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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 278 / 321
Sitaxentan Approved DB06268
small molecule | CAS: 184036-34-8

Sitaxentan was marketed under the trade name Thelin for the treatment of pulmonary arterial hypertension (PAH) by Encysive Pharmaceuticals until Pfizer purchased Encysive in February 2008. In 2010, Pfizer voluntarily removed sitaxentan from the market over co…

Kategori:
Antihypertensive AgentsAntihypertensives for Pulmonary Arterial HypertensionCytochrome P-450 CYP2C19 Inhibitors +12
Target Protein:
Endothelin-1 receptorEndothelin receptor type B
Waktu Paruh10 hours
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biotech | CAS: 898830-54-1

Sitimagene ceradenovec is a novel gene-based product for the treatment of patients with operable high grade glioma, a type of malignant brain tumour, given in addition to standard surgery and radiotherapy/chemotherapy. It is being developed by Ark Therapeutic…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsAntineoplastic cell and gene therapy +6
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Sitravatinib DB15036
small molecule | CAS: 1123837-84-2

Sitravatinib is under investigation in clinical trial NCT03680521 (Neoadjuvant Sitravatinib in Combination With Nivolumab in Patients With Clear Cell Renal Cell Carcinoma).

Kategori:
AmidesAminesAniline Compounds +3
Target Protein:
Hepatocyte growth factor receptorVascular endothelial growth factor receptor 3Vascular endothelial growth factor receptor 2 +1
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Sivelestat DB12863
small molecule | CAS: 127373-66-4

Sivelestat has been used in trials studying the treatment of Acute Lung Injury and Respiratory Distress Syndrome, Adult.

Kategori:
AmidesAmino AcidsAmino Acids, Peptides, and Proteins +5
Target Protein:
Neutrophil elastaseChymotrypsin-like elastase family member 1
Waktu Paruh-
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Sivifene DB05686
small molecule | CAS: 2675-35-6

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesHydrazines
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Sivopixant DB18816
small molecule | CAS: 2414285-40-6

Deskripsi belum tersedia.

Kategori:
Amines
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Sizofiran DB13128
small molecule | CAS: 9050-67-3

A beta-D-glucan obtained from the Aphyllophoral fungus Schizophyllum commune. It is used as an immunoadjuvant in the treatment of neoplasms, especially tumors found in the stomach. Sizofiran has been used in trials studying the treatment of Cervical Cancer.

Kategori:
Adjuvants, ImmunologicAntineoplastic AgentsAntineoplastic Agents, Phytogenic +6
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SJ-733 DB12659
small molecule | CAS: 1424799-20-1

SJ-733 has been used in trials studying Malaria.

Kategori:
Heterocyclic Compounds, Fused-Ring
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SJG-136 DB11965
small molecule | CAS: 232931-57-6

SJG-136 has been used in trials studying the treatment of Recurrent Fallopian Tube Cancer, Secondary Acute Myeloid Leukemia, de Novo Myelodysplastic Syndromes, Recurrent Ovarian Epithelial Cancer, and Secondary Myelodysplastic Syndromes, among others.

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
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Skf 107457 DB04191
small molecule | CAS: 144285-77-8

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
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SKF-91488 DB07106
small molecule | CAS: 68643-23-2

Deskripsi belum tersedia.

Kategori:
AmidesHistamine AgentsHistamine Agonists +4
Target Protein:
Histamine N-methyltransferase
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small molecule | CAS: 162849-90-3

SKF-96365 is a receptor-mediated calcium entry (RMCE) inhibitor structurally different from other calcium antagonists.[A253132]

Kategori:
Antiarrhythmic agentsAntiplatelet agentsCalcium Channel Blockers +4
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biotech

Skin-derived ABCB5-positive Mesenchymal Stem cells are under investigation in clinical trial NCT04971161 (Allogeneic Abcb5-positive Dermal Mesenchymal Stromal Cells for Treatment of CVU (Phase Iib)).

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SKL-27969 DB18168
small molecule | CAS: 2634762-24-4

Deskripsi belum tersedia.

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SLC-0111 DB18815
small molecule | CAS: 178606-66-1

Deskripsi belum tersedia.

Kategori:
AmidesAntineoplastic AgentsBenzene Derivatives +2
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SLC-391 DB18814
small molecule | CAS: 1783825-18-2

Deskripsi belum tersedia.

