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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
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14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 278 / 282
Zanolimumab DB17376
biotech | CAS: 652153-01-0

Zanolimumab is a fully human monoclonal antibody directed against CD4.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
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Zansecimab DB16389
biotech | CAS: 2415205-37-5

Zansecimab is under investigation in clinical trial NCT04342897 (A Study of LY3127804 in Participants With COVID-19).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +9
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Zanubrutinib Approved DB15035
small molecule | CAS: 1691249-45-2

Zanubrutinib is a novel Bruton's tyrosine kinase (BTK) inhibitor used for the treatment of adult patients with mantle cell lymphoma (MCL) who have received at least one prior therapy.[L10163] Mantle cell lymphoma is an aggressive mature B-cell non-Hodgkin lym…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBruton's tyrosine kinase (BTK) inhibitors +19
Target Protein:
Tyrosine-protein kinase BTKEpidermal growth factor receptorReceptor tyrosine-protein kinase erbB-2 +12
Waktu ParuhFollowing administr…
Vol. DistribusiThe geometric mean …
KlirensThe mean (%CV) appa…
Genetik -
Zanzalintinib DB17525
small molecule | CAS: 2367004-54-2

Deskripsi belum tersedia.

Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
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Zapnometinib DB18244
small molecule | CAS: 303175-44-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAminesAminobenzoates +4
Waktu Paruh-
Vol. Distribusi-
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Zardaverine DB02918
small molecule | CAS: 101975-10-4

Deskripsi belum tersedia.

Kategori:
Anti-Asthmatic AgentsAutonomic AgentsBronchodilator Agents +4
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4D
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Zasocitinib DB19278
small molecule | CAS: 2272904-53-5

Deskripsi belum tersedia.

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Zastumotide DB14926
biotech | CAS: 949885-73-8

Zastumotide is a recombinant MAGE-A3 Antigen-Specific Cancer Immunotherapeutic (MAGE-A3 ASCI) also known as astuprotimut-R. It is under investigation in clinical trial NCT00257738 (0804 GCC: MAGE-A3/HPV 16 Vaccine for Squamous Cell Carcinoma of the Head and N…

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Zatolmilast DB14790
small molecule | CAS: 1606974-33-7

BPN-14770 is under investigation in clinical trial NCT02840279 (A Multiple Ascending Dose Study of BPN14770 in Healthy Young and Elderly Male or Female Subjects).

Kategori:
Acids, AcyclicEnzyme InhibitorsFatty Acids +5
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4D
Waktu Paruh-
Vol. Distribusi-
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Zavegepant Approved DB15688
small molecule | CAS: 1337918-83-8

Zavegepant (BHV-3500) is a calcitonin gene-related peptide (CGRP) receptor antagonist.[L45505] CGRP is released from sensory nerves and acts as a strong vasodilator, and thanks to these properties, it is involved in pain pathways. CGRP receptors are expressed…

Kategori:
Antimigraine PreparationsCalcitonin Gene-Related Peptide (CGRP) AntagonistsCalcitonin Gene-Related Peptide Receptor Antagonists +14
Target Protein:
Calcitonin gene-related peptide type 1 receptor
Waktu ParuhFollowing a 10 mg d…
Vol. DistribusiIntranasal zavegepa…
KlirensIntranasal zavegepa…
Genetik -
ZD-6126 DB11872
small molecule | CAS: 219923-05-4

ZD6126 has been used in trials studying the treatment of Kidney Neoplasms, Colorectal Neoplasms, Metastases, Neoplasm, and Carcinoma, Renal Cell.

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ZD4407 DB06539
small molecule | CAS: 166882-70-8

The drug ZD4407, an antiasthmatic developed by AstraZeneca, functions as a 5-lipoxygenase inhibitor. It entered Phase 1 clinical trials for chronic obstructive pulmonary disease (COPD) in the United Kingdom but was discontinued during this phase in March 2003

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Zeatin DB11337
small molecule | CAS: 1637-39-4

An aminopurine factor in plant extracts that induces cell division. (Grant & Hackh's Chemical Dict, 5th ed)

Kategori:
CytokininsGrowth SubstancesHeterocyclic Compounds, Fused-Ring +2
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Zebularine DB03068
small molecule | CAS: 3690-10-6

A chemically stable, cytidine analog that displays anti-tumor properties. It acts as a transition state analog inhibitor of cytidine deaminase by binding to the active site as covalent hydrates. Also shown to inhibit DNA methylation and tumor growth both in v…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosidesPyrimidine Nucleosides +2
Target Protein:
Cytidine deaminase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ZED-1227 DB19208
small molecule | CAS: 1542132-88-6

ZED-1227 is under investigation in clinical trial NCT05305599 (Different Doses of ZED1227 vs. Placebo in NAFLD).

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Zelasudil DB19315
small molecule | CAS: 2365193-22-0

Deskripsi belum tersedia.

