetik -
Quinidine barbiturate Approved DB01346
small molecule

The administration of quinidine derivatives helps to observe various skin and mucosal reactions. A papulopurpuric eruption in a patient (without thrombopenia) can be developed who is taking quinidine phenylethyl barbiturate intermittently and at reintroducti…

Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit alpha-2Sodium channel protein type 5 subunit alpha +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quinine Approved DB00468
small molecule | CAS: 130-95-0

An alkaloid derived from the bark of the cinchona tree. It is used as an antimalarial drug, and is the active ingredient in extracts of the cinchona that have been used for that purpose since before 1633. Quinine is also a mild antipyretic and analgesic and h…

Kategori:
Agents that produce neuromuscular block (indirect)Agents that reduce seizure thresholdAlkaloids +57
Target Protein:
Fe(II)-protoporphyrin IXPlatelet glycoprotein IXIntermediate conductance calcium-activated potassium channel protein 4
Waktu ParuhApproximately 18 ho…
Vol. Distribusi* 1.43 ± 0.18 L/kg …
Klirens* 0.17 L/h/kg [heal…
Genetik -
Quinisocaine DB13683
small molecule | CAS: 86-80-6

Deskripsi belum tersedia.

Kategori:
AnestheticsAnesthetics for Topical UseAnesthetics, Local +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quinoline DB18050
small molecule | CAS: 91-22-5

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 8004-92-0

Deskripsi belum tersedia.

Kategori:
Agents causing angioedemaAgents that produce hypertensionHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quinolinic Acid DB01796
small molecule | CAS: 89-00-9

A metabolite of tryptophan with a possible role in neurodegenerative disorders. Elevated CSF levels of quinolinic acid are correlated with the severity of neuropsychological deficits in patients who have AIDS. [PubChem]

Kategori:
PyridinesQuinolinic Acids
Target Protein:
Nicotinate-nucleotide pyrophosphorylase [carboxylating]Nicotinate-nucleotide pyrophosphorylase [carboxylating]
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 79647-29-3

Deskripsi belum tersedia.

Target Protein:
Phenylalanine-4-hydroxylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quinupramine Approved DB13246
small molecule | CAS: 31721-17-2

Quinupramine has been approved in France under the brand name Kinupril, as an antidepressant [A175003].

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quinupristin Approved DB01369
small molecule | CAS: 120138-50-3

Quinupristin/dalfopristin is a combination of two antibiotics used to treat infections by staphylococci and by vancomycin-resistant Enterococcus faecium. Dalfopristin inhibits the early phase of protein synthesis in the bacterial ribosome and quinupristin inh…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +9
Target Protein:
23S ribosomal RNA50S ribosomal protein L1050S ribosomal protein L22
Waktu Paruh3.1 hours
Vol. Distribusi-
Klirens-
Genetik -
Quisinostat DB12985
small molecule | CAS: 875320-29-9

Quisinostat has been used in trials studying the treatment of Lymphoma, Neoplasms, Myelodysplastic Syndromes, and Advanced or Refractory Leukemia.

Kategori:
AminesHydroxy AcidsHydroxylamines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quisovalimab DB16482
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quisqualic acid DB02999
small molecule | CAS: 52809-07-1

Quisqualic acid is an agonist at two subsets of excitatory amino acid receptors, ionotropic receptors that directly control membrane channels and metabotropic receptors that indirectly mediate calcium mobilization from intracellular stores. The compound is ob…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsExcitatory Amino Acid Agents +4
Target Protein:
Metabotropic glutamate receptor 1Glutamate receptor ionotropic, kainate 1Metabotropic glutamate receptor 2 +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quizartinib Approved DB12874
small molecule | CAS: 950769-58-1

Quizartinib is an oral and potent fms-like tyrosine kinase 3 (FLT3) inhibitor and it is the first drug developed specifically targeting FLT3, as other agents with FLT3 inhibition activities were investigated with other targets in mind.[A260641] Additionally, …

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +17
Target Protein:
Receptor-type tyrosine-protein kinase FLT3
Waktu ParuhThe mean (SD) effec…
Vol. DistribusiVolume of distribut…
KlirensTotal body clearanc…
Genetik -
QXL138AM DB18552
biotech

QXL138AM is a masked immunocytokine (MIC) comprised of an anti-CD138 immunoglobulin G1 antibody fused to interferon alpha 2a. It binds the CD138 protein on the surface of the tumour cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 37571-78-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-1487 DB06518
small molecule | CAS: 449811-92-1

Deskripsi belum tersedia.

Kategori:
Mitogen-Activated Protein Kinase 14, antagonists & inhibitorsPyridines
Target Protein:
Mitogen-activated protein kinase 14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Stromelysin-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-30490 DB09179
small molecule | CAS: 60618-49-7

R-30490 is an opioid related to carfentanil used as an animal tranquilizer. It was first synthesized by Janssen Pharmaceutica as part of a structure-activity relationship study of fentanly and its derivatives. R-30490 was found to be the most selective agonis…

Kategori:
Piperidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-306465 DB12382
small molecule | CAS: 604769-01-9

R306465 has been used in trials studying the treatment of Neoplasms.