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SLN124 DB18646
biotech

SLN124 is a synthetic double-stranded siRNA oligonucleotide directed against TMPRSS6 mRNA and covalently linked to a ligand containing 3 N-acetylgalactosamine residues.

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SLN500 DB18636
biotech

SLN500 is a synthetic double-strand small interfering ribonucleic acid (siRNA) oligonucleotide drug directed against C3 messenger RNA

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SLV-334 DB15356
small molecule | CAS: 182821-33-6

SLV-334 is under investigation in clinical trial NCT00735085 (A Phase 2a Dose Escalation Study With SLV334 in Patients With Traumatic Brain Injury.).

Target Protein:
Neprilysin
Waktu Paruh-
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SLx-2101 DB05615
small molecule

SLx-2101 is an oral, long-acting PDE5 inhibitor developed by Surface Logix Inc. to treat Hypertension.

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SLx-4090 DB05678
small molecule | CAS: 913541-47-6

SLx-4090 is a microsomal triglyceride transfer protein (MTTP) inhibitor potentially for the treatment of type 2 diabetes. [A33218]

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Target Protein:
Microsomal triglyceride transfer protein large subunit
Waktu Paruh-
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SM-1997 DB18670
biotech

SM-1997 is a protein-free solution derived from calf's blood comprising electrolytes, trace minerals, amino acids, peptides, nucleosides, and nucleotides.[A261816] It is under investigation for the treatment of cutaneous sulfur mustard-induced injury.

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SM-337 DB17112
small molecule | CAS: 1071992-61-4

Deskripsi belum tersedia.

Target Protein:
E3 ubiquitin-protein ligase XIAP
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Genetik -
biotech

The New York City Board of Health strain of _Vaccinia_ is a viral strain used as a component of some smallpox vaccinations.[L12747] ACAM2000, a percutaneously administered smallpox vaccine that was approved by the FDA in 2007, contains live antigens of this s…

Kategori:
Actively Acquired ImmunityBiological ProductsComplex Mixtures +4
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biotech

Deskripsi belum tersedia.

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SMART101 DB18370
biotech

SMART101 is an investigational cell therapy comprising human allogeneic CD34-CD7+ T cell progenitors that were cultured ex vivo.

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Smilagenin DB05450
small molecule | CAS: 126-18-1

Smilagenin is a novel non-peptide, orally bioavailable neurotrophic factor inducer that readily reverses free radical neurotoxicity produced by 1-ethyl-4- phenylpyridium (MPP+) in dopaminergic neurones and reverses the decrease of neuronal growth factors and …

Kategori:
CholestanesDrugs, Chinese HerbalFused-Ring Compounds +4
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SN-38 DB05482
small molecule | CAS: 86639-52-3

7-ethyl-10-hydroxycamptothecin (SN 38) is a liposomal formulation of the active metabolite of Irinotecan [DB00762], a chemotherapeutic pro-drug approved for the treatment of advanced colorectal cancer. SN 38 has been used in trials studying the treatment of …

Kategori:
AlkaloidsAntineoplastic AgentsCytochrome P-450 CYP3A Inhibitors +9
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
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small molecule | CAS: 59734-15-5

Deskripsi belum tersedia.

Kategori:
GlycerophosphatesGlycerophospholipidsLipids +3
Target Protein:
Annexin A5
Waktu Paruh-
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Genetik -
small molecule | CAS: 17989-41-2

Deskripsi belum tersedia.

Target Protein:
Fructose-bisphosphate aldolase BPyridoxine 5'-phosphate synthaseTriosephosphate isomerase +1
Waktu Paruh-
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Snail, unspecified Approved DB14245
biotech

Snail, unspecified is an animal extract used in some OTC (over-the-counter) products. It is not an approved drug.

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SNP-ACTH (1-39) DB18544
biotech

SNP-ACTH (1-39) is a synthetic porcine Corticotropin (ACTH)

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SNS-032 DB05969
small molecule | CAS: 345627-80-7

Deskripsi belum tersedia.

