Hasil Filter

2279

Total database: 17430
Struktur (SMILES)
866 (38.0%)
Target
1100 (48.3%)
Genomik
31 (1.4%)
Referensi
2279 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (2279)

Halaman 28 / 46
Methapyrilene DB04819
small molecule | CAS: 91-80-5

Methapyrilene, formerly marketed in many drug products, was shown to be a potent carcinogen. Manufacturers voluntarily withdrew methapyriline drug products from the market in May and June 1979.

Kategori:
AminesAminopyridinesAnti-Allergic Agents +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methaqualone DB04833
small molecule | CAS: 72-44-6

Methaqualone is a sedative-hypnotic drug that is similar in effect to barbiturates, a general central nervous system depressant. The sedative-hypnotic activity was first noted by Indian researchers in the 1950s and in 1962 methaqualone itself was patented in …

Kategori:
Central Nervous System AgentsCentral Nervous System DepressantsCytochrome P-450 CYP3A Substrates +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methenamine Approved DB06799
small molecule | CAS: 100-97-0

Methenamine is a heterocyclic organic compound with a cage-like structure similar to adamantane. In salt form it is used for the treatment of urinary tract infection (Example: methenamine hippurate which is the hippuric acid salt of methenamine).

Kategori:
Acids, CarbocyclicAmidesAmines +14
Waktu ParuhElimination half-li…
Vol. Distribusi-
Klirens70-90% of a single…
Genetik -
Methimazole Approved DB00763
small molecule | CAS: 60-56-0

Methimazole is a thionamide antithyroid agent that inhibits the synthesis of thyroid hormones.[A184559,A184733,A184694] It was first introduced as an antithyroid agent in 1949[A184502] and is now commonly used in the management of hyperthyroidism, particularl…

Kategori:
Antithyroid agentsCytochrome P-450 CYP1A2 InhibitorsCytochrome P-450 CYP1A2 Inhibitors (strength unknown) +30
Target Protein:
Thyroid peroxidase
Waktu ParuhFollowing a single …
Vol. DistribusiThe apparent volume…
KlirensFollowing a single …
Genetik -
Methionine Approved DB00134
small molecule | CAS: 63-68-3

A sulfur containing essential amino acid that is important in many body functions. It is a chelating agent for heavy metals.

Kategori:
Amino AcidsAmino Acids, EssentialAmino Acids, Neutral +7
Target Protein:
Methionine synthase reductaseMethionine synthaseMethionine aminopeptidase 2 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 25281-48-5

Deskripsi belum tersedia.

Target Protein:
Mannose-binding protein C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methyl salicylate Approved DB09543
small molecule | CAS: 119-36-8

Methyl salicylate (oil of wintergreen or wintergreen oil) is an organic ester naturally produced by many species of plants, particularly wintergreens. The compound was first extracted and isolated from plant species Gaultheria procumbens in 1843. It can be ma…

Kategori:
Acids, CarbocyclicAnalgesicsAntirheumatic Agents +16
Target Protein:
Transient receptor potential cation channel subfamily A member 1
Waktu ParuhThe plasma half-lif…
Vol. DistribusiAfter absorption, m…
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Hemagglutinin-neuraminidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Endoplasmic reticulum mannosyl-oligosaccharide 1,2-alpha-mannosidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methylchloroisothiazolinone Approved DB14197
small molecule | CAS: 26172-55-4

Methylchloroisothiazolinone (MCI) is an isothiazolinone commonly used as a preservative with antibacterial and antifungal properties. It is found within many commercially available cosmetics, lotions, and makeup removers. It is also a known dermatological sen…

Kategori:
Anti-Infective AgentsCell-mediated ImmunityCompounds used in a research, industrial, or household setting +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methyldopa Approved DB00968
small molecule | CAS: 555-30-6

Methyldopa, or ?-methyldopa, is a centrally acting sympatholytic agent and an antihypertensive agent.[A231784] It is an analog of DOPA (3,4?hydroxyphenylanine), and it is a prodrug, meaning that the drug requires biotransformation to an active metabolite for …