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Zelavespib DB12638
small molecule | CAS: 873436-91-0

Zelavespib (PU-H71) has been used in trials studying the treatment of LYMPHOMA, Solid Tumors, Metastatic Solid Tumor, and Myeloproliferative Neoplasms (MPN).

Kategori:
Antineoplastic AgentsDioxolesHeterocyclic Compounds, Fused-Ring
Target Protein:
Heat shock protein HSP 90-beta
Waktu Paruh-
Vol. Distribusi-
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Zelpultide alfa DB18587
biotech | CAS: 2245003-06-7

Zelpultide alfa is a recombinant human surfactant protein D.

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Zelquistinel DB19336
small molecule | CAS: 2151842-64-5

Zelquistinel is under investigation in clinical trial NCT06547489 (GATE-251 or Placebo for the Reduction of Symptoms of Major Depressive Disorder).

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Zeluvalimab DB18868
biotech | CAS: 2315361-37-4

Zeluvalimab is under investigation in clinical trial NCT04631601 (Safety and Efficacy of Therapies for Metastatic Castration-resistant Prostate Cancer (Mcrpc)).

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Zemirciclib DB18823
small molecule | CAS: 2057509-72-3

Deskripsi belum tersedia.

Target Protein:
Cyclin-dependent kinase 9
Waktu Paruh-
Vol. Distribusi-
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ZEN-012 DB06042
small molecule

ZEN-012 is a novel small molecule and the first anti-cancer drug in development involving two mechanisms of action: tubulin and topoisomerase II inhibition. ZEN-012 also expresses additional modes of action such as pro-apoptotic and anti-angiogenic properties…

Target Protein:
Tubulin beta chainTubulin beta-1 chainTubulin beta-3 chain +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Zenarestat DB02132
small molecule | CAS: 112733-06-9

Deskripsi belum tersedia.

Kategori:
Aldehyde Reductase, antagonists & inhibitorsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring
Target Protein:
Aldo-keto reductase family 1 member B1
Waktu Paruh-
Vol. Distribusi-
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Zenocutuzumab Approved DB15559
biotech | CAS: 1969309-56-5

Zenocutuzumab is under investigation in clinical trial NCT03321981 (MCLA-128 With Trastuzumab/chemotherapy in HER2+ and With Endocrine Therapy in ER+ and Low HER2 Breast Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
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Zeranol DB11478
small molecule | CAS: 26538-44-3

Zeranol is a non-steroidal estrogen agonist. It is a mycotoxin, derived from fungi in the Fusarium family, and may be found as a contaminant in fungus-infected crops. It is 3-4x more potent as an estrogen agonist than the related compound zearalenone.

Kategori:
Benzene DerivativesEstrogensEstrogens, Non-Steroidal +6
Target Protein:
Estrogen receptorSex hormone-binding globulin
Waktu Paruh-
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Zetomipzomib DB16070
small molecule | CAS: 1629677-75-3

Zetomipzomib is under investigation in clinical trial NCT04033926 (A Phase 2 Study of KZR-616 to Evaluate Safety and Efficacy in Patients With Active Polymyositis or Dermatomyositis).

Kategori:
Oxazines
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biotech

Deskripsi belum tersedia.

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Zibotentan DB06629
small molecule | CAS: 186497-07-4

Deskripsi belum tersedia.

Target Protein:
Endothelin-1 receptor
Waktu Paruh-
Vol. Distribusi-
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Ziconotide Approved DB06283
biotech | CAS: 107452-89-1

Ziconotide (also known as SNX-111) is a neurotoxic peptide derived from the cone snail _Conus magus_ comprising 25 amino acids with three disulphide bonds.[A202835, L13389] Other such peptides, collectively termed conotoxins, exist, and some have shown effica…

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAntiarrhythmic agents +22
Target Protein:
Voltage-dependent N-type calcium channel subunit alpha-1BVoltage-dependent P/Q-type calcium channel subunit alpha-1A
Waktu ParuhIn patients adminis…
Vol. DistribusiIn patients adminis…
KlirensZiconotide CSF clea…
Genetik -
Zicronapine DB12188
small molecule | CAS: 170381-16-5

Zicronapine has been used in trials studying the treatment of Schizophrenia.

Target Protein:
D(2) dopamine receptorD(1A) dopamine receptor5-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zidebactam DB13090
small molecule | CAS: 1436861-97-0

Zidebactam is under investigation in clinical trial NCT02674347 (MAD Study to Evaluate the Safety, Tolerability and Pharmacokinetics of Intravenous Zidebactam in Healthy Adults).

Kategori:
Aza CompoundsCycloparaffins
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 106060-89-3

Deskripsi belum tersedia.

Kategori:
DeoxyribonucleosidesDeoxyribonucleotidesDideoxynucleosides +6
Target Protein:
Nucleoside diphosphate kinase A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 29706-85-2

Deskripsi belum tersedia.

Kategori:
DeoxyribonucleosidesDeoxyribonucleotidesDideoxynucleosides +6
Target Protein:
Thymidylate kinaseThymidylate kinase
Waktu Paruh-
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Zifibancimig DB19332
biotech | CAS: 2517939-46-5

Zifibancimig is under investigation in clinical trial NCT04567303, focusing on participants with neovascular age-related macular degeneration.