Kategori:
Sulfur Compounds
Target Protein:
Cyclin-dependent kinase 9Cyclin-dependent kinase 2Cyclin-dependent kinase 7 +1
Waktu Paruh-
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SNS-314 DB06134
small molecule | CAS: 1057249-41-8

SNS-314 is a potent and selective inhibitor of Aurora kinases A, B, and C. Proliferating cells treated with SNS-314 bypass the mitotic spindle checkpoint and fail to undergo cytokinesis, leading to multiple rounds of endoreduplication and eventually cell deat…

Kategori:
AmidesBenzene DerivativesProtein Kinase Inhibitors +1
Target Protein:
Aurora kinase BAurora kinase CAurora kinase A
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SNS01-T DB17302
biotech

SNS01-T is a gene therapy nanoparticle. It is composed of three components: a B cell-specific plasmid expressing eIF5AK50R; an siRNA that targets the native eIF5A that promotes growth/anti-apoptosis of cancer cells; and polyethylenimine.[A254706]

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small molecule | CAS: 1226795-18-1

Snubh-nm-333 F-18 is under investigation in clinical trial NCT02149017 (Phase 1 and Phase 2 Clinical Trials of SNUBH-NM-333(18F)).

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SNX-2112 DB17055
small molecule | CAS: 908112-43-6

SNX-2112 is a heat shock protein 90 (Hsp90) inhibitor.[A253137]

Kategori:
Heterocyclic Compounds, Fused-RingHSP90 Heat-Shock Proteins, antagonists & inhibitors
Target Protein:
Heat shock protein HSP 90-alpha
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SNX-5422 DB06070
small molecule | CAS: 908115-27-5

SNX-5422 is a synthetic, novel, small molecule Hsp90 Inhibitor. As an oral formulation that demonstrates strong efficacy and tolerability, SNX-5422 is positioned as a breakthrough therapy with broad applicability across a wide range of cancers.

Kategori:
Acids, CarbocyclicAmidesAmino Acids +5
Target Protein:
Heat shock protein HSP 90-alphaHeat shock protein HSP 90-beta
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SO-101 DB05345
small molecule

SO-101(Silenor) is a low-dose oral tablet formulation of doxepin hydrochloride that is patent protected for its use in insomnia. Doxepin has been prescribed for more than 40 years for the treatment of depression and anxiety at dosages typically ranging from 7…

Target Protein:
Histamine H1 receptor
Waktu Paruh-
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Sobetirome DB07425
small molecule | CAS: 211110-63-3

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicBenzene DerivativesFatty Acids +2
Target Protein:
Muscarinic acetylcholine receptor M1Thyroid hormone receptor, alpha isoform 1 variantThyroid hormone receptor beta
Waktu Paruh-
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SOBI-003 DB15451
biotech

SOBI-003 is a chemically modified variant of a recombinant human sulfamidase. It is under investigation in clinical trial NCT03811028 (A Study to Assess the Safety, Tolerability, and Efficacy of Long-term SOBI003 Treatment in Pediatric MPS IIIA Patients).

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Soblidotin DB12677
small molecule | CAS: 149606-27-9

Soblidotin has been used in trials studying the treatment of Sarcoma, Lung Cancer, and Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsPeptides
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Sobrerol DB13315
small molecule | CAS: 42370-41-2

Deskripsi belum tersedia.

Kategori:
Cough and Cold PreparationsExpectorantsRespiratory System Agents
Waktu Paruh-
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Socazolimab DB18845
biotech | CAS: 2305043-30-3

Socazolimab is under investigation in clinical trial NCT04878016 (A Study of Carboplatin Plus Etoposide With or Without ZKAB001 (Anti-pd-l1 Antibody) in Patients With ES-SCLC).

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Sodelglitazar DB16332
small molecule | CAS: 447406-78-2

Sodelglitazar is under investigation in clinical trial NCT00196989 (Study in People With Type 2 Diabetes).

Target Protein:
Peroxisome proliferator-activated receptor deltaPeroxisome proliferator-activated receptor gammaPeroxisome proliferator-activated receptor alpha
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small molecule | CAS: 200880-41-7

Deskripsi belum tersedia.

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Sodium acetate Approved DB09395
small molecule | CAS: 127-09-3

Sodium Acetate is chemically designated CH3COONa, a hygroscopic powder very soluble in water. Sodium acetate could be used as additives in food, industry, concrete manufacture, heating pads and in buffer solutions. Medically, sodium acetate is important compo…

Kategori:
AcetatesAcids, AcyclicBlood and Blood Forming Organs +5
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small molecule | CAS: 1344-00-9

Deskripsi belum tersedia.

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Sodium apolate DB13477
small molecule | CAS: 25053-27-4

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicAlkenes +12
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Sodium arsenite DB18508
small molecule | CAS: 7784-46-5

Deskripsi belum tersedia.

Kategori:
AnionsArsenicalsElectrolytes +3
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