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +28
Target Protein:
D(2) dopamine receptorAromatic-L-amino-acid decarboxylaseAlpha-2A adrenergic receptor
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe apparent volume…
KlirensThe renal clearance…
Genetik -
Metreleptin Approved DB09046
biotech | CAS: 186018-45-1

Metreleptin, a recombinant analog of the human hormone leptin, is an orphan drug used to treat complications of leptin deficiency in people with lipodystrophy. Lipodystrophies include a range of disorders characterized by the reduction, absence, or altered di…

Kategori:
AdipokinesAlimentary Tract and MetabolismAmino Acids and Derivatives +11
Target Protein:
Leptin receptor
Waktu ParuhFollowing subcutane…
Vol. DistribusiFollowing intraveno…
KlirensThe clearance of me…
Genetik -
Metronidazole Approved DB00916
small molecule | CAS: 443-48-1

Metronidazole is a commonly used antibiotic, belonging to the nitroimidazole class of antibiotics.[L3754] It is frequently used to treat gastrointestinal infections as well as trichomoniasis and giardiasis, and amebiasis which are parasitic infections.[A18103…

Kategori:
Agents that reduce seizure thresholdAlimentary Tract and MetabolismAnti-Bacterial Agents +38
Target Protein:
Oxygen-insensitive NADPH nitroreductaseAnaerobic bacterial DNAProtozoal DNA
Waktu ParuhThe elimination hal…
Vol. DistribusiMetronidazole is wi…
KlirensDose adjustments ma…
Genetik -
Mevonlerbart DB19416
biotech | CAS: 2453195-99-6

Mevonlerbart is under investigation in clinical trial NCT06602726 (A Study to Demonstrate How Well REGN1908-1909 Works in Reducing Ocular Allergy Signs and Symptoms in Adult Participants With Cat Allergy).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mezagitamab DB16370
biotech | CAS: 2227490-52-8

Mezagitamab is under investigation in clinical trial NCT04278924 (Study to Evaluate Safety, Tolerability, and Efficacy of TAK-079 in Participants With Persistent/chronic Primary Immune Thrombocytopenia).

Target Protein:
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MG98 DB06544
biotech

MG98, a second-generation antisense oligodeoxynucleotide inhibitor of human DNMT1, was investigated in the completed clinical trial NCT00003890 for treating patients with advanced solid tumors.

Target Protein:
DNA (cytosine-5)-methyltransferase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Microcrystalline cellulose Approved DB14158
small molecule | CAS: 9004-34-6

A polysaccharide with glucose units linked as in CELLOBIOSE. It is the chief constituent of plant fibers, cotton being the purest natural form of the substance. As a raw material, it forms the basis for many derivatives used in chromatography, ion exchange ma…

Kategori:
BiopolymersCarbohydratesCellulose +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Miglustat Approved DB00419
small molecule | CAS: 72599-27-0

Miglustat, commonly marketed under the trade name Zavesca, is a drug used to treat Gaucher disease. It inhibits the enzyme glucosylceramide synthase, an essential enzyme for the synthesis of most glycosphingolipids. It is only used for patients who cannot be …

Kategori:
Alimentary Tract and MetabolismAlkaloidsAnti-HIV Agents +14
Target Protein:
Ceramide glucosyltransferase
Waktu ParuhThe effective half-…
Vol. Distribusi-
Klirens-
Genetik -
Milnacipran Approved DB04896
small molecule | CAS: 92623-85-3

Milnacipran is a selective serotonin and norepinephrine reuptake inhibitor (SNRI) and like many agents in this category was originally developed for and continues to be approved and indicated for the treatment of depression [F3928, F3934, A175786, A175951]. F…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAgents producing tachycardia +30
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporterNMDA receptor
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe mean volume of …
KlirensThe total plasma cl…
Genetik -
Miltefosine Approved DB09031
small molecule | CAS: 58066-85-6