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Ziftomenib DB17171
small molecule | CAS: 2134675-36-6

Deskripsi belum tersedia.

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Zigakibart DB18892
biotech | CAS: 2642175-46-8

Zigakibart is under investigation in clinical trial NCT05852938 (A Study of BION-1301 in Adults With Iga Nephropathy).

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biotech | CAS: 2220231-04-7

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
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Zilebesiran DB18929
biotech | CAS: 2380166-33-4

Zilebesiran is under investigation in clinical trial NCT06272487 (Zilebesiran as Add-on Therapy in Patients With High Cardiovascular Risk and Hypertension Not Adequately Controlled by Standard of Care Antihypertensive Medications (KARDIA-3)).

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Zileuton Approved DB00744
small molecule | CAS: 111406-87-2

Leukotrienes are substances that induce numerous biological effects including augmentation of neutrophil and eosinophil migration, neutrophil and monocyte aggregation, leukocyte adhesion, increased capillary permeability, and smooth muscle contraction. These …

Kategori:
Agents to Treat Airway DiseaseAmidesAnalgesics +19
Target Protein:
Polyunsaturated fatty acid 5-lipoxygenase
Waktu Paruh2.5 hours
Vol. Distribusi* 1.2 L/kg
Klirens* Apparent oral cl=…
Genetik -
Zilganersen DB18161
biotech | CAS: 2305355-56-8

Deskripsi belum tersedia.

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Zilovertamab DB18403
biotech | CAS: 2485779-13-1

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Genetik -
biotech | CAS: 2376463-48-6

Zilovertamab vedotin is an Antibody-drug conjugate (ADC) comprising an anti-ROR1 monoclonal antibody (UC-961), a proteolytically cleavable maleimidocaproyl-valine-citrulline-para-aminobenzoate linker (mc-vc-PAB), and a monomethyl auristatin E (MMAE) cytotoxin.

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Zilpaterol DB11479
small molecule | CAS: 119520-05-7

Zilpaterol is a ?2 adrenergic agonist sold under the trade name, Zilmax, produced by Intervet, a subsidiary of Merck & Co. Zilpaterol is typically fed to cattle in the last three to six weeks of life with a brief washout period to clear the drug from the tiss…

Kategori:
Heterocyclic Compounds, Fused-RingOrganosilicon CompoundsReceptors, Adrenergic, beta
Waktu Paruh-
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Ziltivekimab DB18836
biotech | CAS: 2226654-05-1

Ziltivekimab is under investigation in clinical trial NCT06200207 (A Research Study Looking Into How Ziltivekimab Works Compared to Placebo in Participants With Heart Failure and Inflammation).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Zilucoplan Approved DB15636
small molecule | CAS: 1841136-73-9

Zilucoplan is a 15 amino-acid, synthetic macrocyclic peptide. It is a complement inhibitor that works to prevent the activation of C5, which is a complement protein involved in the innate immune system to initiate inflammatory responses.[A261841] On October 1…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating AgentsBlood Proteins +5
Target Protein:
Complement C5
Waktu ParuhThe mean plasma ter…
Vol. DistribusiThe mean volume of …
KlirensNo information is a…
Genetik -
Zilurgisertib DB18152
small molecule | CAS: 2173389-57-4

Deskripsi belum tersedia.

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Zimberelimab DB17505
biotech | CAS: 2259860-24-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zimelidine Approved DB04832
small molecule | CAS: 56775-88-3

Zimelidine has been banned worldwide due to serious, sometimes fatal, cases of central and/or peripheral neuropathy known as Guillain-Barré syndrome and due to a peculiar hypersensitivity reaction involving many organs including skin exanthema, flu-like sympt…

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsCytochrome P-450 CYP3A Inhibitors +16
Target Protein:
Sodium-dependent serotonin transporterAmine oxidase [flavin-containing] BAmine oxidase [flavin-containing] A
Waktu Paruh8.4 +/- 2.0 hours f…
Vol. Distribusi-
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Zinc Approved DB01593
small molecule | CAS: 7440-66-6

A metallic element of atomic number 30 and atomic weight 65.38. It is a necessary trace element in the diet, forming an essential part of many enzymes, and playing an important role in protein synthesis and in cell division. Zinc deficiency is associated with…

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseDiet, Food, and NutritionElements +12
Target Protein:
B1 bradykinin receptorMethylated-DNA--protein-cysteine methyltransferaseFructose-bisphosphate aldolase A +121
Waktu ParuhThe half-life of zi…
Vol. DistribusiA pharmacokinetic s…
KlirensIn one study of hea…
Genetik -
Zinc ascorbate Approved DB14485
small molecule | CAS: 331242-75-2

Deskripsi belum tersedia.

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseMetal cationsMetal divalent cations +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 13851–13900 dari 14063
Sebelumnya Halaman 278 / 282 Berikutnya