Kategori:
AminesAntineoplastic AgentsEnzyme Inhibitors +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-348 DB06321
small molecule | CAS: 916742-11-5

Deskripsi belum tersedia.

Target Protein:
Tyrosine-protein kinase JAK3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-82913 DB08598
small molecule | CAS: 126347-69-1

Deskripsi belum tersedia.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +7
Target Protein:
Gag-Pol polyproteinGag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-851 DB05747
small molecule

R-851 is part of the family of immune response modifier (IRM) and it acts in a novel way to stimulate the human body's immnune system to attack virus-infected cells and tumor cells. It is expected to be topical treatment for cervical displasia and cervical hi…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 14047-28-0

Deskripsi belum tersedia.

Target Protein:
Thymidine kinase, cytosolicThymidine kinaseThymidine kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-95845 DB07327
small molecule | CAS: 163435-77-6

R-95845 is an inhibitor of HIV-1 reverse transcriptase.

Kategori:
AcetatesAcids, AcyclicAmides +1
Target Protein:
Gag-Pol polyproteinGag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-azabisabolene DB03985
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R048-8071 DB02016
small molecule | CAS: 161582-11-2

Deskripsi belum tersedia.

Target Protein:
Lanosterol synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R107474 DB06553
small molecule | CAS: 214548-46-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R112 DB06252
small molecule | CAS: 575474-82-7

R112 is an investigational compound developed to treat Allergic Rhinitis. It's mechanism of action is to inhibit SYK kinase.

Target Protein:
Tyrosine-protein kinase SYK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R1204 DB05118
small molecule

R1204 is G-protein-coupled receptor modulator. It is developed for the treatment of depression.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R1295 DB05122
small molecule

R1295 is an integrin antagonist currently in clinical trials for the treatment of rheumatoid arthritis. Integrins are associated to the pathology seen in some of the autoimmune diseases such as rheumatoid arthritis.

Target Protein:
Integrin alpha-4Integrin beta-4Integrin beta-7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R1626 DB05060
small molecule

R1626 is one of a new class of hepatitis C therapies called polymerase inhibitors. It achieves significant reductions in viral load in chronic hepatitis C patients infected with the difficult to treat genotype 1 virus. R1626 is very effective in inhibiting vi…

Kategori:
CarbohydratesGlycosidesNucleic Acids, Nucleotides, and Nucleosides
Target Protein:
RNA-dependent RNA-polymerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R343 DB06316
small molecule | CAS: 575484-78-5

R343, was investigated in clinical trial NCT01591044 to evaluate its safety and efficacy in patients with mild to moderate asthma.

Target Protein:
Tyrosine-protein kinase SYK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R3R01 DB18078
small molecule

R3R01 is an investigational lipid-modifying drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R411 DB05468
small molecule

R411 is a non-steroid oral medicine for the treatment of asthma. It is not immunosuppressive, but blocks the activation and recruitment of cells involved in respiratory inflammation. It is a dual-acting competitive integrin antagonist (as compared to previous…

Target Protein:
Integrin alpha-4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R450 DB05469
small molecule

R450 is an alpha 1 antagonist that acts to tighten the muscle tone in the bladder. It is being considered for treatment of stress-related urinary incontinence. Phase IIa data for the drug show it reduced the number of incontinent episodes compared to placebo …

Target Protein:
Alpha-1A adrenergic receptorAlpha-1B adrenergic receptorAlpha-1D adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R673 DB05466
small molecule

R673 is a novel NK1 antagonist that penetrates the blood-brain barrier, has excellent safety and tolerability and shows low P450-based drug interaction potential. The phase II program for treatment of depression and anxiety is ongoing in the US and EU.It is n…

Target Protein:
Substance-P receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R906289 DB19126
small molecule | CAS: 2602614-45-7

R906289 is under investigation in clinical trial NCT05308264 (Study of R289 in Participants With Lower-risk Myelodysplastic Syndromes (LR MDS)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
rAAV1-CB-hAAT DB18724
biotech

rAAV1-CB-hAAT is a recombinant adeno-associated virus alpha 1-antitrypsin vector.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
rAAV9-hNAGLU DB18415
biotech

rAAV9-hNAGLU consists of a recombinant AAV9 expressing human alpha-N-acetylglucosaminidase.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
rAAV9-rsATP7A DB17664
biotech

A recombinant adeno-associated viral vector gene therapy under investigation for the treatment of Menkes disease.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rabacfosadine DB12762
small molecule | CAS: 859209-74-8

Rabacfosadine has been used in trials studying the treatment of Multiple Myeloma, Non-Hodgkin's Lymphoma, and Chronic Lymphocytic Leukemia.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsHeterocyclic Compounds, Fused-Ring
Target Protein:
DNA polymerase catalytic subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rabbit Approved DB10415
biotech

Rabbit allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 14001–14050 dari 17430
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