Miltefosine is a broad spectrum antimicrobial, anti-leishmanial, phospholipid drug that was originally developed in the 1980s as an anti-cancer agent. It is currently the only recognized oral agent used to treat visceral, cutaneous, and mucosal forms of leish…

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAminesAnti-Infective Agents +9
Target Protein:
Phospholipase A2ATP-dependent translocase ABCB1
Waktu ParuhThe primary elimina…
Vol. DistribusiRadioactivity studi…
KlirensPlasma clearance is…
Genetik -
Mineral oil Approved DB11057
small molecule | CAS: 8042-47-5

Mineral oil, or paraffin oil, is a mixture of higher alkanes from a mineral source, such as petroleum. Petroleum mineral oil is manufactured from crude oils by vacuum distillation to produce several distillates and a residual oil that are then further refined…

Kategori:
Alimentary Tract and MetabolismBasic Ointments and ProtectantsDermatologicals +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mirikizumab Approved DB14910
biotech | CAS: 1884201-71-1

Mirikizumab is a monoclonal antibody developed by Eli Lilly intended to treat ulcerative colitis. It inhibits the actions of interleukin-23 (IL-23), a pro-inflammatory cytokine that activates pathways contributing to the development of inflammatory diseases.[…

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAnti-Inflammatory Agents +16
Target Protein:
Interleukin-23 subunit alpha
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Mirococept DB06492
biotech | CAS: 507453-82-9

Mirococept (APT070) is a complement inhibitor currently under development for treatment of rheumatoid arthritis and I/RI. It is a truncated form of the human Complement Receptor 1 (CR1) linked to a unique Prodaptin™ construct that regulates the over-productio…

Target Protein:
Complement C3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mirtazapine Approved DB00370
small molecule | CAS: 85650-52-8

Mirtazapine is a tetracyclic _piperazino-azepine_ antidepressant agent that was initially approved for the treatment of major depressive disorder (MDD) in the Netherlands in 1994.[A177946] This drug was first manufactured by Organon Inc., and received FDA app…

Kategori:
Adrenergic AgentsAdrenergic alpha-2 Receptor AntagonistsAdrenergic alpha-Antagonists +38
Target Protein:
5-hydroxytryptamine receptor 2A5HT3 serotonin receptorAlpha-2A adrenergic receptor +4
Waktu Paruh20-40 hours [FDA la…
Vol. DistribusiThe volume of distr…
KlirensTotal body clearanc…
Genetik -
Mirvetuximab DB16235
biotech | CAS: 1453084-36-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Misoprostol Approved DB00929
small molecule | CAS: 59122-46-2

Misoprostol is a prostaglandin analog used to reduce the risk of NSAID related ulcers, manage miscarriages, prevent post partum hemorrhage, and also for first trimester abortions.[L7616,L7619,A181589,A181583,A181697] The stimulation of prostaglandin receptors…

Kategori:
Abortifacient AgentsAbortifacient Agents, NonsteroidalAlimentary Tract and Metabolism +24
Target Protein:
Prostacyclin receptorProstaglandin E2 receptor EP3 subtypeProstaglandin E2 receptor EP2 subtype +2
Waktu ParuhThe half life of an…
Vol. DistribusiData regarding the …
KlirensBecause of the rapi…
Genetik -
Mitazalimab DB15225
biotech | CAS: 2055640-86-1

Mitazalimab is under investigation in clinical trial NCT02379741 (ADC-1013 First-in-Human Study).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mitotane Approved DB00648
small molecule | CAS: 53-19-0

Mitotane is an adrenolytic isomer of the insecticide dichlorodiphenyldichloroethane (DDD) - itself a metabolite of dichlorodiphenyltrichloroethane (DDT) - that inhibits cells of the adrenal cortex and their production of hormones. It has been in use since 195…

Kategori:
Adrenal Cytotoxic AgentsAntineoplastic AgentsAntineoplastic Agents, Hormonal +15
Target Protein:
Cytochrome P450 11B1, mitochondrialEstrogen receptorProgesterone receptor +2
Waktu ParuhThe plasma terminal…
Vol. DistribusiMitotane is extensi…
Klirens-
Genetik -
Mitsugumin-53 DB16969
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0482 DB17453
biotech

MK-0482 is a novel humanized IgG4 monoclonal antibody targeting the immunoglobulin-like transcript (ILT) 3.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-2225 DB18240
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-4721 DB05933
biotech

MK-4721 is a fully human monoclonal antibody directed to Agensys’ proprietary target Prostate Stem Cell Antigen (PSCA), an antigen expressed at significant levels on tumor cells from the majority of patients with all stages of prostate, pancreatic and bladder…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Prostate stem cell antigen
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MM-093 DB05512
biotech

MM-093 is a recombinant version of human alpha-fetoprotein (hAFP), an immunomodulatory serum protein normally produced at very high levels by the fetus and present in low levels in the blood of adults and children. Research on AFP suggests that it may play a …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mobocertinib Approved DB16390
small molecule | CAS: 1847461-43-1

Mobocertinib is a kinase inhibitor targeted against human epidermal growth factor receptor (EGFR). It is used specifically in the treatment of non-small cell lung cancer (NSCLC) caused by exon 20 insertion mutations in the _EGFR_ gene,[L38368] which are typic…

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +15
Target Protein:
Epidermal growth factor receptor
Waktu ParuhAt steady-state, th…
Vol. DistribusiThe mean apparent v…
KlirensAt steady-state, th…
Genetik -
Moclobemide Approved DB01171
small molecule | CAS: 71320-77-9

A reversible monoamine oxidase inhibitor (MAOI) selective for isoform A (RIMA) used to treat major depressive disorder. Most meta-analyses and most studies indicate that in the acute management of depression, moclobemide is more efficacious than placebo medic…

Kategori:
Acids, CarbocyclicAgents that produce hypertensionAgents that reduce seizure threshold +28
Target Protein:
Amine oxidase [flavin-containing] AMonoamine oxidaseAmine oxidase [flavin-containing] B
Waktu Paruh1-2 hours (4 hours …
Vol. Distribusi1-1.5 L/Kg [L1350]
KlirensClearance of 30-78 …
Genetik -
Mogamulizumab Approved DB12498
biotech | CAS: 1159266-37-1

Mogamulizumab is a humanized monoclonal antibody (mAb) directed against CC chemokine receptor 4 (CCR4) for the treatment of Mycosis Fungoides (MF) and Sézary Syndrome (SS), the most common subtypes of cutaneous T-cell lymphoma. Cutaneous T-cell lymphomas occu…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
C-C chemokine receptor type 4
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe central volume …
KlirensClearance is 12 mL/…
Genetik -
Molnupiravir DB15661
small molecule | CAS: 2349386-89-4

Molnupiravir (EIDD-2801, MK-4482) is the isopropylester prodrug of [N4-hydroxycytidine].[A193014,A193026] With improved oral bioavailability in non-human primates, it is hydrolyzed _in vivo_, and distributes into tissues where it becomes the active 5’-triphos…

Kategori:
AminesAnti-Infective AgentsAntiinfectives for Systemic Use +13
Waktu ParuhThe half life of th…
Vol. Distribusi-
Klirens-
Genetik -
Momelotinib Approved DB11763
small molecule | CAS: 1056634-68-4

Momelotinib is a Janus Kinase 1 (JAK1) and 2 (JAK2) inhibitor. It is a competitive inhibitor of JAK ATP binding.[A261566] First approved by the FDA on September 15, 2023,[L48206] momelotinib is used to treat myelofibrosis.[L48186] Myelofibrosis (MF) is a grou…

Kategori:
Acids, CarbocyclicAmidesAntineoplastic Agents +24
Target Protein:
Tyrosine-protein kinase JAK1Tyrosine-protein kinase JAK2Tyrosine-protein kinase JAK3 +3
Waktu ParuhThe elimination hal…
Vol. DistribusiThe mean (%CV) appa…
KlirensThe mean (%CV) clea…
Genetik -
Mometasone furoate Approved DB14512
small molecule | CAS: 83919-23-7

Mometasone furoate is a corticosteroid drug that can be used for the treatment of asthma, rhinitis, and certain skin conditions[FDA Label][F4292,F4295]. It has a glucocorticoid receptor binding affinity 22 times stronger than [dexamethasone] and higher than m…

Kategori:
Adrenal Cortex HormonesAdrenalsAdrenergics, Inhalants +28
Target Protein:
Glucocorticoid receptorProgesterone receptor
Waktu ParuhThe terminal half l…
Vol. DistribusiSteady state volume…
KlirensThe clearance rate …
Genetik -
Monobenzone Approved DB00600
small molecule | CAS: 103-16-2

Monobenzone is the monobenzyl ether of hydroquinone used medically for depigmentation. Monobenzone occurs as a white, almost tasteless crystalline powder, soluble in alcohol and practically insoluble in water. It exerts a depigmenting effect on skin of mammal…

Kategori:
alpha-Galactosidase, antagonists & inhibitorsBenzene DerivativesDepigmenting Agents +3
Target Protein:
Tyrosinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MOR-22 DB17790
biotech

MOR-22, a Natural human lymphoblastoid interferon-alpha, is currently being investigated to treat papillomavirus warts in the oral cavity of HIV-positive patients.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MORAb-066 DB17347
biotech

MORAb-066 is a humanized antibody directed against tissue factor (TF). It is being investigated in pancreatic cancer.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Moroctocog alfa Approved DB13999
biotech | CAS: 284036-24-4

Moroctocog alfa, also known as BDDrFVIII (B domain deleted recombinant factor VIII), is a recombinant DNA-based drug with functional characteristics comparable to those of endogenous coagulation Factor VIII, the essential human blood clotting protein that is …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +5
Target Protein:
Coagulation factor XCoagulation factor IXvon Willebrand factor +8
Waktu ParuhMean terminal elimi…
Vol. DistribusiMean steady-state v…
KlirensMean clearance = 4.…
Genetik -
Mosunetuzumab Approved DB15434
biotech | CAS: 1905409-39-3

Mosunetuzumab is a humanized anti-CD20/CD3 bispecific antibody.[L42230] It can recognize and bind two different targets simultaneously, CD20 on cancer B-cells and CD3 on T-cells, allowing it to redirect T-cell cytotoxic activity to cancer cells.[A249320] The …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +13
Target Protein:
B-lymphocyte antigen CD20T-cell surface glycoprotein CD3 epsilon chain
Waktu ParuhMosunetuzumab has a…
Vol. DistribusiThe estimated centr…
KlirensThe mean steady-sta…
Genetik -
MRG-003 DB17407
biotech

MRG-003 is a recombinant humanized anti-human epidermal growth factor receptor monoclonal antibody conjugated to monomethyl auristatin E.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
mRNA-3745 DB18554
biotech

mRNA-3745 is a lipid nanoparticle (LNP) encapsulated with nucleoside-modified, codon-optimized mRNAs encoding human glucose 6-phosphatase (G6Pase).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MRT5005 DB18260
biotech

MRT5005 is a human cystic fibrosis transmembrane conductance regulator (hCFTR) messenger RNA (mRNA) complexed with branched polyethyleneimine (bPEI).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MRx-4DP0004 DB15751
biotech

MRx-4DP0004 is a lyophilised formulation of the Bifidobacterium breve strain of commensal bacteria. It is a live biotherapeutic derived from the microbiota of a healthy human infant.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MT-0169 DB17430
biotech

MT-0169 is a usion protein comprised of an enzymatically active Shiga-like toxin-I A1 subunit fused to a human single chain variable fragment with affinity for human CD38 cell surface protein.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 1351–1400 dari 2279
Sebelumnya Halaman 28 / 46 Berikutnya